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3253

Total database: 17430
Struktur (SMILES)
2451 (75.3%)
Target
1833 (56.3%)
Genomik
35 (1.1%)
Referensi
3253 (100.0%)

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Hasil Pencarian (3253)

Halaman 65 / 66
WP-1066 DB12679
small molecule | CAS: 857064-38-1

WP1066 has been used in trials studying the treatment of Melanoma, Brain Cancer, Solid Tumors, and Central Nervous System Neoplasms.

Kategori:
Benzene DerivativesBenzylidene CompoundsHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Signal transducer and activator of transcription 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
WP-1122 DB17192
small molecule

WP-1122 is a prodrug of 2-deoxy-D-glucose (2-DG). It was granted FDA orphan designation for the treatment of glioblastoma multiforme.[L47361]

Kategori:
CarbohydratesDeoxy Sugars
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
WRR-112 DB03691
small molecule

Deskripsi belum tersedia.

Target Protein:
CruzipainCathepsin F
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
WT-1 122 long DB17353
biotech | CAS: 952720-86-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
WZB-117 DB16764
small molecule | CAS: 1223397-11-2

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Xamoterol Approved DB13781
small molecule | CAS: 81801-12-9

Xamoterol is a ?1-adrenoceptor partial agonist that has shown to improve systolic and diastolic function in studies with heart failure patients. It modulates the sympathetic control of the heart but has no agonist action on ?2-adrenoceptors.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-1 Receptor Agonists +14
Target Protein:
Beta-3 adrenergic receptorBeta-1 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Xanthan gum Approved DB11253
small molecule | CAS: 11138-66-2

Xanthan gum is a polysaccharide gum derived from* Xanthomonas campestris* by a pure-culture fermentation process and purified by recovery with isopropyl alcohol. The major constituents include D-glucose, D-mannose, and D-glucuronic acid. Xanthan gum is a dire…

Kategori:
AntigensAntigens, BacterialBiological Factors +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Xempritolimod DB19412
biotech | CAS: 2639319-18-7

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
XEN-2174 DB05012
small molecule | CAS: 701909-57-1

XEN-2174 is a synthetic drug modeled on a peptide from the venom of a cone shell found on Australia's Great Barrier Reef. XEN-2174 represents a new class of molecules, called the chi conopeptides that selectively inhibit the Norepinephrine Transporter (NET). …

Kategori:
Amino Acids, Peptides, and Proteins
Target Protein:
Sodium-dependent noradrenaline transporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Xenon Xe-127 Approved DB09461
small molecule | CAS: 13994-19-9

Deskripsi belum tersedia.

Kategori:
ElementsGasesInhalation Diagnostic Agent +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Xenon Xe-129 Approved DB17386
small molecule | CAS: 13965-99-6

Hyperpolarized Xenon-129 (Xe-129) is a contrast agent used in the lung's clinical magnetic resonance imaging (MRI). Lung MRIs are challenging due to the low proton density of this tissue, as well as the presence of artifacts due to respiration and cardiovascu…

Kategori:
Contrast MediaDiagnostic Uses of ChemicalsHyperpolarized Contrast Agent +3
Waktu ParuhXenon-129 in a 75% …
Vol. DistribusiXenon is readily di…
KlirensNot available.
Genetik -
XL-888 DB12981
small molecule | CAS: 1149705-71-4

XL888 has been used in trials studying the treatment of Cancer and Melanoma.

Kategori:
Acids, CarbocyclicAza CompoundsHSP90 Heat-Shock Proteins, antagonists & inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
XL820 DB05146
small molecule | CAS: 1123889-88-2

XL820 is investigated for use/treatment in solid tumors. XL820 is a solid. The proteins that XL820 inhibit include platelet-derived growth factor receptor beta (PDGFR), mast/stem cell growth factor receptor KIT, vascular endothelial growth factor receptor 2, …

Target Protein:
Vascular endothelial growth factor receptor 2Mast/stem cell growth factor receptor KitPlatelet-derived growth factor receptor alpha +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
XL999 DB05014
small molecule | CAS: 921206-68-0

XL999 has the potential to provide benefit to patients with lung cancer and acute myelogenous leukemia. XL999 is a new chemical entity that inhibits a spectrum of receptor tyrosine kinases (RTKs) with growth promoting and angiogenic properties, including FGFR…

Target Protein:
Fibroblast growth factor receptor 3Fibroblast growth factor receptor 1Vascular endothelial growth factor receptor 2 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
XP12B DB04928
small molecule

XP12B is being developed by Xanodyne Pharmaceuticals for the treatment of menorrhagia (heavy menstrual bleeding). It was granted Fast Track status for this indication by the FDA in November 2004.

Waktu Paruh-
Vol. Distribusi-
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XP21279 DB06319
small molecule

XP21279 is a prodrug of [Levodopa], a dopamine precursor used in the management of Parkinson's disease. XP21279 was under investigation in clinical trial NCT00914602 (An Exploratory Study of XP21279 (With Lodosyn®) and Sinemet® in Parkinson's Disease Subjects…

Target Protein:
Aromatic-L-amino-acid decarboxylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
YA-101 DB18121
small molecule | CAS: 151602-49-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Z-160 DB12743
small molecule | CAS: 41332-24-5

Z160 has been used in trials studying the treatment of Postherpetic Neuralgia and Lumbosacral Radiculopathy.

Kategori:
Antiarrhythmic agentsBenzene DerivativesCalcium Channel Blockers +3
Target Protein:
Voltage-dependent calcium channel subunit alpha-2/delta-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zabofloxacin DB12479
small molecule | CAS: 219680-11-2

Zabofloxacin has been used in trials studying the treatment of Community Acquired Pneumonia and Chronic Obstructive Pulmonary Disease.

Kategori:
4-QuinolonesHeterocyclic Compounds, Fused-RingQuinolines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zalutumumab DB12202
biotech | CAS: 667901-13-5

Zalutumumab is a fully human IgG1 monoclonal antibody designed to bind with selectivity to the epidermal growth factor receptor (EGFR). Zalutumumab has been investigated for the treatment of Squamous Cell Cancer and Head and Neck Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Target Protein:
Epidermal growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zalypsis DB12454
small molecule | CAS: 308359-57-1

Zalypsis has been used in trials studying the treatment of Lymphoma, Solid Tumors, Ewing's Sarcoma, Endometrial Cancer, and Uterine Cervical Cancer, among others.

Kategori:
AlkaloidsHeterocyclic Compounds, Fused-RingIsoquinolines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zamicastat DB12389
small molecule | CAS: 1080028-80-3

Zamicastat has been used in trials studying the treatment of Hypertension and Chronic Heart Failure.

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingPyrans
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zansecimab DB16389
biotech | CAS: 2415205-37-5

Zansecimab is under investigation in clinical trial NCT04342897 (A Study of LY3127804 in Participants With COVID-19).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zanubrutinib Approved DB15035
small molecule | CAS: 1691249-45-2

Zanubrutinib is a novel Bruton's tyrosine kinase (BTK) inhibitor used for the treatment of adult patients with mantle cell lymphoma (MCL) who have received at least one prior therapy.[L10163] Mantle cell lymphoma is an aggressive mature B-cell non-Hodgkin lym…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBruton's tyrosine kinase (BTK) inhibitors +19
Target Protein:
Tyrosine-protein kinase BTKEpidermal growth factor receptorReceptor tyrosine-protein kinase erbB-2 +12
Waktu ParuhFollowing administr…
Vol. DistribusiThe geometric mean …
KlirensThe mean (%CV) appa…
Genetik -
ZD-6126 DB11872
small molecule | CAS: 219923-05-4

ZD6126 has been used in trials studying the treatment of Kidney Neoplasms, Colorectal Neoplasms, Metastases, Neoplasm, and Carcinoma, Renal Cell.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ZED-1227 DB19208
small molecule | CAS: 1542132-88-6

ZED-1227 is under investigation in clinical trial NCT05305599 (Different Doses of ZED1227 vs. Placebo in NAFLD).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Zelavespib DB12638
small molecule | CAS: 873436-91-0

Zelavespib (PU-H71) has been used in trials studying the treatment of LYMPHOMA, Solid Tumors, Metastatic Solid Tumor, and Myeloproliferative Neoplasms (MPN).

Kategori:
Antineoplastic AgentsDioxolesHeterocyclic Compounds, Fused-Ring
Target Protein:
Heat shock protein HSP 90-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ZEN-012 DB06042
small molecule

ZEN-012 is a novel small molecule and the first anti-cancer drug in development involving two mechanisms of action: tubulin and topoisomerase II inhibition. ZEN-012 also expresses additional modes of action such as pro-apoptotic and anti-angiogenic properties…

Target Protein:
Tubulin beta chainTubulin beta-1 chainTubulin beta-3 chain +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zenarestat DB02132
small molecule | CAS: 112733-06-9

Deskripsi belum tersedia.

Kategori:
Aldehyde Reductase, antagonists & inhibitorsEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring
Target Protein:
Aldo-keto reductase family 1 member B1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zenocutuzumab Approved DB15559
biotech | CAS: 1969309-56-5

Zenocutuzumab is under investigation in clinical trial NCT03321981 (MCLA-128 With Trastuzumab/chemotherapy in HER2+ and With Endocrine Therapy in ER+ and Low HER2 Breast Cancer).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zicronapine DB12188
small molecule | CAS: 170381-16-5

Zicronapine has been used in trials studying the treatment of Schizophrenia.

Target Protein:
D(2) dopamine receptorD(1A) dopamine receptor5-hydroxytryptamine receptor 2A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zimberelimab DB17505
biotech | CAS: 2259860-24-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zinc ascorbate Approved DB14485
small molecule | CAS: 331242-75-2

Deskripsi belum tersedia.

Kategori:
Agents for Treatment of Hemorrhoids and Anal Fissures for Topical UseMetal cationsMetal divalent cations +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zinc gluconate Approved DB11248
small molecule | CAS: 4468-02-4

Zinc gluconate is a zinc salt of gluconic acid comprised of two gluconic acid molecules for each zinc cation (2+). Zinc gluconate is a generally recognized as safe (GRAS) substance by FDA [L2081]. It is available as a trace mineral supplement and over the cou…

Kategori:
Acids, AcyclicAgents for Treatment of Hemorrhoids and Anal Fissures for Topical UseAlimentary Tract and Metabolism +8
Waktu Paruh280 days [L2091]
Vol. DistribusiStored primarily in…
KlirensPlease refer to Dru…
Genetik -
small molecule | CAS: 14354-67-7

Deskripsi belum tersedia.

Kategori:
Biological FactorsCoordination ComplexesHeterocyclic Compounds, Fused-Ring +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zinc phenolsulfonate Approved DB15793
small molecule | CAS: 127-82-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Zinc sulfate is a common zinc supplement in parenteral nutrition.[A216916,L12888]

Kategori:
Agents for Treatment of Hemorrhoids and Anal Fissures for Topical UseMetal cationsMetal divalent cations +2
Target Protein:
B1 bradykinin receptorMethylated-DNA--protein-cysteine methyltransferaseFructose-bisphosphate aldolase A +94
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zingerone DB15589
small molecule | CAS: 122-48-5

Zingerone is a pungent component of ginger.

Kategori:
Benzene DerivativesCatecholsEthers +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zk-806450 DB02112
small molecule

Deskripsi belum tersedia.

Target Protein:
Serine protease 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zoledronic acid Approved DB00399
small molecule | CAS: 118072-93-8

Zoledronic acid, or CGP 42'446,[A203120] is a third generation, nitrogen containing bisphosphonate similar to [ibandronic acid], [minodronic acid], and [risedronic acid].[A203111] Zoledronic acid is used to treat and prevent multiple forms of osteoporosis, hy…

Kategori:
BisphosphonatesBone Density Conservation AgentsDrugs Affecting Bone Structure and Mineralization +5
Target Protein:
Geranylgeranyl pyrophosphate synthaseHydroxylapatiteFarnesyl pyrophosphate synthase
Waktu ParuhZoledronic acid has…
Vol. Distribusi-
KlirensZoledronic acid has…
Genetik -
Zoliflodacin DB12817
small molecule | CAS: 1620458-09-4

Zoliflodacin has been used in trials studying the basic science and treatment of Gonorrhoea.

Kategori:
Antineoplastic AgentsEnzyme InhibitorsOxazines +5
Target Protein:
DNA gyrase subunit ADNA gyrase subunit B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zolimidine DB13593
small molecule | CAS: 1222-57-7

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismDrugs for Acid Related DisordersDrugs for Peptic Ulcer and Gastro-Oesophageal Reflux Disease (Gord)
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zolmitriptan Approved DB00315
small molecule | CAS: 139264-17-8

Zolmitriptan is a member of the triptan class of 5-hydroxytryptamine(5-HT)<sub>1B/1D/(1F)</sub> receptor agonists used to treat acute migraine.[A462, L12978] [Sumatriptan] was the first triptan to be developed, but had poor oral bioavailability and lipophilic…

Kategori:
Agents that produce hypertensionAminesAnalgesics +24
Target Protein:
5-hydroxytryptamine receptor 1B5-hydroxytryptamine receptor 1D5-hydroxytryptamine receptor 1F +5
Gen Terkait:
GNB3
Waktu ParuhZolmitriptan has a …
Vol. DistribusiZolmitriptan has a …
KlirensZolmitriptan has a …
Genetik 1 Varian
small molecule | CAS: 139570-93-7

Zoptarelin doxorubicin has been used in trials studying the treatment of Breast Cancer, Ovarian Cancer, Prostate Cancer, Endometrial Cancer, and Urothelial Carcinoma, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAnthracyclinesCarbohydrates +12
Target Protein:
Gonadotropin-releasing hormone receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zorevunersen DB16912
biotech | CAS: 2415330-04-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zotiraciclib DB16656
small molecule | CAS: 1204918-72-8

Zotiraciclib is under investigation in clinical trial NCT02942264 (Zotiraciclib (TG02) Plus Dose-dense or Metronomic Temozolomide Followed by Randomized Phase II Trial of Zotiraciclib (TG02) Plus Temozolomide Versus Temozolomide Alone in Adults With Recurrent…

Kategori:
Cyclin-Dependent Kinases, antagonists & inhibitorsHeterocyclic Compounds, Fused-Ring
Target Protein:
Cyclin-dependent kinase 2Cyclin-dependent kinase 9Tyrosine-protein kinase Fyn +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zotizalkib DB19238
small molecule | CAS: 2648641-36-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ZSTK-474 DB12904
small molecule | CAS: 475110-96-4

ZSTK474 has been used in trials studying the treatment of Neoplasms.

Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zucapsaicin Approved DB09120
small molecule | CAS: 25775-90-0

Zucapsaicin, the cis-isomer of capsaicin, is a topical analgesic used to treat osteoarthritis of the knee and other neuropathic pain. It is a modulator of transient receptor potential cation channel subfamily V member 1 (TRPV-1), also known as the vanilloid o…

Kategori:
AlkaloidsAlkenesAlkynes +25
Target Protein:
Transient receptor potential cation channel subfamily V member 1
Waktu ParuhIn rats, the elimin…
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 29584-22-3

Zuretinol acetate has been used in trials studying the treatment of Impaired Dark Adaptation, RP (Retinitis Pigmentosa), Retinitis Pigmentosa (RP), and LCA (Leber Congenital Amaurosis).

Kategori:
Adjuvants, ImmunologicAlkenesAnticarcinogenic Agents +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 3201–3250 dari 3253
Sebelumnya Halaman 65 / 66 Berikutnya