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3253

Total database: 17430
Struktur (SMILES)
2451 (75.3%)
Target
1833 (56.3%)
Genomik
35 (1.1%)
Referensi
3253 (100.0%)

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Halaman 64 / 66
Velusetrag DB12702
small molecule | CAS: 866933-46-2

Velusetrag has been used in trials studying the treatment of Gastroparesis and Alzheimer's Disease. It is a highly selective serotonin receptor agonist effective in patients with chronic constipation. It is being developed by Theravance. Velusetrag was discov…

Kategori:
Aza Compounds
Target Protein:
5-hydroxytryptamine receptor 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vemircopan DB18012
small molecule | CAS: 2086178-00-7

Deskripsi belum tersedia.

Target Protein:
Complement factor D
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vemurafenib Approved DB08881
small molecule | CAS: 918504-65-1

Vemurafenib is a competitive kinase inhibitor with activity against BRAF kinase with mutations like V600E.[A31269] It exerts its function by binding to the ATP-binding domain of the mutant BRAF.[A31270] Vemurafenib was co-developed by Roche and Plexxikon and …

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +41
Target Protein:
Serine/threonine-protein kinase B-raf
Waktu ParuhThe elimination hal…
Vol. DistribusiThe estimation of t…
KlirensThe total body clea…
Genetik -
Venetoclax Approved DB11581
small molecule | CAS: 1257044-40-8

Venetoclax is a BCL-2 inhibitor that was initially approved by the FDA in April 2016 [FDA label]. Proteins in the B cell CLL/lymphoma 2 (BCL-2) family are important regulators of the apoptotic (programmed cell death) process [A18565], [A18566]. Venetoclax is…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +19
Target Protein:
Apoptosis regulator Bcl-2
Waktu ParuhThe half-life of ve…
Vol. DistribusiThe population esti…
KlirensMainly hepatic [FDA…
Genetik -
Vepafestinib DB18779
small molecule | CAS: 2129515-96-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Verdinexor DB12207
small molecule | CAS: 1392136-43-4

Kpt 335 is under investigation in clinical trial NCT02431364 (Trial of Safety and Tolerability of Oral Verdinexor (Verdinexor) in Healthy Adults).

Kategori:
Acids, AcyclicAcrylatesAmides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Verdiperstat DB12440
small molecule | CAS: 890655-80-8

Verdiperstat has been used in trials studying the basic science and treatment of Multiple System Atrophy (MSA).

Kategori:
Pyrimidines
Target Protein:
Myeloperoxidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Verteporfin Approved DB00460
small molecule | CAS: 129497-78-5

Verteporfin, marketed as Visudyne, is a benzoporphyrin derivative comprising a 50:50 mixture of two isomers: [CL-315555] and [CL-315585]. It is used as a photosensitizer in photodynamic therapy to eliminate abnormal blood vessels in wet form macular degenerat…

Kategori:
Antineovascularisation AgentsDermatologicalsEENT Drugs, Miscellaneous +10
Waktu ParuhFollowing intraveno…
Vol. Distribusi-
Klirens-
Genetik -
Verubecestat DB12285
small molecule | CAS: 1286770-55-5

Verubecestat is under investigation for the treatment of Alzheimer's Disease, Prodromal Alzheimer's disease, and Amnestic Mild Cognitive Impairment. Verubecestat is Merck’s investigational oral ?-site amyloid precursor protein cleaving enzyme (BACE1 or ? …

Kategori:
Sulfur CompoundsThiazines
Target Protein:
Beta-secretase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Verucerfont DB12512
small molecule | CAS: 885220-61-1

Verucerfont has been used in trials studying the treatment of Congenital Adrenal Hyperplasia.

Kategori:
Aza CompoundsOxazolesReceptors, Corticotropin-Releasing Hormone, antagonists & inhibitors
Target Protein:
Corticotropin-releasing factor receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vesatolimod DB12687
small molecule | CAS: 1228585-88-3

Vesatolimod has been used in trials studying the treatment of Hepatitis B and Chronic Hepatitis B.

Kategori:
Anti-Infective AgentsAntiviral AgentsHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Toll-like receptor 7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vesencumab DB15428
biotech | CAS: 1205533-60-3

Vesencumab is under investigation in clinical trial NCT00747734 (A Study of MNRP1685A in Patients With Locally Advanced or Metastatic Solid Tumors).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vesnarinone DB12082
small molecule | CAS: 81840-15-5

Vesnarinone has been used in trials studying the treatment of HIV Infections and Sarcoma, Kaposi.

Kategori:
Adjuvants, ImmunologicAnti-Infective AgentsAntineoplastic Agents +8
Target Protein:
cGMP-inhibited 3',5'-cyclic phosphodiesterase 3AVoltage-gated inwardly rectifying potassium channel KCNH2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vestronidase alfa Approved DB12366
biotech | CAS: 1638194-78-1

Vestronidase alfa, or vestronidase alfa-vjbk, is a recombinant human lysosomal beta glucuronidase that is a purified enzyme produced by recombinant DNA technology in a Chinese hamster ovary cell line. The enzyme is a homotetramer consisted of 4 monomers with …

Kategori:
Alimentary Tract and MetabolismEnzymesEnzymes and Coenzymes +3
Waktu ParuhAfter repeated dosi…
Vol. DistribusiAfter repeated dosi…
KlirensAfter repeated dosi…
Genetik -
VG161 DB18469
biotech

VG161 is an oncolytic virus therapy under investigation for the treatment of cholangiocarcinoma.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vibecotamab DB18872
biotech | CAS: 2138442-13-2

Vibecotamab is under investigation in clinical trial NCT05285813 (A Phase II Study of Vibecotamab (Xmab14045) for MRD- Positive AML and MDS After Hypomethylating Agent Failure).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vibegron Approved DB14895
small molecule | CAS: 1190389-15-1

Vibegron is a potent, selective beta-3 adrenergic receptor (?3) agonist that relaxes the detrusor smooth muscle of the bladder, thereby increasing bladder capacity.[L28305] Vibegron was first approved in Japan in September 2018 for the treatment of overactive…

Kategori:
Adrenergic AgonistsAdrenergic beta-3 Receptor AgonistsAdrenergic beta-Agonists +10
Target Protein:
Beta-3 adrenergic receptor
Waktu ParuhThe terminal plasma…
Vol. DistribusiThe mean apparent v…
KlirensThere is limited in…
Genetik -
biotech | CAS: 1704499-30-8

_Vibrio cholerae_ CVD 103-HgR strain live antigen is a component of Vaxchora, an oral vaccine for immunization against _Vibrio cholerae_ serogroup O1.[L12801] Cholera is an acute bacterial disease of the small intestine caused by _Vibrio cholerae_, which is g…

Kategori:
Bacterial VaccinesBiological ProductsComplex Mixtures +3
Waktu ParuhPharmacokinetic inf…
Vol. DistribusiPharmacokinetic inf…
KlirensPharmacokinetic inf…
Genetik -
Vidupiprant DB12272
small molecule | CAS: 1169483-24-2

Vidupiprant has been used in trials studying the treatment and basic science of Asthma.

Kategori:
Acids, CarbocyclicAmidesSulfones +1
Target Protein:
Prostaglandin D2 receptor 2Prostaglandin D2 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vigabatrin Approved DB01080
small molecule | CAS: 68506-86-5

Vigabatrin is an analog of gamma-aminobutyric acid ([GABA]), the main inhibitory neurotransmitter in the central nervous system, used in the treatment of refractory seizures and infantile spasms.[L13616] It irreversibly inhibits the enzyme responsible for GAB…

Kategori:
Acids, AcyclicAminobutyratesAnti-epileptic Agent +15
Target Protein:
4-aminobutyrate aminotransferase, mitochondrial
Waktu ParuhThe terminal half-l…
Vol. DistribusiVigabatrin is widel…
KlirensThe oral clearance …
Genetik -
Vilaprisan DB11971
small molecule | CAS: 1262108-14-4

Vilaprisan has been used in trials studying the treatment of Leiomyoma and Clinical Trial, Phase I.

Kategori:
Fused-Ring Compounds
Target Protein:
Progesterone receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vilastobart DB19327
biotech | CAS: 2760549-50-4

Vilastobart is under investigation in clinical trial NCT04896697 (Vilastobart (XTX101) Monotherapy and Vilastobart and Atezolizumab Combination Therapy in Advanced Solid Tumors).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vilazodone Approved DB06684
small molecule | CAS: 163521-12-8

Vilazodone is a novel compound with combined high affinity and selectivity for the 5-hydroxytryptamine (5-HT) transporter and 5-HT(1A) receptors[Label,A177622]. Vilazodone may also be associated with less sexual dysfunction and weight gain[A6947]. Vilazodone …

Kategori:
Agents that produce hypertensionAntidepressive AgentsAntidepressive Agents Indicated for Depression +26
Target Protein:
Sodium-dependent serotonin transporter5-hydroxytryptamine receptor 1A
Waktu Paruh25 hours[Label,A384…
Vol. DistribusiVilazodone's volume…
KlirensClearance of vilazo…
Genetik -
Viltolarsen Approved DB15005
biotech | CAS: 2055732-84-6

Duchenne muscular dystrophy (DMD) is an X-linked recessive allelic disorder characterized by a lack of functional dystrophin protein, which leads to progressive ambulatory, pulmonary, and cardiac function and is invariably fatal. A related, albeit a less seve…

Kategori:
Antisense OligonucleotidesMorpholinesMusculo-Skeletal System +5
Target Protein:
DMD gene (exon 53 viltolarsen target site)
Waktu ParuhViltolarsen has a r…
Vol. DistribusiViltolarsen has a s…
KlirensViltolarsen has a r…
Genetik -
Vinbarbital DB13377
small molecule | CAS: 125-42-8

Deskripsi belum tersedia.

Kategori:
Barbiturates, PlainCentral Nervous System DepressantsHypnotics and Sedatives +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vinpocetine DB12131
small molecule | CAS: 42971-09-5

Vinpocetine has been investigated for the treatment of Epilepsy.

Kategori:
Agents causing hyperkalemiaAlkaloidsAntiarrhythmic agents +25
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Violaxanthin DB03460
small molecule | CAS: 126-29-4

Deskripsi belum tersedia.

Kategori:
AlkenesBiological FactorsCarotenoids +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vipoglanstat DB18126
small molecule | CAS: 1360622-01-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Visilizumab DB12053
biotech | CAS: 219716-33-3

Visilizumab has been investigated for the treatment of Ulcerative Colitis.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vismodegib Approved DB08828
small molecule | CAS: 879085-55-9

Vismodegib is an orally active small molecule that inhibits the hedgehog signaling pathway by binding to and inhibiting the transmembrane protein smoothened homologue (SMO).[A258613,A258618,L45803] It was discovered by high-throughput screening of a library o…

Kategori:
AmidesAminesAniline Compounds +18
Target Protein:
Protein smoothened
Waktu ParuhThe half-life of vi…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
small molecule | CAS: 15713-12-9

Deskripsi belum tersedia.

Target Protein:
5-methyltetrahydrofolate--homocysteine S-methyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Voacamine DB04877
small molecule | CAS: 3371-85-5

Voacamine is an alkaloid isolated from the bark of the _Pescheria fuchsiae folia_ tree. It is an antimalarial drug approved for use in several African countries. Voacamine is also under investigation for use in modulating multidrug-resistance in tumor cells.

Kategori:
AlkaloidsHeterocyclic Compounds, Fused-RingIndole Alkaloids +5
Target Protein:
ATP-dependent translocase ABCB1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Voclosporin Approved DB11693
small molecule | CAS: 515814-01-4

Lupus nephritis (LN) is a type of glomerulonephritis occurring in patients with systemic lupus erythematosus (SLE). LN is a significant cause of renal failure, morbidity, and death in patients with SLE. Within 10 years of being diagnosed with SLE, 5-20% of …

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating AgentsCalcineurin Inhibitor Immunosuppressant +16
Target Protein:
Guided entry of tail-anchored proteins factor CAMLGProtein phosphatase 3 catalytic subunit alphaCalcineurin subunit B type 1 +1
Waktu ParuhThe average termina…
Vol. DistribusiThe apparent volume…
KlirensThe mean apparent s…
Genetik -
Vofatamab DB14781
biotech | CAS: 1312305-12-6

Vofatamab is under investigation in clinical trial NCT02401542 (Dose Escalation, Expansion Study of Vofatamab (B-701) in Treatment of Locally Advanced or Metastatic Urothelial Cell Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vofopitant DB12436
small molecule | CAS: 168266-90-8

Vofopitant has been used in trials studying the treatment of PTSD, Primary Insomnia, and Sleep Initiation and Maintenance Disorders.

Kategori:
AntiemeticsAutonomic AgentsCentral Nervous System Agents +4
Target Protein:
Substance-P receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Volagidemab DB16421
biotech | CAS: 1233956-13-2

Volagidemab is under investigation in clinical trial NCT03117998 (Multiple Dose Study to Evaluate the Efficacy, Safety and Pharmacodynamics of REMD-477 in Subjects With Type 1 Diabetes Mellitus).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Volasertib DB12062
small molecule | CAS: 755038-65-4

Volasertib has been used in trials studying the treatment of Leukemia, Neoplasms, Leukemia, Myeloid, Acute, Myelodysplastic Syndromes, and Leukemia, Monocytic, Acute, among others.

Kategori:
Antineoplastic AgentsHeterocyclic Compounds, Fused-Ring
Target Protein:
Serine/threonine-protein kinase PLK1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Volixibat DB13914
small molecule | CAS: 1025216-57-2

Volixibat, also known as SHP626 or LUM002, is an investigational drug that will potentially be used for the treatment of Non-Alcoholic Steatohepatitis (NASH). If approved for use, it will be the first available agent for the treatment of NASH. Volixibat is…

Kategori:
CarbohydratesHeterocyclic Compounds, Fused-RingLipid Regulating Agents +1
Target Protein:
Ileal sodium/bile acid cotransporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vonicog alfa Approved DB12872
biotech

Vonicog alfa is a recombinant human von Willebrand factor (rVWF) produced from Chinese hamster ovary cells.[A264444] Used to treat von Willebrand Disease (vWD), it mimics the biological actions of endogenous VWF,[L51274] which is a critical plasma glycoprotei…

Kategori:
von Willebrand Factor
Target Protein:
Coagulation factor VIIICollagen alpha-1(I) chain
Waktu ParuhIn Study 071001, th…
Vol. Distribusi-
KlirensIn Study 071001, th…
Genetik -
Vorozole DB13767
small molecule | CAS: 129731-10-8

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsAromatase Inhibitors +8
Target Protein:
Aromatase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Voxilaprevir Approved DB12026
small molecule | CAS: 1535212-07-7

Voxilaprevir is a Direct-Acting Antiviral (DAA) medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized i…

Kategori:
Acids, AcyclicAmidesAmino Acids +36
Target Protein:
Genome polyproteinGenome polyprotein
Waktu Paruh33 hr [FDA Label]
Vol. Distribusi-
Klirens-
Genetik -
Voxtalisib DB12400
small molecule | CAS: 934493-76-2

Voxtalisib has been used in trials studying the treatment of Cancer, Melanoma, Lymphoma, Glioblastoma, and Breast Cancer, among others.

Kategori:
AmidesHeterocyclic Compounds, Fused-RingPhosphatidylinositol 3-Kinases, antagonists & inhibitors +2
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformSerine/threonine-protein kinase mTOR
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VP-14637 DB12195
small molecule | CAS: 235106-62-4

MDT-637 has been investigated for the treatment of Drug Safety.

Kategori:
Benzene DerivativesHydrazines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VPO-227 DB18004
small molecule | CAS: 1314873-02-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VS-5584 DB12986
small molecule | CAS: 1246560-33-7

VS-5584 has been used in trials studying the treatment of Lymphoma, Metastatic Cancer, and Non Hematologic Cancers.

Kategori:
Heterocyclic Compounds, Fused-RingOxazines
Target Protein:
Target of rapamycin complex 2 subunit MAPKAP1Serine/threonine-protein kinase mTORPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VTP-201227 DB05652
small molecule

VTP-201227 has a novel mechanism of action and is being developed as a topical agent for the treatment of psoriasis with potential extensions into other dermatological indications. It is being developed by Vitae Pharmaceuticals.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VTP-27999 DB12416
small molecule | CAS: 942142-51-0

VTP-27999 has been used in trials studying the basic science of Renal Function.

Kategori:
Acids, AcyclicAgents Acting on the Renin-Angiotensin SystemRenin Inhibitors
Target Protein:
Renin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Willardiine DB04129
small molecule | CAS: 21416-43-3

Willardiine is a compound isolated from seeds of _Acacia willariana_.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsPyrimidines +1
Target Protein:
Glutamate receptor 1Glutamate receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
WIN 55212-2 DB13950
small molecule | CAS: 131543-22-1

WIN 55,212-2 is a chemical described as an aminoalkylindole derivative, which produces effects similar to those of cannabinoids such as tetrahydrocannabinol (THC) but has an entirely different chemical structure. It is a potent cannabinoid receptor agonist th…

Kategori:
Agents causing hyperkalemiaAgents producing tachycardiaAnalgesics +21
Target Protein:
Cannabinoid receptor 1Cannabinoid receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
WNT-974 DB12561
small molecule | CAS: 1243244-14-5

WNT974 has been used in trials studying the treatment of Metastatic Colorectal Cancer and Squamous Cell Carcinoma, Head And Neck.

Kategori:
Enzyme Inhibitors
Target Protein:
Protein-serine O-palmitoleoyltransferase porcupine
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 3151–3200 dari 3253
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