Hasil Filter

6694

Total database: 17430
Struktur (SMILES)
4518 (67.5%)
Target
3751 (56.0%)
Genomik
81 (1.2%)
Referensi
6694 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (6694)

Halaman 62 / 134
Golvatinib DB11977
small molecule | CAS: 928037-13-2

Golvatinib has been investigated for the treatment of Platinum-Resistant Squamous Cell Carcinoma of the Head and Neck.

Kategori:
AminesPyridinesVascular Endothelial Growth Factor Receptor-2, antagonists & inhibitors
Target Protein:
Vascular endothelial growth factor receptor 2Hepatocyte growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gondoic acid DB14073
small molecule | CAS: 5561-99-9

Deskripsi belum tersedia.

Kategori:
Fatty AcidsFatty Acids, UnsaturatedLipids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gontivimab DB16179
biotech | CAS: 1257358-38-5

Gontivimab is under investigation in clinical trial NCT03468829 (Efficacy and Safety of ALX-0171 in Adult Hematopoietic Stem Cell Transplant (HSCT) Recipients Who Present With Respiratory Syncytial Virus (RSV) Infection).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntiviral Agents +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gosogliptin DB08382
small molecule | CAS: 869490-23-3

Gosogliptin has been used in trials studying the treatment of Renal Insufficiency, Chronic.

Kategori:
Agents causing angioedemaBlood Glucose Lowering AgentsDiabetes Mellitus, Type 2, drug therapy +1
Target Protein:
Dipeptidyl peptidase 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GP-100 antigen DB14800
biotech

GP-100 antigen is under investigation in clinical trial NCT00006385 (Vaccine Therapy With or Without Biological Therapy in Treating Patients With Metastatic Melanoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntigensAntigens, Neoplasm +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GP2 peptide DB16180
biotech | CAS: 160790-21-6

GP2 peptide is under investigation in clinical trial NCT00524277 (Vaccine Therapy in Treating Patients With Breast Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GPI-0100 DB05929
small molecule

GPI-0100 is Avantogen’s lead adjuvanat-immunopotentiator, a key component of vaccines for boosting the immune response. The GPI-0100 adjuvant, which has been shown to significantly enhance the immune response with a variety of vaccines, has been shown to hav…

Kategori:
CarbohydratesGlycosides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GRAd-COV2 DB16428
biotech

GRAd-COV2 is a COVID-19 vaccine candidate being developed by ReiThera[L30420, L30423]. This therapy is based on a novel replication-incompetent simian adenoviral vector that encodes the full-length SARS-CoV-2 spike protein (GRAd-COV2)[L30420, L30423]. Preclin…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gramicidin D Approved DB00027
small molecule | CAS: 1405-97-6

Gramcidin D is a heterogeneous mixture of three antibiotic compounds, gramicidins A, B and C, making up 80%, 6%, and 14% respectively all of which are obtained from the soil bacterial species Bacillus brevis and called collectively gramicidin D. Gramcidins ar…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +9
Target Protein:
Dihydropteroate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Granaticin B DB17273
small molecule | CAS: 19879-03-9

Deskripsi belum tersedia.

Kategori:
BenzopyransBenzoquinonesChromans +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Grapefruit Approved DB10534
biotech

Grapefruit allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityCytochrome P-450 CYP3A InhibitorsCytochrome P-450 CYP3A4 Inhibitors +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Grapefruit oil DB15663
biotech | CAS: 8016-20-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Grapiprant DB12836
small molecule | CAS: 415903-37-6

Grapiprant, also known as AT-001 and CJ-023, is a drug from the piprant class. These molecules were derived from acylsulfonamide and are characterized to be a novel series of para-N-acylaminomethylbenzoic acid known to be prostaglandin receptor antagonists.[A…

Kategori:
AmidesBenzene DerivativesP-glycoprotein substrates +3
Target Protein:
Prostaglandin E2 receptor EP4 subtype
Waktu ParuhThe reported elimin…
Vol. DistribusiThe reported volume…
KlirensThe reported cleara…
Genetik -
Grazoprevir Approved DB11575
small molecule | CAS: 1350514-68-9

Grazoprevir is a direct acting antiviral medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized into nin…

Kategori:
Acids, AcyclicAmidesAnti-Infective Agents +24
Target Protein:
Genome polyprotein
Waktu ParuhThe geometric mean …
Vol. DistribusiGrazoprevir has an …
KlirensThe clearance of Gr…
Genetik -
Grepafloxacin Approved DB00365
small molecule | CAS: 119914-60-2

Grepafloxacin is an oral broad-spectrum quinoline antibacterial agent used to treat bacterial infections. Due to the QTc-prolonging potential, as indicated by the changes in the QT interval on the electrocardiogram, and the risk for cardiovascular adverse eve…

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +22
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +1
Waktu Paruh15 ± 3 hours
Vol. Distribusi-
Klirens-
Genetik -
Gresonitamab DB18210
biotech | CAS: 2413817-97-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Grn163l DB05036
small molecule

GRN163L is a novel anti-cancer drug. It has been characterized preclinically and shown to inhibit telomerase in human tumor cells of many cancer types (including lung, breast, prostate, liver, and early stage of human breast cancer), in both cell culture syst…

Target Protein:
Telomerase-binding protein EST1AN-terminal kinase-like proteinProstaglandin E synthase 3 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GS-100 DB18337
biotech

GS-100 is an adeno-associated virus serotype 9 virus particle containing viral DNA that includes an expression cassette containing the human NGLY1 gene coding sequence

Kategori:
CyclohexanesCycloparaffinsLipids +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GSK-356278 DB12542
small molecule | CAS: 720704-34-7

Gsk356278 has been used in trials studying the treatment and basic science of Anxiety Disorders, Huntington Disease, Depressive Disorder, Huntingtons Disease, and Depressive Disorder, Major, among others.

Kategori:
OxazolesSulfur Compounds
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4A3',5'-cyclic-AMP phosphodiesterase 4D3',5'-cyclic-AMP phosphodiesterase 4B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GSK-364735 DB13119
small molecule | CAS: 863434-13-3

GSK-364735 (Naphthyridinone) has been used in trials studying the treatment of HIV-1 Infection and Infection, Human Immunodeficiency Virus.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GSK-424887 DB12219
small molecule

Gsk424887 has been used in trials studying the basic science and treatment of Depressive Disorder and Anxiety Disorder.

Kategori:
AcetatesAcids, AcyclicAmides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GSK-923295 DB06097
small molecule

GSK-923295 is a small-molecule inhibitor of the mitotic kinesin centromere-associated protein E (CENP-E), and the third novel drug candidate to arise from Cytokinetics' broad strategic alliance with GlaxoSmithKline (GSK). GSK-923295 demonstrated a broad spect…

Target Protein:
Centromere-associated protein E
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GSK-945237 DB15345
small molecule | CAS: 944406-54-6

GSK-945237 is under investigation in clinical trial NCT01039610 (A Single Center Four Part Study in Healthy Adult Subjects to Evaluate: the Safety, Tolerability and Pharmacokinetics of a Single Oral Dose and Repeat Escalating Oral Doses of GSK945237; the Effe…

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GSK2798745 DB16033
small molecule | CAS: 1419609-94-1

GSK2798745 is under investigation in clinical trial NCT03372603 (A Study to Assess the Effectiveness and Side Effects of GSK2798745 in Participants With Chronic Cough).

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GT-AS DB17883
biotech

GT-AS recombinant adeno-associated virus serotype 9 vector containing the transgene UBE3A encoding for ubiquitin protein ligase E3A/E6-AP.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GTB-3550 DB18494
biotech

GTB-3550 is a single-chain, tri-specific scFv recombinant fusion protein conjugate composed of the variable regions of the heavy and light chains of anti-CD16 and anti-CD33 antibodies and a modified form of Interleukin 15 (IL-15).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GTI-2040 DB15030
biotech | CAS: 236391-66-5

GTI-2040 is under investigation in clinical trial NCT00084643 (GTI-2040, Oxaliplatin, and Capecitabine in Treating Patients With Locally Advanced or Metastatic Colorectal Cancer or Other Solid Tumors).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GTP-506 DB17682
biotech

GTP-506 is a gene therapy formed by two vectors, a nuclease vector targeting gene editing in the well-characterized PCSK9 gene locus and a therapeutic donor vector that inserts the OTC gene to provide the desired genetic correction.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GTX-758 DB14969
small molecule | CAS: 938067-78-8

GTX-758 is under investigation in clinical trial NCT01420861 (GTx-758 on Serum Prostate-specific Antigen (PSA) in Men With Castrate Resistant Prostate Cancer).

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Guadecitabine DB11918
small molecule | CAS: 929901-49-5

Guadecitabine is under investigation for the treatment of Previously Treated Metastatic Colorectal Cancer.

Kategori:
Antineoplastic AgentsAza CompoundsImmunologic Factors +5
Target Protein:
DNA (cytosine-5)-methyltransferase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Guaiacol Approved DB11359
small molecule | CAS: 90-05-1

Guaiacol is an agent thought to have disinfectant properties and used as an expectorant. Guaiacol is a phenolic natural product first isolated from Guaiac resin and the oxidation of lignin. Guaiacol is also present in wood smoke, as a product of pyrolysis of …

Kategori:
Benzene DerivativesCatecholsEthers +4
Target Protein:
Albumin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Guaifenesin Approved DB00874
small molecule | CAS: 93-14-1

Guaifenesin possesses a storied history, having been originally formally approved by the US FDA in 1952 and continues to be one of very few - if not perhaps the only drug that is readily available and used as an expectorant [F4525]. Since that time the agent …

Kategori:
Benzene DerivativesCatecholsCough and Cold Preparations +6
Target Protein:
NMDA receptor
Waktu ParuhThe half-life in pl…
Vol. DistribusiThe geometric mean …
KlirensThe mean clearance …
Genetik -
Guanethidine Approved DB01170
small molecule | CAS: 55-65-2

An antihypertensive agent that acts by inhibiting selectively transmission in post-ganglionic adrenergic nerves. It is believed to act mainly by preventing the release of norepinephrine at nerve endings and causes depletion of norepinephrine in peripheral sym…

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAmidines +16
Target Protein:
Sodium-dependent noradrenaline transporter
Waktu Paruh1.5 days
Vol. Distribusi-
Klirens* Renal cl=56 ml/min
Genetik -
Guanfacine Approved DB01018
small molecule | CAS: 29110-47-2

Guanfacine, or BS 100-141,[A189838,A189841] is a selective alpha-A2 adrenergic receptor agonist initially indicated for the treatment of hypertension[L11274] but is now indicated as an extended release tablet for the treatment of ADHD.[L11277] Guanfacine was …

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +26
Target Protein:
Alpha-2A adrenergic receptorAlpha-2B adrenergic receptor
Waktu ParuhGuanfacine has a ha…
Vol. DistribusiGuanfacine has a vo…
KlirensGuanfacine has a to…
Genetik -
small molecule | CAS: 77482-44-1

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicDicarboxylic Acids
Target Protein:
Carboxypeptidase D
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 117-68-0

Deskripsi belum tersedia.

Kategori:
Guanine NucleotidesHeterocyclic Compounds, Fused-RingIsomerism +5
Target Protein:
RibonucleaseBifunctional protein PyrR
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 33503-72-9

Guanosine tetraphosphate is a guanine nucleotide containing four phosphate groups. Two phosphate groups are esterified to the sugar moiety in the 5' position and the other two in the 2' or 3' position. This nucleotide serves as a messenger to turn off the syn…

Kategori:
Guanine NucleotidesHeterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and Nucleosides +4
Target Protein:
Hypoxanthine-guanine-xanthine phosphoribosyltransferaseXanthine phosphoribosyltransferaseGTPase Obg
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 130-50-7

Deskripsi belum tersedia.

Kategori:
Guanine NucleotidesHeterocyclic Compounds, Fused-RingIsomerism +5
Target Protein:
Guanyl-specific ribonuclease Sa
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Guanoxan Approved DB13211
small molecule | CAS: 2165-19-7

Guanoxan is an antihypertensive agent similar in its mechanism of action to guanethidine; may cause liver damage. Guanoxan was approved in the UK but was withdrawn from the market due to hepatotoxicity.

Kategori:
AmidinesAntiadrenergic Agents, Peripherally ActingAntihypertensive Agents +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gusacitinib DB15670
small molecule | CAS: 1425381-60-7

Gusacitinib is under investigation in clinical trial NCT02550678 (A Study of the Efficacy and Safety of ASN-002 in Adult Patients With Low-risk Nodular Basal Cell Carcinoma).

Kategori:
Nitriles
Target Protein:
Tyrosine-protein kinase SYK
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Guvacine DB08848
small molecule | CAS: 498-96-4

Guvacine is a pyridine alkaloid found in the Areca nut (also known as the Betel nut). It is an experimental drug with no approved indication. Experimental studies are still being investigated to determine all of the physiological effects and mechanisms of act…

Kategori:
Pyridines
Target Protein:
Sodium- and chloride-dependent GABA transporter 2Sodium- and chloride-dependent GABA transporter 1Sodium- and chloride-dependent GABA transporter 3 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GVAX DB17276
biotech

GVAX is a granulocyte-macrophage colony-stimulating factor (GM-CSF) gene-transfected tumor cell vaccine.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GW 468816 DB05417
small molecule

GW 468816 is glycine receptor antagonist. It is designed to aid abstinence in people who have just quit smoking, delaying the time to relapse. It was undergoing phase II trials since December 2003.

Kategori:
Heterocyclic Compounds, Fused-RingReceptors, N-Methyl-D-Aspartate, antagonists & inhibitors
Target Protein:
Glycine receptor subunit alpha-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GW-468816 DB15099
small molecule | CAS: 476689-77-7

GW-468816 is under investigation in clinical trial NCT00218465 (Effectiveness of GW468816, an NMDA Glycine Site Antagonist, for Prevention of Relapse to Smoking).

Kategori:
Heterocyclic Compounds, Fused-RingReceptors, N-Methyl-D-Aspartate, antagonists & inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GX-19 Vaccine DB15891
biotech

The GX-19 vaccine is a DNA vaccine created by Genexine, Inc. Company in Gyeonggi, Korea[A219758]. As of June 2020, the vaccine candidate is undergoing Phase I and Phase IIa trials to determine dose levels for safety and efficacy[A219758,L16488].

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
H-89 DB07995
small molecule | CAS: 127243-85-0

Deskripsi belum tersedia.

Kategori:
AmidesEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring +3
Target Protein:
cAMP-dependent protein kinase catalytic subunit alphacAMP-dependent protein kinase inhibitor alphaSerine/threonine-protein kinase haspin +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
H3B-8800 DB14017
small molecule | CAS: 1825302-42-8

H3B-8800 is a novel spliceosome inhibitor developed by H3 Biomedicine [L2551]. It offers the benefit of preferentially killing spliceosome-mutant cancer cells whereas other splicesome inhibitors, such as the pladienolide analogue E7107, show no such preferent…

Target Protein:
Splicing factor 3B subunit 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Hachimycin DB13302
small molecule | CAS: 1394-02-1

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntifungals for Dermatological UseAntifungals for Topical Use +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Hadacidin DB02109
small molecule | CAS: 689-13-4

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAntibiotics, Antineoplastic +4
Target Protein:
Inosine-5'-monophosphate dehydrogenase 1Adenylosuccinate synthetaseAdenylosuccinate synthetase +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Haemophilus influenzae type b capsular polysaccharide meningococcal outer membrane protein conjugate antigen is a vaccine containing outer membrane antigen extracted from *Haemophilus influenzae*.

Kategori:
Actively Acquired ImmunityHaemophilus VaccinesInactivated Haemophilus Influenzae B Vaccine
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 3051–3100 dari 6694
Sebelumnya Halaman 62 / 134 Berikutnya