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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 62 / 236
Brigimadlin DB18578
small molecule | CAS: 2095116-40-6

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brilacidin DB12997
small molecule | CAS: 1224095-98-0

Brilacidin is under investigation for the supportive care of Mucositis, Stomatitis, Mouth Diseases, and Head and Neck Neoplasms.

Kategori:
AmidinesAnti-Infective Agents
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brilaroxazine DB09226
small molecule | CAS: 1239729-06-6

Brilaroxazine (RP5063) is an investigational atypical antipsychotic which is under development by Reviva Pharmaceuticals for the treatment of schizophrenia and schizoaffective disorder. Reviva Pharmaceuticals also intends to investigate RP5063 for the treatme…

Kategori:
Antidepressive AgentsAntipsychotic AgentsAntipsychotic Agents (Second Generation [Atypical]) +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brilliant green cation Approved DB11279
small molecule | CAS: 18198-35-1

Brilliant green, or ethanaminium, is a derivative of triarylmethane dye that has been used as a dye to color silk and wool. Due to its inhibitory actions against Gram positive microorganisms, brilliant green can be found in antiseptic products such as solutio…

Kategori:
AminesAmmonium CompoundsAnti-Infective Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brimapitide DB15231
small molecule | CAS: 1445179-97-4

Brimapitide is under investigation in clinical trial NCT01570205 (Safety, Tolerability and PK of a Single iv Infusion of 10, 40, and 80 µg/kg XG-102 Administered to Healthy Volunteers).

Kategori:
Amino Acids, Peptides, and ProteinsNeuroprotective Agents
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brimonidine Approved DB00484
small molecule | CAS: 59803-98-4

Brimonidine is an alpha-adrenergic agonist and 2-imidazoline derivative that was first introduced in 1996.[A178951] It is considered to be a third generation alpha-2 aadrenergic receptor agonist, since it displays preferential binding at alpha-2 adrenoceptors…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +14
Target Protein:
Alpha-2A adrenergic receptorAlpha-2B adrenergic receptorAlpha-2C adrenergic receptor
Waktu ParuhFollowing ocular ad…
Vol. DistribusiThe volume of distr…
KlirensThe apparent cleara…
Genetik -
Brincidofovir Approved DB12151
small molecule | CAS: 444805-28-1

Brincidofovir is an oral antiviral drug used in the treatment of human smallpox infections. It is a lipid conjugate pro-drug of the acyclic nucleotide analogue [cidofovir][L34404,A235725] - this lipid conjugate improves drug delivery to the target cells and s…

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +27
Target Protein:
DNA polymerase nuDNA polymerase delta subunit 4DNA polymerase delta catalytic subunit +7
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe apparent volume…
KlirensThe apparent cleara…
Genetik -
Brinzolamide Approved DB01194
small molecule | CAS: 138890-62-7

Brinzolamide is a highly specific, non-competitive, reversible carbonic anhydrase II (CA-II) inhibitor indicated to reduce ocular pressure in patients with ocular hypertension or open-angle glaucoma.[L35310] Although the exact pathophysiology of glaucoma is s…

Kategori:
AmidesAntiglaucoma Preparations and MioticsCarbonic Anhydrase Inhibitors +17
Target Protein:
Carbonic anhydrase 2Carbonic anhydrase 1Carbonic anhydrase 4 +2
Waktu ParuhDue to its affinity…
Vol. Distribusi-
Klirens-
Genetik -
Briquilimab DB18136
biotech | CAS: 2574591-89-0

Briquilimab is a humanized aglycosylated IgG1 kappa monoclonal antibody targeting CD117 (cKit).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Brivanib DB11958
small molecule | CAS: 649735-46-6

Brivanib is under investigation for the treatment of HepatoCellular Carcinoma. Brivanib has been investigated for the treatment of Solid Tumors, Hepato Cellular Carcinoma (HCC), and Metastatic Colorectal Cancer (MCRC).

Kategori:
Amino AcidsAmino Acids, Peptides, and Proteins
Target Protein:
Vascular endothelial growth factor receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 649735-63-7

Brivanib alaninate has been investigated for the treatment of Colorectal Cancer.

Kategori:
Amino AcidsAmino Acids, Peptides, and Proteins
Target Protein:
Fibroblast growth factor receptor 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brivaracetam Approved DB05541
small molecule | CAS: 357336-20-0

Brivaracetam is a racetam derivative of levetiracetam used in the treatment of partial-onset seizures. Brivaracetam binds SV2A with 20 times higher affinity than levetiracetam [A19184]. It is available under the brand name Briviact made by UCB. Briviact recei…

Kategori:
AnticonvulsantsCentral Nervous System AgentsCentral Nervous System Depressants +11
Target Protein:
Synaptic vesicle glycoprotein 2ASodium channel protein
Waktu Paruh7-8h [A19180].
Vol. Distribusi0.5L/kg [FDA Label].
KlirensCL/F of 0.7-1.07 mL…
Genetik -
Brivoligide DB16116
biotech | CAS: 1803075-42-4

Brivoligide is under investigation in clinical trial NCT04104919 (Study to Evaluate a Preop Dose of Brivoligide Injection for Pain After Mastectomy in Patients With High PCS Scores).

Waktu Paruh-
Vol. Distribusi-
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Brivudine Approved DB03312
small molecule | CAS: 69304-47-8

Brivudine is used in the treatment of herpes zoster. Although not approved in the U.S. or Canada, it is approved in several European countries.

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +9
Target Protein:
Thymidine kinase 2, mitochondrialThymidine kinase, cytosolicDNA polymerase +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brodalumab Approved DB11776
biotech | CAS: 1174395-19-7

Brodalumab has been used in trials studying the treatment of Asthma, Psoriasis, Crohn's Disease, Psoriatic Arthritis, and Rheumatoid Arthritis. Brodalumab was FDA approved in February, 2017 as Siliq for the treatment of moderate-to-severe plaque psoriasis.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +13
Target Protein:
Interleukin-17 receptor A
Waktu Paruh-
Vol. Distribusi4.62 L.
Klirens0.223 L/day.
Genetik -
Brodimoprim DB13795
small molecule | CAS: 56518-41-3

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntibacterials for Systemic UseAntiinfectives for Systemic Use +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brofaromine DB13876
small molecule | CAS: 63638-91-5

Deskripsi belum tersedia.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsEnzyme Inhibitors +3
Target Protein:
Amine oxidase [flavin-containing] A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brolucizumab Approved DB14864
biotech | CAS: 1531589-13-5

Brolucizumab, also known as RTH258 or ESBA1008,[A187211] is a monoclonal antibody indicated to treat neovascular age related macular degeneration.[L9089] Brolucizumab was granted FDA approval in October 2019.[L9089]

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAntibodies +14
Target Protein:
Vascular endothelial growth factor A, long form
Waktu ParuhThe systemic half l…
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik -
Bromamphenicol DB07492
small molecule | CAS: 16803-75-1

Deskripsi belum tersedia.

Kategori:
AlcoholsBenzene DerivativesGlycols +3
Target Protein:
Dr hemagglutinin structural subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bromelains DB13281
biotech | CAS: 9001-00-7

Bromelain is a protease enzyme derived from the stems of pineapples that is composed of a mixture of different thiol endopeptidases and other components like phosphatase, glucosidase, peroxidase, cellulase, escharase, and several protease inhibitors [A27198].…

Kategori:
Cysteine EndopeptidasesCysteine ProteasesDermatologicals +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bromfenac Approved DB00963
small molecule | CAS: 91714-94-2

Bromfenac is a nonsteroidal anti-inflammatory drug (NSAID) for ophthalmic use. Ophthalmic NSAIDs are becoming a cornerstone for the management of ocular pain and inflammation. Their well-characterized anti-inflammatory activity, analgesic property, and establ…

Kategori:
Agents causing hyperkalemiaAnalgesicsAnalgesics, Non-Narcotic +16
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bromhexine Approved DB09019
small molecule | CAS: 3572-43-8

Bromhexine is mucolytic agent used for a variety of respiratory conditions associated with increased mucus secretion. It is derived from the Adhatoda vasica plant and aids in the clearance of excess mucus, improving breathing and reducing cough. It was introd…

Kategori:
AminesAniline CompoundsCough and Cold Preparations +5
Target Protein:
Transmembrane protease serine 2Angiotensin-converting enzyme 2
Waktu ParuhFollowing single or…
Vol. DistribusiAfter intravenous a…
KlirensThe clearance of br…
Genetik -
Bromisoval DB13370
small molecule | CAS: 496-67-3

Deskripsi belum tersedia.

Kategori:
AmidesCentral Nervous System AgentsCentral Nervous System Depressants +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bromo-WR99210 DB04007
small molecule

Deskripsi belum tersedia.

Target Protein:
Peptide deformylase, mitochondrialDihydrofolate reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 3679-64-9

Deskripsi belum tersedia.

Kategori:
Antifungals for Dermatological UseAntifungals for Topical UseDermatologicals
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bromocriptine Approved DB01200
small molecule | CAS: 25614-03-3

Bromocriptine mesylate is a semisynthetic ergot alkaloid derivative with potent dopaminergic activity. It inhibits prolactin secretion and may be used to treat dysfunctions associated with hyperprolactinemia. Bromocriptine is also indicated for the management…

Kategori:
Adrenergic AgonistsAdrenergic alpha-1 Receptor AgonistsAdrenergic alpha-1 Receptor Antagonists +41
Target Protein:
D(2) dopamine receptorD(3) dopamine receptor5-hydroxytryptamine receptor 1D +15
Waktu Paruh2-8 hours
Vol. Distribusi-
Klirens-
Genetik -
Bromodiphenhydramine Approved DB01237
small molecule | CAS: 118-23-0

Bromodiphenhydramine is an ethanolamine antihistamine with antimicrobial property. Bromodiphenhydramine is used in the control of cutaneous allergies. Ethanolamine antihistamines produce marked sedation in most patients.

Kategori:
AminesAminoalkyl EthersAntihistamines for Systemic Use +5
Target Protein:
Histamine H1 receptor
Waktu Paruh1 to 4 hours
Vol. Distribusi-
Klirens-
Genetik -
Bromoform DB03054
small molecule | CAS: 75-25-2

Deskripsi belum tersedia.

Kategori:
CarcinogensHydrocarbons, HalogenatedNoxae +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bromopyruvate DB17135
small molecule | CAS: 1113-59-3

Deskripsi belum tersedia.

Kategori:
Affinity LabelsCompounds used in a research, industrial, or household settingEnzyme Inhibitors +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bromothalonil Approved DB14199
small molecule | CAS: 35691-65-7

Bromothalonil, also known as Methyldibromo glutaronitrile (MDBGN), is a widely used preservative that can be found in many personal hygiene and industrial products. It is also a known allergen and dermatological irritant that has been banned in many EU countr…

Kategori:
AllergensAntigensBiological Factors +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bromotheophylline Approved DB14018
small molecule | CAS: 10381-75-6

Bromotheophylline is the active moiety of pamabrom, a mixture of 2-amino-2-methyl-propanol and bromotheophylline. From this mixture, bromotheophylline acts as a weak diuretic that has been used along with some analgesics to relieve the symptoms of premenstrua…

Kategori:
AlcoholsAlkaloidsAmines +11
Target Protein:
Adenosine receptor
Waktu ParuhThe apparent elimin…
Vol. DistribusiThis pharmacokineti…
KlirensThis pharmacokineti…
Genetik -
Bromperidol Approved DB12401
small molecule | CAS: 10457-90-6

Bromperidol has been used in trials studying the treatment of Dementia, Depression, Schizophrenia, Anxiety Disorders, and Psychosomatic Disorders, among others.

Kategori:
Antipsychotic AgentsButyrophenone DerivativesButyrophenones +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bronopol Approved DB13960
small molecule | CAS: 52-51-7

Bronopol, or 2-Bromo-2-nitro-1,3-propanediol, is an organic compound with wide-spectrum antimicrobial properties. First synthesized in 1897, bronopol was primarily used as a preservative for pharmaceuticals and was registered in the United States in 1984 for …

Kategori:
AlcoholsAnti-Infective AgentsAnti-Infective Agents, Local +9
Target Protein:
Thiol groups
Waktu ParuhThe half-life of br…
Vol. DistribusiThe highest concent…
KlirensNo data available.
Genetik -
Brontictuzumab DB12737
biotech | CAS: 1447814-75-6

Brontictuzumab has been used in trials studying the treatment of Adenoid Cystic Carcinoma, Relapsed or Refractory Solid Tumors, and Relapsed or Refractory Lymphoid Malignancies.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bropirimine DB04168
small molecule | CAS: 56741-95-8

Deskripsi belum tersedia.

Kategori:
Adjuvants, ImmunologicAntineoplastic AgentsImmunologic Factors +3
Target Protein:
Dihydroneopterin aldolase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brotizolam DB09017
small molecule | CAS: 57801-81-7

Brotizolam is a sedative-hypnotic thienodiazepine drug which is a benzodiazepine analog. It demonstrates anxiolytic, anticonvulsant, hypnotic, sedative and skeletal muscle relaxant effects. Brotizolam has similar effects to short-acting benzodiazepines such a…

Kategori:
Benzodiazepine hypnotics and sedativesBenzodiazepines and benzodiazepine derivativesCentral Nervous System Agents +7
Target Protein:
GABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu Paruh4.4 hours.
Vol. Distribusi0.63 l/kg.
KlirensTotal clearance: 10…
Genetik -
biotech

Broussonetia papyrifera pollen is the pollen of the Broussonetia papyrifera plant. Broussonetia papyrifera pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brovanexine DB14720
small molecule | CAS: 54340-61-3

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brown iron oxide Approved DB14567
small molecule | CAS: 52357-70-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Broxyquinoline DB13536
small molecule | CAS: 521-74-4

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAntidiarrheals, Intestinal Antiinflammatory/antiinfective AgentsAntiparasitic Products, Insecticides and Repellents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bryostatin 1 DB11752
small molecule | CAS: 83314-01-6

Bryostatin 1 has been investigated for the treatment of HIV Infection and Alzheimer's Disease.

Kategori:
Adjuvants, ImmunologicAnti-Bacterial AgentsAntineoplastic Agents +15
Target Protein:
Protein kinase C epsilon typeProtein kinase C alpha typeCaspase-8 +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BS-001 DB17415
biotech

BS-001 is a recombinant oncolytic herpes simplex virus type II (OH2) therapeutic injection (Vero cell) for human use (rHSV2hGM-CSF).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BSK02 DB17434
biotech

BSK02 is a Sperm Protein-17 oral microparticle vaccine

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BTA798 DB05181
small molecule

BTA798 is an antiviral for the treatment of HRV, the common cold virus, known to cause significant clinical complications in sufferers of Asthma and Chronic Obstructive Pulmonary Disease.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BTRX-246040 DB16048
small molecule | CAS: 1307245-86-8

BTRX-246040 is under investigation in clinical trial NCT03193398 (BTRX-246040 Administered Once Daily to Patients With Major Depressive Disorder).

Target Protein:
Nociceptin receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BTZ-043 DB17737
small molecule | CAS: 1161233-85-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bucelipase alfa DB16664
biotech | CAS: 9026-00-0

Bucelipase alfa is under investigation in clinical trial NCT00743483 (Efficacy of Bucelipase Alfa (BSSL) in Patients With Cystic Fibrosis and Pancreatic Insufficiency).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bucetin Approved DB13278
small molecule | CAS: 1083-57-4

Bucetin is an analgesic and antipyretic medication which was approved for use in Germany but was withdrawn from the market in 1986 due to renal toxicity caused by the medication.[A175636]

Kategori:
AminesAminophenolsAnalgesics +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bucillamine DB12160
small molecule | CAS: 65002-17-7

Bucillamine has been used in trials studying the treatment and prevention of Gout and Rheumatoid Arthritis.

Kategori:
Amino AcidsAmino Acids, NeutralAmino Acids, Peptides, and Proteins +17
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bucindolol DB12752
small molecule | CAS: 71119-11-4

Bucindolol has been investigated in Heart Failure.

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +17
Target Protein:
Beta-2 adrenergic receptorBeta-1 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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