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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 62 / 252
BI-K0376 DB05858
biotech

BI-K0376 is investigated for use/treatment in acne. BI-K0376 is a solid. It is under investigation by Pfizer and has gone through phase I of the clinical trails.

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Bibenzonium DB13630
small molecule | CAS: 59866-76-1

Deskripsi belum tersedia.

Kategori:
Cough and Cold Preparations
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Bibrocathol DB13818
small molecule | CAS: 6915-57-7

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsBenzene DerivativesOphthalmologicals +2
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Bicalutamide Approved DB01128
small molecule | CAS: 90357-06-5

Bicalutamide is an oral non-steroidal anti-androgen for prostate cancer. It is comprised of a racemic mixture that is a 50:50 composition of the (R)-bicalutamide and (S)-bicalutamide enantionmers. Bicalutamide binds to the androgen receptor.

Kategori:
AmidesAminesAndrogen Receptor Antagonists +31
Target Protein:
Androgen receptor
Waktu Paruh5.9 days
Vol. Distribusi-
Klirens* Apparent oral cl=…
Genetik -
Bicifadine DB04889
small molecule | CAS: 71195-57-8

Bicifadine (DOV-220075) is a nonopioid analgesic. It is an inhibitor of both the norepinephrine and serotonin transporters and an NMDA antagonist with a non-narcotic profile. Bicifadine was shown to have potent analgesic activity in vivo and was chosen for fu…

Kategori:
AnalgesicsCytochrome P-450 CYP1A2 SubstratesCytochrome P-450 CYP2D6 Substrates +2
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporterD(2) dopamine receptor
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Bicine DB03709
small molecule | CAS: 150-25-4

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, Peptides, and Proteins
Target Protein:
PlasminogenMembrane-bound lytic murein transglycosylase BUDP-galactopyranose mutase
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Bicisate Approved DB11164
small molecule | CAS: 121251-02-3

Bicisate, also known as ethyl cysteinate dimer (ECD), is a N,N'-1,2-ethylene-di-yl-bis-L-cysteinate diethyl ester. It is used in conjunction with technetium Tc99m as a tracer to measure cerebral blood flow with single-photon emission computed tomography (SPEC…

Kategori:
Diagnostic AgentsDrugs that are Mainly Renally ExcretedRadioactive Diagnostic Agent
Waktu ParuhThe stability of bi…
Vol. DistribusiAfter intravenous a…
KlirensThe clearance of bi…
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Bicuculline DB11562
small molecule | CAS: 485-49-4

Bicuculline is a light-sensitive competitive antagonist of GABAA receptors. It was originally identified in 1932 in plant alkaloid extracts and has been isolated from Dicentra cucullaria, Adlumia fungosa, Fumariaceae, and several Corydalis species.

Kategori:
AlkaloidsBenzylisoquinolinesCentral Nervous System Agents +8
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Bicyclol DB16014
small molecule | CAS: 118159-48-1

Bicyclol is under investigation in clinical trial NCT02944552 (The Multi Center, Randomized, Double-blind, Positive Controlled Study of Bicyclol in the Treatment of Acute DILI).

Kategori:
Benzene Derivatives
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Bietaserpine DB13575
small molecule | CAS: 53-18-9

Deskripsi belum tersedia.

Kategori:
AlkaloidsAntiadrenergic Agents, Centrally ActingAntihypertensive Agents +7
Waktu Paruh-
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Bifemelane DB13550
small molecule | CAS: 90293-01-9

Deskripsi belum tersedia.

Kategori:
Antidepressive AgentsBenzene DerivativesCentral Nervous System Agents +5
Target Protein:
Amine oxidase [flavin-containing] A
Waktu Paruh-
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Bifenthrin DB15056
small molecule | CAS: 82657-04-3

Bifenthrin is under investigation in clinical trial NCT01560247 (Percutaneous Recanalization in Ischemic Stroke Management in Europe Observational Registry).

Kategori:
Cyclopentane MonoterpenesMonoterpenesSarcoma, Experimental, chemically induced +1
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Bifeprunox DB04888
small molecule | CAS: 350992-10-8

Bifeprunox is a novel atypical antipsychotic agent which, along with SLV313, [aripiprazole] and SSR-181507 combines minimal D2 receptor agonism with 5-HT receptor agonism.

Kategori:
Antipsychotic AgentsAntipsychotic Agents (Second Generation [Atypical])Central Nervous System Depressants +2
Target Protein:
5-hydroxytryptamine receptor 1AD(2) dopamine receptor
Waktu Paruh-
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biotech

Deskripsi belum tersedia.

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Bifidobacterium bifidum Approved DB16538
biotech

Deskripsi belum tersedia.

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biotech

Deskripsi belum tersedia.

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biotech

Bifidobacterium Longum Infantis 35624 is a probiotic being investigated for the treatment of gastrointestinal disorders, such as Crohn's disease and irritable bowel syndrome.[A259872, A259877]

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biotech

Deskripsi belum tersedia.

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Bifikafusp alfa DB19185
biotech | CAS: 1957239-90-5

Bifikafusp alfa is under investigation in clinical trial NCT05329792 (L19IL2/L19TNF in Skin Cancer Patients).

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biotech

Bifunctional epoxide hydrolase 2 is under investigation in clinical trial NCT00654966 (Evaluation of the Effects of Urotensin-II and Soluble Epoxide Hydrolase Inhibitors on Skin Microvessel Tone in Patients With Heart Failure, and in Healthy Volunteers).

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Biguanide Approved DB13100
small molecule | CAS: 56-03-1

Biguanide has been investigated for the treatment of Diabetes Mellitus.

Kategori:
AmidinesBlood Glucose Lowering AgentsGuanidines
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BIIB015 DB06304
biotech

BIIB015 is a humanized, IgG1 [immunoglobulin G 1], DM4-Conjugated, anti-cripto, monoclonal antibody. It has been investigated for the treatment of subjects with relapsed or refractory solid tumours.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +6
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BIIB021 DB12359
small molecule | CAS: 848695-25-0

BIIB021 has been investigated for the treatment of Tumors and Lymphoma.

Kategori:
Heterocyclic Compounds, Fused-RingHSP90 Heat-Shock Proteins, antagonists & inhibitorsPurines
Target Protein:
Heat shock protein HSP 90-alpha
Waktu Paruh-
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BIIB115 DB18418
biotech

BIIB115 is an investigational antisense oligonucleotide in development for spinal muscular atrophy.

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Bilastine Approved DB11591
small molecule | CAS: 202189-78-4

Bilastine is a novel new-generation antihistamine that is highly selective for the H1 histamine receptor, has a rapid onset and prolonged duration of action.

Kategori:
Antihistamines for Systemic UseDecongestants and AntiallergicsHeterocyclic Compounds, Fused-Ring +8
Target Protein:
Histamine H1 receptor
Waktu ParuhThe mean half life …
Vol. Distribusi-
KlirensBilastine has a tot…
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Bilberry Approved DB14235
biotech

Deskripsi belum tersedia.

Kategori:
AngiospermsBenzopyransBiological Factors +21
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small molecule | CAS: 114-25-0

Deskripsi belum tersedia.

Target Protein:
Heme oxygenase 1MyoglobinFlavin reductase (NADPH)
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Bimagrumab DB12584
biotech | CAS: 1356922-05-8

Bimagrumab has been used in trials studying the treatment and supportive care of Sarcopenia, Skeletal Muscle, Mechanical Ventilation, Sporadic Inclusion Body Myositis, and Sporadic Inclusion Body Myositis (sIBM), among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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Bimatoprost Approved DB00905
small molecule | CAS: 155206-00-1

Bimatoprost, also known as Latisse or Lumigan, belongs to a group of drugs called prostamides, which are synthetic structural analogs of prostaglandin. Bimatoprost, marketed by Allergan, is administered in both the ophthalmic solution and implant form. It has…

Kategori:
AmidesAntiglaucoma Preparations and MioticsAntihypertensive Agents +19
Target Protein:
Prostaglandin F2-alpha receptorProstaglandin E2 receptor EP1 subtypeProstaglandin E2 receptor EP3 subtype
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance was m…
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Bimekizumab Approved DB12917
biotech | CAS: 1418205-77-2

Bimekizumab is a humanized monoclonal antibody directed towards IL-17, which was approved for use in the EU on August 20, 2021, for the treatment of plaque psoriasis.[L39665,L39680] It is the first IL-17 inhibitor to target both IL-17A and IL-17F.[A244455] It…

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAntibodies +11
Target Protein:
Interleukin-17AInterleukin-17F
Waktu ParuhThe mean terminal e…
Vol. DistribusiIn patients with pl…
KlirensThe median apparent…
Genetik -
Bimiralisib DB14846
small molecule | CAS: 1225037-39-7

Bimiralisib is under investigation in clinical trial NCT02723877 (PQR309 and Eribulin in Metastatic HER2 Negative and Triple-negative Breast Cancer (PIQHASSO)).

Target Protein:
Serine/threonine-protein kinase mTORPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Bimoclomol DB06258
small molecule | CAS: 130493-03-7

Bimoclomol is an investigational drug that induces stress proteins and has cytoprotective effects.

Target Protein:
Heat shock 70 kDa protein 1BHeat shock 70 kDa protein 1AHeat shock factor protein 1
Waktu Paruh-
Vol. Distribusi-
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Bimosiamose DB06197
small molecule | CAS: 187269-40-5

Deskripsi belum tersedia.

Kategori:
AlkanesBenzene DerivativesCarbohydrates +3
Target Protein:
E-selectin
Waktu Paruh-
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Binetrakin DB12182
biotech | CAS: 207137-56-2

Binetrakin has been used in trials studying the treatment of HIV Infections, Sarcoma, Kaposi, Non-Hodgkin's Lymphoma (NHL), Myelodysplastic Syndrome (MDS), and Leukemia, Acute Myelogenous (AML), among others.

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntineoplastic Agents +9
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Binimetinib Approved DB11967
small molecule | CAS: 606143-89-9

Binimetinib, also known as _Mektovi_, is a potent and selective oral mitogen-activated protein kinase 1/2 (MEK 1/2) inhibitor which is combined with [Encorafenib].[A34275,L3335] On June 27, 2018, the Food and Drug Administration approved the combination of…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +16
Target Protein:
Dual specificity mitogen-activated protein kinase kinase 2Dual specificity mitogen-activated protein kinase kinase 1
Waktu ParuhThe mean (CV%) term…
Vol. DistribusiThe geometric mean …
KlirensThe apparent cleara…
Genetik -
Binodenoson DB04853
small molecule | CAS: 144348-08-3

Binodenoson is a pharmacologic stress agent specific to the only adenosine receptor necessary for increased cardiac blood flow, the A<sub>2A</sub> receptor. This specificity allows Binodenoson to deliver - in a single injection - a more effective dose of medi…

Kategori:
Heterocyclic Compounds, Fused-RingNeurotransmitter AgentsNucleic Acids, Nucleotides, and Nucleosides +7
Target Protein:
Adenosine receptor A2a
Waktu Paruh10 &plusmn; 4 minut…
Vol. Distribusi-
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Bintrafusp alfa DB15387
biotech | CAS: 1918149-01-5

Bintrafusp alfa is under investigation in clinical trial NCT03833661 (M7824 Monotherapy in Locally Advanced or Metastatic Second Line (2L) Biliary Tract Cancer (Cholangiocarcinoma and Gallbladder Cancer)).

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Bioallethrin Approved DB13746
small molecule | CAS: 584-79-2

Bioallethrin refers to a mixture of two of the allethrin isomers (1R,trans;1R and 1R,trans;1S) in an approximate ratio of 1:1, where both isomers are active ingredients. A mixture of the two same stereoisomers, but in an approximate ratio of R:S in 1:3, is ca…

Kategori:
Agents causing hyperkalemiaAgrochemicalsAntiarrhythmic agents +21
Target Protein:
Sodium channel proteinVoltage-gated sodium channel alpha subunitVoltage-dependent calcium channel +3
Waktu Paruh-
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Biochanin A DB15334
small molecule | CAS: 491-80-5

Biochanin A is under investigation in clinical trial NCT02174666 (Isoflavone Treatment for Postmenopausal Osteopenia.).

Kategori:
Anticarcinogenic AgentsAntineoplastic AgentsBenzopyrans +12
Target Protein:
Steroid hormone receptor ERR1AromataseFatty acid synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Biomed 101 DB05851
small molecule

Biomed 101 is investigated for use/treatment in adverse effects (chemotherapy) and renal cell carcinoma. Biomed 101 is a solid. Biomed 101 binds to the leukotriene B4 receptor, but does not affect interleukin-2 antitumor activity.

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Biomodulin T DB16529
biotech

Biomodulin T is a polypeptide fraction from bovine thymus with immunomodulatory effects.

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Biotin Approved DB00121
small molecule | CAS: 58-85-5

A water-soluble, enzyme co-factor present in minute amounts in every living cell. It occurs mainly bound to proteins or polypeptides and is abundant in liver, kidney, pancreas, yeast, and milk.

Kategori:
Alimentary Tract and MetabolismCoenzymesDiet, Food, and Nutrition +10
Target Protein:
Propionyl-CoA carboxylase beta chain, mitochondrialBiotin--protein ligaseMethylcrotonoyl-CoA carboxylase beta chain, mitochondrial +5
Waktu Paruh-
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BIOTINOL-5-AMP DB04651
small molecule

Deskripsi belum tersedia.

Target Protein:
Bifunctional ligase/repressor BirA
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Streptavidin
Waktu Paruh-
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Bioymifi DB17493
small molecule | CAS: 1420071-30-2

Bioymifi is a small molecule that acts as a tumor necrosis factor-related apoptosis-induced ligand (TRAIL) mimetic. Upon binding to the death receptor 5 (DR5) on cancer cells, bioymifi triggers apoptosis, possibly through a caspase-dependent pathway. Bioymifi…

Kategori:
Acids, CarbocyclicHeterocyclic Compounds, Fused-RingImides +5
Target Protein:
Tumor necrosis factor receptor superfamily member 10B
Waktu Paruh-
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Biperiden Approved DB00810
small molecule | CAS: 514-65-8

A muscarinic antagonist that has effects in both the central and peripheral nervous systems. It has been used in the treatment of arteriosclerotic, idiopathic, and postencephalitic parkinsonism. It has also been used to alleviate extrapyramidal symptoms induc…

Kategori:
Agents producing tachycardiaAnti-Dyskinesia AgentsAnti-Parkinson Drugs +18
Target Protein:
Muscarinic acetylcholine receptor M1
Waktu Paruh-
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small molecule | CAS: 792-74-5

Nissel has been investigated for the treatment of Chronic Liver Disease.

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Birabresib DB15189
small molecule | CAS: 202590-98-5

Birabresib is under investigation in clinical trial NCT02698176 (A Dose Exploration Study With MK-8628 in Participants With Selected Advanced Solid Tumors (MK-8628-006)).

Kategori:
AmidesAminesAnilides +2
Target Protein:
Bromodomain-containing protein 2Bromodomain-containing protein 4
Waktu Paruh-
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Birch bark extract Approved DB16536
small molecule | CAS: 84012-15-7

Birch bark extract is rich in triterpenoids with beneficial biological and pharmacological activities. Some of the compounds identified in it include betulin, [lupeol], [betulinic acid], oleanolic acid, and erythrodiol.[A249945] Birch bark extract is obtained…

Kategori:
Anti-Inflammatory AgentsAnti-inflammatory Agents, MiscellaneousBiological Products +7
Waktu ParuhThis pharmacokineti…
Vol. DistribusiThis pharmacokineti…
KlirensThis pharmacokineti…
Genetik -
Biricodar DB04851
small molecule | CAS: 159997-94-1

The pipecolinate derivative biricodar (VX-710) is a clinically applicable modulator of P-glycoprotein (Pgp) and multidrug resistance protein (MRP-1).

Kategori:
P-glycoprotein inhibitors
Target Protein:
ATP-dependent translocase ABCB1ATP-binding cassette sub-family B member 5Multidrug resistance-associated protein 1 +1
Waktu Paruh-
Vol. Distribusi-
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