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3253

Total database: 17430
Struktur (SMILES)
2451 (75.3%)
Target
1833 (56.3%)
Genomik
35 (1.1%)
Referensi
3253 (100.0%)

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Hasil Pencarian (3253)

Halaman 62 / 66
Trilaciclib Approved DB15442
small molecule | CAS: 1374743-00-6

Trilaciclib, or G1T28, is a CDK4 and CDK6 inhibitor, indicated to reduce the incidence of chemotherapy induced myelosuppression in patients before topotecan-containing or platinum and etoposide-containing chemotherapy for extensive stage small cell lung cance…

Kategori:
BCRP/ABCG2 SubstratesCyclin-dependent Kinase 4 InhibitorsCyclin-dependent Kinase 6 Inhibitors +16
Target Protein:
Cyclin-dependent kinase 4Cyclin-dependent kinase 6Cyclin-dependent kinase 9 +3
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of tr…
Genetik -
Trimegestone DB13129
small molecule | CAS: 74513-62-5

Trimegestone has been used in trials studying the treatment of Postmenopause.

Kategori:
Fused-Ring CompoundsGenito Urinary System and Sex HormonesNorpregnadienes +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trimethadione Approved DB00347
small molecule | CAS: 127-48-0

An anticonvulsant effective in absence seizures, but generally reserved for refractory cases because of its toxicity. (From AMA Drug Evaluations Annual, 1994, p378)

Kategori:
Agents causing hyperkalemiaAnti-epileptic AgentAntiarrhythmic agents +18
Target Protein:
Voltage-dependent T-type calcium channel subunit alpha-1G
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trimetrexate Approved DB01157
small molecule | CAS: 52128-35-5

A nonclassical folic acid inhibitor through its inhibition of the enzyme dihydrofolate reductase. It is being tested for efficacy as an antineoplastic agent and as an antiparasitic agent against pneumocystis pneumonia in AIDS patients. Myelosuppression is its…

Kategori:
Acids, AcyclicAcids, AldehydicAnti-Infective Agents +18
Target Protein:
Peptide deformylase, mitochondrialDihydrofolate reductase
Waktu Paruh11 to 20 hours
Vol. Distribusi* 20 ± 8 L/m2 * 36…
Klirens* 38 +/- 15 mL/min/…
Genetik -
Triphendiol DB06588
small molecule | CAS: 1213777-80-0

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesFlavonoids +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Triprolidine Approved DB00427
small molecule | CAS: 486-12-4

First generation histamine H1 antagonist used in allergic rhinitis; asthma; and urticaria. It is a component of cough and cold medicines. It may cause drowsiness.

Kategori:
Anti-Allergic AgentsAntihistamines for Systemic UseCentral Nervous System Depressants +7
Target Protein:
Histamine H1 receptor
Waktu Paruh4 to 6 hours.
Vol. Distribusi-
Klirens-
Genetik -
Triptolide DB12025
small molecule | CAS: 38748-32-2

Triptolide has been used in trials studying the treatment of HIV, Crohn's Disease, Intestinal Diseases, Gastrointestinal Diseases, and Digestive System Diseases, among others.

Kategori:
Adrenal Cortex HormonesAlkylating DrugsAntineoplastic Agents +10
Target Protein:
Transcription factor RelBNuclear factor NF-kappa-B p105 subunitNuclear factor NF-kappa-B p100 subunit +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trofosfamide DB12902
small molecule | CAS: 22089-22-1

Trofosfamide has been used in trials studying the treatment of Ependymomas, Medulloblastomas, Sarcoma, Soft Tissue, Supratentorial PNETs, and Recurrent Brain Tumors.

Kategori:
Alkylating DrugsAntineoplastic AgentsAntineoplastic Agents, Alkylating +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Troxerutin DB13124
small molecule | CAS: 7085-55-4

Troxerutin has been used in trials studying the treatment of Chronic Venous Insufficiency.

Kategori:
AnticoagulantsBenzopyransCapillary Stabilizing Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TRV-120027 DB12199
small molecule | CAS: 1234510-46-3

TRV120027 has been used in trials studying the treatment of Heart Failure and Kidney Disease.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Target Protein:
Type-1 angiotensin II receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trypsin Approved DB11237
small molecule | CAS: 9002-07-7

Trypsin is a serine protease that plays an essential role in protein hydrolysis and absorption in mammals. When converted from its zymogen trypsinogen, trypsin is available as an active peptide hydrolase (EC 3.4.21.4) form to cleave peptide chains, mainly at …

Kategori:
Blood and Blood Forming OrgansDermatologicalsEndopeptidases +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tryptophan Approved DB00150
small molecule | CAS: 73-22-3

An essential amino acid that is necessary for normal growth in infants and for nitrogen balance in adults. It is a precursor of indole alkaloids in plants. It is a precursor of serotonin (hence its use as an antidepressant and sleep aid). It can be a precurso…

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +14
Target Protein:
Indoleamine 2,3-dioxygenase 1Tryptophan--tRNA ligase, cytoplasmicTryptophan--tRNA ligase +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TSHA-120 DB16985
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TSN-084 DB18306
small molecule | CAS: 2412309-60-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TT-232 DB12088
small molecule | CAS: 147159-51-1

Tln 232 is under investigation in clinical trial NCT00422786 (Phase II Study of CAP-232 in Patients With Refractory Metastatic Renal Cell Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +8
Target Protein:
Pyruvate kinase PKM
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TT-301 DB12899
small molecule | CAS: 886208-76-0

TT301 has been used in trials studying the treatment of Traumatic Brain Injury.

Target Protein:
Interleukin-1 beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TU-100 DB12467
small molecule | CAS: 1310907-71-1

TU-100 has been used in trials studying the treatment of Abdominal Pain, Colonic Transit, Crohn's Disease, Rectal Sensation, and Gastric Emptying, among others.

Kategori:
DNA Topoisomerases, Type IINaphthalenesQuinones +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tuaminoheptane DB13238
small molecule | CAS: 123-82-0

Deskripsi belum tersedia.

Kategori:
Nasal PreparationsSympathomimetics, Plain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 92129-86-7

Tuberculin Purified Protein Derivative (PPD) is a sterile aqueous solution of a purified protein fraction for intradermal administration as an aid in the diagnosis of tuberculosis. The diagnostic test is commonly referred to as the Mantoux test which serves t…

Kategori:
Amino Acids, Peptides, and ProteinsAntigensAntigens, Bacterial +12
Target Protein:
Toll-like receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tubocurarine Approved DB01199
small molecule | CAS: 57-95-4

Tubocurarine is a non-depolarizing neuromuscular blocking agent and the first identified curare alkaloid.[A216008] Curare is one of the names used to describe plant-derived poisons used by indigenous South Americans to coat the tips of hunting arrows and dart…

Kategori:
AlkaloidsAminesAnticholinergic Agents +23
Target Protein:
Neuronal acetylcholine receptor subunit alpha-25-hydroxytryptamine receptor 3AAcetylcholinesterase +1
Waktu Paruh1-2 hours
Vol. Distribusi-
Klirens-
Genetik -
Tucatinib Approved DB11652
small molecule | CAS: 937263-43-9

Tucatinib is a kinase inhibitor drug used with [trastuzumab] and [capecitabine] in the treatment of unresectable or metastatic HER-2 positive breast cancer. It was developed by Seattle Genetics and approved by the FDA on April 17, 2020.[L12951] Tucatinib is a…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +18
Target Protein:
Receptor tyrosine-protein kinase erbB-2Receptor tyrosine-protein kinase erbB-3
Waktu ParuhA pharmacokinetic s…
Vol. DistribusiThe volume of distr…
KlirensThe apparent cleara…
Genetik -
Tulobuterol DB12248
small molecule | CAS: 41570-61-0

Tulobuterol has been used in trials studying the treatment of Chronic Obstructive Pulmonary Disease.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-Agonists +17
Target Protein:
Beta-2 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TUM012 DB18652
biotech

TUM012 is a synthetic polymer PEG conjugated to a phospholipid anchor (2-dipalmitoyl-sn-glycerol-3-phosphatidylethanolamine)

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tuparstobart DB19118
biotech | CAS: 2649466-03-3

Tuparstobart is under investigation in clinical trial NCT05287113 (Study of Retinfanlimab in Combination With INCAGN02385 and INCAGN02390 as First-line Treatment in Participants With Pd-l1-positive (CPS ? 1) Recurrent/metastatic Squamous Cell Carcinoma of the…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 629664-81-9

Fxr 450 is under investigation in clinical trial NCT00509756 (Study Evaluating Turofexorate isopropyl in Healthy Japanese Men).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Bile acid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Turpentine Approved DB11120
small molecule | CAS: 9005-90-7

Turpentine, also known as spirit of turpentine, oil of turpentine, and wood turpentine, is a liquid extracted from live trees, mainly pine, through distillation of resin. It is used as a solvent and base material in organic synthesis reactions. Turpentine is …

Kategori:
Biological ProductsComplex MixturesCompounds used in a research, industrial, or household setting +9
Target Protein:
Mitogen-activated protein kinase 1
Waktu ParuhEight male voluntee…
Vol. DistribusiTurpentine, as a li…
Klirens-
Genetik -
Tylvalosin DB11554
small molecule | CAS: 63409-12-1

Deskripsi belum tersedia.

Kategori:
Anti-Bacterial AgentsLactonesMacrolides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tyrosine Approved DB00135
small molecule | CAS: 60-18-4

Tyrosine is a non-essential amino acid. In animals it is synthesized from [phenylalanine]. It is also the precursor of [epinephrine], thyroid hormones, and melanin.

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +4
Target Protein:
Tyrosine 3-monooxygenaseTyrosine--tRNA ligase, mitochondrialTyrosine--tRNA ligase, cytoplasmic +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tyvelose DB04028
small molecule | CAS: 5658-12-8

Deskripsi belum tersedia.

Kategori:
CarbohydratesMonosaccharides
Target Protein:
Tail fiber protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TZP-102 DB16129
small molecule | CAS: 1008993-65-4

TZP-102 is under investigation in clinical trial NCT01452815 (Affects of Once-daily Oral Administration of TZP-102 on the Treatment of Symptoms Associated With Diabetic Gastroparesis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
U-0126 DB17060
small molecule | CAS: 218601-62-8

U-0126 is a direct inhibitor of the mitogen-activated protein-kinase kinase family members, MEK-1 and MEK-2.[A253162]

Kategori:
AlkadienesAlkenesEnzyme Inhibitors +2
Target Protein:
Mitogen-activated protein kinase kinase kinase 2Mitogen-activated protein kinase kinase kinase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
UB-612 DB16444
biotech

The UB-612 COVID-19 vaccine was developed by United Biomedical Inc Asia in Taipei as the first COVID-19 “multi-tope” protein-peptide vaccine made up of eight rationally designed components[L30653]. The vaccine incorporates a strong S1-RBD component linked to …

Kategori:
Biological ProductsComplex MixturesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ublituximab Approved DB11850
biotech | CAS: 1174014-05-1

CD20, an antigen expressed by various B and T cells, is an attractive therapeutic target in various cancers and autoimmune conditions.[A244195, A244200, A244205] Monoclonal antibodies for B cell depletion rely on their binding affinity and ability to clear bo…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Target Protein:
B-lymphocyte antigen CD20
Waktu ParuhThe estimated mean …
Vol. DistribusiThe estimated centr…
Klirens-
Genetik -
UK-396,082 DB12099
small molecule | CAS: 400044-47-5

UK-396,082 has been used in trials studying the basic science of Safety, Phase 1, Toleration, Multiple Dose, and Pharmacokinetic.

Kategori:
Amino Acids, Peptides, and Proteins
Target Protein:
Carboxypeptidase B2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
UK-432097 DB12691
small molecule | CAS: 380221-63-6

UK-432,097 has been used in trials studying the treatment of Pulmonary Disease, Chronic Obstructive.

Kategori:
Adenosine A receptor agonistsAdenosine A2 Receptor AgonistsHeterocyclic Compounds, Fused-Ring +5
Target Protein:
Adenosine receptor A2a
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
UK-500001 DB12837
small molecule | CAS: 582332-31-8

UK-500,001 has been used in trials studying the treatment of Pulmonary Disease, Chronic Obstructive.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ukrain cation DB17150
small molecule | CAS: 732958-87-1

Deskripsi belum tersedia.

Kategori:
Adjuvants, ImmunologicAlkaloidsAntineoplastic Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ularitide DB05034
small molecule | CAS: 118812-69-4

Ularitide is a synthetic form of urodilatin, a naturally occurring human natriuretic peptide that is involved in regulating blood pressure and the excretion of water and sodium from the kidneys. Urodilatin is produced in the kidney and excreted into the urine…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Asthmatic AgentsAutonomic Agents +10
Target Protein:
Atrial natriuretic peptide receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ulimorelin DB12128
small molecule | CAS: 842131-33-3

Ulimorelin is a novel small molecule ghrelin agonist being developed by Tranzyme Pharma as a first-in-class treatment for both POI and diabetic gastroparesis, serious medical conditions in which motility of the GI tract is severely impaired.

Target Protein:
Growth hormone secretagogue receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ulinastatin DB12038
biotech | CAS: 80449-31-6

Ulinastatin has been investigated for the prevention of Cardiovascular Disease and Adverse Reaction to Drug.

Kategori:
Amino Acids, Peptides, and ProteinsAntifibrinolytic AgentsBlood and Blood Forming Organs +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ulocuplumab DB12018
biotech | CAS: 1375830-34-4

Ulocuplumab is under investigation in Solid Tumor.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Target Protein:
C-X-C chemokine receptor type 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ulodesine DB12353
small molecule | CAS: 548486-59-5

Ulodesine has been used in trials studying the treatment of Gout, Arthritis, Hyperuricemia, and Joint Disease.

Kategori:
CarbohydratesIminesImino Sugars +3
Target Protein:
Purine nucleoside phosphorylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ulviprubart DB18281
biotech | CAS: 2569434-60-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Umifenovir DB13609
small molecule | CAS: 131707-25-0

Umifenovir is an indole-based, hydrophobic, dual-acting direct antiviral/host-targeting agent used for the treatment and prophylaxis of influenza and other respiratory infections.[A191475] It has been in use in Russia for approximately 25 years and in China s…

Kategori:
AnionsAntiinfectives for Systemic UseAntiviral Agents +19
Waktu ParuhThe half-life of um…
Vol. DistribusiData regarding the …
KlirensIn a study involvin…
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Lysozyme C
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Undecanal DB04093
small molecule | CAS: 112-44-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Undecanoic acid DB16857
small molecule | CAS: 112-37-8

Deskripsi belum tersedia.

Kategori:
Lipids
Target Protein:
G-protein coupled receptor 84
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Undecylenic acid Approved DB11117
small molecule | CAS: 112-38-9

Undecylenate, or undecylenic acid, is an unsaturated fatty acid with a terminal double bond that is derived from castor oil. Undecylenic acid is also found naturally in the human sweat. It is used as a precursor in the manufacture of aromatic chemicals, polym…

Kategori:
Antifungals for Dermatological UseAntifungals for Topical UseDermatologicals +4
Target Protein:
Calpain-1 catalytic subunit
Waktu ParuhNo information rega…
Vol. DistribusiNo information rega…
KlirensNo information rega…
Genetik -
Unoprostone Approved DB06826
small molecule | CAS: 120373-36-6

Unoprostone isopropyl is a prostaglandin analogue. Ophthalmic Solution 0.15% is a synthetic docosanoid. Unoprostone isopropyl has the chemical name isopropyl (+)-(Z)-7-[(1R,2R,3R,5S)-3,5 dihydroxy-2-(3-oxodecyl)cyclopentyl]-5-heptenoate. The main indication …

Kategori:
Antiglaucoma Preparations and MioticsAntihypertensive AgentsAutacoids +12
Waktu ParuhHalf-life of Unopr…
Vol. DistribusiIntended for local …
KlirensIntended for local …
Genetik -
Uproleselan DB14829
small molecule | CAS: 1983970-12-2

Uproleselan is a novel, specific E-Selectin antagonist under investigation in clinical trial NCT02306291 (Study to Determine Safety, Pharmacokinetics and Efficacy of GMI-1271 in Combination With Chemotherapy in AML).

Kategori:
CarbohydratesE-Selectin, antagonists & inhibitorsGlycoconjugates +1
Target Protein:
E-selectin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 3051–3100 dari 3253
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