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6694

Total database: 17430
Struktur (SMILES)
4518 (67.5%)
Target
3751 (56.0%)
Genomik
81 (1.2%)
Referensi
6694 (100.0%)

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Hasil Pencarian (6694)

Halaman 61 / 134
Glatiramer Approved DB05259
biotech | CAS: 28704-27-0

Glatiramer acetate is a mix of synthetic polypeptides that includes L-glutamic acid, L-alanine, L-tyrosine, and L-lysine at an average molar fraction of 0.141, 0.427, 0.095, and 0.338, respectively.[L41940] Since glatiramer acetate is a heterogeneous drug, th…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating Agents +5
Target Protein:
MHC class II protein complex
Waktu ParuhNot available.
Vol. DistribusiNot available.
KlirensNot available.
Genetik -
Glecaprevir Approved DB13879
small molecule | CAS: 1365970-03-1

Glecaprevir is a direct acting antiviral agent and Hepatitis C virus (HCV) NS3/4A protease inhibitor that targets the the viral RNA replication. In combination with [DB13878], glecaprevir is a useful therapy for patients who experienced therapeutic failure fr…

Kategori:
Acids, AcyclicAmidesAmino Acids +37
Target Protein:
NS3 proteaseGenome polyprotein
Waktu ParuhThe elimination hal…
Vol. Distribusi-
Klirens-
Genetik -
Glecirasib DB18744
small molecule | CAS: 2657613-87-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Glenzocimab DB16175
biotech | CAS: 2101829-58-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gleptoferron DB11417
small molecule | CAS: 57680-55-4

Colloid solution of ferric hydroxide, dextran & glucoheptonic acid.

Kategori:
Acids, AcyclicCarbohydratesCompounds used in a research, industrial, or household setting +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gliclazide Approved DB01120
small molecule | CAS: 21187-98-4

Gliclazide is an oral antihyperglycemic agent used for the treatment of non-insulin-dependent diabetes mellitus (NIDDM). It has been classified differently according to its drug properties in which based on its chemical structure, gliclazide is considered a f…

Kategori:
Alimentary Tract and MetabolismAmidesBenzene Derivatives +15
Target Protein:
ATP-binding cassette sub-family C member 8Vascular endothelial growth factor A, long form
Gen Terkait:
CYP2C19 CYP2C19
Waktu Paruh10.4 hours. Duratio…
Vol. Distribusi-
Klirens-
Genetik 2 Varian
Glimepiride Approved DB00222
small molecule | CAS: 93479-97-1

First introduced in 1995, glimepiride is a member of the second-generation sulfonylurea (SU) drug class used for the management of type 2 diabetes mellitus (T2DM) to improve glycemic control. Type 2 diabetes is a metabolic disorder with increasing prevalences…

Kategori:
Alimentary Tract and MetabolismAmidesBlood Glucose Lowering Agents +12
Target Protein:
ATP-binding cassette sub-family C member 9ATP-sensitive inward rectifier potassium channel 11ATP-sensitive inward rectifier potassium channel 1 +1
Waktu ParuhThe elimination hal…
Vol. DistribusiFollowing intraveno…
KlirensA single-dose, cros…
Genetik -
Glipizide Approved DB01067
small molecule | CAS: 29094-61-9

Glipizide is an oral hypoglycemic agent in the second-generation sulfonylurea drug class that is used to control blood sugar levels in patients with type 2 diabetes mellitus. It was first introduced in 1984 [A179491] and is available in various countries incl…

Kategori:
Alimentary Tract and MetabolismBlood Glucose Lowering AgentsBSEP/ABCB11 Substrates +11
Target Protein:
ATP-binding cassette sub-family C member 8ATP-sensitive inward rectifier potassium channel 10Peroxisome proliferator-activated receptor gamma
Gen Terkait:
CYP2C9
Waktu ParuhThe mean terminal e…
Vol. DistribusiThe mean volume of …
KlirensThe mean total body…
Genetik 1 Varian
Glisoxepide DB01289
small molecule | CAS: 25046-79-1

Glisoxepide is one of the sulphonamide-derived oral antidiabetic drugs. It inhibits the uptake of bile acids into isolated rat hepatocytes. However it inhibits taurocholate uptake only in the absence of sodium ions. Glisoxepide uptake could be further inhibit…

Kategori:
Alimentary Tract and MetabolismAmidesBlood Glucose Lowering Agents +8
Target Protein:
ATP-sensitive inward rectifier potassium channel 10ATP-sensitive inward rectifier potassium channel 8Insulin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Glofitamab Approved DB16371
biotech | CAS: 2229047-91-8

Glofitamab is a full-length bispecific monoclonal antibody with affinity for both CD20 and CD3 surface antigens found on B- and T-cells, respectively. It has a 2:1 configuration, with bivalency towards CD20 and monovalency towards CD3, and works by recruiting…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
B-lymphocyte antigen CD20T-cell surface glycoprotein CD3
Waktu ParuhThe transition from…
Vol. DistribusiFollowing intraveno…
KlirensGlofitamab's serum …
Genetik -
Glucagon Approved DB00040
biotech | CAS: 16941-32-5

Glucagon is a 29 amino acid hormone used as a diagnostic aid in radiologic exams to temporarily inhibit the movement of the gastrointestinal tract and to treat severe hypoglycemia.[L7634,L7637,L7640,L7643,L8519] Glucagon raises blood sugar through activation …

Kategori:
Amino Acids, Peptides, and ProteinsAntihypoglycemic AgentDecreased GI Motility +19
Target Protein:
Glucagon receptorGlucagon-like peptide 2 receptorGlucagon-like peptide 1 receptor
Waktu ParuhThe half life of gl…
Vol. DistribusiThe volume of distr…
KlirensA 1mg intravenous d…
Genetik -
biotech | CAS: 223460-79-5

Glucagon-like peptide II is under investigation for the basic science of Short Bowel Syndrome.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Glucaric acid DB03603
small molecule | CAS: 87-73-0

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicCarbohydratesHydroxy Acids +1
Target Protein:
Glucarate dehydratase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Glucarpidase Approved DB08898
biotech | CAS: 9074-87-7

Glucarpidase is a recombinant carboxypeptidase G2 produced by genetically modified _Escherichia coli_ bacteria. It is a 390-amino acid homodimer protein.[L39855] High-dose [methotrexate], an antifolate agent, has been widely and safely used for many decades i…

Kategori:
Amino Acids, Peptides, and ProteinsAntidotesCarboxypeptidases +8
Waktu ParuhFollowing intraveno…
Vol. DistribusiIn healthy adults w…
KlirensThe mean systemic c…
Genetik -
Gluconic Acid Approved DB13180
small molecule | CAS: 526-95-4

Commonly found in salts with sodium and calcium. Gluconic acid or gluconate is used to maintain the cation-anion balance on electrolyte solutions.

Kategori:
Acids, AcyclicCarbohydratesChelating Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gluconolactone Approved DB04564
small molecule | CAS: 90-80-2

Gluconolactone is a naturally-occurring food additive used as a sequestrant, an acidifier, or a curing, pickling, or leavening agent. It is a cyclic ester of D-gluconic acid. Pure gluconolactone is a white odorless crystalline powder.

Kategori:
Acids, AcyclicCalculi Dissolution AgentCarbohydrates +3
Target Protein:
Lactase/phlorizin hydrolase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 56-73-5

An ester of glucose with phosphoric acid, made in the course of glucose metabolism by mammalian and other cells. It is a normal constituent of resting muscle and probably is in constant equilibrium with fructose-6-phosphate. (Stedman, 26th ed)

Kategori:
CarbohydratesGlucosephosphatesHexosephosphates +1
Target Protein:
Glutamine--fructose-6-phosphate aminotransferase [isomerizing]Glucose-6-phosphate isomerase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Glutamic acid Approved DB00142
small molecule | CAS: 56-86-0

A peptide that is a homopolymer of glutamic acid.

Kategori:
Acid PreparationsAlimentary Tract and MetabolismAmino Acids +11
Target Protein:
Metabotropic glutamate receptor 1Metabotropic glutamate receptor 4Glutamate receptor ionotropic, kainate 4 +59
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1955-67-5

Deskripsi belum tersedia.

Kategori:
AminesAmino AcidsAmino Acids, Acidic +5
Target Protein:
Glutamine--fructose-6-phosphate aminotransferase [isomerizing]
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Glutaral DB03266
small molecule | CAS: 111-30-8

One of the protein CROSS-LINKING REAGENTS that is used as a disinfectant for sterilization of heat-sensitive equipment and as a laboratory reagent, especially as a fixative.

Kategori:
AldehydesAnti-Infective AgentsCompounds used in a research, industrial, or household setting +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Glutaric Acid DB03553
small molecule | CAS: 110-94-1

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicDicarboxylic AcidsOAT1/SLC22A6 inhibitors +3
Target Protein:
Organic anion transporter 3Aspartate aminotransferaseBranched-chain-amino-acid aminotransferase +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Glutathione Approved DB00143
small molecule | CAS: 70-18-8

A tripeptide with many roles in cells. It conjugates to drugs to make them more soluble for excretion, is a cofactor for some enzymes, is involved in protein disulfide bond rearrangement and reduces peroxides.

Kategori:
Amino Acids, Peptides, and ProteinsAntidotesDietary Supplements +4
Target Protein:
Aldo-keto reductase family 1 member B1Matrix metalloproteinase-9Cytochrome P450 3A4 +38
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 3773-07-7

Deskripsi belum tersedia.

Target Protein:
Glutathione S-transferase Mu 4Glutathione S-transferase A1Glutathione S-transferase P +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Glyburide Approved DB01016
small molecule | CAS: 10238-21-8

Glyburide is a second generation sulfonylurea used to treat patients with diabetes mellitus type II.[L8123] It is typically given to patients who cannot be managed with the standard first line therapy, [metformin].[L8123] Glyburide stimulates insulin secretio…

Kategori:
Alimentary Tract and MetabolismAmidesBCRP/ABCG2 Substrates +28
Target Protein:
ATP-binding cassette sub-family C member 8Sulfonylurea receptor 1, Kir6.2ATP-binding cassette sub-family C member 9 +6
Waktu ParuhElderly patients ha…
Vol. DistribusiElderly patients ha…
KlirensElderly patients ha…
Genetik -
small molecule | CAS: 17181-54-3

Deskripsi belum tersedia.

Kategori:
AlcoholsCarbohydratesLipids +5
Target Protein:
Triosephosphate isomerase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 111-03-5

Deskripsi belum tersedia.

Kategori:
Lipids
Target Protein:
Glucose-dependent insulinotropic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 27215-38-9

Deskripsi belum tersedia.

Kategori:
Cariostatic AgentsCompounds used in a research, industrial, or household settingFatty Acids +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Glyceryl monocaprylate Approved DB19362
small molecule | CAS: 26402-26-6

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicFatty AcidsLipids +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 31566-31-1

Glycerol monostearate, commonly known as GMS, is the glycerol ester of stearic acid . It is commonly used as an emulsifier in foods.

Kategori:
Lipids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Glycinamide DB03636
small molecule | CAS: 598-41-4

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, Peptides, and Proteins
Target Protein:
Neutrophil collagenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsNucleic Acids, Nucleotides, and Nucleosides +1
Target Protein:
Phosphoribosylglycinamide formyltransferase 2Phosphoribosylglycinamide formyltransferaseTrifunctional purine biosynthetic protein adenosine-3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Glycine Approved DB00145
small molecule | CAS: 56-40-6

A non-essential amino acid. It is found primarily in gelatin and silk fibroin and used therapeutically as a nutrient. It is also a fast inhibitory neurotransmitter.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsBlood and Blood Forming Organs +7
Target Protein:
Glutamate receptor ionotropic, NMDA 2A2-amino-3-ketobutyrate coenzyme A ligase, mitochondrial5-aminolevulinate synthase, non-specific, mitochondrial +22
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 640-79-9

A bile salt formed in the liver from chenodeoxycholate and glycine, usually as the sodium salt. It acts as a detergent to solubilize fats for absorption and is itself absorbed. It is a cholagogue and choleretic. [PubChem]

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsBile Acids and Salts +12
Target Protein:
7-alpha-hydroxysteroid dehydrogenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 475-31-0

The glycine conjugate of cholic acid. It acts as a detergent to solubilize fats for absorption and is itself absorbed.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsBile Acids and Salts +11
Target Protein:
Gastrotropin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Glycocyamine DB02751
small molecule | CAS: 352-97-6

Deskripsi belum tersedia.

Kategori:
Affinity LabelsAmino AcidsAmino Acids, Peptides, and Proteins +3
Target Protein:
Guanidinoacetate N-methyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Glycol salicylate Approved DB11323
small molecule | CAS: 87-28-5

Glycol salicylate, also known as _2-hydroxyethyl salicylate_, is a benzoate ester formed from the condensation of the carboxy group of salicylic acid with one of the hydroxy groups of ethylene glycol. It is found as an active ingredient and topical analgesic …

Kategori:
Acids, CarbocyclicAnti-Inflammatory AgentsAnti-Inflammatory Agents, Non-Steroidal +5
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu ParuhThe serum half-life…
Vol. Distribusi-
Klirens-
Genetik -
Glycolic acid Approved DB03085
small molecule | CAS: 79-14-1

Deskripsi belum tersedia.

Kategori:
AcetatesAcids, AcyclicDermatologicals +2
Target Protein:
Glucose-6-phosphate 1-dehydrogenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Glycopyrronium Approved DB00986
small molecule | CAS: 740028-90-4

Glycopyrronium, also known as NVA237 or glycopyrrolate, is a racemic mixture of two enantiomers.[L33110] They are both quaternary ammonium compounds and long acting muscarinic antagonists.[L33110] It is one of the most commonly prescribed anticholinergic medi…

Kategori:
Adjuvants, AnesthesiaAdrenergics, InhalantsAgents producing tachycardia +30
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M2 +2
Waktu ParuhThe half life after…
Vol. DistribusiThe mean volume of …
KlirensA 6 µg/kg intraveno…
Genetik -
Glycyrrhizic acid Approved DB13751
small molecule | CAS: 1405-86-3

Glycyrrhizic acid is extracted from the root of the licorice plant; _Glycyrrhiza glabra_.[F79] It is a triterpene glycoside with glycyrrhetinic acid that possesses a wide range of pharmacological and biological activities. When extracted from the plant, it ca…

Kategori:
Alimentary Tract and MetabolismAnti-Inflammatory AgentsBile and Liver Therapy +6
Target Protein:
11-beta-hydroxysteroid dehydrogenase 1Tumor necrosis factorCaspase-3 +2
Waktu ParuhDepending on the do…
Vol. DistribusiThe apparent volume…
KlirensThe constant reabso…
Genetik -
Glymidine Approved DB01382
small molecule | CAS: 339-44-6

Glycodiazine is used with diet to lower blood glucose by increasing the secretion of insulin from pancreas and increasing the sensitivity of peripheral tissues to insulin. The mechanism of action of glycodiazine in lowering blood glucose appears to be depende…

Kategori:
Alimentary Tract and MetabolismAmidesBlood Glucose Lowering Agents +7
Target Protein:
ATP-sensitive inward rectifier potassium channel 1ATP-sensitive inward rectifier potassium channel 10ATP-binding cassette sub-family C member 8
Waktu Paruh4 hours.
Vol. Distribusi-
Klirens-
Genetik -
Glyoxylic acid DB04343
small molecule | CAS: 298-12-4

Deskripsi belum tersedia.

Kategori:
Acids, Aldehydic
Target Protein:
Malate synthase GIsocitrate lyaseMalate synthase G +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Glypromate DB05633
small molecule | CAS: 32302-76-4

Neuren Pharmaceuticals was developing Glypromate (glycine-proline glutamate), a naturally occurring small-molecule neuroprotectant derived from IGF-1 which inhibits caspase III dependent apoptosis, for the potential treatment of neurodegenerative diseases by …

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GMK DB06661
biotech

GMK vaccine (a ganglioside conjugate vaccine coupled to keyhole limpet hemocyanin and formulated with the adjuvant QS-21) for the potential treatment of melanoma

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GMX1777 DB05217
small molecule

GMX1777 is a water-soluble prodrug of the cyanoguanidine compound GMX1778 with potential antineoplastic activity. In vivo, apoptosis inducer GMX1777 is rapidly converted into GMX1778 through hydrolytic cleavage of a carbonate ester bond. Although the exact me…

Kategori:
Amidines
Target Protein:
Nicotinamide phosphoribosyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

The GnRH pharmaccine consists of synthetic peptides (constructed to "look like" GnRH), which are bound chemically to a carrier and suspended in a proprietary "delivery vehicle". The pharmaccine is administered intramuscularly to the patient by injection and i…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Go-6976 DB17029
small molecule | CAS: 136194-77-9

An inhibitor of calcium-dependent isoforms of protein kinase C.[A253002,A253007]

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingIndoles +1
Target Protein:
Transcription factor RelBNuclear factor NF-kappa-B p105 subunitNuclear factor NF-kappa-B p100 subunit +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Golidocitinib DB18057
small molecule | CAS: 2091134-68-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Golimumab Approved DB06674
biotech | CAS: 476181-74-5

Golimumab is a human IgG1? monoclonal antibody derived from immunizing genetically engineered mice with human TNF?. Golimumab binds and inhibits soluble and transmembrane human TNF?. Increased TNF? is associated with chronic inflammation. Thus golimumab is in…

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAnti-Inflammatory Agents +17
Target Protein:
Tumor necrosis factor
Waktu ParuhGolimumab has a lon…
Vol. DistribusiAfter IV administra…
KlirensAfter one IV dose o…
Genetik -
Golodirsen Approved DB15593
biotech | CAS: 1422959-91-8

Golodirsen is a morpholino antisense oligomer designed to treat about 8% of patients with Duchenne Muscular Dystrophy (DMD). This is an X-linked condition leading to progressive muscle degeneration that begins in early childhood, rendering many patients wheel…

Kategori:
Antisense Elements (Genetics)Antisense OligonucleotidesCompounds used in a research, industrial, or household setting +10
Target Protein:
Dystrophin
Waktu ParuhIn a pharmacokineti…
Vol. DistribusiThe volume of distr…
KlirensThis drug is rapidl…
Genetik -
Golotimod DB05475
small molecule | CAS: 229305-39-9

SCV-07 (g -D-glutamyl-L-tryptophan) is a novel synthetic dipeptide that acts broadly on the Toll-like receptor pathway. It has been shown to stimulate T-lymphocyte differentiation, macrocytic phagocytosis, and specific immune responses, and enhance IL-2 and …

Kategori:
Amino Acids, Peptides, and ProteinsOligopeptidesPeptides
Target Protein:
Signal transducer and activator of transcription 3Toll-like receptor 2Toll-like receptor 4 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 3001–3050 dari 6694
Sebelumnya Halaman 61 / 134 Berikutnya