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11778

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8554 (72.6%)
Target
6383 (54.2%)
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96 (0.8%)
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11778 (100.0%)

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Halaman 61 / 236
Bopindolol DB08807
small molecule | CAS: 62658-63-3

Bopindolol (INN) is an ester prodrug for the beta blocker [pindolol].

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +12
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptorBeta-3 adrenergic receptor +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Bordetella pertussis filamentous hemagglutinin antigen (formaldehyde inactivated) is a vaccine that contains inactivated acellular pertussis antigen that is isolated from Bordetella pertussis culture.

Kategori:
Actively Acquired ImmunityInactivated Bordetella Pertussis Vaccine
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Bordetella pertussis fimbriae 2/3 antigen is a vaccine for the prophylaxis of the disease caused by Bordetella pertussis which is a a Gram-negative coccobacillus that expresses two serologically distinct fimbriae (Fim2 and Fim3).

Kategori:
Actively Acquired ImmunityInactivated Bordetella Pertussis Vaccine
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Bordetella pertussis pertactin antigen is a vaccine for the prophylaxis of whooping cough that contains pertactin, a membrane-associated antigen of Bordetella pertussis [A31248].

Kategori:
Amino Acids, Peptides, and ProteinsBacterial ProteinsBacterial Toxins +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Kategori:
Actively Acquired ImmunityInactivated Bordetella Pertussis Vaccine
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Borneol DB11288
small molecule | CAS: 507-70-0

Deskripsi belum tersedia.

Kategori:
Bicyclic MonoterpenesBridged-Ring CompoundsMonoterpenes +3
Target Protein:
Transient receptor potential cation channel subfamily V member 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bornyl acetate DB14665
small molecule | CAS: 76-49-3

Deskripsi belum tersedia.

Kategori:
Bicyclic MonoterpenesBridged-Ring CompoundsMonoterpenes +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Borocaptate DB17408
small molecule

Deskripsi belum tersedia.

Kategori:
BoranesBoron CompoundsBoron Neutron Capture Therapy +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Boron DB11203
small molecule | CAS: 7440-42-8

Boron (B) is a chemical element with an atomic number 5 that belongs in the Period 2 and Group 13 in the periodic table. It is a low-abundant metalloid that is a poor electrical conductor at room temperature. Natural boron exists in 2 stable isotopes however …

Kategori:
Diet, Food, and NutritionElementsFood +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bortezomib Approved DB00188
small molecule | CAS: 179324-69-7

Bortezomib is a dipeptide boronic acid derivative and proteasome inhibitor used to treat multiple myeloma and mantle cell lymphoma.[A204083] The 26S proteasome is a protein complex that degrades ubiquitinated proteins in the ubiquitin-proteasome pathway: reve…

Kategori:
AcidsAcids, NoncarboxylicAntineoplastic Agents +36
Target Protein:
Proteasome subunit beta type-5Serine protease 1Proteasome subunit beta type-1
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe mean distributi…
KlirensFollowing the admin…
Genetik -
Bortezomib D-mannitol Approved DB16741
small molecule | CAS: 444576-08-3

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsProteasome Inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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BOS172722 DB15498
small molecule | CAS: 1578245-44-9

BOS172722 is a novel and selective Monopolar spindle 1 (Mps1) kinase inhibitor identified as a potential anticancer agent.[A187123] Normally, Mps1 supports the proper division of cancer cells, ensuring survival and replication. The key role of Mps1 in the gro…

Target Protein:
Dual specificity protein kinase TTK
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bosakitug DB19101
biotech | CAS: 2762183-23-1

Bosakitug (BSI-045B) is under investigation in clinical trial NCT05932654 (POC Study to Evaluate BSI-045B Monotherapy and BSI-045B Add-on Therapy With Dupilumab in Atopic Dermatitis).

Waktu Paruh-
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Boscalid Approved DB12792
small molecule | CAS: 188425-85-6

Boscalid has been investigated for the treatment of OSDI, Glaucoma, Staining, Schirmers, and Disease Severity, among others.

Kategori:
Benzene DerivativesNicotinic AcidsPyridines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bosentan Approved DB00559
small molecule | CAS: 147536-97-8

Bosentan is a dual endothelin receptor antagonist marketed under the trade name Tracleer by Actelion Pharmaceuticals. Bosentan is used to treat pulmonary hypertension by blocking the action of endothelin molecules that would otherwise promote narrowing of the…

Kategori:
AmidesAntihypertensive AgentsAntihypertensives for Pulmonary Arterial Hypertension +24
Target Protein:
Endothelin receptor type BEndothelin-1 receptor
Waktu ParuhTerminal eliminatio…
Vol. Distribusi* 18 L
Klirens* 4 L/h [patients w…
Genetik -
Boserolimab DB17452
biotech | CAS: 2444297-08-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bosutinib Approved DB06616
small molecule | CAS: 380843-75-4

Bosutinib is a 7-alkoxy-3-quinolinecarbonitrile that functions as a potent, dual SRC and ABL tyrosine kinase inhibitor indicated for chronic myelogenous leukemia (CML), specifically Philadelphia chromosome-positive (Ph+) CML. Philadelphia chromosome is a hall…

Kategori:
AminesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +22
Target Protein:
Tyrosine-protein kinase ABL1Tyrosine-protein kinase LynProto-oncogene tyrosine-protein kinase Src +8
Waktu ParuhThe mean (SD) bosut…
Vol. DistribusiThe mean (SD) appar…
KlirensThe mean (SD) appar…
Genetik -
biotech | CAS: 2417551-39-2

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Botensilimab DB16651
biotech | CAS: 2408310-37-0

Botensilimab is under investigation in clinical trial NCT03860272 (Fc-engineered Anti-ctla-4 Monoclonal Antibody in Advanced Cancer).

Waktu Paruh-
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Genetik -
Bouteloua gracilis pollen Approved DB10715
biotech

Bouteloua gracilis pollen is the pollen of the Bouteloua gracilis plant. Bouteloua gracilis pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityGrass Pollen Allergen ExtractsIncreased Histamine Release +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1383710-57-3

Bovhyaluronidase azoximer is under investigation in clinical trial NCT06458543 (Optimization of Bacterial Vaginosis Treatment in Women of Reproductive Age).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bovine type I collagen Approved DB10771
biotech | CAS: 9050-08-2

Bovine collagen alpha-1 is a naturally occurring extracellular matrix protein which is found in tendons and other connective tissues. It plays a vital role in cell growth, differentiation, attachment, and migration [L2481]. Often combined with other ingredie…

Kategori:
Allogeneic Cultured Cell Scaffold
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BP-14979 DB16302
small molecule | CAS: 1000036-77-0

BP-14979 is under investigation in clinical trial NCT01785147 (Efficacy and Safety of BP1.4979 in Smoking Cessation).

Waktu Paruh-
Vol. Distribusi-
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BPC-157 DB11882
small molecule | CAS: 137525-51-0

Bepecin is under investigation in clinical trial NCT02637284 (PCO-02 - Safety and Pharmacokinetics Trial).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Ulcer AgentsGastrointestinal Agents +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BPH-608 DB07404
small molecule

Deskripsi belum tersedia.

Target Protein:
Farnesyl pyrophosphate synthaseDitrans,polycis-undecaprenyl-diphosphate synthase ((2E,6E)-farnesyl-diphosphate specific)
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BPR-0L075 DB17155
small molecule | CAS: 613679-11-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BQ-788 DB17984
small molecule | CAS: 156161-89-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntihypertensive AgentsCardiovascular Agents +3
Target Protein:
Endothelin receptor type B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BR-007 DB18408
small molecule | CAS: 2409546-40-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BR101801 DB17387
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Bradanicline DB06090
small molecule | CAS: 639489-84-2

Bradanicline, a novel small molecule that modulates the activity of the neuronal nicotinic receptor (NNR) subtype known as alpha7(?7). Bradanicline belongs to a new class of drugs for the treatment of central nervous system diseases and disorders.

Kategori:
Heterocyclic Compounds, Fused-RingReceptors, Nicotinic
Target Protein:
Neuronal acetylcholine receptor subunit alpha-7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Branaplam DB14918
small molecule | CAS: 1562338-42-4

Branaplam is under investigation in clinical trial NCT02268552 (An Open Label Study of LMI070 (Branaplam) in Type 1 Spinal Muscular Atrophy (SMA)).

Target Protein:
Survival motor neuron protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Branebrutinib DB15347
small molecule | CAS: 1912445-55-6

Branebrutinib is under investigation in clinical trial NCT02705989 (Safety, Tolerability and Relative Bioavailability Study of BMS-986195 in Healthy Subjects).

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingProtein Kinase Inhibitors
Target Protein:
Tyrosine-protein kinase BTK
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brasofensine DB04857
small molecule | CAS: 171655-91-7

Brasofensine is an orally administered dopamine reuptake inhibitor being developed for the treatment of Parkinson's Disease. Phase I/II trials for brasofensine have been completed in the U.K. In November 2001, NeuroSearch confirmed that the drug's development…

Kategori:
AminesHeterocyclic Compounds, Fused-RingHydroxylamines
Target Protein:
Sodium-dependent serotonin transporterD(2) dopamine receptor
Waktu ParuhPlasma terminal eli…
Vol. Distribusi-
Klirens-
Genetik -
Brazikumab DB16115
biotech | CAS: 1610353-18-8

Brazikumab is under investigation in clinical trial NCT03759288 (An Active and Placebo-controlled Study of Brazikumab in Participants With Moderately to Severely Active Crohn's Disease).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brecanavir DB04887
small molecule | CAS: 313682-08-5

Brecanavir (VX-385) an orally active aspartic protease inhibitor (PI), under investigation by Vertex and GlaxoSmithKline for the treatment of HIV. In July 2006, Vertex indicated that it expected GSK to initiate phase III trials of the drug in 2007. In Decembe…

Kategori:
Acids, AcyclicDioxolesHeterocyclic Compounds, Fused-Ring
Target Protein:
Gag-Pol polyproteinPol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brefeldin A DB07348
small molecule | CAS: 20350-15-6

A metabolite from Penicillium brefeldianum that exhibits a wide range of antibiotic activity.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsCytochrome P-450 CYP3A Inhibitors +9
Target Protein:
Cytohesin-2ADP-ribosylation factor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bremelanotide Approved DB11653
biotech | CAS: 189691-06-3

Bremelanotide is a 7 amino acid peptide used to treat hypoactive sexual desire disorder in premenopausal women.[L9635] Bremelanotide does not interact with alcohol.[A179686] The mechanism by which bremelanotide's action on receptors translates to a clinical e…

Kategori:
Amino Acids, Peptides, and ProteinsGenito Urinary System and Sex HormonesHormones +16
Target Protein:
Melanocyte-stimulating hormone receptorMelanocortin receptor 4Melanocortin receptor 3 +2
Waktu ParuhThe half life of br…
Vol. DistribusiThe mean volume of …
KlirensThe mean clearance …
Genetik -
Bremzalerbart DB19417
biotech | CAS: 2456307-07-4

Bremzalerbart is under investigation in clinical trial NCT06602739 (A Study to Demonstrate the Effect of REGN5713-5715 on Reducing Ocular Allergy Signs and Symptoms in Adult Participants With Birch Pollen Allergy).

Waktu Paruh-
Vol. Distribusi-
Klirens-
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Brenetafusp DB19441
biotech | CAS: 2736407-54-6

Brenetafusp is under investigation in clinical trial NCT04262466 (Safety and Efficacy of IMC-F106C as a Single Agent and in Combination With Checkpoint Inhibitors).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brensocatib DB15638
small molecule | CAS: 1802148-05-5

Brensocatib is under investigation in clinical trial NCT03218917 (Assessment of INS1007 in Subjects With Non-cystic Fibrosis Bronchiectasis).

Kategori:
AzepinesHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brentuximab vedotin Approved DB08870
biotech | CAS: 914088-09-8

Brentuximab vedotin, also known as Adcetris®, is an antibody-drug conjugate that combines an anti-CD30 antibody with the drug monomethyl auristatin E (MMAE). It is an anti-neoplastic agent used in the treatment of Hodgkin's lymphoma and systemic anaplastic la…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +35
Target Protein:
Tumor necrosis factor receptor superfamily member 8
Waktu ParuhThe terminal half-l…
Vol. DistribusiMMAE is unlikely to…
KlirensThe liver is the pr…
Genetik -
Brequinar DB03523
small molecule | CAS: 96187-53-0

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsBenzene DerivativesEnzyme Inhibitors +5
Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brevenal DB17865
small molecule | CAS: 776331-34-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brexanolone Approved DB11859
small molecule | CAS: 516-54-1

As of March 2019, brexanolone - developed and made available commercially by Sage Therapeutics Inc. as the brand name product Zulresso - is the first drug to have ever been approved by the US FDA specifically for the treatment of postpartum depression (PPD) i…

Kategori:
AnestheticsAnticonvulsantsAntidepressive Agents +28
Target Protein:
Gamma-aminobutyric acid receptor subunit deltaGamma-aminobutyric acid receptor subunit gamma-3GABA(A) Receptor +3
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe volume of distr…
KlirensThe total plasma cl…
Genetik -
Brexpiprazole Approved DB09128
small molecule | CAS: 913611-97-9

Brexpiprazole is an atypical antipsychotic and a novel D2 dopamine and serotonin 1A partial agonist called serotonin-dopamine activity modulator (SDAM). It has a high affinity for serotonin, dopamine and alpha (?)-adrenergic receptors.[L46417] Although it is …

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +30
Target Protein:
5-hydroxytryptamine receptor 1AD(2) dopamine receptorD(3) dopamine receptor +9
Waktu ParuhAfter multiple once…
Vol. DistribusiThe volume of distr…
KlirensApparent oral clear…
Genetik -
BRG01 DB18173
biotech

BRG01 is a genetically modified autologous CAR-T cell therapy under investigation for the treatment of nasopharyngeal carcinoma.[L48111]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Briciclib DB12004
small molecule | CAS: 865783-99-9

Briciclib has been used in trials studying the treatment of Lymphoma, Neoplasms, Advanced Solid Tumor, and Acute Lymphocytic Leukemia.

Target Protein:
G1/S-specific cyclin-D1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brifentanil DB09172
small molecule | CAS: 101345-71-5

Brifentanil (also known as A-3331) is an analog of fentanyl, a potent opioid. This drug is classified as an opioid analgesic and was developed in the early 1990s. The effects of brifentanil are very similar to those of alfentanil, with strong but short lastin…

Kategori:
Piperidines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brigatinib Approved DB12267
small molecule | CAS: 1197953-54-0

Brigatinib, originally named AP26113, is a reversible dual inhibitor of anaplastic lymphoma kinase (ALK) and epidermal growth factor receptor (EGFR). It presents selectivity against the mutant forms of EGFR compared to the wild-type.[A31311] It also exhibits …

Kategori:
Anaplastic lymphoma kinase (ALK) inhibitorsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +18
Target Protein:
ALK tyrosine kinase receptorEpidermal growth factor receptorTyrosine-protein kinase ABL1 +6
Waktu ParuhThe half-life of br…
Vol. DistribusiThe apparent volume…
KlirensAfter oral administ…
Genetik -
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