Hasil Filter

3253

Total database: 17430
Struktur (SMILES)
2451 (75.3%)
Target
1833 (56.3%)
Genomik
35 (1.1%)
Referensi
3253 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (3253)

Halaman 61 / 66
TNP-2092 DB16312
small molecule | CAS: 922717-97-3

TNP-2092 is under investigation in clinical trial NCT03964493 (TNP-2092 to Treat Acute Bacterial Skin and Skin Structure Infection).

Kategori:
Heterocyclic Compounds, Fused-RingLactams, MacrocyclicQuinolines
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA topoisomerase 4 subunit A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TNP-470 DB08633
small molecule | CAS: 129298-91-5

O-(chloroacetylcarbamoyl)fumagillol (TNP-470) has been used in trials studying the treatment of HIV Infections, Sarcoma, Kaposi, and Pancreatic Neoplasms.

Kategori:
Angiogenesis InhibitorsAngiogenesis Modulating AgentsAntibiotics, Antineoplastic +7
Target Protein:
Methionine aminopeptidase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tobevibart DB18986
biotech | CAS: 2645440-65-7

Tobevibart is under investigation in clinical trial NCT05612581 (A Platform Study to Evaluate Investigational Therapies in Chronic Hepatitis B Infection).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tocilizumab Approved DB06273
biotech | CAS: 375823-41-9

Tocilizumab is a recombinant humanized monoclonal antibody IL-6 receptor inhibitor used to treat inflammatory and autoimmune conditions.[L12789] It was first described in the literature in 2003 when Chugai, a subsidiary of Roche began developing IL-6 inhibiti…

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAntibodies +21
Target Protein:
Interleukin-6 receptor subunit alpha
Waktu ParuhThe half life of to…
Vol. DistribusiIn rheumatoid arthr…
KlirensThe linear clearanc…
Genetik -
Tocofersolan Approved DB11635
small molecule | CAS: 9002-96-4

D-Alpha-tocopheryl polyethylene glycol 1000 succinate (Tocofersolan, Vedrop), has been developed in Europe as an orally bioavailable source of vitamin E in children suffering from cholestasis [L2371]. Cholestasis is the reduction or stoppage of bile flow, eit…

Kategori:
Alimentary Tract and MetabolismBenzopyransCompounds used in a research, industrial, or household setting +9
Target Protein:
ATP-dependent translocase ABCB1
Waktu Paruh29.7 h [L2371]
Vol. DistribusiLocated principally…
Klirens-
Genetik -
Tocopherol Approved DB11251
small molecule | CAS: 1406-66-2

Tocopherol exists in four different forms designated as ?, ?, ?, and ?. They present strong antioxidant activities, and it is determined as the major form of vitamin E. Tocopherol, as a group, is composed of soluble phenolic compounds that consist of a chroma…

Kategori:
Alimentary Tract and MetabolismAntioxidantsBenzopyrans +16
Target Protein:
Free radicals
Waktu ParuhThe elimination hal…
Vol. DistribusiThe apparent volume…
KlirensClearance ranged fr…
Genetik -
Tocotrienol DB12647
small molecule | CAS: 6829-55-6

Tocotrienol has been investigated for the treatment of Cholesterol Lowering.

Kategori:
AntioxidantsBenzopyransBiological Factors +11
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tolbutamide Approved DB01124
small molecule | CAS: 64-77-7

Tolbutamide is an oral antihyperglycemic agent used for the treatment of non-insulin-dependent diabetes mellitus (NIDDM). It is structurally similar to acetohexamide, chlorpropamide and tolazamide and belongs to the sulfonylurea class of insulin secretagogues…

Kategori:
Alimentary Tract and MetabolismAmidesBenzene Derivatives +25
Target Protein:
ATP-binding cassette sub-family C member 9ATP-binding cassette sub-family C member 8ATP-sensitive inward rectifier potassium channel 1
Gen Terkait:
CYP2C9
Waktu ParuhApproximately 7 hou…
Vol. Distribusi-
Klirens-
Genetik 1 Varian
Tolfenamic acid Approved DB09216
small molecule | CAS: 13710-19-5

Tolfenamic acid, with the formula N-(2-methyl-3-chlorphenyl)-anthranilic acid, is a nonsteroidal anti-inflammatory agent.[A31824] It was discovered by scientists at Medica Pharmaceutical Company in Finland. It is used in the UK as a treatment for migraine und…

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +29
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu ParuhThe estimated half-…
Vol. DistribusiThe volume of distr…
KlirensThe estimated clear…
Genetik -
Tolterodine Approved DB01036
small molecule | CAS: 124937-51-5

Tolterodine is an antimuscarinic drug that is used to treat urinary incontinence. Tolterodine acts on M2 and M3 subtypes of muscarinic receptors.

Kategori:
Agents producing tachycardiaAlcoholsAmines +26
Target Protein:
Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M5 +2
Waktu Paruh1.9-3.7 hours
Vol. Distribusi* 113 ± 26.7 L
Klirens-
Genetik -
Tolu balsam DB11223
small molecule | CAS: 9000-64-0

Deskripsi belum tersedia.

Kategori:
Biological ProductsBiopolymersComplex Mixtures +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tolvaptan Approved DB06212
small molecule | CAS: 150683-30-0

Tolvaptan is used to treat low blood sodium levels (hyponatremia) associated with various conditions like congestive heart failure, cirrhosis, and syndrome of inappropriate antidiuretic hormones (SIADH). FDA approved on May 19, 2009.

Kategori:
Agents causing hyperkalemiaAntidiuretic Hormone Receptor AntagonistsBenzazepines +14
Target Protein:
Vasopressin V2 receptorVasopressin V1a receptor
Waktu ParuhTerminal half life,…
Vol. DistribusiHealthy subjects: 3…
Klirens4 mL/min/kg (post-o…
Genetik -
Tonapofylline DB12569
small molecule | CAS: 340021-17-2

Tonapofylline has been used in trials studying the treatment of Heart Failure, Renal Insufficiency, and Congestive Heart Failure.

Kategori:
AlkaloidsHeterocyclic Compounds, Fused-RingPurines +2
Target Protein:
Adenosine receptor A1Adenosine receptor A2aAdenosine receptor A3 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TOP-1288 DB14839
small molecule | CAS: 1630202-02-6

TOP-1288 is under investigation in clinical trial NCT02888379 (Phase 2a Study to Evaluate the Safety/Tolerability and Efficacy of TOP1288 200 mg Rectal Solution Once Daily for 4 Weeks in Ulcerative Colitis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Topiramate Approved DB00273
small molecule | CAS: 97240-79-4

Topiramate is a anti-epileptic drug used to manage seizures and prevent migraines.[A175249] It was initially approved by the FDA in 1996. In 2004, topiramate was approved for the prevention of migraine in adults.[A188309,L10544,L43478] Since 2012, the extende…

Kategori:
Alimentary Tract and MetabolismAnti-Obesity AgentsAnticonvulsants +23
Target Protein:
Glutamate receptor ionotropic, kainate 1Gamma-aminobutyric acid receptor subunit alpha-1Voltage-gated sodium channel alpha subunit +7
Waktu ParuhThe elimination hal…
Vol. DistribusiThe mean apparent v…
KlirensThe mean oral plasm…
Genetik -
Topotecan Approved DB01030
small molecule | CAS: 123948-87-8

An antineoplastic agent used to treat ovarian cancer. It works by inhibiting DNA topoisomerases, type I.

Kategori:
AlkaloidsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +21
Target Protein:
DNA topoisomerase 1DNADNA topoisomerase I, mitochondrial
Waktu Paruh2-3 hours
Vol. Distribusi-
Klirens-
Genetik -
Topsalysin DB05160
small molecule | CAS: 917121-25-6

Topsalysin is being developed for the treatment of localized prostate cancer and also benign prostatic hyperplasia. Topsalysin is delivered locally to the prostate under ultrasound guidance.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsMembrane Proteins +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Toreforant DB12522
small molecule | CAS: 952494-46-1

Toreforant has been used in trials studying the treatment of Asthma, Psoriasis, Hepatic Impairment, and Rheumatoid Arthritis.

Kategori:
Heterocyclic Compounds, Fused-RingHistamine AgentsHistamine Antagonists +1
Target Protein:
Histamine H4 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tovetumab DB12609
biotech | CAS: 1243266-04-7

Tovetumab has been used in trials studying the treatment of Cancer, Glioblastoma Multiforme, and Advanced Solid Malignancies.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tozadenant DB12203
small molecule | CAS: 870070-55-6

Tozadenant has been investigated for the basic science of Cocaine Dependence.

Kategori:
Heterocyclic Compounds, Fused-RingThiazoles
Target Protein:
Adenosine receptor A2a
Waktu ParuhFollowing the oral …
Vol. Distribusi-
Klirens-
Genetik -
TP-1287 DB18104
small molecule | CAS: 2044686-42-0

Deskripsi belum tersedia.

Target Protein:
Cyclin-dependent kinase 9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TP-252 DB17912
small molecule | CAS: 1841444-50-5

TP-252 consists of magnesium L-lysinate bis-eicosapentaenoate, an ionizable salt of eicosapentaenoic acid (EPA), currently being investigated to treat familial adenomatous polyposis.[A259956]

Kategori:
Dietary FatsDietary Fats, UnsaturatedEicosanoids +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TP-271 DB15040
small molecule | CAS: 1207284-17-0

TP-271 is under investigation in clinical trial NCT02724085 (A Phase 1 Study to Assess the Safety, Tolerability and PK of IV TP-271).

Kategori:
Naphthacenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trabodenoson DB13122
small molecule | CAS: 871108-05-3

Trabodenoson has been used in trials studying the treatment of Ocular Hypertension (OHT) and Primary Open-Angle Glaucoma (POAG).

Kategori:
Adenosine A receptor agonistsAdenosine A1 Receptor AgonistsAnions +9
Target Protein:
Adenosine receptor A1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tradipitant DB12580
small molecule | CAS: 622370-35-8

Tradipitant has been used in trials studying the treatment and prevention of Eczema, Pruritus, Gastroparesis, Chronic Pruritus, and Atopic Dermatitis, among others.

Target Protein:
Substance-P receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tralokinumab Approved DB12169
biotech | CAS: 1044515-88-9

Atopic dermatitis (AD) is an inflammatory skin disorder that causes skin inflammation, skin barrier dysfunction, and chronic pruritus.[A242432] It is estimated to affect up to 20% of adults and children worldwide, and is frequently associated with other atopi…

Kategori:
Agents for Dermatitis, Excluding CorticosteroidsAmino Acids, Peptides, and ProteinsAntibodies +9
Target Protein:
Interleukin-13
Waktu ParuhThe half-life of tr…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of tr…
Genetik -
Tranilast DB07615
small molecule | CAS: 53902-12-8

Tranilast is an antiallergic drug developed by Kissei Pharmaceuticals. In 1982, it was approved in Japan and South Korea for the management of bronchial asthma. Indications for keloid and hypertrophic scar were added in 1993. It has been used for the treatmen…

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAminobenzoates +23
Target Protein:
Steryl-sulfataseHistamine H1 receptorHematopoietic prostaglandin D synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Transfluthrin DB15117
small molecule | CAS: 118712-89-3

Transfluthrin is under investigation in clinical trial NCT02394522 (Spatial Repellent Products for Control of Vector Borne Diseases - Malaria - Zambia (SR-M-ZM)).

Kategori:
AgrochemicalsBenzene DerivativesCompounds used in a research, industrial, or household setting +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trastuzumab Approved DB00072
biotech | CAS: 180288-69-1

Produced in CHO cell cultures, trastuzumab is a recombinant IgG1 kappa, humanized monoclonal antibody [A40276] that selectively binds with high affinity in a cell-based assay (Kd = 5 nM) to the extracellular domain of the human epidermal growth factor recepto…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +21
Target Protein:
Receptor tyrosine-protein kinase erbB-2
Gen Terkait:
ERBB2
Waktu ParuhThe terminal half-l…
Vol. Distribusi-
KlirensThe predicted stead…
Genetik 1 Varian
Traxoprodil DB18795
small molecule | CAS: 134234-12-1

Deskripsi belum tersedia.

Target Protein:
Glutamate receptor ionotropic, NMDA 2B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trebananib DB12056
biotech | CAS: 894356-79-7

Trebananib is under investigation for the treatment of Ovarian Cancer, Peritoneal Cancer, and Fallopian Tube Cancer. Trebananib has been investigated for the treatment of Cancer, Oncology, Carcinoma, Metastases, and Colon Cancer, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trefentanil DB09181
small molecule | CAS: 120656-74-8

Trefentanil (A-3665) is a fentanyl analogue opioid developed in 1992. It is more potent and shorter acting than alfentanil. Trefentanil is not used in clinics due to the severity of its respiratory depression, though it is still used in research.

Target Protein:
Mu-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tregalizumab DB13073
biotech | CAS: 1207446-68-1

Tregalizumab has been used in trials studying the treatment of Rheumatoid Arthritis.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trehalose DB12310
small molecule | CAS: 99-20-7

Cabaletta has been used in trials studying the treatment of Oculopharyngeal Muscular Dystrophy.

Kategori:
CarbohydratesCompounds used in a research, industrial, or household settingDisaccharides +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tremelimumab Approved DB11771
biotech | CAS: 745013-59-6

Tremelimumab, formerly known as ticilimumab, is a fully human IgG2 monoclonal antibody directed against cytotoxic T-lymphocyte-associated antigen 4 (CTLA-4). CTLA-4 is a cell surface receptor expressed on activated T cells to act as a negative regulator for T…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Target Protein:
Cytotoxic T-lymphocyte protein 4
Waktu ParuhThe geometric mean …
Vol. DistribusiThe geometric mean …
KlirensThe geometric mean …
Genetik -
Trenonacog alfa DB13201
biotech | CAS: 1232401-60-3

Human coagulation factor IX (EC 3.4.21.22, Christmas factor, plasma thromboplastin component), produced in CHO cells.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Triamcinolone Approved DB00620
small molecule | CAS: 124-94-7

Triamcinolone is a corticosteroid used to treat various inflammatory conditions in the body from allergic rhinitis to acute exacerbations of multiple sclerosis.[L8255] Triamcinolone can be used as a one time adjunct treatment of osteoarthritic knee pain,[L826…

Kategori:
Adrenal Cortex HormonesAdrenalsAgents Causing Muscle Toxicity +44
Target Protein:
Glucocorticoid receptor
Waktu ParuhThe half life of tr…
Vol. DistribusiThe apparent volume…
KlirensThe clearance of tr…
Genetik -
Triazavirin DB15622
small molecule | CAS: 123606-06-4

Triazavirin is a guanine nucleotide analog antiviral originally developed in Russia that has shown efficacy against influenza A and B, including the H5N1 strain.[A191709,A191625,A191916] It appears that Triazavirin has shown promise in reducing influenza dise…

Kategori:
Antiviral AgentsExperimental Unapproved Treatments for COVID-19Guanine Nucleotides
Waktu ParuhIn rabbits, intraga…
Vol. DistribusiIn rabbits, intraga…
KlirensIn rabbits, intraga…
Genetik -
small molecule | CAS: 101200-48-0

Deskripsi belum tersedia.

Kategori:
Arylsulfonic AcidsSulfonic AcidsSulfur Acids +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tributyrin DB12709
small molecule | CAS: 60-01-5

Tributyrin has been used in trials studying the treatment of Prostate Cancer and Unspecified Adult Solid Tumor, Protocol Specific.

Kategori:
GlyceridesLipids
Target Protein:
Caspase-3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tricaprylin DB12176
small molecule | CAS: 538-23-8

Tricaprilin has been used in trials studying the supportive care and treatment of Alzheimer's Disease.

Kategori:
Acids, AcyclicAlzheimer Disease, drug therapyCompounds used in a research, industrial, or household setting +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trichophyton verrucosum Approved DB11295
small molecule

Trichophyton verrucosum is a fungus which can provoke allergic reactions. Trichophyton verrucosum extract is used in allergenic testing.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Triciribine DB12405
small molecule | CAS: 35943-35-2

Triciribine has been used in trials studying the treatment of Leukemia, Ovarian Cancer, HER2/Neu Negative, Breast Adenocarcinoma, and Stage IV Breast Cancer, among others.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleosides
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Triclabendazole Approved DB12245
small molecule | CAS: 68786-66-3

Triclabendazole, manufactured by Novartis pharmaceuticals, is an antihelminthic drug that was approved by the FDA in February 2019 for the treatment of fascioliasis in humans.[FDA label, L5452] Fascioliasis is a parasitic infection often caused by the helmi…

Kategori:
AnthelminticsAnti-Infective AgentsAntihelminthic +34
Target Protein:
CruzipainExcretory Secretory (ES) proteins
Waktu ParuhThe plasma eliminat…
Vol. DistribusiThe apparent volume…
Klirens-
Genetik -
small molecule | CAS: 2943-75-1

Deskripsi belum tersedia.

Kategori:
NaphthalenesQuinonesSilicon Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 112-27-6

Deskripsi belum tersedia.

Kategori:
AlcoholsCompounds used in a research, industrial, or household settingEthylene Glycols +3
Target Protein:
Acetolactate synthase, catabolicArabinogalactan endo-beta-1,4-galactanasePhosphoserine aminotransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Triethylenetetramine Approved DB06824
small molecule | CAS: 112-24-3

Triethylenetatramine (TETA), also known as trientine, is a potent and selective copper (II)-selective chelator. It is a structural analog of linear polyamine compounds, [spermidine] and [spermine]. TETA was first developed in Germany in 1861 and its chelating…

Kategori:
Alimentary Tract and MetabolismAminesChelating Agents +11
Target Protein:
Carbonic anhydrase 14
Waktu ParuhThe mean terminal h…
Vol. DistribusiTETA is widely dist…
KlirensIn healthy adult vo…
Genetik -
Trifarotene Approved DB12808
small molecule | CAS: 895542-09-3

Trifarotene is a topical retinoid cream used in the treatment of acne vulgaris that was first approved for use in the United States in October 2019.[L9013] Retinoids are a class of medications structurally and functionally analogous to [vitamin A], though lat…

Kategori:
AlkenesAnti-Acne PreparationsAnti-Acne Preparations for Topical Use +11
Target Protein:
Retinoic acid receptor gammaRetinoic acid receptor betaRetinoic acid receptor alpha
Waktu ParuhThe terminal half-l…
Vol. Distribusi-
Klirens-
Genetik -
Triglyme DB02078
small molecule | CAS: 112-49-2

Triethylene glycol dimethyl ether (also called triglyme) is a glycol ether used as a solvent.

Kategori:
AlcoholsCompounds used in a research, industrial, or household settingEthylene Glycols +3
Target Protein:
Tyrosine-protein kinase FynProfilin-2Outer-membrane lipoprotein LolB +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Triheptanoin Approved DB11677
small molecule | CAS: 620-67-7

Triheptanoin is a source of heptanoate fatty acids, which can be metabolized without the enzymes of long chain fatty acid oxidation.[L14612] In clinical trials, patients with long chain fatty acid oxidation disorders (lc-FAODs) treated with triheptanoin are l…

Kategori:
Alimentary Tract and MetabolismCaloric AgentsGlycerides +5
Waktu ParuhDue to multiple pea…
Vol. Distribusi-
KlirensA single dose of 0.…
Genetik -
Menampilkan 3001–3050 dari 3253
Sebelumnya Halaman 61 / 66 Berikutnya