Hasil Filter

6694

Total database: 17430
Struktur (SMILES)
4518 (67.5%)
Target
3751 (56.0%)
Genomik
81 (1.2%)
Referensi
6694 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (6694)

Halaman 60 / 134
Gatifloxacin Approved DB01044
small molecule | CAS: 112811-59-3

Gatifloxacin is an antibiotic agent and a member of the fourth-generation fluoroquinolone family. It works by inhibiting the bacterial enzymes DNA gyrase and topoisomerase IV. It was first introduced by Bristol-Myers Squibb in 1999 under the brand name Tequin…

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +23
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +3
Waktu Paruh7-14 hours
Vol. Distribusi-
Klirens-
Genetik -
Gatipotuzumab DB18861
biotech | CAS: 1264737-26-9

Gatipotuzumab is under investigation in clinical trial NCT01899599 (Pankomab-gex™ Versus Placebo as Maintenance Therapy in Advanced Ovarian Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gavestinel DB06741
small molecule | CAS: 153436-22-7

Highly potent and selective non-competitive antagonist acting at the strychnine-insensitive glycine binding site of the NMDA receptor-channel complex (Kd = 0.8 nM). Gavestinel displays > 1000-fold selectivity over NMDA, AMPA and kainate binding sites and is o…

Kategori:
Excitatory Amino Acid AgentsExcitatory Amino Acid AntagonistsGlycine Agents +5
Target Protein:
Glycine receptor subunit alpha-1Glycine receptor subunit alpha-2Glycine receptor subunit alpha-3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gavorestat DB16707
small molecule | CAS: 2170729-29-8

Gavorestat is under investigation in clinical trial NCT04902781 (Clinical Benefit, Safety, PK and PD Study of AT-007 in Pediatric Subjects With Classic Galactosemia).

Target Protein:
Aldo-keto reductase family 1 member B1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GC-373 DB15797
small molecule

GC-373 is a peptide aldehyde which is metabolized from the bisulfide adduct, [GC-376 free acid][A219031,A219036]. It is an inhibitor of M<sup>pro</sup> (otherwise known as 3CL<sup>pro</sup>), a viral encoded protease that cleaves and activates functional prot…

Kategori:
AmidesAmino AcidsAmino Acids, Branched-Chain +3
Target Protein:
Replicase polyprotein 1abReplicase polyprotein 1aReplicase polyprotein 1ab +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1417031-79-8

GC-376 is a 3C-like protease (3CL<sup>pro</sup> or M<sup>pro</sup>) inhibitor that stops the cleavage and activation of functional viral proteins required for replication and transcription in host cells[A219036]. The compound is known as a direct acting antiv…

Kategori:
AcidsAcids, NoncarboxylicAlkalies +15
Target Protein:
Replicase polyprotein 1abReplicase polyprotein 1aReplicase polyprotein 1ab +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GDC-0425 DB14791
small molecule | CAS: 1627539-18-7

GDC-0425 is under investigation in clinical trial NCT01359696 (A Study Evaluating the Safety, Tolerability, and Pharmacokinetics of GDC-0425 Administered With and Without Gemcitabine in Patients With Refractory Solid Tumors or Lymphoma).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Serine/threonine-protein kinase Chk1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GDC-0810 DB12253
small molecule | CAS: 1365888-06-7

ARN-810 has been used in trials studying the basic science and treatment of Breast Cancer.

Kategori:
Acids, CarbocyclicHeterocyclic Compounds, Fused-RingPyrazoles
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
GDP-mannose 6-dehydrogenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gedatolisib DB11896
small molecule | CAS: 1197160-78-3

Gedatolisib has been used in trials studying the basic science and treatment of Neoplasm, Ovary Cancer, Breast Cancer, Advanced Cancer, and Endometrial Cancer, among others.

Kategori:
Enzyme InhibitorsOxazinesProtein Kinase Inhibitors
Target Protein:
Serine/threonine-protein kinase mTORPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gefapixant Approved DB15097
small molecule | CAS: 1015787-98-0

It has been estimated that 5-10% of adults globally suffer from chronic cough, which is defined as a cough lasting longer than eight weeks.[L48601] A subset of these patients remain symptomatic despite thorough investigation and treatment, termed refractory c…

Kategori:
AmidesBCRP/ABCG2 SubstratesBenzene Derivatives +8
Target Protein:
P2X purinoceptor 3P2X purinoceptor 2
Waktu ParuhThe terminal half-l…
Vol. DistribusiBased on population…
KlirensPopulation pharmaco…
Genetik -
Gefurulimab DB18928
biotech | CAS: 2456407-94-4

Gefurulimab is under investigation in clinical trial NCT05556096 (Safety and Efficacy of ALXN1720 in Adults With Generalized Myasthenia Gravis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gelatin Approved DB11242
small molecule | CAS: 9000-70-8

Gelatin is a multifunctional ingredient that is used in foods, pharmaceuticals, cosmetics, and photographic films as a gelling agent, stabilizer, thickener, emulsifier, as well as film former.[A32432] As a thermoreversible hydrocolloid with a small gap bet…

Kategori:
Amino Acids, Peptides, and ProteinsBlood and Blood Forming OrgansBlood and Related Products +4
Waktu ParuhHalf-life is about …
Vol. Distribusi-
KlirensA large percentage …
Genetik -
Geldanamycin DB02424
small molecule | CAS: 30562-34-6

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Infective AgentsAntibiotics, Antineoplastic +7
Target Protein:
Heat shock protein HSP 90-alphaEndoplasminHeat shock protein HSP 90-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gemcitabine Approved DB00441
small molecule | CAS: 95058-81-4

Gemcitabine is a nucleoside analog and a chemotherapeutic agent. It was originally investigated for its antiviral effects, but it is now used as an anticancer therapy for various cancers.[A233135] Gemcitabine is a cytidine analog with two fluorine atoms repla…

Kategori:
AntimetabolitesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +23
Target Protein:
DNARibonucleoside-diphosphate reductase subunit M2Ribonucleoside-diphosphate reductase large subunit +2
Gen Terkait:
RRM1
Waktu ParuhFollowing intraveno…
Vol. DistribusiIn patients with va…
KlirensFollowing intraveno…
Genetik 1 Varian
small molecule | CAS: 210829-30-4

Gemcitabine elaidate has been used in trials studying the treatment of Solid Tumor, Lung Cancer, Non-small-cell Lung Cancer, and Metastatic Pancreatic Adenocarcinoma.

Kategori:
DeoxyribonucleosidesNucleic Acids, Nucleotides, and NucleosidesNucleosides +2
Target Protein:
Ribonucleoside-diphosphate reductase subunit M2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gemfibrozil Approved DB01241
small molecule | CAS: 25812-30-0

Gemfibrozil is a fibric acid agent, similar to [clofibrate], used to treat Type IIb, IV, and V hyperlipidemias.[A185777,L8525] Gemfibrozil is not a first line treatment and is prescribed to patients who have not responded adequately to weight loss, diet, exer…

Kategori:
Acids, AcyclicAgents Causing Muscle ToxicityBenzene Derivatives +53
Target Protein:
Peroxisome proliferator-activated receptor alphaLipoprotein lipaseSolute carrier organic anion transporter family member 1B1 +3
Waktu ParuhGemfibrozil has a p…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of ge…
Genetik -
Gemifloxacin Approved DB01155
small molecule | CAS: 175463-14-6

Gemifloxacin is a quinolone antibacterial agent with a broad-spectrum activity that is used in the treatment of acute bacterial exacerbation of chronic bronchitis and mild-to-moderate pneumonia. It is available in oral formulations. Gemifloxacin acts by inhib…

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +16
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +1
Waktu Paruh7 (&plusmn; 2) hours
Vol. Distribusi* 1.66 to 12.12 L/kg
Klirens* renal cl=11.6+/- …
Genetik -
Gemigliptin DB12412
small molecule | CAS: 911637-19-9

Gemigliptin is under investigation in Type 2 Diabetes Mellitus. Gemigliptin has been investigated for the treatment of Cancer and Cisplatin Adverse Reaction.

Kategori:
Agents causing angioedemaAlimentary Tract and MetabolismBlood Glucose Lowering Agents +5
Target Protein:
Dipeptidyl peptidase 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Gemogenovatucel-T is a bi-shRNA furin/Granulocyte Macrophage Colony Stimulating Factor (GMCSF) Augmented autologous tumour cell vaccine. Furin is a convertase involved in the activation of TGF?-1 and TGF?-2.[A255163] Gemogenovatucel-T is being investigated in…

Kategori:
Biological ProductsComplex MixturesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gemtuzumab ozogamicin Approved DB00056
biotech | CAS: 220578-59-6

Gemtuzumab ozogamicin is a recombinant humanized IgG4 kappa antibody which is conjugated with calicheamicin derivative, a cytotoxic antitumor antibiotic isolated from fermentation of Micromonospora echinospora ssp. calichensis. Gemtuzumab ozogamicin has appro…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +28
Target Protein:
Myeloid cell surface antigen CD33Low affinity immunoglobulin gamma Fc region receptor III-BLow affinity immunoglobulin gamma Fc region receptor III-A +1
Waktu ParuhIn pediatric patien…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik -
Geneticin DB04263
small molecule | CAS: 49863-47-0

Geneticin (also known as G418) is an aminoglycoside antibiotic similar in structure to gentamicin B1, produced by Micromonospora rhodorangea. Geneticin blocks polypeptide synthesis by inhibiting the elongation step in both prokaryotic and eukaryotic cells and…

Kategori:
Agents that produce neuromuscular block (indirect)AmebicidesAminoglycoside Antibacterials +8
Target Protein:
Ornithine decarboxylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Genipin DB19124
small molecule | CAS: 6902-77-8

Genipin is under investigation in clinical trial NCT05755750 (Intratendinous Genipin Injection in Horses With Tendon Injuries).

Kategori:
AdhesivesCholagogues and CholereticsCycloparaffins +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gentamicin Approved DB00798
small molecule | CAS: 1403-66-3

Gentamicin is a bactericidal aminoglycoside that was discovered and isolated from _Micromonospora purpurea_ in 1963.[A234349] It is one of the most frequently prescribed aminoglycosides due to its spectrum of activity, low cost, and availability.[A234339,A234…

Kategori:
Agents that produce neuromuscular block (indirect)alpha-Galactosidase, antagonists & inhibitorsAminoglycoside Antibacterials +21
Target Protein:
30S ribosomal protein S1216S ribosomal RNA23S ribosomal RNA +4
Waktu ParuhOne study assessing…
Vol. Distribusi-
KlirensThe renal clearance…
Genetik -
Gentamicin C1a DB04729
small molecule | CAS: 26098-04-4

Deskripsi belum tersedia.

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +6
Target Protein:
30S ribosomal protein S1216S ribosomal RNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gentamicin C2 DB17884
small molecule | CAS: 25876-11-3

Deskripsi belum tersedia.

Kategori:
Aminoglycoside AntibacterialsAnti-Bacterial AgentsCarbohydrates +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gepirone Approved DB12184
small molecule | CAS: 83928-76-1

Gepirone, an azapirone, is a pharmacologic analog of [buspirone] that acts selectively on the pre- and post-synaptic 5HT<sub>1A</sub> receptors. Although earlier clinical trials showed promising results for gepirone, its formulation as an immediate-release ta…

Kategori:
Anti-Anxiety AgentsAntidepressive AgentsCentral Nervous System Agents +12
Target Protein:
5-hydroxytryptamine receptor 1A
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe apparent volume…
KlirensAfter the administr…
Genetik -
Gepotidacin DB12134
small molecule | CAS: 1075236-89-3

Gepotidacin has been used in trials studying the treatment of Gonorrhea, Infections, Bacterial, and Infections, Respiratory Tract.

Kategori:
Antineoplastic AgentsEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring +2
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Geraniol Approved DB14183
small molecule | CAS: 106-24-1

Geraniol is a monoterpene that is found within many essential oils of fruits, vegetables, and herbs including rose oil, citronella, lemongrass, lavender, and other aromatic plants. It is emitted from the flowers of many species of plant and is commonly used b…

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseMonoterpenes +2
Target Protein:
Transient receptor potential cation channel subfamily M member 8
Waktu ParuhIn vitro measuremen…
Vol. Distribusi-
Klirens-
Genetik -
GI-101 DB17243
biotech

GI-101 is a bi-specific fragment crystallizable region (Fc) fusion protein containing a cluster of differentiation 80 ectodomain as an N-terminal moiety and interleukin-2 variant as a C-terminal moiety conjugated with human immunoglobulin G4 Fc.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GI-4000 DB05698
biotech

A vaccine containing a heat-killed recombinant <em>Saccharomyces cerevisiae</em> yeast transfected with mutated forms of Ras, an oncogene frequently found in solid tumors, with potential immunostimulant and antitumor activity. [L112]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GI-5005 DB05942
biotech | CAS: 1001913-27-4

GI-5005 is GlobeImmune's lead infectious disease product from its proprietary Tarmogen active immunotherapy platform for the treatment of chronic hepatitis C infection. GI-5005 is whole, heat-killed recombinant yeast genetically modified to express HCV-specif…

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBiological Factors +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gibberella fujikuroi Approved DB15511
biotech

Gibberella fujikuroi allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 77-06-5

Deskripsi belum tersedia.

Kategori:
AlkaloidsDiterpene AlkaloidsDiterpenes +5
Target Protein:
Arylacetamide deacetylase-like 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gibberellin A4 DB07815
small molecule | CAS: 468-44-0

Deskripsi belum tersedia.

Kategori:
AlkaloidsDiterpene AlkaloidsDiterpenes +2
Target Protein:
Arylacetamide deacetylase-like 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Giloralimab DB18862
biotech | CAS: 2226292-20-0

Giloralimab is under investigation in clinical trial NCT04807972 (Study to Evaluate Adverse Events and Change in Disease Activity When Intravenous (IV) Infusion of ABBV-927 Is Administered in Combination With IV Modified FOLFIRINOX (Mffx) With or Without IV B…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gimatecan DB06721
small molecule | CAS: 292618-32-7

Gimatecan is an orally available 7-t-butoxyiminomethyl-substituted lipophilic camptothecin derivative.

Kategori:
AlkaloidsOATP1B1/SLCO1B1 Substrates
Target Protein:
DNA topoisomerase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gimeracil Approved DB09257
small molecule | CAS: 103766-25-2

Gimeracil is an adjunct to antineoplastic therapy, used to increase the concentration and effect of the main active componets within chemotherapy regimens. Approved by the European Medicines Agency (EMA) in March 2011, Gimeracil is available in combination wi…

Kategori:
Drugs that are Mainly Renally Excreted
Target Protein:
Dihydropyrimidine dehydrogenase [NADP(+)]
Waktu ParuhFollowing a single …
Vol. DistribusiAlthough no intrave…
Klirens-
Genetik -
Ginger oil Approved DB14690
biotech | CAS: 8007-08-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ginisortamab DB18863
biotech | CAS: 2390147-17-6

Ginisortamab is under investigation in clinical trial NCT04393298 (A Study to Assess the Safety, Pharmacokinetics and Anti Tumor Activity of UCB6114 Administered Intravenously to Participants With Advanced Solid Tumors).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ginkgo biloba Approved DB01381
biotech | CAS: 90045-36-6

_Ginkgo biloba_ extract contains a group of terpene lactones (notably, ginkgolides and diterpenes) and ginkgo flavone glycosides (notably, ginkgetin, bilobetin, and sciadopitysin) that have antioxidant and vasoactive properties.[A232389] Most of the studies t…

Kategori:
Anti-Dementia DrugsBiological ProductsBlood Circulation +27
Target Protein:
Sodium-dependent noradrenaline transporterPhospholipase A2, membrane associatedGlycine receptor subunit alpha-1 +5
Waktu ParuhUnpublished human d…
Vol. DistribusiNo data available.
KlirensNo data available.
Genetik -
Ginseng DB01404
biotech | CAS: 50647-08-0

Ginseng is promoted as an adaptogen (a product that increases the body's resistance to stress), one which can to a certain extent be supported with reference to its anticarcinogenic and antioxidant properties. Ginseng is also known to contain phytoestrogens.

Kategori:
AngiospermsAraliaceaeBiological Products +11
Target Protein:
Aryl hydrocarbon receptorInterleukin-6Prostaglandin G/H synthase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Giredestrant DB19125
small molecule | CAS: 1953133-47-5

Giredestrant is under investigation in clinical trial NCT06065748 (A Study to Evaluate Efficacy and Safety of Giredestrant Compared With Fulvestrant (Plus a CDK4/6 Inhibitor), in Participants With Er-positive, Her2-negative Advanced Breast Cancer Resistant to…

Kategori:
Heterocyclic Compounds, Fused-RingIndole AlkaloidsIndoles +1
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Girentuximab DB05304
biotech | CAS: 916138-87-9

Girentuximab is a monoclonal chimeric (mouse/human) antibody directed against carbonic anhydrase IX, an antigen expressed in 95% of clear cell renal cell carcinomas (RCC).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Target Protein:
Carbonic anhydrase 9Interleukin-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1011710-99-8

Girentuximab I-124 is under investigation in clinical trial NCT01762592 (REDECT 2: REnal Masses: Pivotal Trial to DEteCT Clear Cell Renal Cell Carcinoma With PET/CT).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2166101-71-7

Giroctocogene fitelparvovec is under investigation in clinical trial NCT04370054 (Study to Evaluate the Efficacy and Safety of PF-07055480 in Moderately Severe to Severe Hemophilia a Adults).

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Givastomig DB18618
biotech

Givastomig is an anti-Claudin 18.2 and 4.1BB bispecific antibody.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Givosiran Approved DB15066
biotech | CAS: 1639325-43-1

Givosiran is a small interfering RNA (siRNA) directed towards 5-aminolevulinic acid synthase, a critical enzyme in the heme biosynthesis pathway.[L10202] It is manufactured by Alnylam Pharmaceuticals and was first approved for use in the United States in Nove…

Kategori:
Alimentary Tract and MetabolismAmino SugarsAminolevulinate Synthase 1-directed RNA Interaction +13
Target Protein:
ALAS1 mRNA5-aminolevulinate synthase, non-specific, mitochondrial
Waktu ParuhBoth givosiran and …
Vol. DistribusiThe apparent centra…
KlirensThe apparent cleara…
Genetik -
Glafenine DB08963
small molecule | CAS: 3820-67-5

An anthranilic acid derivative with analgesic properties used for the relief of all types of pain. Glafenine is withdrawn from the American market.

Kategori:
Acids, CarbocyclicAminobenzoatesAnalgesics +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Glasdegib Approved DB11978
small molecule | CAS: 1095173-27-5

Glasdegib, also known as PF-04449913, is a small-molecule hedgehog signaling inhibitor selected under the group of benzimidazoles. In early research, benzimidazoles attracted large interest as they represented a class of inhibitors with low molecular weight, …

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +19
Target Protein:
Protein smoothenedSerine/threonine-protein kinase mTOR
Waktu ParuhThe reported half-l…
Vol. DistribusiGlasdegib reported …
KlirensThe clearance rate …
Genetik -
Menampilkan 2951–3000 dari 6694
Sebelumnya Halaman 60 / 134 Berikutnya