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3253

Total database: 17430
Struktur (SMILES)
2451 (75.3%)
Target
1833 (56.3%)
Genomik
35 (1.1%)
Referensi
3253 (100.0%)

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Hasil Pencarian (3253)

Halaman 60 / 66
Tetrasul DB12838
small molecule | CAS: 2227-13-6

Tetrasul has been used in trials studying the treatment of Erythematous (Type One) Rosacea.

Kategori:
Benzene DerivativesHydrocarbons, ChlorinatedHydrocarbons, Halogenated
Target Protein:
Alpha-2C adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tetrofosmin Approved DB11180
small molecule | CAS: 127502-06-1

Tetrofosmin was developed to overcome the non-target uptake of radioligands by the generation of hetero-atomic compounds. It presents a molecular formula of 1,2-bis(bis(2-ethoxyethyl)phosphino)ethane. Tetrofosmin is part of the group of diphosphines. Tetrofos…

Kategori:
Radioactive Diagnostic Agent
Waktu ParuhRefer to [DB09160]
Vol. DistribusiThis pharmacokineti…
KlirensRefer to [DB09160]
Genetik -
small molecule

Betalutin has been used in trials studying the treatment of Non-Hodgkin Lymphoma and Relapsed, Diffuse Large B-cell Lymphoma.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Teverelix DB05624
small molecule | CAS: 151272-78-5

A synthetic decapeptide, water-soluble Gonadotropin-releasing hormone antagonist. It has reached phase II clinical trials.

Kategori:
Amino Acids, Peptides, and ProteinsHormone AntagonistsHormones, Hormone Substitutes, and Hormone Antagonists +1
Target Protein:
Gonadotropin-releasing hormone receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tezacaftor Approved DB11712
small molecule | CAS: 1152311-62-0

Tezacaftor is a drug of the cystic fibrosis transmembrane conductance regulator (CFTR) potentiator class.[L1595] It was developed by Vertex Pharmaceuticals and FDA approved in combination with [ivacaftor] to manage cystic fibrosis.[L6814] This drug was approv…

Kategori:
BCRP/ABCG2 InhibitorsBCRP/ABCG2 SubstratesCytochrome P-450 CYP1A2 Inhibitors +33
Target Protein:
Cystic fibrosis transmembrane conductance regulator
Waktu ParuhThe apparent half-l…
Vol. DistribusiThe apparent volume…
KlirensThe apparent cleara…
Genetik -
Tezepelumab Approved DB15090
biotech | CAS: 1572943-04-4

Asthma is a heterogeneous chronic obstructive respiratory disease with both "type 2" (T2) and T2-low endotypes characterized by reduced airflow, chronic inflammation, and airway remodelling.[A243764, A243769] Thymic stromal lymphopoietin (TSLP), an innate ple…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Target Protein:
Thymic stromal lymphopoietin
Waktu ParuhTezepelumab has an …
Vol. DistribusiTezepelumab has a c…
KlirensTezepelumab has an …
Genetik -
TG01 vaccine DB17123
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1373958-68-9

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingXanthenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thalidomide Approved DB01041
small molecule | CAS: 50-35-1

A piperidinyl isoindole originally introduced as a non-barbiturate hypnotic, thalidomide was withdrawn from the market due to teratogenic effects. It has been reintroduced and used for a number of inflammatory disorders and cancers. Thalidomide displays immun…

Kategori:
Angiogenesis InhibitorsAngiogenesis Modulating AgentsAntineoplastic Agents +38
Target Protein:
Tumor necrosis factorProtein cereblonDNA +1
Waktu ParuhThe half-life of th…
Vol. DistribusiThe volume of distr…
KlirensThe oral clearance …
Genetik -
Thallous chloride Approved DB09316
small molecule | CAS: 7791-12-0

Thallous chloride (also known as Thallium(I) chloride) is a colourless solid intermediate in the isolation of thallium from its ores. It is created from the treatment of thallium(I) sulfate with hydrochloric acid. This solid crystallizes in the caesium chlori…

Kategori:
ElementsMetalsMetals, Heavy +1
Waktu Paruh91% of the blood ra…
Vol. Distribusi3–10 L/kg
KlirensApproximately 4-8% …
Genetik -
Theanine DB12444
small molecule | CAS: 3081-61-6

Theanine, a precursor of ethylamine, is found in green tea. It is under investigation in clinical trial NCT00291070 (Effects of L-Theanine in Boys With ADHD).

Kategori:
Amino AcidsAmino Acids, AcidicAmino Acids, Dicarboxylic +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thenalidine Approved DB04826
small molecule | CAS: 86-12-4

Withdrawn from the Canadian, US, and UK markets in 1963 due to concerns involving neutropenia.

Kategori:
Antihistamines for Systemic UseAntihistamines for Topical UseAntipruritics, Incl. Antihistamines, Anesthetics, Etc. +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Theobromine DB01412
small molecule | CAS: 83-67-0

Theobromine (3,7-dimethylxanthine) is the principle alkaloid in Theobroma cacao (the cacao bean) and other plants. A xanthine alkaloid that is used as a bronchodilator and as a vasodilator. It has a weaker diuretic activity than theophylline and is also a les…

Kategori:
AlkaloidsAnti-Asthmatic AgentsAutonomic Agents +15
Target Protein:
Adenosine receptor A15'-nucleotidaseAdenosine receptor A2a +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Theodrenaline DB12927
small molecule | CAS: 13460-98-5

Theodrenaline is under investigation in clinical trial NCT01311414 (Effect of Cafedrine/Theodrenaline and Urapidil on Cerebral Oxygenation).

Kategori:
Adrenergic and Dopaminergic AgentsAgents that produce hypertensionAlcohols +20
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thiamine Approved DB00152
small molecule | CAS: 70-16-6

Thiamine or thiamin, also known as vitamin B1, is a colorless compound with the chemical formula C12H17N4OS. It is soluble in water and insoluble in alcohol. Thiamine decomposes if heated. Thiamine was first discovered by Umetaro Suzuki in Japan when research…

Kategori:
Alimentary Tract and MetabolismDiet, Food, and NutritionFood +10
Target Protein:
Thiamine pyrophosphokinase 1Pyruvate dehydrogenase E1 component
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thioredoxin Approved DB11298
small molecule | CAS: 52500-60-4

Thioredoxin is a small dithiol protein and specific reductant for major allergenic proteins present in foods from animal and plant products. It is a 12-kD oxidoreductase enzyme encoded by TXN and TXN2 genes that contains a dithiol-disulfide active site. It pl…

Kategori:
Amino Acids, Peptides, and ProteinsProteinsThioredoxins +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thonzylamine Approved DB11235
small molecule | CAS: 91-85-0

Thonzylamine is an antihistamine and anticholinergic drug. It is available as combination products with [DB04837] or [DB00388] for temporary relief of symptoms of common cold, hay fever (allergic rhinitis) or other upper respiratory allergies.

Kategori:
Agents producing tachycardiaAntiallergic Agents, Excl. CorticosteroidsAnticholinergic Agents +11
Target Protein:
Histamine H1 receptorMuscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Threonic acid DB14228
small molecule | CAS: 3909-12-4

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thrombomodulin Alfa Approved DB05777
biotech | CAS: 120313-91-9

Thrombomodulin Alfa is a novel, recombinant and soluble thrombomodulin (ART-123). It is a human protein with both thrombin inhibiting and protein C stimulating activities, for the potential treatment of thromboembolism and blood clotting disorders, such as di…

Kategori:
Amino Acids, Peptides, and ProteinsCarbohydratesGlycoconjugates +7
Target Protein:
ProthrombinCoagulation factor V
Waktu Paruh2–3 days after sc i…
Vol. Distribusi-
Klirens7-10 days
Genetik -
Thymosin beta-4 DB12003
biotech | CAS: 77642-24-1

Thymosin Beta 4 has been investigated for the treatment of STEMI, Dry Eye, Diabetes, Pressure Ulcers, and Dry Eye Syndrome, among others.

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thyrotropin alfa Approved DB00024
biotech | CAS: 194100-83-9

Thyrotropin alfa is a recombinant form of thyroid stimulating hormone used in performing certain tests in patients who have or have had thyroid cancer. It is also used along with a radioactive agent to destroy remaining thyroid tissue in certain patients who …

Kategori:
Agents used to treat hypothyroidismAnterior Pituitary Lobe Hormones and AnaloguesHormones +7
Target Protein:
Thyrotropin receptor
Waktu Paruh25 ± 10 hours
Vol. Distribusi-
Klirens-
Genetik -
Tiapride DB13025
small molecule | CAS: 51012-32-9

Tiapride is a selective D2 and D3 dopamine receptor blocker in the brain.

Kategori:
Acids, CarbocyclicAminesAntipsychotic Agents +16
Target Protein:
Sodium channel protein type 10 subunit alphaD(2) dopamine receptorD(3) dopamine receptor +3
Waktu Paruh2.9–3.6 hours
Vol. DistribusiTiapride distribute…
Klirens16.6 l/h.
Genetik -
Ticagrelor Approved DB08816
small molecule | CAS: 274693-27-5

Ticagrelor, or AZD6140, was first described in the literature in 2003.[A204170,A2903] Ticagrelor is an ADP derivative developed for its P2Y<sub>12</sub> receptor antagonism.[A2903] Unlike [clopidogrel], ticagrelor is not a prodrug.[A2903] It is marketed by As…

Kategori:
AnticoagulantsAntiplatelet agentsBlood and Blood Forming Organs +37
Target Protein:
P2Y purinoceptor 12
Waktu ParuhTicagrelor has a pl…
Vol. DistribusiThe steady state vo…
KlirensThe renal clearance…
Genetik -
biotech

Tick-borne encephalitis (TBE) is a disease caused by the TBE virus (TBEV), transmitted by ticks from the genus _Ixodes_. The disease course is variable. Some patients will be asymptomatic or experience a mild febrile illness, while others will experience the …

Kategori:
VaccinesViral Vaccines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tideglusib DB12129
small molecule | CAS: 865854-05-3

Tideglusib is under the investigation for the development of treatments for Alzheimer's disease and for progressive supranuclear palsy. It is reported to be a potent anti-inflammatory and neuroprotective that is a non-ATP competitive inhibitor of glycogen syn…

Kategori:
Glycogen Synthase Kinase 3, antagonists & inhibitorsSulfur CompoundsThiazoles
Target Protein:
Glycogen synthase kinase-3 beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 144-12-7

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAnticholinergic Agents +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tifuvirtide DB05413
biotech | CAS: 251562-00-2

Tifuvirtide is the first members of a new class of anti-HIV drugs which is also called fusion inhibitors. It has received fast-track designation from the FDA and is in Phase I/II clinical testing.

Kategori:
Amino Acids, Peptides, and ProteinsAntigensAntigens, Viral +14
Target Protein:
Plasma serine protease inhibitor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tigatuzumab DB15101
biotech | CAS: 918127-53-4

Tigatuzumab is under investigation in clinical trial NCT00991796 (CS-1008 With Carboplatin/Paclitaxel in Chemotherapy naïve Subjects With Metastatic or Unresectable Non-small Cell Lung Cancer (NSCLC)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tigecycline Approved DB00560
small molecule | CAS: 220620-09-7

Tigecycline is a glycylcycline antibiotic developed and marketed by Wyeth under the brand name Tygacil. It was developed in response to the growing prevalence of antibiotic resistance in bacteria such as Staphylococcus aureus. It was granted fast-track approv…

Kategori:
Agents that produce neuromuscular block (indirect)Anti-Bacterial AgentsAnti-Infective Agents +7
Target Protein:
16S ribosomal RNA30S ribosomal protein S930S ribosomal protein S12 +3
Waktu Paruh27-43 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 943001-56-7

Deskripsi belum tersedia.

Kategori:
Terpenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tigulixostat DB18799
small molecule | CAS: 1287766-55-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tildrakizumab Approved DB14004
biotech | CAS: 1326244-10-3

Tildrakizumab is a high-affinity, humanized, IgG1 ? antibody targeting interleukin 23 p19 that shows promise in the evolution of treatment strategy in chronic plaque psoriasis [A32255]. The Food and Drug Administration (FDA) approved ILUMYA (tildrakizumab-…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Target Protein:
Interleukin-23
Waktu ParuhThe half-life is ap…
Vol. DistribusiThe geometric mean …
KlirensThe mean (CV%) syst…
Genetik -
TILT-123 DB17519
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Timcodar DB12761
small molecule | CAS: 179033-51-3

Timcodar has been used in trials studying the treatment of Unspecified Adult Solid Tumor, Protocol Specific.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Timonacic DB12856
small molecule | CAS: 444-27-9

Timonacic has been used in trials studying the treatment of HIV Infections.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 14325-05-4

Deskripsi belum tersedia.

Kategori:
Biological FactorsCoordination ComplexesEnzyme Inhibitors +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tinoridine DB13001
small molecule | CAS: 24237-54-5

Tinoridine is under investigation in clinical trial NCT01224756 (Efficacy of Tinoridine in Treating Pain and Inflammation in Adults).

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tinostamustine DB15147
small molecule | CAS: 1236199-60-2

Tinostamustine is under investigation in clinical trial NCT03452930 (Tinostamustine With or Without Radiation Therapy in Treating Patients With Newly Diagnosed MGMT-Unmethylated Glioblastoma).

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tipelukast DB12435
small molecule | CAS: 125961-82-2

Tipelukast is under investigation for the treatment of IPF and Idiopathic pulmonary fibrosis.

Target Protein:
Polyunsaturated fatty acid 5-lipoxygenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tipiracil Approved DB09343
small molecule | CAS: 183204-74-2

Tipiracil is a thymidine phosphorylase inhibitor. It is used in combination with trifluridine, in a ratio of 1:0.5, to form TAS-102. The main function of Tipiracil in TAS-102 is to increase trifluridine bioavailability by inhibiting its catabolism.[A31255] TA…

Kategori:
MATE 1 SubstratesMATE 1 Substrates with a Narrow Therapeutic IndexMATE substrates +6
Target Protein:
Thymidine phosphorylase
Waktu ParuhAfter administratio…
Vol. DistribusiFollowing a single …
KlirensFollowing a single …
Genetik -
Tiplimotide DB12738
biotech | CAS: 178823-49-9

Tiplimotide has been used in trials studying the treatment of Multiple Sclerosis.

Kategori:
Amino Acids, Peptides, and ProteinsMembrane ProteinsMyelin Proteins +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tirasemtiv DB12209
small molecule | CAS: 1005491-05-3

Tirasemtiv has been used in trials studying the treatment of Myasthenia Gravis, Intermittent Claudication, and Amyotrophic Lateral Sclerosis.

Target Protein:
Troponin C, skeletal muscle
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tiropramide DB13091
small molecule | CAS: 55837-29-1

Tiropramide is under investigation in clinical trial NCT01629212 (Comparison of the Efficacy and Safety of Tiropramide and Octylonium in the Treatment of Irritable Bowel Syndrome).

Kategori:
Alimentary Tract and MetabolismAmino AcidsAmino Acids, Aromatic +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tivantinib DB12200
small molecule | CAS: 905854-02-6

Tivantinib has been investigated in Solid Tumors.

Kategori:
Heterocyclic Compounds, Fused-RingProto-Oncogene Proteins c-met, antagonists & inhibitorsPyrrolidines
Target Protein:
Hepatocyte growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TK-112690 DB18822
small molecule | CAS: 22423-26-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TLY-012 DB18336
biotech

TLY-012 is a PEGylated recombinant human tumor necrosis factor-related apoptosis-inducing ligand (PEGylated TRAIL).[L48166]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TMC-310911 DB15623
small molecule | CAS: 1000287-05-7

TMC-310911 (also known as ASC-09) is a novel investigational protease inhibitor (PI) that is structurally similar to the currently available [darunavir].[L12045] It is being investigated for use in HIV-1 infections. TMC-310911 has shown marked activity agains…

Kategori:
Acids, AcyclicAmidesAnti-HIV Agents +10
Target Protein:
Gag-Pol polyproteinHIV-1 protease
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TMC-647055 DB11822
small molecule | CAS: 1204416-97-6

TMC647055 has been used in trials studying the treatment of Hepatitis C, Chronic Hepatitis C, Hepatitis C, Chronic, and Chronic Hepatitis C Virus.

Kategori:
AmidesHeterocyclic Compounds, Fused-RingSulfones +1
Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TMC-649128 DB15152
small molecule | CAS: 1019639-33-8

TMC-649128 is under investigation in clinical trial NCT01391117 (TMC649128HPC1002 - a Trial inGenotype 1 Hepatitis C Virus (HCV) - Infected Participants to Determine the Safety, Tolerability, Pharmacokinetics and Antiviral Activity of TMC649128, Alone and Com…

Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 2951–3000 dari 3253
Sebelumnya Halaman 60 / 66 Berikutnya