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Total database: 17430
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191 (65.6%)
Target
206 (70.8%)
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Halaman 6 / 6
Sulesomab Approved DB13976
biotech | CAS: 167747-19-5

Market product is Tc99m-labeled murine antibody fragment for nuclear imaging of activated granulocytes.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Susoctocog alfa Approved DB11606
biotech | CAS: 1339940-90-7

Intravenous susoctocog alfa is a recombinant, B-domain deleted, porcine sequence antihaemophilic factor VIII (FVIII) product that has recently been approved for the treatment of bleeding episodes in adults with acquired haemophilia A (AHA). AHA is a rare blee…

Kategori:
Blood and Blood Forming OrgansBlood Coagulation FactorsHemostatics
Target Protein:
von Willebrand factor
Waktu ParuhThe terminal half-l…
Vol. DistribusiFollowing intraveno…
KlirensFollowing intraveno…
Genetik -
biotech

A version of [tabituximab barzuxetan] radiolabeled with yttrium-90.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tamsulosin Approved DB00706
small molecule | CAS: 106133-20-4

Tamsulosin is a selective alpha-1A and alpha-1B adrenoceptor antagonist that exerts its greatest effect in the prostate and bladder, where these receptors are most common.[Label] It is indicated for the treatment of signs and symptoms of benign prostatic hype…

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +22
Target Protein:
Alpha-1A adrenergic receptorAlpha-1D adrenergic receptorAlpha-1B adrenergic receptor
Waktu ParuhThe half life in fa…
Vol. Distribusi16L after intraveno…
Klirens2.88L/h.[Label]
Genetik -
Taurine Approved DB01956
small molecule | CAS: 107-35-7

Taurine, whose chemical name is 2-aminoethanesulfonic acid, is one of the most abundant amino acids in several organs. It plays important role in essential biological processes.[A31396] This conditional amino acid can be either be manufactured by the body or …

Kategori:
AlkanesAlkanesulfonic AcidsAmino Acids +5
Target Protein:
Glutamate receptor ionotropic, NMDA 2BGlycine receptor subunit betaGlycine receptor subunit alpha-2 +6
Waktu ParuhOral administration…
Vol. DistribusiThe distribution of…
KlirensThe clearance rate …
Genetik -
Tazobactam Approved DB01606
small molecule | CAS: 89786-04-9

Tazobactam is an antibiotic of the beta-lactamase inhibitor class that prevents the breakdown of other antibiotics by beta-lactamase enzyme producing organisms. It is combined with [Piperacillin] and [Ceftolozane] for the treatment of a variety of bacterial i…

Kategori:
AmidesAnti-Infective AgentsAntibacterials for Systemic Use +15
Target Protein:
Beta-lactamaseBeta-lactamase TEMBeta-lactamase Ohio-1 +1
Waktu ParuhPiperacillin-tazoba…
Vol. Distribusi18.2 L when given w…
KlirensBecause tazobactam …
Genetik -
biotech | CAS: 154361-49-6

Reduced Fab fragment of the murine IgG1 monoclonal antibody IMMU-4 (also called NP-4) with specificity for carcinoembryonic antigen (CEA) covalently labeled with Technitium 99. The molecule has a molecular weight of ~54,000 Daltons.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +9
Target Protein:
Cell adhesion molecule CEACAM1
Waktu ParuhApproximately 1 hour
Vol. Distribusi-
Klirens-
Genetik -
biotech

Technetium Tc-99m epratuzumab is under investigation in clinical trial NCT00003337 (Radiolabeled Monoclonal Antibody in the Detection and Staging of Patients With Non-Hodgkin's Lymphoma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 99944-78-2

Technetium Tc-99m exametazime is a radiopharmaceutical sold under the trade name Ceretec used in the detection of altered regional cerebral perfusion in stroke and other cerebrovascular diseases. It can also be used for the labelling of leukocytes to localise…

Kategori:
AminesCentral Nervous SystemCompounds used in a research, industrial, or household setting +13
Waktu Paruh-
Vol. DistribusiThe activity not as…
Klirens-
Genetik -
small molecule | CAS: 165942-79-0

Technetium Tc-99m nofetumomab merpentan (Tc-99m nm) consists of a Fab fragment of an IgG2b of the pancarcinoma murine antibody NR-LU-10.[A32115] The NR-LU-10 antibody is directed against a 40 kDa glycoprotein antigen expressed in a variety of cancers and some…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Epithelial cell adhesion moleculeB-lymphocyte antigen CD20
Waktu ParuhThe radioactive hal…
Vol. Distribusi-
Klirens-
Genetik -
biotech

Technetium Tc-99m red blood cells is a radiopharmaceutical diagnostic agent that is intravenously administered to be used in blood pool imaging, including cardiac first pass and gated equilibrium imaging and for detection of sites of gastrointestinal bleeding…

Kategori:
Radioactive Diagnostic AgentRadiopharmaceutical Activity
Waktu ParuhTechnetium Tc 99m d…
Vol. DistribusiFollowing intraveno…
Klirens-
Genetik -
small molecule | CAS: 1262984-82-6

Technetium Tc-99m tilmanocept is a radiopharmaceutical diagnostic imaging agent approved by the U.S. Food and Drug Administration (FDA) for the imaging of lymph nodes with or without scintigraphic imaging. It is a macromolecule consisting of multiple units of…

Kategori:
Diagnostic RadiopharmaceuticalsRadioactive Diagnostic AgentRadiopharmaceutical Activity +2
Target Protein:
Macrophage mannose receptor 1
Waktu ParuhTechnetium Tc99m ti…
Vol. Distribusi-
KlirensIn dose-ranging cli…
Genetik -
Telaprevir Approved DB05521
small molecule | CAS: 402957-28-2

Telaprevir is a direct acting antiviral medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized into nine…

Kategori:
Amino Acids, Peptides, and ProteinsAntiinfectives for Systemic UseAntiviral Agents +21
Target Protein:
Genome polyproteinGenome polyproteinSolute carrier organic anion transporter family member 1B1 +1
Waktu ParuhTelaprevir has a ha…
Vol. DistribusiThe estimated appar…
KlirensTelaprevir has an e…
Genetik -
Temoporfin Approved DB11630
small molecule | CAS: 122341-38-2

Temoporfin is a photosensitizing agent used in the treatment of squamous cell carcinoma of the head and neck [FDA Label]. It was first authorized for market by the European Medicines Agency in October 2001. It is currently available under the brand name Fosca…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBiological Factors +8
Waktu ParuhTerminal plasma hal…
Vol. DistribusiThe volume of distr…
KlirensTemoporfin is clear…
Genetik -
Tenofovir disoproxil Approved DB00300
small molecule | CAS: 201341-05-1

Tenofovir disoproxil fumarate (a prodrug of tenofovir), marketed by Gilead Sciences under the trade name _Viread_, belongs to a class of antiretroviral drugs known as nucleotide analogue reverse transcriptase inhibitors (nRTIs). This drug is prescribed in co…

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +19
Target Protein:
Gag-Pol polyproteinReverse transcriptase/RNaseHProtein P
Waktu ParuhWhen a single oral …
Vol. DistribusiThe volume of distr…
KlirensThe clearance of te…
Genetik -
Terazosin Approved DB01162
small molecule | CAS: 63590-64-7

Terazosin is a quinazoline derivative alpha-1-selective adrenergic blocking agent indicated for benign prostatic hyperplasia and hypertension[FDA Label][A176831]. Terazosin blocks adrenaline's action on alpha-1 adrenergic receptors, causing relaxation of smoo…

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +14
Target Protein:
Alpha-1A adrenergic receptorAlpha-1B adrenergic receptorAlpha-1D adrenergic receptor +4
Waktu ParuhTerazosin has a mea…
Vol. Distribusi25L to 30L[A176831].
KlirensPlasma clearance is…
Genetik -
Terconazole Approved DB00251
small molecule | CAS: 67915-31-5

Terconazole is an anti-fungal drug that is mainly used to treat vaginal yeast infections (or vaginal candidiasis). It is classified as a _triazole ketal derivative_.[A178096] Terconazole was initially approved by the FDA in 1987.[FDA label] This drug is avail…

Kategori:
Anti-Infective AgentsAntifungal AgentsAntifungal Agents (Vaginal) +4
Target Protein:
Lanosterol 14-alpha demethylase
Waktu Paruh6.9 hours (range 4.…
Vol. Distribusi-
Klirens-
Genetik -
Teriflunomide Approved DB08880
small molecule | CAS: 163451-81-8

Teriflunomide is the active metabolite of leflunomide, and it acts as an immunomodulatory agent by inhibiting pyrimidine synthesis. It is marketed under the name Aubagio® and is indicated for the treatment of multiple sclerosis, specifically relapsing forms. …

Kategori:
Acids, AcyclicAminesAnalgesics +32
Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrial3-hydroxy-3-methylglutaryl-coenzyme A reductaseDihydroorotate dehydrogenase (quinone), mitochondrial
Waktu ParuhThe median half-lif…
Vol. DistribusiAfter a single intr…
KlirensAfter a single IV d…
Genetik -
biotech

Tetanus Immune Globulin is manufactured from human plasma [FDA Label]. It contains antibodies against tetanus toxoid and is primarily used as prophylaxis against tetanus in wounded patients.

Kategori:
Amino Acids, Peptides, and ProteinsAntiinfectives for Systemic UseBlood Proteins +7
Target Protein:
Tetanus toxin
Waktu ParuhHalf life is about …
Vol. Distribusi-
Klirens-
Genetik -
Thrombin Approved DB11300
biotech

Also known as coagulation factor II, thrombin is a serine protease that plays a physiological role in regulating hemostasis and maintaining blood coagulation. Once converted from prothrombin, thrombin converts fibrinogen to fibrin, which, in combination with …

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +18
Target Protein:
Coagulation factor XICoagulation factor XIII A chainCoagulation factor XIII B chain +7
Waktu ParuhUnfortunately, litt…
Vol. DistribusiLittle has been rep…
KlirensAlthough little has…
Genetik -
Ticlopidine Approved DB00208
small molecule | CAS: 55142-85-3

Ticlopidine is an effective inhibitor of platelet aggregation. It is a prodrug that is metabolised to an active form, which blocks the ADP receptor that is involved in GPIIb/IIIa receptor activation leading to platelet aggregation. Ticlopidine is marketed und…

Kategori:
Antiplatelet agentsBlood and Blood Forming OrgansCardiovascular Agents +36
Target Protein:
Platelet-activating factor receptorP2Y purinoceptor 12
Waktu ParuhHalf-life following…
Vol. DistribusiThe volume of distr…
KlirensTiclopidine clearan…
Genetik -
Tizanidine Approved DB00697
small molecule | CAS: 51322-75-9

Tizanidine is a fast-acting drug used for the management of muscle spasm, which may result from the effects of multiple sclerosis, stroke, an acquired brain injury, or a spinal cord injury [T574]. It may also be caused by musculoskeletal injury [A177583]. R…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +24
Target Protein:
Alpha-1 adrenergic receptorsAlpha-2 adrenergic receptorsNischarin
Waktu ParuhApproximately 2.5 h…
Vol. DistribusiExtensively distrib…
Klirens**A note on renal i…
Genetik -
Trastuzumab emtansine Approved DB05773
biotech | CAS: 1018448-65-1

Trastuzumab emtansine, formerly called Trastuzumab-DM1 (T-DM1) is a first-in-class HER2 antibody drug conjugate (ADC) comprised of Genentech's trastuzumab antibody linked to ImmunoGen's cell-killing agent, DM1. T-DM1 combines two strategies-- anti-HER2 activi…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +42
Target Protein:
Receptor tyrosine-protein kinase erbB-2
Waktu ParuhTrastuzumab emtansi…
Vol. DistribusiThe volume of distr…
KlirensAfter IV infusion, …
Genetik -
Triclabendazole Approved DB12245
small molecule | CAS: 68786-66-3

Triclabendazole, manufactured by Novartis pharmaceuticals, is an antihelminthic drug that was approved by the FDA in February 2019 for the treatment of fascioliasis in humans.[FDA label, L5452] Fascioliasis is a parasitic infection often caused by the helmi…

Kategori:
AnthelminticsAnti-Infective AgentsAntihelminthic +34
Target Protein:
CruzipainExcretory Secretory (ES) proteins
Waktu ParuhThe plasma eliminat…
Vol. DistribusiThe apparent volume…
Klirens-
Genetik -
Urea C-13 Approved DB09510
small molecule | CAS: 58069-82-2

Urea 13C is a urea molecule radiolabelled with the non-radioactive element carbon-13. It is currently used for the Urea Breath Test (UBT) and is available as a rapid diagnostic test (marketed as Pranactin-Citric) for the detection of Helicobacter pylori infec…

Kategori:
Diagnostic AgentsHelicobacter pylori Diagnostic
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Urea C-14 Approved DB09513
small molecule | CAS: 594-05-8

Urea 14C is a urea molecule radiolabelled with a radioactive carbon-14. It is currently used for the Urea Breath Test (UBT) and is available as a rapid diagnostic test (marketed as PyTest) for the detection of Helicobacter pylori infections. H pylori is a com…

Kategori:
Radioactive Diagnostic Agent
Waktu Paruh14C-urea that is no…
Vol. Distribusi-
Klirens-
Genetik -
Vaborbactam Approved DB12107
small molecule | CAS: 1360457-46-0

Vaborbactam is a ?-lactamase inhibitor based on a cyclic boronic acid pharmacophore.[A32053] It has been used in trials investigating the treatment of bacterial infections in subjects with varying degrees of renal insufficiency. In August 2017, a combination …

Kategori:
AcidsAcids, NoncarboxylicAnti-Infective Agents +6
Target Protein:
Beta-lactamaseBeta-lactamaseCarbapenem-hydrolyzing beta-lactamase KPC +7
Waktu ParuhThe half life of va…
Vol. DistribusiThe steady-state vo…
KlirensThe mean renal clea…
Genetik -
Valaciclovir Approved DB00577
small molecule | CAS: 124832-26-4

Valaciclovir (valacyclovir), also known as _Valtrex_, is an antiviral drug that has been used to manage and treat various herpes infections for more than 2 decades. It was initially approved by the FDA in 1995 [FDA label] and marketed by GlaxoSmithKline [L56…

Kategori:
Acyclovir and prodrugAmino AcidsAmino Acids, Branched-Chain +19
Target Protein:
Thymidine kinaseDNA polymerase catalytic subunit
Waktu ParuhThe plasma eliminat…
Vol. DistribusiCerebrospinal fluid…
KlirensRenal clearance of …
Genetik -
Valbenazine Approved DB11915
small molecule | CAS: 1025504-45-3

Valbenazine is a modified metabolite of [tetrabenazine], and it is currently being approved for the treatment of various movement disorders, particularly tardive dyskinesia and chorea associated with Huntington's disease.[L47885,A261135] Tardive dyskinesia ha…

Kategori:
Amino AcidsAmino Acids, Branched-ChainAmino Acids, Peptides, and Proteins +11
Target Protein:
Synaptic vesicular amine transporter
Waktu ParuhBoth Valbenazine an…
Vol. DistribusiThe mean steady-sta…
KlirensValbenazine has a m…
Genetik -
biotech

Recombinant zoster vaccine, manufactured as the product Shingrix by GlaxoSmithKline, is an adjuvanted non-live recombinant vaccine indicated for prevention of shingles. First approved in October 2017 by the Food and Drug Administration, Shingrix is the prefer…

Kategori:
VaccinesVaricella Zoster Vaccines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Venetoclax Approved DB11581
small molecule | CAS: 1257044-40-8

Venetoclax is a BCL-2 inhibitor that was initially approved by the FDA in April 2016 [FDA label]. Proteins in the B cell CLL/lymphoma 2 (BCL-2) family are important regulators of the apoptotic (programmed cell death) process [A18565], [A18566]. Venetoclax is…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +19
Target Protein:
Apoptosis regulator Bcl-2
Waktu ParuhThe half-life of ve…
Vol. DistribusiThe population esti…
KlirensMainly hepatic [FDA…
Genetik -
Venlafaxine Approved DB00285
small molecule | CAS: 93413-69-5

Venlafaxine is an antidepressant and a serotonin and norepinephrine reuptake inhibitor (SNRI). Its active metabolite, [desvenlafaxine], works by blocking the reuptake of serotonin and norepinephrine, which are key neurotransmitters in mood regulation. Venlafa…

Kategori:
Agents producing tachycardiaAgents that reduce seizure thresholdAmines +39
Target Protein:
Sodium-dependent serotonin transporterSodium-dependent noradrenaline transporterSodium-dependent dopamine transporter
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +2
Waktu ParuhThe apparent elimin…
Vol. DistribusiThe apparent volume…
KlirensMean ± SD plasma ap…
Genetik 5 Varian
Vestronidase alfa Approved DB12366
biotech | CAS: 1638194-78-1

Vestronidase alfa, or vestronidase alfa-vjbk, is a recombinant human lysosomal beta glucuronidase that is a purified enzyme produced by recombinant DNA technology in a Chinese hamster ovary cell line. The enzyme is a homotetramer consisted of 4 monomers with …

Kategori:
Alimentary Tract and MetabolismEnzymesEnzymes and Coenzymes +3
Waktu ParuhAfter repeated dosi…
Vol. DistribusiAfter repeated dosi…
KlirensAfter repeated dosi…
Genetik -
Vilazodone Approved DB06684
small molecule | CAS: 163521-12-8

Vilazodone is a novel compound with combined high affinity and selectivity for the 5-hydroxytryptamine (5-HT) transporter and 5-HT(1A) receptors[Label,A177622]. Vilazodone may also be associated with less sexual dysfunction and weight gain[A6947]. Vilazodone …

Kategori:
Agents that produce hypertensionAntidepressive AgentsAntidepressive Agents Indicated for Depression +26
Target Protein:
Sodium-dependent serotonin transporter5-hydroxytryptamine receptor 1A
Waktu Paruh25 hours[Label,A384…
Vol. DistribusiVilazodone's volume…
KlirensClearance of vilazo…
Genetik -
Vitamin E Approved DB00163
small molecule | CAS: 59-02-9

In 1922, vitamin E was demonstrated to be an essential nutrient[A32448]. Vitamin E is a term used to describe 8 different fat soluble tocopherols and tocotrienols, alpha-tocopherol being the most biologically active[A176104]. Vitamin E acts as an antioxidant,…

Kategori:
AntioxidantsBasic Ointments and ProtectantsBenzopyrans +23
Target Protein:
SEC14-like protein 4SEC14-like protein 3SEC14-like protein 2 +7
Waktu Paruh44 hours in prematu…
Vol. Distribusi0.41L/kg in prematu…
Klirens6.5mL/hr/kg in prem…
Genetik -
VM4-037 DB15319
small molecule | CAS: 1071470-72-8

VM4-037 is under investigation in clinical trial NCT00884520 (An Exploratory, Open Label, Multi-Center, Non-Randomized Study of [F-18]VM4-037).

Kategori:
AmidesAmino Acids, Peptides, and ProteinsFluorine Radioisotopes +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Voxilaprevir Approved DB12026
small molecule | CAS: 1535212-07-7

Voxilaprevir is a Direct-Acting Antiviral (DAA) medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized i…

Kategori:
Acids, AcyclicAmidesAmino Acids +36
Target Protein:
Genome polyproteinGenome polyprotein
Waktu Paruh33 hr [FDA Label]
Vol. Distribusi-
Klirens-
Genetik -
Yellow fever vaccine Approved DB10805
biotech

Yellow fever vaccine prevents against Yellow Fever, a viral hemorrhagic disease caused by the transmission of a _flavivirus_ through the bite of an infected mosquito. Symptoms of Yellow fever can range from asymptomatic, to mild flu-like illness, to more seve…

Kategori:
Actively Acquired ImmunityAntiinfectives for Systemic UseBiological Products +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2377668-38-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Zirconium panitumumab Zr-89 is under investigation in clinical trial NCT05423197 (Study Evaluating Zr-panitumumab for Assessment of Suspected Metastatic Lesions on 18F-FDG-PET/CT in Head and Neck Squamous Cell Carcinoma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zolpidem Approved DB00425
small molecule | CAS: 82626-48-0

Zolpidem, also known as _Ambien_, is a hypnotic drug that was initially approved by the FDA in 1992 [FDA label]. Zolpidem improves sleep in patients with insomnia. It is aimed for use in patients with difficulties initiating sleep. This drug decreases the ti…

Kategori:
Benzodiazepine hypnotics and sedativesCentral Nervous System AgentsCentral Nervous System Depressants +21
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Gamma-aminobutyric acid receptor subunit gamma-3Gamma-aminobutyric acid receptor subunit alpha-2 +2
Waktu ParuhThe average zolpide…
Vol. Distribusi0.54 to 0.68 L/kg (…
KlirensIn a clinical trial…
Genetik -
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