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2279

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Halaman 6 / 46
Atibuclimab DB06546
biotech | CAS: 2417175-94-9

Atibuclimab (IC14) is a chimeric CD14 antibody investigated for the treatment of patients with severe sepsis.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Target Protein:
Monocyte differentiation antigen CD14
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Atidarsagene autotemcel Approved DB17538
biotech

Atidarsagene autotemcel, sold under the brand name Libmeldy, is a gene therapy comprising genetically modified autologous CD34+ enriched hematopoietic stem and progenitor cells transduced _ex vivo_ using a lentiviral vector encoding the human arylsulfatase A …

Kategori:
Alimentary Tract and MetabolismAutologous Cultured CellAutologous Hematopoietic Stem Cell-Based Gene Therapy +2
Target Protein:
Human Arylsulfatase A mRNA
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Atipamezole DB11481
small molecule | CAS: 104054-27-5

Atipamezole is a synthetic ?2 adrenoceptor antagonistused to reverse the sedative and analgesic effects of dexmedetomidine and medetomidine in dogs. It has also been undergone research as a potential anti-Parkinsonian drug for humans.

Kategori:
Adrenergic AgentsAdrenergic alpha-2 Receptor AntagonistsAdrenergic alpha-Antagonists +3
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Atoltivimab Approved DB15898
biotech | CAS: 2135632-29-8

Ebola virus (EBOV) remains an important human pathogen within the _Ebolavirus_ genus, having been responsible for at least 17 known outbreaks with an average case fatality rate of 43.92%.[A221825] Immune therapy using monoclonal antibodies (mAbs) is becoming …

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +10
Target Protein:
Envelope glycoprotein
Waktu ParuhAtoltivimab adminis…
Vol. DistribusiAtoltivimab adminis…
KlirensAtoltivimab adminis…
Genetik -
Atomoxetine Approved DB00289
small molecule | CAS: 83015-26-3

Atomoxetine is a selective norepinephrine (NE) reuptake inhibitor used for the treatment of attention deficit hyperactivity disorder (ADHD). Also known as the marketed product Strattera, atomoxetine is used with other treatment modalities (psychological, educ…

Kategori:
Adrenergic AgentsAgents producing tachycardiaAgents that produce hypertension +17
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporterNMDA receptor +2
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +3
Waktu ParuhThe reported half-l…
Vol. DistribusiThe reported volume…
KlirensThe clearance rate …
Genetik 6 Varian
Atorvastatin Approved DB01076
small molecule | CAS: 134523-00-5

Atorvastatin (Lipitor®), is a lipid-lowering drug included in the statin class of medications. By inhibiting the endogenous production of cholesterol in the liver, statins lower abnormal cholesterol and lipid levels, and ultimately reduce the risk of cardiova…

Kategori:
Agents Causing Muscle ToxicityAnticholesteremic AgentsBSEP/ABCB11 Substrates +37
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductaseDipeptidyl peptidase 4Aryl hydrocarbon receptor +2
Gen Terkait:
KIF6 HMGCR CYP3A4
Waktu ParuhThe half-life of at…
Vol. DistribusiThe reported volume…
KlirensThe registered tota…
Genetik 3 Varian
Atrazine DB07392
small molecule | CAS: 1912-24-9

Atrazine is a selective triazine herbicide. Inhalation hazard is low and there are no apparent skin manifestations or other toxicity in humans. Acutely poisoned sheep and cattle may show muscular spasms, fasciculations, stiff gait, increased respiratory rates…

Kategori:
AgrochemicalsCompounds used in a research, industrial, or household settingHerbicides +3
Target Protein:
Photosynthetic reaction center cytochrome c subunitReaction center protein H chainReaction center protein L chain +1
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ATSN-101 DB18327
biotech

ATSN-101 is a adeno-associated virus serotype 5 encoding human retinal guanylate cyclase 1 gene (AAV5-GUCY2D)

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ATX-101 DB05780
small molecule

ATX-101 (medical), sodium deoxycholate for subcutaneous injection, is being evaluated as a treatment for the reduction of localized fat deposits. This includes treatment of superficial lipomas (benign tumors of soft tissue composed of mature fat cells), fat d…

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ATYR-1940 DB16991
biotech

Deskripsi belum tersedia.

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Aurothioglucose Approved DB09121
small molecule | CAS: 12192-57-3

Aurothioglucose, also known as gold thioglucose, was formerly used to treat rheumatoid arthritis. Contemporary research on the effect of gold salts treatment began in 1935, primarily to reduce inflammation and to slow disease progression in patients with r…

Kategori:
Antiinflammatory and Antirheumatic ProductsAntirheumatic AgentsDrugs that are Mainly Renally Excreted +5
Target Protein:
Adenylate cyclase type 1Adenylate cyclase type 2Adenylate cyclase type 5
Waktu ParuhThe biological half…
Vol. DistribusiReadily accessible …
KlirensWhen a standard wee…
Genetik -
biotech

Deskripsi belum tersedia.

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biotech

Deskripsi belum tersedia.

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Avalglucosidase alfa Approved DB16099
biotech | CAS: 1802558-87-7

Avalglucosidase alfa, or NeoGAA, is a drug for enzyme replacement therapy specifically designed for Pompe disease, a rare inherited neuromuscular disorder caused by the deficiency of the alpha-glucosidase (GAA) enzyme. GAA is an essential enzyme that hydrolyz…

Kategori:
Alimentary Tract and MetabolismEnzyme Replacement TherapyEnzymes +2
Target Protein:
Cation-independent mannose-6-phosphate receptor
Waktu ParuhThe mean avalglucos…
Vol. DistribusiThe volume of distr…
KlirensThe mean avalglucos…
Genetik -
biotech | CAS: 2227000-30-6

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
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small molecule | CAS: 435327-40-5

Avasopasem manganese, also known as GC4419, is a highly-selective small molecule mimetic of superoxide dismutase (SOD) being investigated for the reduction of radiation-induced severe oral mucositis.[L27246, L27256] This drug has potential application for rad…

Kategori:
AntioxidantsFree Radical Scavengers
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AVB-001 DB18452
biotech

AVB-001 is an encapsulated, engineered human ARPE-19 cell line that constitutively expresses the native human IL-2 cytokine

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AVB-101 DB18416
biotech

AVB-101 is a recombinant AAV9 vector encoding the human progranulin (PGRN) gene.

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Avelumab Approved DB11945
biotech | CAS: 1537032-82-8

Avelumab is a human IgG1 lambda monoclonal antibody that binds programmed cell death ligand-1 (PD-L1) to block its interaction with its receptors found on T cells and antigen-presenting cells.[A261496] Avelumab was first approved by the FDA on March 23, 2017.…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +19
Target Protein:
Programmed cell death 1 ligand 1
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe geometric mean …
KlirensThe total systemic …
Genetik -
AVI-014 DB17086
biotech

AVI-014 is a glycosylated, recombinant human granulocyte colony-stimulating factor (G-CSF).

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AVID-200 DB18454
biotech | CAS: 2269485-28-9

AVID-200 is an Anti-transforming growth factor beta (TGF-?) trap fusion protein.

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Avizakimab DB18842
biotech | CAS: 2229685-51-0

Avizakimab is under investigation in clinical trial NCT03371251 (Study of BOS161721 in Systemic Lupus Erythematosus (SLE) Patients on a Background of Limited Standard of Care).

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Avobenzone Approved DB09495
small molecule | CAS: 70356-09-1

Avobenzone is dibenzoyl methane derivative. It is oil soluble ingredient. Avobenzone has the ability to absorb ultraviolet light over wider range of wavelengths. It is included in many commercially available sunscreens which are used as wide spectrum sunscree…

Kategori:
Compounds used in a research, industrial, or household settingCosmeticsDermatologicals +4
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AVP-21D9 DB17798
biotech

AVP-21D9 is a fully human anthrax monoclonal antibody that is being investigated as an anthrax antitoxin.[A259522]

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
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AVR-RD-01 DB17651
biotech

AVR-RD-01 is an investigational _ex vivo_ lentiviral gene therapy developed by AVROBIO Inc. It consists of autologous CD34+ cells that transduced with Lentiviral Vector/alpha-galactosidase A (AGA) encoding for the human AGA complementary deoxyribonucleic acid…

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AVR-RD-02 DB17650
biotech

AVR-RD-02 is an investigational _ex vivo_ lentiviral gene therapy developed by AVROBIO Inc. It consists of autologous CD34+ enriched hematopoietic stem cells (HSCs) that have been genetically modified _ex vivo_ with a lentiviral vector (LV) to contain a ribon…

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AVR-RD-04 DB18644
biotech

AVR-RD-04 is an investigational gene therapy for cystinosis. It consists of autologous CD34+ enriched cells transduced with a lentiviral vector containing RNA resulting in codon-optimized cDNA encoding for functional human cystinosin.

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AVR-RD-05 DB18631
biotech

AVR-RD-05 is a gene therapy comprising genetically modified autologous stem cells transduced _ex vivo_ with a lentiviral vector encoding the human iduronate-2-sulfatase (IDS) enzyme. It is under investigation for the treatment of Hunter Syndrome (Mucopolysacc…

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AVR118 DB04979
biotech

AVR118 represents a new type of biopolymer chemistry that also possesses novel immunomodulator activity. This non-toxic peptide-nucleic acid, which to date has shown no indication of human toxicity, appears to stimulate the proinflammatory responses required …

Kategori:
HIVNucleic Acids, Nucleotides, and NucleosidesNucleotides +2
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biotech

Axalimogene filolisbac is under investigation in clinical trial NCT02853604 (Study of ADXS11-001 in Subjects With High Risk Locally Advanced Cervical Cancer).

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Axatilimab Approved DB16388
biotech | CAS: 2155851-88-8

Axatilimab is a humanized IgG4 monoclonal antibody produced in Chinese hamster ovary cells.[L51194] It is targeted against macrophage colony-stimulating factor 1 receptor (CSF-1R), causing a reduction in circulating levels of monocytes and macrophages respons…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Macrophage colony-stimulating factor 1 receptor
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe volume of distr…
KlirensThe total clearance…
Genetik -
Azadirachtin DB19419
small molecule | CAS: 11141-17-6

Azadirachtin is under investigation in clinical trial NCT06617026 (Short-term Outcome of Medical vs. Surgical Management of Chronic Anal Fissure).

Kategori:
AgrochemicalsAzadirachtaCompounds used in a research, industrial, or household setting +5
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Azaperone DB11376
small molecule | CAS: 1649-18-9

Azaperone is a pyridinylpiperazine and butyrophenone agent that is capable of eliciting neuroleptic sedative and antiemetic effects. It is subsequently employed predominantly as a veterinary tranquilizer and mainly for pigs and elephants. At the same time, th…

Kategori:
Antipsychotic AgentsAntipsychotic Agents (First Generation [Typical])Butyrophenones +11
Target Protein:
D(3) dopamine receptorD(2) dopamine receptor
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AZD-8330 DB06061
small molecule | CAS: 869357-68-6

AZD-8330 is a potent, selective, orally active MEK inhibitor that blocks signal transduction pathways implicated in cancer cell proliferation and survival. AZD-8330 has shown tumor suppressive activity in multiple preclinical models of human cancer including …

Kategori:
Protein Kinase InhibitorsPyridines
Target Protein:
Mitogen-activated protein kinase kinase kinase 1
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Azelaic acid Approved DB00548
small molecule | CAS: 123-99-9

Azelaic acid is a saturated dicarboxylic acid found naturally in wheat, rye, and barley. It is also produced by _Malassezia furfur_, also known as _Pityrosporum ovale_, which is a species of fungus that is normally found on human skin. Azelaic acid is effecti…

Kategori:
Acids, AcyclicAnti-Acne PreparationsAnti-Acne Preparations for Topical Use +5
Target Protein:
Thioredoxin reductasePolyprenal reductase3-oxo-5-alpha-steroid 4-dehydrogenase 1 +4
Waktu ParuhThe observed half-l…
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Azelnidipine DB09230
small molecule | CAS: 123524-52-7

Azelnidipine is a dihydropyridine calcium channel blocker. It is marketed by Daiichi-Sankyo pharmaceuticals, Inc. in Japan. It has a gradual onset of action and produces a long-lasting decrease in blood pressure, with only a small increase in heart rate, unl…

Kategori:
Acids, AcyclicAgents causing hyperkalemiaAmino Acids +14
Target Protein:
Voltage-dependent L-type calcium channel subunit beta-1
Waktu Paruh16 –28 hours [L1383…
Vol. DistribusiIn a Chinese study …
Klirens-
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Azilsartan medoxomil Approved DB08822
small molecule | CAS: 863031-21-4

Azilsartan medoxomil is a prodrug that is broken down to azilsartan, which belongs in the angiotensin-receptor blocking (ARB) drug class. It is a selective AT1 subtype angiotensin II receptor antagonist. Azilsartan medoxomil is a relatively recently-developed…

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +18
Target Protein:
Type-1 angiotensin II receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensRenal clearance of …
Genetik -
biotech

Bacillus Calmette-Guerin (BCG) substrain Russian BCG-I is a live BCG vaccine administered directly into the bladder for the adjuvant treatment of papillary urothelial cell carcinoma of the bladder. Live BCG vaccines administered intravesically have been a gol…

Kategori:
Antineoplastic AgentsLive vaccinesVaccines
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biotech | CAS: 68038-66-4

Deskripsi belum tersedia.

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Baclofen Approved DB00181
small molecule | CAS: 1134-47-0

Baclofen is a gamma-aminobutyric acid (GABA) agonist used as a skeletal muscle relaxant. Although originally designed in 1962 to treat epilepsy, baclofen was not effective in treating this condition but instead was shown to reduce spasticity in selected patie…

Kategori:
Agents Causing Muscle ToxicityAmino AcidsAmino Acids, Peptides, and Proteins +15
Target Protein:
Gamma-aminobutyric acid type B receptor subunit 2C-X-C chemokine receptor type 4Gamma-aminobutyric acid type B receptor subunit 1
Waktu ParuhThe half-life is 2-…
Vol. DistribusiThe volume of distr…
KlirensThe systemic cleara…
Genetik -
Baloramotide DB17986
biotech | CAS: 2207581-19-7

Deskripsi belum tersedia.

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Bamlanivimab Approved DB15718
biotech | CAS: 2423943-37-5

Bamlanivimab (LY-CoV555, also known as LY3819253), is a synthetic monoclonal antibody (mAb) derived from one of the first blood samples in the United States from a patient who recovered from COVID-19.[A224039, L15311, L15316] Bamlanivimab is a neutralizing Ig…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +10
Target Protein:
Spike glycoprotein
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Barecetamab DB17479
biotech | CAS: 2275727-74-5

Deskripsi belum tersedia.

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Barium sulfate Approved DB11150
small molecule | CAS: 7727-43-7

Barium sulfate is an inorganic compound with the chemical formula BaSO4 [L1957]. Barium sulfate occurs in nature as the mineral _barite_. It is also used in various manufacturing applications and mixed into heavy concrete to serve as a radiation shield [L1…

Kategori:
Barium CompoundsBarium Sulfate Containing X-Ray Contrast MediaCompounds used in a research, industrial, or household setting +9
Waktu Paruh-
Vol. Distribusi-
KlirensThe rate of excreti…
Genetik -
Barzolvolimab DB18934
biotech | CAS: 2438203-51-9

Barzolvolimab is under investigation in clinical trial NCT06455202 (A Phase 3 Study of Barzolvolimab in Participants With Chronic Spontaneous Urticaria (CSU)).

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biotech | CAS: 106096-93-9

Basic Fibroblast Growth Factor (bFGF) is a single-chain polypeptide growth factor that plays a significant role in the process of wound healing and is a potent inducer of physiologic angiogenesis. Several different forms of the human protein exist ranging fro…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsFibroblast Growth Factor 2, antagonists & inhibitors +4
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Basiliximab Approved DB00074
biotech | CAS: 179045-86-4

A recombinant chimeric (murine/human) monoclonal antibody (IgG1k) that functions as an immunosuppressive agent, specifically binding to and blocking the interleukin-2 receptor a-chain (IL-2R alpha, also known as CD25 antigen) on the surface of activated T-lym…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +14
Target Protein:
Interleukin-2 receptor subunit alphaInterleukin-2 receptor subunit beta
Waktu Paruh7.2 +/- 3.2 days (a…
Vol. Distribusi* 7.8 ± 5.1 L [Pedi…
Klirens* 41 +/- 19 mL/h [A…
Genetik -
Batoclimab DB16104
biotech | CAS: 2187430-05-1

Batoclimab is under investigation in clinical trial NCT04428255 (A Clinical Study on the Efficacy and Safety of HBM9161 in Patients With ITP).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
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Batroxobin DB09005
biotech | CAS: 9039-61-6

Batroxobin is a defibrinogenating hemostatic agent derived from the venom of a pit viper, Bothrops atrox moojeni. In addition to batroxobin, the venom of Bothrops atrox has a composition of 10.2% neutral carbohydrate. Batroxobin is a serine protease, which cl…

Kategori:
Biological FactorsBlood and Blood Forming OrgansCardiovascular Agents +18
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BB-1701 DB17443
biotech

BB-1701 is a humanized IgG1 kappa monoclonal antibody (anti-HER2 antibody) conjugated to eribulin developed by Bliss Biopharmaceutical.

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