Hasil Filter

16749

Total database: 17430
Struktur (SMILES)
11810 (70.5%)
Target
9015 (53.8%)
Genomik
112 (0.7%)
Referensi
16749 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (16749)

Halaman 59 / 335
AGG-523 DB15460
small molecule | CAS: 920289-29-8

AGG-523 is under investigation in clinical trial NCT00380900 (Study Evaluating the Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of Multiple Ascending Doses in Healthy subjects and in subjects with osteoarthritis).

Target Protein:
A disintegrin and metalloproteinase with thrombospondin motifs 5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AGI-1096 DB05840
small molecule

AGI-1096 is a novel oral antioxidant and selective anti-inflammatory agent that is being developed to address the accelerated inflammation of grafted blood vessels, known as transplant arteritis, common in chronic organ transplant rejection.

Kategori:
Acids, AcyclicBenzene DerivativesFatty Acids +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AGI-134 DB19005
small molecule | CAS: 1821461-84-0

AGI-134 is under investigation in clinical trial NCT03593226 (Study to Evaluate Safety & Tolerability of AGI-134 in Solid Tumour).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AGIL-FA DB16973
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Agkistrodon piscivorus antivenin is derived and purified immunoglobulin fragments obtained from other domestic animals such as sheep previously immunized with Agkistrodon piscivorus (_Cottonmouth_ or _Water Moccasin snake_). The final purified antivenin produ…

Kategori:
AntiveninsPassively Acquired ImmunityVenom Neutralization
Target Protein:
Group 10 secretory phospholipase A2
Waktu Paruh12 to 23 hours [FDA…
Vol. Distribusi-
KlirensSystemic clearance …
Genetik -
biotech | CAS: 1621271-62-2

Aglatimagene besadenovec is under investigation in clinical trial NCT00638612 (AdV-tk Therapy With Surgery and Chemoradiation for Pancreas Cancer (PaTK01)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Agmatine DB08838
small molecule | CAS: 306-60-5

Agmantine is a natural metabolite of the amino acid arginine. It is formed when arginine is decarboxylated by the enzyme arginine decarboxylase and is found naturally in ragweed pollen, ergot fungi, octopus muscle, herring sperm, sponges, and the mammalian br…

Kategori:
Agents causing hyperkalemiaAmidinesAntiarrhythmic agents +12
Target Protein:
Alpha-2C adrenergic receptorNischarinAcetylcholine receptor subunit alpha +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AGN-201904 DB13135
small molecule | CAS: 651729-53-2

Agn 201904 has been used in trials studying the prevention of Peptic Ulcer.

Kategori:
2-PyridinylmethylsulfinylbenzimidazolesBenzimidazolesHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Agomelatine Approved DB06594
small molecule | CAS: 138112-76-2

Agomelatine is structurally closely related to melatonin. Agomelatine is a potent agonist at melatonin receptors and an antagonist at serotonin-2C (5-HT2C) receptors, tested in an animal model of depression. Agomelatine was developed in Europe by Servier Labo…

Kategori:
AcetatesAcids, AcyclicAmides +15
Target Protein:
5-hydroxytryptamine receptor 2CMelatonin receptor type 1AMelatonin receptor type 1B
Waktu Paruh<2 hours
Vol. Distribusi-
Klirens-
Genetik -
AGRO100 DB04998
biotech | CAS: 301636-59-9

AGRO100 is an oligonucleotide that functions as an aptamer and binds to nucleolin, a protein found intranuclear in all cells, but uniquely expressed on the surface of tumor cells. Such binding leads to internalization of the complex, and a strong anti-prolife…

Kategori:
Aptamers, NucleotideNucleic Acids, Nucleotides, and NucleosidesNucleotides +2
Target Protein:
NF-kappa-B essential modulator
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Agrostis gigantea pollen Approved DB10403
biotech

Agrostis gigantea pollen is the pollen of the Agrostis gigantea plant. Agrostis gigantea pollen is mainly used in allergenic testing.

Kategori:
Allergenic ExtractsCell-mediated ImmunityGrass Pollen Allergen Extracts +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Agrostis gigantea top Approved DB14757
biotech

Agrostis gigantea top is the flowering part of the Agrostis gigantea plant. Agrostis gigantea top is mainly used in allergenic testing.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Agrostis stolonifera pollen Approved DB10962
biotech

Agrostis stolonifera pollen is the pollen of the Agrostis stolonifera plant. Agrostis stolonifera pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityGrass Pollen Allergen ExtractsIncreased Histamine Release +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AGS-004 DB05742
small molecule

AGS-004 is a personalized RNA-loaded dendritic cellbased immunotherapy that is designed to stimulate the patient’s immune system to target and destroy the patient’s own unique viral burden. Non-personalized HIV immunotherapies are unable to raise cytotoxic T…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AGS-005 DB05741
small molecule

AGS-005 is a personalized dendritic cell-based immunotherapy, with optimized immune response characteristics, that is designed to stimulate the patient's immune system to target and destroy the patient's cancer cells.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AGS-16C3F DB17551
biotech

AGS 16C3F is an intravenously administered, anti-ectonucleotide pyrophosphatase/phosphodiesterase 3 (ENPP3) antibody-drug conjugate. AGS-16C3F is under investigation in clinical trial NCT02639182 (A Study of AGS-16C3F vs. Axitinib in Metastatic Renal Cell Car…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AGS-499 DB18058
small molecule | CAS: 1092372-02-5

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesTelomerase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AGT-182 DB17630
biotech

AGT-182 is an investigational enzyme replacement therapy engineered by the fusion of the iduronate-2-sulfatase (IDS) enzyme and a human insulin receptor monoclonal antibody.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AGTC-401 DB18432
biotech

AGTC-401 is a recombinant adeno-associated virus vector expressing the cyclic nucleotide gated channel beta subunit (rAAV-CNGB3).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AGTC-402 DB18433
biotech

AGTC-402 is a recombinant adeno-associated virus vector expressing the cyclic nucleotide gated channel alpha subunit (CNGA3).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AGuIX DB18189
biotech

AGuIX is an investigational brand product consisting of a polysiloxane matrix and gadolinium chelates. It is under development as a radiosensitizer to be used during radiation treatment of malignant glioma.

Kategori:
ElementsLanthanoid Series ElementsMetals +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2417550-70-8

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AI-128 DB05841
small molecule

AI-128 is the first human demonstration of sustained release drug administration in the lung. AI-128 consists of slowly dissolving microspheres designed to control where drug particles go in the lung and how quickly they release their drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AI-850 DB05842
small molecule

AI-850 is a Cremophor(R)-free formulation of paclitaxel, the active ingredient in Taxol(R), a product used to treat a variety of solid tumors.

Kategori:
CyclodecanesCycloparaffinsDiterpenes +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 3031-94-5

5-Aminoimidazole-4-carboxamide ribonucleotide (AICAR) is an intermediate in the generation of inosine monophosphate and analog of adenosine monophosphate (AMP) that is capable of stimulating AMP-dependent protein kinase (AMPK) activity. AICAR has been used cl…

Kategori:
Blood Glucose Lowering AgentsImidazolesNucleic Acids, Nucleotides, and Nucleosides +1
Target Protein:
Bifunctional purine biosynthesis protein ATIC
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ailanthus altissima pollen Approved DB10452
biotech

Ailanthus altissima pollen is the pollen of the Ailanthus altissima plant. Ailanthus altissima pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AIM-102 DB16176
small molecule | CAS: 551936-17-5

AIM-102 is under investigation in clinical trial NCT01501942 (Efficacy, Safety, Tolerability, Pharmacodynamics and Pharmacokinetics of Oral Administration of AIM-102 in Patients With Mild to Moderate Allergic Asthma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AIT-034 DB06106
small molecule | CAS: 138117-48-3

AIT-034 is a distinct chemical analog of hypoxanthine and pyrollidone that has been demonstrated in animal studies to enhance memory and to reverse memory deficits in severely impaired animals that do not respond to Neotrofin. AIT-034 does not induce the prod…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ajmaline Approved DB01426
small molecule | CAS: 4360-12-7

An alkaloid found in the root of Rauwolfia serpentina, among other plant sources. It is a class Ia antiarrhythmic agent that apparently acts by changing the shape and threshold of cardiac action potentials. Ajmaline produces potent sodium channel blocking eff…

Kategori:
Ajmaline and derivativesAlkaloidsAntiarrhythmic agents +16
Target Protein:
Sodium channel protein type 5 subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ajoene DB17735
small molecule | CAS: 92285-01-3

Deskripsi belum tersedia.

Kategori:
AnionsAnti-Infective AgentsAntifungal Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AK106-001616 DB16058
small molecule | CAS: 590416-75-4

AK106-001616 is under investigation in clinical trial NCT01285752 (A Study of AK106-001616 in Patients With Rheumatoid Arthritis (RA)).

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AK119 DB16423
biotech

AK119 is a humanized anti-CD73 monoclonal antibody being investigated in the clinical trial NCT04516564 (A Study of AK119 (Anti-CD73 Antibody), a Treatment for COVID-19, in Healthy Subjects).[L28315]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AKI-001 DB07266
small molecule | CAS: 925218-37-7

AKI-001 is an aurora kinase inhibitor.

Kategori:
Heterocyclic Compounds, Fused-RingProtein Kinase Inhibitors
Target Protein:
Aurora kinase A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aklavine DB19070
small molecule | CAS: 66676-88-8

Aklavine is under investigation in clinical trial NCT03026842 (Decitabine Versus Conventional Chemotherapy for Maintenance Therapy of Acute Myeloid Leukemia With T(8;21)).

Kategori:
Adjuvants, ImmunologicAminoglycoside AntibacterialsAnthracyclines +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AKN-028 DB12746
small molecule | CAS: 1175017-90-9

AKN-028 has been used in trials studying the treatment of Acute Myeloid Leukemia.

Target Protein:
Receptor-type tyrosine-protein kinase FLT3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AKV-9 DB18061
small molecule | CAS: 1307262-15-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AL-01211 DB17654
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AL-034 DB17471
small molecule

AL-034 (TQ-A3334) is an oral toll-like receptor 7 agonist developed for the treatment of chronic hepatitis B (CHB) viral infection.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Carbonic anhydrase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Carbonic anhydrase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Ala-geninthiocin is a novel thiopeptide antibacterial compound derived from marine _Streptomyces_ species.[A192840] It has exhibited potent _in vitro_ activity against gram-positive bacteria including _Staphylococcus aureus_, _Bacillus subtilis_, _Mycobacteri…

Kategori:
Anti-Bacterial Agents
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alagebrium DB12497
small molecule | CAS: 393121-34-1

Alagebrium has been investigated for the treatment and prevention of Aging, Heart Failure, Physical Activity, Diabetic Nephropathy, and Cardiovascular Disease, among others.

Kategori:
Sulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alamifovir DB06368
small molecule | CAS: 193681-12-8

Alamifovir is an antiviral agent specific for HBV.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alanine DB00160
small molecule | CAS: 56-41-7

Alanine is a non-essential amino acid that occurs in high levels in its free state in plasma. It is produced from pyruvate by transamination. It is involved in sugar and acid metabolism, increases immunity, and provides energy for muscle tissue, brain, and th…

Kategori:
AlanineAmino AcidsAmino Acids, Peptides, and Proteins +3
Target Protein:
4-aminobutyrate aminotransferase, mitochondrialAlanine--glyoxylate aminotransferaseAlanine aminotransferase 1 +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alanosine DB05540
small molecule | CAS: 5854-93-3

An amino acid analogue and antibiotic derived from the bacterium Streptomyces alanosinicus with antimetabolite and potential antineoplastic activities.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAntibiotics, Antineoplastic +4
Target Protein:
Aspartate carbamoyltransferase catalytic subunitAdenylosuccinate synthetase isozyme 2Adenylosuccinate synthetase isozyme 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 39537-23-0

Alanyl Glutamine is under investigation in clinical trial NCT00338221 (Clinical Trial of Alanyl-Glutamine or Glycine in Children With Persistent Diarrhea or Malnutrition).

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsBlood and Blood Forming Organs +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alaproclate DB13233
small molecule | CAS: 60719-82-6

Alaproclate was developed as one of the first selective serotonin reuptake inhibitor (SSRI) antidepressants by Astra AB (now AstraZeneca) in the 1970s. Development was discontinued due to concerns over hepatotoxicity observed in animal studies. Alaproclate ha…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAntidepressive Agents +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alatrofloxacin Approved DB09335
small molecule | CAS: 146961-76-4

Alatrofloxacin is a fluoroquinolone antibiotic developed by Pfizer, delivered as a mesylate salt. It was withdrawn from the U.S. market in 2001.

Kategori:
4-QuinolonesAnti-Infective AgentsEnzyme Inhibitors +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Albaconazole DB12073
small molecule | CAS: 187949-02-6

Albaconazole has been used in trials studying the basic science of Onychomycosis.

Kategori:
Anti-Infective AgentsAntifungal AgentsAzole Antifungals +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Albendazole Approved DB00518
small molecule | CAS: 54965-21-8

A benzimidazole broad-spectrum anthelmintic structurally related to mebendazole that is effective against many diseases. (From Martindale, The Extra Pharmacopoeia, 30th ed, p38)

Kategori:
Acids, AcyclicAnthelminticsAnti-Infective Agents +23
Target Protein:
Tubulin beta-2 chainTubulin alpha-1A chainTubulin beta-4B chain +1
Waktu ParuhTerminal eliminatio…
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 2901–2950 dari 16749
Sebelumnya Halaman 59 / 335 Berikutnya