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11793

Total database: 17430
Struktur (SMILES)
8607 (73.0%)
Target
6418 (54.4%)
Genomik
102 (0.9%)
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11793 (100.0%)

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Hasil Pencarian (11793)

Halaman 59 / 236
BPI-3016 DB15158
biotech

BPI-3016 is under investigation in clinical trial NCT03188848 (Dose Escalating Study of BPI-3016 in Healthy Subjects).

Kategori:
Amino Acids, Peptides, and ProteinsGastrointestinal HormonesGlucagon-Like Peptides +4
Waktu Paruh-
Vol. Distribusi-
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Genetik -
BPR-0L075 DB17155
small molecule | CAS: 613679-11-1

Deskripsi belum tersedia.

Waktu Paruh-
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BQ-123 DB12054
small molecule | CAS: 136553-81-6

BQ-123 has been investigated for the basic science and treatment of Coronary Artery Disease, Aorto-coronary Bypass Grafting, and ST-Elevation Myocardial Infarction.

Kategori:
Amino Acids, Peptides, and ProteinsAntihypertensive AgentsCardiovascular Agents +2
Target Protein:
Endothelin-1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
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BQ-788 DB17984
small molecule | CAS: 156161-89-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntihypertensive AgentsCardiovascular Agents +3
Target Protein:
Endothelin receptor type B
Waktu Paruh-
Vol. Distribusi-
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BR-007 DB18408
small molecule | CAS: 2409546-40-1

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

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Bradanicline DB06090
small molecule | CAS: 639489-84-2

Bradanicline, a novel small molecule that modulates the activity of the neuronal nicotinic receptor (NNR) subtype known as alpha7(?7). Bradanicline belongs to a new class of drugs for the treatment of central nervous system diseases and disorders.

Kategori:
Heterocyclic Compounds, Fused-RingReceptors, Nicotinic
Target Protein:
Neuronal acetylcholine receptor subunit alpha-7
Waktu Paruh-
Vol. Distribusi-
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Bradykinin DB12126
small molecule | CAS: 58-82-2

Bradykinin has been investigated for the basic science and treatment of Hypertension and Diabetes Type 2.

Kategori:
Amino Acids, Peptides, and ProteinsAutacoidsBiological Factors +11
Target Protein:
B2 bradykinin receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Branaplam DB14918
small molecule | CAS: 1562338-42-4

Branaplam is under investigation in clinical trial NCT02268552 (An Open Label Study of LMI070 (Branaplam) in Type 1 Spinal Muscular Atrophy (SMA)).

Target Protein:
Survival motor neuron protein
Waktu Paruh-
Vol. Distribusi-
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Branebrutinib DB15347
small molecule | CAS: 1912445-55-6

Branebrutinib is under investigation in clinical trial NCT02705989 (Safety, Tolerability and Relative Bioavailability Study of BMS-986195 in Healthy Subjects).

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingProtein Kinase Inhibitors
Target Protein:
Tyrosine-protein kinase BTK
Waktu Paruh-
Vol. Distribusi-
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Brasofensine DB04857
small molecule | CAS: 171655-91-7

Brasofensine is an orally administered dopamine reuptake inhibitor being developed for the treatment of Parkinson's Disease. Phase I/II trials for brasofensine have been completed in the U.K. In November 2001, NeuroSearch confirmed that the drug's development…

Kategori:
AminesHeterocyclic Compounds, Fused-RingHydroxylamines
Target Protein:
Sodium-dependent serotonin transporterD(2) dopamine receptor
Waktu ParuhPlasma terminal eli…
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Brazikumab DB16115
biotech | CAS: 1610353-18-8

Brazikumab is under investigation in clinical trial NCT03759288 (An Active and Placebo-controlled Study of Brazikumab in Participants With Moderately to Severely Active Crohn's Disease).

Waktu Paruh-
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Brecanavir DB04887
small molecule | CAS: 313682-08-5

Brecanavir (VX-385) an orally active aspartic protease inhibitor (PI), under investigation by Vertex and GlaxoSmithKline for the treatment of HIV. In July 2006, Vertex indicated that it expected GSK to initiate phase III trials of the drug in 2007. In Decembe…

Kategori:
Acids, AcyclicDioxolesHeterocyclic Compounds, Fused-Ring
Target Protein:
Gag-Pol polyproteinPol polyprotein
Waktu Paruh-
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Brefeldin A DB07348
small molecule | CAS: 20350-15-6

A metabolite from Penicillium brefeldianum that exhibits a wide range of antibiotic activity.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsCytochrome P-450 CYP3A Inhibitors +9
Target Protein:
Cytohesin-2ADP-ribosylation factor 1
Waktu Paruh-
Vol. Distribusi-
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Bremelanotide Approved DB11653
biotech | CAS: 189691-06-3

Bremelanotide is a 7 amino acid peptide used to treat hypoactive sexual desire disorder in premenopausal women.[L9635] Bremelanotide does not interact with alcohol.[A179686] The mechanism by which bremelanotide's action on receptors translates to a clinical e…

Kategori:
Amino Acids, Peptides, and ProteinsGenito Urinary System and Sex HormonesHormones +16
Target Protein:
Melanocyte-stimulating hormone receptorMelanocortin receptor 4Melanocortin receptor 3 +2
Waktu ParuhThe half life of br…
Vol. DistribusiThe mean volume of …
KlirensThe mean clearance …
Genetik -
Bremzalerbart DB19417
biotech | CAS: 2456307-07-4

Bremzalerbart is under investigation in clinical trial NCT06602739 (A Study to Demonstrate the Effect of REGN5713-5715 on Reducing Ocular Allergy Signs and Symptoms in Adult Participants With Birch Pollen Allergy).

Waktu Paruh-
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BREN-02 DB18264
biotech

BREN-02 is a recombinant human homeoprotein Engrailed 1 (rhEN1).

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Brenetafusp DB19441
biotech | CAS: 2736407-54-6

Brenetafusp is under investigation in clinical trial NCT04262466 (Safety and Efficacy of IMC-F106C as a Single Agent and in Combination With Checkpoint Inhibitors).

Waktu Paruh-
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Brensocatib DB15638
small molecule | CAS: 1802148-05-5

Brensocatib is under investigation in clinical trial NCT03218917 (Assessment of INS1007 in Subjects With Non-cystic Fibrosis Bronchiectasis).

Kategori:
AzepinesHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
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Brequinar DB03523
small molecule | CAS: 96187-53-0

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsBenzene DerivativesEnzyme Inhibitors +5
Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Bretylium Approved DB01158
small molecule | CAS: 59-41-6

Bretylium blocks the release of noradrenaline from the peripheral sympathetic nervous system, and is used in emergency medicine, cardiology, and other specialties for the acute management of ventricular tachycardia and ventricular fibrillation. The primary mo…

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAmines +13
Target Protein:
Sodium/potassium-transporting ATPase subunit alpha-1Beta-1 adrenergic receptor
Waktu ParuhThe terminal half-l…
Vol. Distribusi-
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Brevenal DB17865
small molecule | CAS: 776331-34-1

Deskripsi belum tersedia.

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Brexanolone Approved DB11859
small molecule | CAS: 516-54-1

As of March 2019, brexanolone - developed and made available commercially by Sage Therapeutics Inc. as the brand name product Zulresso - is the first drug to have ever been approved by the US FDA specifically for the treatment of postpartum depression (PPD) i…

Kategori:
AnestheticsAnticonvulsantsAntidepressive Agents +28
Target Protein:
Gamma-aminobutyric acid receptor subunit deltaGamma-aminobutyric acid receptor subunit gamma-3GABA(A) Receptor +3
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe volume of distr…
KlirensThe total plasma cl…
Genetik -
Brexpiprazole Approved DB09128
small molecule | CAS: 913611-97-9

Brexpiprazole is an atypical antipsychotic and a novel D2 dopamine and serotonin 1A partial agonist called serotonin-dopamine activity modulator (SDAM). It has a high affinity for serotonin, dopamine and alpha (?)-adrenergic receptors.[L46417] Although it is …

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +30
Target Protein:
5-hydroxytryptamine receptor 1AD(2) dopamine receptorD(3) dopamine receptor +9
Waktu ParuhAfter multiple once…
Vol. DistribusiThe volume of distr…
KlirensApparent oral clear…
Genetik -
Brexucabtagene autoleucel Approved DB15699
biotech

Mantle cell lymphoma is a heterogeneous sub-category of non-Hodgkin's lymphoma that can be classified as either an aggressive nodal or an indolent leukemic non-nodal variant. Despite the introduction of Bruton's tyrosine kinase (BTK) inhibitors such as [ibrut…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsAntineoplastic Agents, Immunological +16
Target Protein:
B-lymphocyte antigen CD19
Waktu Paruh-
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Briakinumab DB05459
biotech | CAS: 339308-60-0

Briakinumab is a human anti-IL-12 monoclonal antibody being developed for the treatment of a number of T-cell driven autoimmune diseases. It targets and neutralize interleukin-12 and interleukin-23, two proteins associated with inflammation, such as pro-infla…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Target Protein:
Interleukin-12 subunit betaInterleukin-23 subunit alpha
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Briciclib DB12004
small molecule | CAS: 865783-99-9

Briciclib has been used in trials studying the treatment of Lymphoma, Neoplasms, Advanced Solid Tumor, and Acute Lymphocytic Leukemia.

Target Protein:
G1/S-specific cyclin-D1
Waktu Paruh-
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Brigatinib Approved DB12267
small molecule | CAS: 1197953-54-0

Brigatinib, originally named AP26113, is a reversible dual inhibitor of anaplastic lymphoma kinase (ALK) and epidermal growth factor receptor (EGFR). It presents selectivity against the mutant forms of EGFR compared to the wild-type.[A31311] It also exhibits …

Kategori:
Anaplastic lymphoma kinase (ALK) inhibitorsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +18
Target Protein:
ALK tyrosine kinase receptorEpidermal growth factor receptorTyrosine-protein kinase ABL1 +6
Waktu ParuhThe half-life of br…
Vol. DistribusiThe apparent volume…
KlirensAfter oral administ…
Genetik -
Brigimadlin DB18578
small molecule | CAS: 2095116-40-6

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
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Brilaroxazine DB09226
small molecule | CAS: 1239729-06-6

Brilaroxazine (RP5063) is an investigational atypical antipsychotic which is under development by Reviva Pharmaceuticals for the treatment of schizophrenia and schizoaffective disorder. Reviva Pharmaceuticals also intends to investigate RP5063 for the treatme…

Kategori:
Antidepressive AgentsAntipsychotic AgentsAntipsychotic Agents (Second Generation [Atypical]) +7
Waktu Paruh-
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Brilliant blue G Approved DB15594
small molecule | CAS: 6104-58-1

Brilliant Blue G is used in an ophthalmic solution for staining the internal limiting membrane (ILM) of the eye during ophthalmic procedures.[A188841,A188844] This membrane is thin and translucent, making it difficult to identify during eye surgeries that req…

Kategori:
AminesAniline CompoundsCompounds used in a research, industrial, or household setting +3
Target Protein:
Internal limiting membrane (ILM)
Waktu Paruh-
Vol. DistribusiThis drug is admini…
Klirens-
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Brimonidine Approved DB00484
small molecule | CAS: 59803-98-4

Brimonidine is an alpha-adrenergic agonist and 2-imidazoline derivative that was first introduced in 1996.[A178951] It is considered to be a third generation alpha-2 aadrenergic receptor agonist, since it displays preferential binding at alpha-2 adrenoceptors…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +14
Target Protein:
Alpha-2A adrenergic receptorAlpha-2B adrenergic receptorAlpha-2C adrenergic receptor
Waktu ParuhFollowing ocular ad…
Vol. DistribusiThe volume of distr…
KlirensThe apparent cleara…
Genetik -
Brinzolamide Approved DB01194
small molecule | CAS: 138890-62-7

Brinzolamide is a highly specific, non-competitive, reversible carbonic anhydrase II (CA-II) inhibitor indicated to reduce ocular pressure in patients with ocular hypertension or open-angle glaucoma.[L35310] Although the exact pathophysiology of glaucoma is s…

Kategori:
AmidesAntiglaucoma Preparations and MioticsCarbonic Anhydrase Inhibitors +17
Target Protein:
Carbonic anhydrase 2Carbonic anhydrase 1Carbonic anhydrase 4 +2
Waktu ParuhDue to its affinity…
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Briquilimab DB18136
biotech | CAS: 2574591-89-0

Briquilimab is a humanized aglycosylated IgG1 kappa monoclonal antibody targeting CD117 (cKit).

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Brivanib DB11958
small molecule | CAS: 649735-46-6

Brivanib is under investigation for the treatment of HepatoCellular Carcinoma. Brivanib has been investigated for the treatment of Solid Tumors, Hepato Cellular Carcinoma (HCC), and Metastatic Colorectal Cancer (MCRC).

Kategori:
Amino AcidsAmino Acids, Peptides, and Proteins
Target Protein:
Vascular endothelial growth factor receptor 2
Waktu Paruh-
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small molecule | CAS: 649735-63-7

Brivanib alaninate has been investigated for the treatment of Colorectal Cancer.

Kategori:
Amino AcidsAmino Acids, Peptides, and Proteins
Target Protein:
Fibroblast growth factor receptor 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brivaracetam Approved DB05541
small molecule | CAS: 357336-20-0

Brivaracetam is a racetam derivative of levetiracetam used in the treatment of partial-onset seizures. Brivaracetam binds SV2A with 20 times higher affinity than levetiracetam [A19184]. It is available under the brand name Briviact made by UCB. Briviact recei…

Kategori:
AnticonvulsantsCentral Nervous System AgentsCentral Nervous System Depressants +11
Target Protein:
Synaptic vesicle glycoprotein 2ASodium channel protein
Waktu Paruh7-8h [A19180].
Vol. Distribusi0.5L/kg [FDA Label].
KlirensCL/F of 0.7-1.07 mL…
Genetik -
Brivoligide DB16116
biotech | CAS: 1803075-42-4

Brivoligide is under investigation in clinical trial NCT04104919 (Study to Evaluate a Preop Dose of Brivoligide Injection for Pain After Mastectomy in Patients With High PCS Scores).

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Brivudine Approved DB03312
small molecule | CAS: 69304-47-8

Brivudine is used in the treatment of herpes zoster. Although not approved in the U.S. or Canada, it is approved in several European countries.

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +9
Target Protein:
Thymidine kinase 2, mitochondrialThymidine kinase, cytosolicDNA polymerase +1
Waktu Paruh-
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small molecule | CAS: 80860-82-8

Deskripsi belum tersedia.

Target Protein:
Thymidine kinase
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BRM-421 DB18364
biotech

Deskripsi belum tersedia.

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Brodalumab Approved DB11776
biotech | CAS: 1174395-19-7

Brodalumab has been used in trials studying the treatment of Asthma, Psoriasis, Crohn's Disease, Psoriatic Arthritis, and Rheumatoid Arthritis. Brodalumab was FDA approved in February, 2017 as Siliq for the treatment of moderate-to-severe plaque psoriasis.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +13
Target Protein:
Interleukin-17 receptor A
Waktu Paruh-
Vol. Distribusi4.62 L.
Klirens0.223 L/day.
Genetik -
Brodimoprim DB13795
small molecule | CAS: 56518-41-3

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntibacterials for Systemic UseAntiinfectives for Systemic Use +5
Waktu Paruh-
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small molecule

Brodimoprim-4,6-dicarboxylate is a solid. This compound belongs to the anisoles. These are organic compounds contaiing a methoxybenzene or a derivative thereof. This medication is known to target the protein dihydrofolate reductase.

Target Protein:
Peptide deformylase, mitochondrialDihydrofolate reductase
Waktu Paruh-
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Brofaromine DB13876
small molecule | CAS: 63638-91-5

Deskripsi belum tersedia.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsEnzyme Inhibitors +3
Target Protein:
Amine oxidase [flavin-containing] A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brogidirsen DB18884
biotech | CAS: 2409088-11-3

Brogidirsen is under investigation in clinical trial NCT05996003 (NS-089/NCNP-02-201 in Boys With Duchenne Muscular Dystrophy (DMD)).

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Brolucizumab Approved DB14864
biotech | CAS: 1531589-13-5

Brolucizumab, also known as RTH258 or ESBA1008,[A187211] is a monoclonal antibody indicated to treat neovascular age related macular degeneration.[L9089] Brolucizumab was granted FDA approval in October 2019.[L9089]

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAntibodies +14
Target Protein:
Vascular endothelial growth factor A, long form
Waktu ParuhThe systemic half l…
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik -
Bromamphenicol DB07492
small molecule | CAS: 16803-75-1

Deskripsi belum tersedia.

Kategori:
AlcoholsBenzene DerivativesGlycols +3
Target Protein:
Dr hemagglutinin structural subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bromfenac Approved DB00963
small molecule | CAS: 91714-94-2

Bromfenac is a nonsteroidal anti-inflammatory drug (NSAID) for ophthalmic use. Ophthalmic NSAIDs are becoming a cornerstone for the management of ocular pain and inflammation. Their well-characterized anti-inflammatory activity, analgesic property, and establ…

Kategori:
Agents causing hyperkalemiaAnalgesicsAnalgesics, Non-Narcotic +16
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Bromhexine Approved DB09019
small molecule | CAS: 3572-43-8

Bromhexine is mucolytic agent used for a variety of respiratory conditions associated with increased mucus secretion. It is derived from the Adhatoda vasica plant and aids in the clearance of excess mucus, improving breathing and reducing cough. It was introd…

Kategori:
AminesAniline CompoundsCough and Cold Preparations +5
Target Protein:
Transmembrane protease serine 2Angiotensin-converting enzyme 2
Waktu ParuhFollowing single or…
Vol. DistribusiAfter intravenous a…
KlirensThe clearance of br…
Genetik -
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