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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
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12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 59 / 252
Benoxaprofen Approved DB04812
small molecule | CAS: 51234-28-7

The use of benoxaprofen, formerly marketed as Oraflex tablets, was associated with fatal cholestatic jaundice among other serious adverse reactions. The holder of the approved application voluntarily withdrew Oraflex tablets from the market on August 5, 1982.

Kategori:
Acids, AcyclicAgents causing hyperkalemiaAgents that produce hypertension +18
Target Protein:
Acetyl-CoA acetyltransferase, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benproperine DB13309
small molecule | CAS: 2156-27-6

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesCough and Cold Preparations
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benralizumab Approved DB12023
biotech | CAS: 1044511-01-4

Benralizumab is a humanized recombinant monoclonal antibody of the isotype IgG1k immunoglobulin that specifically binds to the alpha chain of the interleukin 5 receptor (IL-5R) expressed on eosinophils and basophils.[A31294] It inhibits the binding of IL-5 as…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Asthmatic AgentsAntibodies +13
Target Protein:
Interleukin-5 receptor subunit alphaLow affinity immunoglobulin gamma Fc region receptor III-A
Waktu ParuhThe half-life of Be…
Vol. DistribusiPharmacokinetic rep…
KlirensFor a subject weigh…
Genetik -
Benserazide Approved DB12783
small molecule | CAS: 322-35-0

When levodopa is used by itself as a therapy for treating Parkinson's disease, its ubiquitous metabolism into dopamine is responsible for a resultant increase in the levels of circulating dopamine in the blood and to various extracerebral tissues. This can re…

Kategori:
Anti-Dyskinesia AgentsAnti-Parkinson DrugsAromatic L-amino Acid Decarboxylase Inhibitors +6
Target Protein:
Aromatic-L-amino-acid decarboxylase
Waktu ParuhThe half-life of be…
Vol. DistribusiReadily accessible …
KlirensReadily accessible …
Genetik -
Bentamapimod DB16851
small molecule | CAS: 848344-36-5

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingThiazoles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bentiromide DB00522
small molecule | CAS: 37106-97-1

Bentiromide is a dipeptide that is used in the bentiromide test, which is a screening test for evaluating pancreatic exocrine function and monitoring the adequacy of supplemental pancreatic therapy. It is typically administered orally. Cases of headache and g…

Kategori:
Acids, CarbocyclicAminobenzoatesBenzene Derivatives +7
Target Protein:
Serine protease hepsin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bentoquatam Approved DB00516
small molecule | CAS: 1340-69-8

Bentoquatam is a topical medication intended to act as a shield against exposure to the irritating substance urushiol, found in plants such as poison ivy or poison oak. Bentoquatam contains bentonite, a clay, and is only effective as long as the film is visib…

Kategori:
Aluminium CompoundsAluminum SilicatesDermatologicals +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bentracimab DB16659
biotech | CAS: 2260568-31-6

Bentracimab is under investigation in clinical trial NCT04286438 (Bentracimab (PB2452) in Ticagrelor-treated Patients With Uncontrolled Major or Life-threatening Bleeding or Requiring Urgent Surgery or Invasive Procedure).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Neutralizing +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benzalkonium Approved DB11105
small molecule

Benzalkonium is a quaternary ammonium compound used as a biocide, a cationic surfactant, and as a phase transfer agent [FDA Label]. Benzalkonium is more commonly contained in consumer products in its salt form, benzalkonium chloride [FDA Label]. This salt is …

Kategori:
AminesAnti-Infective AgentsAnti-Infective Agents, Local +18
Waktu Paruh-
Vol. DistribusiWhen applied as a t…
Klirens-
Genetik -
Benzatropine Approved DB00245
small molecule | CAS: 86-13-5

Benztropine, with the chemical formula 3alpha-diphenylmethoxytropane, is a tropane-based dopamine inhibitor used for the symptomatic treatment of Parkinson's disease. It is a combination molecule between a tropane ring, similar to cocaine, and a diphenyl ethe…

Kategori:
Agents producing tachycardiaAlkaloidsAnti-Dyskinesia Agents +23
Target Protein:
Muscarinic acetylcholine receptor M1Sodium-dependent dopamine transporterHistamine H1 receptor +2
Waktu ParuhThe elimination hal…
Vol. DistribusiBenztropine is expe…
KlirensExtensive pharmacod…
Genetik -
Benzbromarone DB12319
small molecule | CAS: 3562-84-3

Benzbromarone has been used in trials studying the basic science and treatment of Heart Failure, Hyperuricemia, Chronic Kidney Disease, Abnormal Renal Function, and Gout and Asymptomatic Hyperuricemia.

Kategori:
Antigout PreparationsAntirheumatic AgentsBenzofurans +12
Target Protein:
Anoctamin-1Solute carrier family 22 member 12Multidrug resistance-associated protein 1 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 517-60-2

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicBenzene Derivatives
Target Protein:
Phosphoglycerate mutase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benzethidine DB01518
small molecule | CAS: 3691-78-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benzethonium Approved DB11125
small molecule | CAS: 10172-60-8

Benzethonium is a synthetic quaternary ammonium salt with surfactant, antiseptic, and broad spectrum antimicrobial properties. Its salt form, benzethonium chloride, is primarily used as a skin disinfectant at concentrations of 0.1-0.2 %, which are safe and ef…

Kategori:
AminesAnti-Infective AgentsAnti-Infective Agents, Local +7
Waktu ParuhPharmacokinetic stu…
Vol. DistribusiPharmacokinetic stu…
KlirensPharmacokinetic stu…
Genetik -
Benzgalantamine Approved DB19353
small molecule | CAS: 224169-27-1

Benzgalantamine is a prodrug of [galantamine]. Gastrointestinal adverse effects are the most frequently reported side effects in patients undergoing treatment with cholinesterase inhibitors, including galantamine, and are often a reason for treatment disconti…

Kategori:
AlkaloidsAlzheimer Disease, drug therapyAmaryllidaceae Alkaloids +11
Target Protein:
AcetylcholinesteraseCholinesteraseNeuronal acetylcholine receptor subunit alpha-7 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benzhydrocodone Approved DB15465
small molecule | CAS: 1259440-61-3

Benzhydrocodone is a benzylic prodrug of hydrocodone.[L4894] It was developed in an effort to reduce parenteral bioavailability of the active metabolite as a deterrent to abuse.[A182177] Benzhydrocodone is indicated for use in the short-term management of pai…

Kategori:
Opioids
Target Protein:
Mu-type opioid receptor
Waktu ParuhThe hydrocodone met…
Vol. DistribusiThe hydrocodone met…
KlirensThe apparent cleara…
Genetik -
small molecule | CAS: 495-18-1

Deskripsi belum tersedia.

Kategori:
AminesBenzoatesHydroxy Acids +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benzilone DB13369
small molecule | CAS: 16175-92-1

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAnticholinergic Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benzimate DB05170
small molecule

Benzimate is the lead compound selected from a series of compounds known as benzimidazoles. The anti-cancer and anti-viral activity of the benzimidazoles was originally investigated by the Proctor & Gamble Company beginning in the 1990's. It is currently unde…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benzimidazole DB02962
small molecule | CAS: 51-17-2

Deskripsi belum tersedia.

Kategori:
AnthelminticsAnti-Infective AgentsAntiparasitic Agents +1
Target Protein:
Dual specificity tyrosine-phosphorylation-regulated kinase 1ANicotinate-nucleotide--dimethylbenzimidazole phosphoribosyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benziodarone Approved DB13277
small molecule | CAS: 68-90-6

Benziodarone is a uricostatic and a uricosuric agent which is sold also under the name Amplivex-Labaz. It is used in the treatment of gout [A175630]. It was withdrawn from France markets and British markets due to its effects causing Jaundice in patients [T48…

Kategori:
Antigout PreparationsAntirheumatic AgentsCardiac Therapy +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benznidazole Approved DB11989
small molecule | CAS: 22994-85-0

Benznidazole was granted accelerated approval for the treatment of Chagas disease in children 2-12 years of age by the FDA on August 29, 2017.[L939] It is the first treatment made available in the United States for Chagas disease.

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAnti-Infective AgentsAntiparasitic Agents +12
Waktu ParuhThe half life of el…
Vol. DistribusiThe apparent volume…
KlirensThe apparent oral c…
Genetik -
Benzocaine Approved DB01086
small molecule | CAS: 94-09-7

Benzocaine is an ester local anesthetic that acts by preventing transmission of impulses along nerve fibers and at nerve endings.[A231219] It is commonly used for local anesthesia in many over the counter products.[L32454,L32459,L32464] Benzocaine was first u…

Kategori:
Acids, CarbocyclicAgents for Treatment of Hemorrhoids and Anal Fissures for Topical UseAminobenzoates +29
Target Protein:
Sodium channel protein type 10 subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benzododecinium DB13282
small molecule | CAS: 10328-35-5

Benzododecinium is used as an antiseptic/disinfectant compound. It has been marketed as a tincture for antiseptic product for wounds in the Czech Republic.

Kategori:
AminesAnti-Infective AgentsAnti-Infective Agents, Local +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benzoic acid Approved DB03793
small molecule | CAS: 65-85-0

A fungistatic compound that is widely used as a food preservative. It is conjugated to GLYCINE in the liver and excreted as hippuric acid. As the sodium salt form, sodium benzoate is used as a treatment for urea cycle disorders due to its ability to bind amin…

Kategori:
Acids, CarbocyclicAlimentary Tract and MetabolismAmmonium Ion Binding Activity +18
Target Protein:
Ras-related protein Rab-9ASolute carrier family 15 member 1Cocaine esterase +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benzoin Approved DB14020
small molecule | CAS: 119-53-9

Benzoin is a white crystalline compound prepared by condensation of benzaldehyde in potassium cyanide, and is used in organic syntheses. This should not be confused with benzoin gum from STYRAX (see [DB11222]). Benzoin is an FDA-approved colour additive used …

Kategori:
AcetophenonesAnti-Infective Agents, LocalKetones
Target Protein:
Liver carboxylesterase 1
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Benzoin resin Approved DB11222
biotech | CAS: 9000-05-9

Benzoin resin is a balsamic resin obtained from the bark of several species of trees in the genus _Styrax_. There are two common kinds of benzoin, benzoin Siam and benzoin Sumatra, that are obtained from different species of the _Styrax_ tree. While benzoin r…

Kategori:
AngiospermsAnti-Infective Agents, LocalBiological Products +11
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Benzonatate Approved DB00868
small molecule | CAS: 104-31-4

Benzonatate is an oral antitussive drug used in the relief and suppression of cough in patients older than ten years of age.[A5790] Currently, benzonatate is the only non-narcotic antitussive available as a prescription drug.[A189519] It works to reduce the a…

Kategori:
AlkanesAminesAntitussive Agents +8
Target Protein:
Sodium channel protein type 5 subunit alpha
Waktu ParuhThe half life of be…
Vol. DistribusiThere is limited in…
KlirensThere is limited in…
Genetik -
Benzoxonium DB13565
small molecule | CAS: 23884-64-2

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAminesAntiinfectives and Antiseptics for Local Oral Treatment +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benzoyl peroxide Approved DB09096
small molecule | CAS: 94-36-0

Benzoyl peroxide is a commonly used drug in topical treatments for acne.[L33249,L33264,L33269,L33299,L33314] It has been formulated as products with either a single active ingredient,[L33249,L33299] or with [erythromycin],[L33264] [clindamycin],[L33269] or [a…

Kategori:
Acids, CarbocyclicAnti-Acne PreparationsAnti-Acne Preparations for Topical Use +5
Target Protein:
CatalaseGlutathione peroxidaseAntizyme inhibitor 2 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Cathepsin F
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benzoylecgonine DB01515
small molecule | CAS: 519-09-5

Benzoylecgonine is the major metabolite of cocaine. It is formed by hydrolysis of cocaine in the liver, catalysed by carboxylesterases. It is excreted in the urine of cocaine users after processing in the liver. It is the main pharmaceutical ingredient in the…

Kategori:
AlkaloidsAza CompoundsAzabicyclo Compounds +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 18481-26-0

Deskripsi belum tersedia.

Kategori:
PyrimidinesSulfur CompoundsThiazoles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benzoylpas DB19382
small molecule | CAS: 13898-58-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benzphetamine Approved DB00865
small molecule | CAS: 156-08-1

A sympathomimetic agent with properties similar to dextroamphetamine. It is used in the treatment of obesity. (From Martindale, The Extra Pharmacopoeia, 30th ed, p1222)

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +28
Target Protein:
Synaptic vesicular amine transporterAlpha-2A adrenergic receptorAlpha-1A adrenergic receptor +1
Waktu Paruh16 to 31 hours
Vol. Distribusi-
Klirens-
Genetik -
Benzthiazide Approved DB00562
small molecule | CAS: 91-33-8

Benzthiazide is used to treat hypertension and edema. Like other thiazides, benzthiazide promotes water loss from the body (diuretics). They inhibit Na+/Cl- reabsorption from the distal convoluted tubules in the kidneys. Thiazides also cause loss of potassium…

Kategori:
DiureticsGenito Urinary System and Sex HormonesGynecological Antiinfectives and Antiseptics +8
Target Protein:
Solute carrier family 12 member 3Carbonic anhydraseCarbonic anhydrase 2 +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Collagenase 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benzyl alcohol Approved DB06770
small molecule | CAS: 100-51-6

Deskripsi belum tersedia.

Kategori:
AlcoholsAnestheticsAnesthetics, Local +18
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benzyl benzoate Approved DB00676
small molecule | CAS: 120-51-4

Benzyl benzoate is one of the older preparations used to treat scabies. Scabies is a skin infection caused by the mite sarcoptes scabiei. It is characterised by severe itching (particularly at night), red spots, and may lead to a secondary infection. Benzyl b…

Kategori:
AcaricidesAcids, CarbocyclicAgrochemicals +8
Target Protein:
Hormone-sensitive lipase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benzyl formate DB04569
small molecule | CAS: 104-57-4

Deskripsi belum tersedia.

Kategori:
Acids, Acyclic
Target Protein:
Thermolysin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Cathepsin FCruzipain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 94-44-0

Deskripsi belum tersedia.

Kategori:
Pyridines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benzylfentanyl DB09182
small molecule | CAS: 1474-02-8

Benzylfentanyl (R-4129) is a fentanyl analog opioid that was on the list of Schedule I drugs in America in 1985 due to its structural similarity to fentanyl. In 2010 it was removed from the list after it was found to have minimal opioid activity. Benzylfentan…

Kategori:
Piperidines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benzylmorphine DB01573
small molecule | CAS: 14297-87-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benzylpenicillin Approved DB01053
small molecule | CAS: 61-33-6

Benzylpenicillin (Penicillin G) is narrow spectrum antibiotic used to treat infections caused by susceptible bacteria. It is a natural penicillin antibiotic that is administered intravenously or intramuscularly due to poor oral absorption. Penicillin G may al…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +18
Target Protein:
Peptidoglycan synthase FtsIPenicillin-binding protein 1APenicillin-binding protein 1B +5
Waktu ParuhIn adults with norm…
Vol. Distribusi0.53–0.67 L/kg in a…
Klirens560ml/min in health…
Genetik -
Benzylpenicilloyl polylysine Approved DB00895
small molecule | CAS: 31855-75-1

Benzylpenicilloyl polylysine is used as a skin-testing reagent to detect immunoglobulin E antibodies in people with a history of penicillin allergy. The quantitation of in vitro IgE antibodies to the benzylpenicilloyl determinant is a useful tool for evaluati…

Kategori:
AcetamidesAmidesAnti-Bacterial Agents +9
Target Protein:
High affinity immunoglobulin epsilon receptor subunit gammaHigh affinity immunoglobulin epsilon receptor subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 6336-50-1

Deskripsi belum tersedia.

Kategori:
Antithyroid agentsPyrimidinesPyrimidinones +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bepotastine Approved DB04890
small molecule | CAS: 125602-71-3

Bepotastine is a non-sedating, selective antagonist of the histamine 1 (H1) receptor. Bepotastine was approved in Japan for use in the treatment of allergic rhinitis and uriticaria/puritus in July 2000 and January 2002, respectively, and is marketed by Tanabe…

Kategori:
Anti-Allergic AgentsDrugs that are Mainly Renally ExcretedHistamine Antagonists +2
Target Protein:
Histamine H1 receptor
Waktu ParuhElimination half li…
Vol. Distribusi-
Klirens-
Genetik -
Bepranemab DB17945
biotech | CAS: 2244960-75-4

Bepranemab is a recombinant humanized Igg4P monoclonal antibody directed against human Tau.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bepridil Approved DB01244
small molecule | CAS: 64706-54-3

A long-acting, non selective, calcium channel blocker with significant anti-anginal activity. The drug produces significant coronary vasodilation and modest peripheral effects. It has antihypertensive and selective anti-arrhythmia activities and acts as a cal…

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsAntihypertensive Agents +20
Target Protein:
Voltage-dependent P/Q-type calcium channel subunit alpha-1AVoltage-dependent T-type calcium channel subunit alpha-1HVoltage-dependent calcium channel subunit alpha-2/delta-2 +7
Waktu Paruh24-50 hours
Vol. Distribusi-
Klirens-
Genetik -
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