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14494

Total database: 17430
Struktur (SMILES)
9687 (66.8%)
Target
7525 (51.9%)
Genomik
112 (0.8%)
Referensi
14494 (100.0%)

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Hasil Pencarian (14494)

Halaman 58 / 290
AZ-3102 DB18502
small molecule

AZ-3102 is a Biphenyl-substituted L-ido configured deoxynojirimycin derivative

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Azacitidine Approved DB00928
small molecule | CAS: 320-67-2

Azacitidine is a pyrimidine nucleoside analogue with anti-neoplastic activity. It differs from cytosine by the presence of nitrogen in the C5-position, key in its hypomethylating activity.[A1406,A1413,A1415] Two main mechanisms of action have been proposed fo…

Kategori:
AntimetabolitesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +17
Target Protein:
DNA (cytosine-5)-methyltransferase 1RNADNA
Waktu ParuhThe mean half-life …
Vol. DistribusiIn patients given a…
KlirensAzacitidine has an …
Genetik -
AZACYCLONOL DB19381
small molecule | CAS: 115-46-8

Deskripsi belum tersedia.

Target Protein:
Histamine H1 receptor
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Azadirachta indica leaf Approved DB14352
biotech

Azadirachta indica leaf is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Azadirachtin DB19419
small molecule | CAS: 11141-17-6

Azadirachtin is under investigation in clinical trial NCT06617026 (Short-term Outcome of Medical vs. Surgical Management of Chronic Anal Fissure).

Kategori:
AgrochemicalsAzadirachtaCompounds used in a research, industrial, or household setting +5
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Azafenidin DB19031
small molecule | CAS: 68049-83-2

Azafenidin is under investigation in clinical trial NCT01726582 (Pancreas Cancer: Molecular Profiling as a Guide to Therapy Before and After Surgery ("Personalized Medicine")).

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Azapentacene DB15951
small molecule | CAS: 3863-80-7

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
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Azaperone DB11376
small molecule | CAS: 1649-18-9

Azaperone is a pyridinylpiperazine and butyrophenone agent that is capable of eliciting neuroleptic sedative and antiemetic effects. It is subsequently employed predominantly as a veterinary tranquilizer and mainly for pigs and elephants. At the same time, th…

Kategori:
Antipsychotic AgentsAntipsychotic Agents (First Generation [Typical])Butyrophenones +11
Target Protein:
D(3) dopamine receptorD(2) dopamine receptor
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Azaribine Approved DB19364
small molecule | CAS: 2169-64-4

Deskripsi belum tersedia.

Kategori:
Aza CompoundsDermatologicalsNucleic Acids, Nucleotides, and Nucleosides +4
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Azatadine Approved DB00719
small molecule | CAS: 3964-81-6

Antihistamines such as azatadine appear to compete with histamine for histamine H1- receptor sites on effector cells. The antihistamines antagonize those pharmacological effects of histamine which are mediated through activation of H1- receptor sites and ther…

Kategori:
Agents that reduce seizure thresholdAnticholinergic AgentsAntihistamines for Systemic Use +10
Target Protein:
Histamine H1 receptor
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Azathioprine Approved DB00993
small molecule | CAS: 446-86-6

Azathioprine is a prodrug of 6-mercaptopurine, first synthesized in 1956 by Gertrude Elion, William Lange, and George Hitchings in an attempt to produce a derivative of 6-mercaptopurine with a better therapeutic index.[A189678,A189687,A189690] Azathioprine is…

Kategori:
AntimetabolitesAntineoplastic and Immunomodulating AgentsAntirheumatic Agents +21
Target Protein:
AmidophosphoribosyltransferaseRas-related C3 botulinum toxin substrate 1
Gen Terkait:
TPMT TPMT TPMT
Waktu ParuhThe half life of az…
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik 3 Varian
AZD 3355 DB05404
small molecule

AZD 3355 is a reflux inhibitor used for the treatment of Gastroesophageal Reflux Disease. It is developed by AstraZeneca and is currently in phase I/II trials.

Kategori:
AcidsAcids, NoncarboxylicAmines +8
Target Protein:
Cellular tumor antigen p53
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AZD-0328 DB12145
small molecule | CAS: 220099-91-2

AZD0328 has been used in trials studying the treatment and basic science of Schizophrenia and Alzheimer's Disease.

Kategori:
Receptors, Nicotinic
Target Protein:
Neuronal acetylcholine receptor subunit alpha-7
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AZD-0424 DB13088
small molecule | CAS: 692054-06-1

AZD0424 has been used in trials studying the treatment of Advanced Solid Tumours.

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingProtein Kinase Inhibitors
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AZD-1236 DB11961
small molecule | CAS: 459814-89-2

AZD1236 has been used in trials studying the basic science and treatment of Cystic Fibrosis and Chronic Obstructive Pulmonary Disease.

Kategori:
AmidesImidazolesImidazolidines +2
Target Protein:
Macrophage metalloelastase
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AZD-1305 DB11766
small molecule | CAS: 872045-91-5

AZD1305 has been used in trials studying the treatment and basic science of Atrial Flutter, Atrial Fibrillation, and Left Ventricle Function.

Kategori:
Acids, AcyclicAza Compounds
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AZD-1386 DB15333
small molecule | CAS: 942937-80-6

AZD-1386 is under investigation in clinical trial NCT00945178 (Double-blind Placebo-controlled 2-part Study Assessing the Safety, Tolerability and PK of AZD1386 in Healthy Volunteers).

Kategori:
Heterocyclic Compounds, Fused-Ring
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AZD-1480 DB12588
small molecule | CAS: 935666-88-9

AZD1480 has been used in trials studying the treatment of Solid Malignancies, Post-Polycythaemia Vera, Primary Myelofibrosis (PMF), and Essential Thrombocythaemia Myelofibrosis.

Kategori:
Janus Kinase 2, antagonists & inhibitorsJanus Kinases, antagonists & inhibitors
Target Protein:
Tyrosine-protein kinase JAK2
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AZD-1656 DB14810
small molecule | CAS: 919783-22-5

AZD-1656 is under investigation in clinical trial NCT00747175 (A Study to Evaluate Safety, Tolerability and P-Glucose After Multiple Ascending Oral Doses of AZD1656 in Type 2 Diabetes).

Kategori:
AzetinesGlucokinase
Target Protein:
Hexokinase-4
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AZD-1940 DB17077
small molecule | CAS: 881413-29-2

Deskripsi belum tersedia.

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AZD-1981 DB11946
small molecule | CAS: 802904-66-1

AZD1981 has been used in trials studying the treatment and basic science of Asthma, Postmenopausal, Pharmakokinetic, Asthma Patients, and Drug Interaction, among others.

Target Protein:
Prostaglandin D2 receptor 2
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AZD-2066 DB12644
small molecule | CAS: 934282-55-0

AZD2066 has been used in trials studying the treatment and basic science of Pain, Chronic Pain, Reflux Episodes, Neuropathic Pain, and Diabetic Neuropathy, among others.

Target Protein:
Metabotropic glutamate receptor 5
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AZD-3043 DB12576
small molecule | CAS: 579494-66-9

AZD3043 has been used in trials studying the treatment and basic science of Safety, Sedation, Tolerability, and Pharmacokinetics.

Kategori:
Acids, CarbocyclicCentral Nervous System DepressantsHypnotics and Sedatives
Target Protein:
Gamma-aminobutyric acid receptor subunit gamma-3
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AZD-3759 DB14795
small molecule | CAS: 1626387-80-1

AZD-3759 is under investigation in clinical trial NCT03360929 (Evaluate Safety, Tolerability, Pharmacokinetics and Anti-tumor Activity of AZD3759).

Kategori:
Heterocyclic Compounds, Fused-Ring
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AZD-3839 DB12368
small molecule | CAS: 1227163-84-9

AZD3839 has been used in trials studying the basic science of Safety, Tolerability, Alzheimer's Disease, and Blood Concentration.

Kategori:
Heterocyclic Compounds, Fused-Ring
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AZD-4017 DB14875
small molecule | CAS: 1024033-43-9

AZD-4017 is under investigation in clinical trial NCT01173471 (A Phase IIa Study to Assess the Tolerability, Safety, and Efficacy of AZD4017 for Raised Intra-ocular Pressure).

Kategori:
11-beta-Hydroxysteroid Dehydrogenase Type 1, antagonists & inhibitorsNicotinic AcidsPyridines
Target Protein:
11-beta-hydroxysteroid dehydrogenase 1
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AZD-4547 DB12247
small molecule | CAS: 1035270-39-3

AZD4547 has been used in trials studying the treatment of Cancer, LYMPHOMA, Gastric Cancer, Adenocarcinoma, and Solid Neoplasm, among others.

Target Protein:
Fibroblast growth factor receptor 1
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AZD-4818 DB12002
small molecule | CAS: 1003566-93-5

AZD4818 has been used in trials studying the treatment of Chronic Obstructive Pulmonary Disease (COPD).

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AZD-4877 DB11671
small molecule | CAS: 1176760-49-8

AZD4877 has been used in trials studying the treatment of NHL, Tumors, Cancer, Lymphoma, and Neoplasms, among others.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +2
Target Protein:
Kinesin-like protein KIF11
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AZD-5423 DB12280
small molecule | CAS: 1034148-04-3

AZD5423 has been used in trials studying the basic science and treatment of Asthma, Bioavailability and AUC, and Chronic Obstructive Pulmonary Disease (COPD).

Kategori:
AcetatesAcids, AcyclicAmides +4
Target Protein:
Glucocorticoid receptor
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AZD-5672 DB11804
small molecule | CAS: 780750-65-4

Azd5672 has been used in trials studying the basic science and treatment of Pharmacokinetics, Renal Impairment, and Rheumatoid Arthritis.

Kategori:
AcetamidesAmidesAnti-HIV Agents +5
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AZD-5991 DB14792
small molecule | CAS: 2143010-83-5

AZD-5991 is under investigation in clinical trial NCT03218683 (Study of AZD5991 in Relapsed or Refractory Haematologic Malignancies.).

Kategori:
Antineoplastic Agents
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AZD-6280 DB12210
small molecule | CAS: 942436-93-3

AZD6280 has been used in trials studying the basic science of Anxiety.

Kategori:
Heterocyclic Compounds, Fused-RingReceptors, Opioid, delta, agonists
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-3
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AZD-6482 DB14980
small molecule | CAS: 1173900-33-8

AZD-6482 is under investigation in clinical trial NCT00688714 (Study to Investigate Safety and Tolerability of a Single Dose of AZD6482).

Kategori:
Acids, CarbocyclicAminobenzoatesBenzene Derivatives +3
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform
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AZD-7268 DB19203
small molecule | CAS: 1018988-00-5

AZD-7268 is under investigation in clinical trial NCT01020799 (AZD7268 Safety and Tolerability Study).

Kategori:
Heterocyclic Compounds, Fused-RingReceptors, Opioid, delta, agonists
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AZD-7295 DB12724
small molecule | CAS: 929890-64-2

AZD7295 has been investigated for the treatment of Hepatitis C.

Target Protein:
Genome polyprotein
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AZD-7325 DB13994
small molecule | CAS: 942437-37-8

AZD7325 is a high affinity, selective modulator of the GABAA receptor system. [L2936]

Kategori:
GABA ModulatorsHeterocyclic Compounds, Fused-Ring
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-3Gamma-aminobutyric acid receptor subunit alpha-2
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AZD-7687 DB14949
small molecule | CAS: 1166827-44-6

AZD-7687 is under investigation in clinical trial NCT01119352 (AZD7687 Multiple Ascending Dose Study).

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +1
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AZD-7762 DB12242
small molecule | CAS: 860352-01-8

AZD7762 has been investigated for the treatment of Cancer, Solid Tumors, and Advanced Solid Malignancies.

Kategori:
AmidesSulfur Compounds
Target Protein:
Serine/threonine-protein kinase Chk1
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AZD-8055 DB12774
small molecule | CAS: 1009298-09-2

AZD8055 has been used in trials studying the treatment of Cancer, Lymphomas, Solid Tumors, MALIGNANT GLIOMA, and brainstem glioma, among others.

Kategori:
Oxazines
Target Protein:
Serine/threonine-protein kinase mTOR
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AZD-8165 DB15132
small molecule | CAS: 1201686-72-7

AZD-8165 is under investigation in clinical trial NCT01150812 (Oral AZD8165 After Single Oral Ascending Doses in Healthy Male Subjects).

Target Protein:
Prothrombin
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AZD-8186 DB15029
small molecule | CAS: 1627494-13-6

AZD-8186 is under investigation in clinical trial NCT03218826 (PI3Kbeta Inhibitor AZD8186 and Docetaxel in Treating Patients Advanced Solid Tumors With PTEN or PIK3CB Mutations That Are Metastatic or Cannot Be Removed by Surgery).

Kategori:
AminesBenzopyransHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform
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AZD-8330 DB06061
small molecule | CAS: 869357-68-6

AZD-8330 is a potent, selective, orally active MEK inhibitor that blocks signal transduction pathways implicated in cancer cell proliferation and survival. AZD-8330 has shown tumor suppressive activity in multiple preclinical models of human cancer including …

Kategori:
Protein Kinase InhibitorsPyridines
Target Protein:
Mitogen-activated protein kinase kinase kinase 1
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AZD-8418 DB13102
small molecule | CAS: 1198309-73-7

Azd8418 is under investigation in clinical trial NCT01027234 (This Study Will Assess the Safety and Tolerability of AZD8418 After Single Increasing Oral Doses).

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AZD-8848 DB14868
small molecule | CAS: 866269-28-5

AZD-8848 is under investigation in clinical trial NCT01818869 (To Assess the Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of Multiple Doses AZD8848 in Healthy Subjects).

Kategori:
Acids, CarbocyclicHeterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and Nucleosides +4
Target Protein:
Toll-like receptor 7
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AZD-9056 DB12594
small molecule | CAS: 345304-65-6

AZD9056 has been used in trials studying the basic science and treatment of Rheumatoid Arthritis.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +3
Target Protein:
P2X purinoceptor 7
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AZD-9164 DB12115
small molecule | CAS: 1034978-04-5

AZD9164 has been used in trials studying the basic science and treatment of Chronic Obstructive Pulmonary Disease.

Kategori:
Receptor, Muscarinic M3, antagonists & inhibitors
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AZD-9496 DB15138
small molecule | CAS: 1639042-08-2

AZD-9496 is under investigation in clinical trial NCT02248090 (AZD9496 First Time in Patients Ascending Dose Study).

Kategori:
Acids, CarbocyclicHeterocyclic Compounds, Fused-Ring
Target Protein:
Estrogen receptor
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AZD-9684 DB05712
small molecule

AZD-9684 is the first member of a new anti-thrombotic class (CPU inhibitors). It is being developed by AstraZeneca.

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +1
Target Protein:
Carboxypeptidase B2
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AZD-9977 DB15418
small molecule | CAS: 1850385-64-6

AZD-9977 is under investigation in clinical trial NCT03843060 (A Phase 1 Study to Assess the Pharmacokinetics of AZD9977 Administered Alone and in Combination With Itraconazole in Healthy Volunteers).

Kategori:
Acids, CarbocyclicBenzene Derivatives
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