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6694

Total database: 17430
Struktur (SMILES)
4518 (67.5%)
Target
3751 (56.0%)
Genomik
81 (1.2%)
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6694 (100.0%)

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Hasil Pencarian (6694)

Halaman 58 / 134
biotech | CAS: 2248111-37-5

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Foreskin fibroblast-like stromal cells (FDSCs) are progenitors isolated from human tissue that can differentiate into various cell types [A32660]. Also known as Dermagraft, this device is a cryopreserved human fibroblast-derived dermal substitute. Composed…

Kategori:
Allogeneic Cultured Cell Scaffold
Target Protein:
Vascular endothelial growth factor receptor 1Interleukin-6Interleukin-1 receptor type 1 +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Foretinib DB12307
small molecule | CAS: 849217-64-7

Foretinib has been used in trials studying the treatment of Cancer, Breast Cancer, Carcinoma, Renal Cell, Recurrent Breast Cancer, and Neoplasms, Head and Neck, among others. Foretinib is an orally available small molecule compound designed to target multiple…

Kategori:
AmidesAminesAniline Compounds +3
Target Protein:
Hepatocyte growth factor receptorVascular endothelial growth factor receptor 2Hepatocyte growth factor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Forimtamig DB19015
biotech | CAS: 2649379-96-2

Forimtamig is under investigation in clinical trial NCT06055075 (A Study Evaluating Safety, Tolerability, and Clinical Activity of Forimtamig-based Treatment Combinations in Participants With Relapsed or Refractory Multiple Myeloma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Formic acid DB01942
small molecule | CAS: 64-18-6

Formic acid (systematically called methanoic acid) is the simplest carboxylic acid. It is an important intermediate in chemical synthesis and occurs naturally, most famously in the venom of bee and ant stings. It is commonly used as a preservative and antibac…

Kategori:
Acids, AcyclicBlood Coagulation FactorsHemostatics
Target Protein:
Nitric oxide synthase 1Hematopoietic prostaglandin D synthaseDelta-aminolevulinic acid dehydratase +51
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Formycin DB02281
small molecule | CAS: 6742-12-7

Deskripsi belum tersedia.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleosidesPyrimidine Nucleosides +2
Target Protein:
S-methyl-5'-thioadenosine phosphorylase5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Formycin B DB04198
small molecule

Deskripsi belum tersedia.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleosidesPyrimidine Nucleosides +2
Target Protein:
Hypoxanthine-guanine-xanthine phosphoribosyltransferasePurine nucleoside phosphorylase DeoD-typeHypoxanthine-guanine phosphoribosyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
AMP nucleosidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Forodesine DB06185
small molecule | CAS: 209799-67-7

Forodesine is a highly potent, orally active, rationally designed PNP inhibitor that has shown activity in preclinical studies with malignant cells and clinical utility against T-cell acute lymphoblastic leukemia and cutaneous T-cell lymphoma. Additional prel…

Kategori:
Heterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and NucleosidesNucleosides +3
Target Protein:
Purine nucleoside phosphorylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fosamprenavir Approved DB01319
small molecule | CAS: 226700-79-4

Fosamprenavir is a prodrug of amprenavir, an inhibitor of human immunodeficiency virus (HIV) protease.

Kategori:
Acids, AcyclicAmidesAmprenavir and Prodrugs +22
Target Protein:
Pol polyproteinGag-Pol polyprotein
Waktu ParuhThe plasma eliminat…
Vol. Distribusi-
Klirens-
Genetik -
Fosaprepitant Approved DB06717
small molecule | CAS: 172673-20-0

Fosaprepitant is an intravenously administered antiemetic drug. It is a prodrug of Aprepitant. It aids in the prevention of acute and delayed nausea and vomiting associated with chemotherapy treatment.

Kategori:
AntiemeticsAprepitant and ProdrugsAutonomic Agents +24
Target Protein:
Substance-P receptor
Waktu Paruh9-13 hours
Vol. Distribusi-
Klirens-
Genetik -
Foscarbidopa Approved DB16171
small molecule | CAS: 1907685-81-7

Foscarbidopa is under investigation in clinical trial NCT04379050 (Extension Study to Evaluate Safety and Tolerability of 24-hour Daily Exposure of Continuous Subcutaneous Infusion of ABBV-951 in Adult Participants With Parkinson's Disease).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Foscarnet Approved DB00529
small molecule | CAS: 4428-95-9

An antiviral agent used in the treatment of cytomegalovirus retinitis. Foscarnet also shows activity against human herpes viruses and HIV.

Kategori:
AcetatesAcids, AcyclicAnti-Infective Agents +17
Target Protein:
DNA polymerase catalytic subunitDNA polymerase catalytic subunit
Waktu Paruh3.3-6.8 hours
Vol. Distribusi-
Klirens* 2.13 +/- 0.71 mL/…
Genetik -
Fosciclopirox DB18772
small molecule | CAS: 1380539-06-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fosdagrocorat DB12198
small molecule | CAS: 1044535-58-1

Fosdagrocorat has been used in trials studying the treatment and basic science of Rheumatoid Arthritis.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fosdenopterin Approved DB16628
small molecule | CAS: 150829-29-1

Molybdenum cofactor deficiency (MoCD) is an exceptionally rare autosomal recessive disorder resulting in a deficiency of three molybdenum-dependent enzymes: sulfite oxidase (SOX), xanthine dehydrogenase, and aldehyde oxidase.[A230088] Signs and symptoms begin…

Kategori:
Alimentary Tract and MetabolismBiological FactorsCyclic Pyranopterin Monophosphate +9
Target Protein:
Molybdenum cofactor biosynthesis protein 1Xanthine dehydrogenase/oxidase
Waktu ParuhThe mean half-life …
Vol. DistribusiThe volume of distr…
KlirensTotal body clearanc…
Genetik -
Fosfomycin Approved DB00828
small molecule | CAS: 23155-02-4

Fosfomycin was discovered in 1969 by scientists at the Spanish Penicillin and Antibiotics Company and is produced by _Streptomyces fradiae_.[A229338,A230348] It may also be produced synthetically and is commercially available as the disodium salt for intraven…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAnti-Infective Agents, Urinary +7
Target Protein:
UDP-N-acetylglucosamine 1-carboxyvinyltransferase
Waktu ParuhThe mean eliminatio…
Vol. DistribusiIn healthy subjects…
KlirensIn one study, the r…
Genetik -
small molecule | CAS: 1562406-27-2

NUC-1031 is under investigation in clinical trial NCT03610100 (Acelarin First Line Randomised Pancreatic Study).

Kategori:
Antineoplastic AgentsCytosine NucleotidesNucleic Acids, Nucleotides, and Nucleosides +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fosinopril Approved DB00492
small molecule | CAS: 98048-97-6

Fosinopril is a phosphinic acid-containing ester prodrug that belongs to the angiotensin-converting enzyme (ACE) inhibitor class of medications. It is rapidly hydrolyzed to fosinoprilat, its principle active metabolite. Fosinoprilat inhibits ACE, the enzyme r…

Kategori:
ACE Inhibitors and DiureticsAgents Acting on the Renin-Angiotensin SystemAgents causing angioedema +17
Target Protein:
Angiotensin-converting enzyme
Waktu Paruh12 hours
Vol. Distribusi-
Klirens* 26 - 39 mL/min [h…
Genetik -
Fosinoprilat DB14207
small molecule | CAS: 95399-71-6

Fosinoprilat is the active phosphinic acid metabolite of prodrug [fosinopril], which is activated by esterases in vivo. It binds zinc with phosphinic acid group.

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Foslevodopa Approved DB16683
small molecule | CAS: 97321-87-4

Foslevodopa is under investigation in clinical trial NCT04750226 (Study to Assess Adverse Events and Change in Disease Activity of 24-hour Continuous Subcutaneous Infusion of ABBV-951 in Adult Participants With Advanced Parkinson's Disease).

Kategori:
Anti-Parkinson DrugsDopa and Dopa DerivativesDopamine Agents +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Foslinanib DB16172
small molecule | CAS: 1256037-60-1

Foslinanib is under investigation in clinical trial NCT03600233 (Study of CVM-1118 for Patients With Advanced Neuroendocrine Tumors).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fosmidomycin DB02948
small molecule | CAS: 66508-53-0

Deskripsi belum tersedia.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsOrganophosphonates +1
Target Protein:
1-deoxy-D-xylulose 5-phosphate reductoisomerase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fosnetupitant Approved DB14019
small molecule | CAS: 1703748-89-3

In April 2018, the U.S. Food and Drug Administration (FDA) and the Swiss company Helsinn approved the intravenous formulation of AKYNZEO® (NEPA, a fixed antiemetic combination of fosnetupitant, 235mg, and palonosetron, 0.25mg) as an alternative treatment opti…

Kategori:
Cytochrome P-450 CYP3A InhibitorsCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Inhibitors +6
Target Protein:
Substance-P receptor
Waktu ParuhNetupitant is elimi…
Vol. DistribusiThe mean SD volume …
KlirensNetupitant has a me…
Genetik -
Fosravuconazole DB15204
small molecule | CAS: 351227-64-0

Fosravuconazole is under investigation in clinical trial NCT03378661 (BENDITA BEnznidazole New Doses Improved Treatment and Associations).

Kategori:
Antifungals for Dermatological UseAntifungals for Systemic UseDermatologicals
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fostamatinib Approved DB12010
small molecule | CAS: 901119-35-5

Fostamatinib has been investigated for the treatment and basic science of Rheumatoid Arthritis and Immune Thrombocytopenic Purpura (ITP). It was approved on April 17, 2018, under the trade name Tavalisse for use in ITP [L2644, FDA Label]. Fostamatinib has als…

Kategori:
AminesBCRP/ABCG2 InhibitorsBlood and Blood Forming Organs +17
Target Protein:
Tyrosine-protein kinase SYKAdenosine receptor A3Synaptic vesicular amine transporter +297
Waktu ParuhR406 has a half-lif…
Vol. DistribusiR406 has an apparen…
KlirensR406 has an apparen…
Genetik -
Fostemsavir Approved DB11796
small molecule | CAS: 864953-29-7

Fostemsavir is the phosphonooxymethyl prodrug of temsavir, a novel HIV-1 attachment inhibitor.[L14867] It binds to and inhibits the activity of gp120, a subunit within the HIV-1 gp160 envelope glycoprotein that facilitates the attachment of HIV-1 to host cell…

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +18
Target Protein:
Envelope glycoprotein gp160
Waktu ParuhThe half-life of te…
Vol. DistribusiThe steady-state vo…
KlirensThe mean clearance …
Genetik -
small molecule | CAS: 2129993-56-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fotemustine DB04106
small molecule | CAS: 92118-27-9

Deskripsi belum tersedia.

Kategori:
Alkylating DrugsAmidesAntineoplastic Agents +3
Target Protein:
Thioredoxin reductase 1, cytoplasmic
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Framycetin Approved DB00452
small molecule | CAS: 119-04-0

A component of neomycin that is produced by Streptomyces fradiae. On hydrolysis it yields neamine and neobiosamine B. (From Merck Index, 11th ed)

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +10
Target Protein:
16S ribosomal RNA30S ribosomal protein S12C-X-C chemokine receptor type 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fremanezumab Approved DB14041
biotech | CAS: 1655501-53-3

Fremanezumab is a humanized monoclonal antibody targeted against human calcitonin gene-related peptide (CGRP) for the prevention of migraine headaches.[L11749] It was developed by Teva Pharmaceuticals USA and approved by the FDA in September 2018.[L11779] Alo…

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAntibodies +12
Target Protein:
Calcitonin gene-related peptide 1Calcitonin gene-related peptide 2
Waktu ParuhThe mean half-life …
Vol. DistribusiFremanezumab has an…
KlirensThe apparent cleara…
Genetik -
Friulimicin B DB06087
small molecule | CAS: 239802-15-4

Friulimicin B is a naturally occurring antibiotic produced by a micro-organism, *Actinoplanes friuliensis*. It shows strong cidal activity against a number of Gram-positive pathogens which commonly cause serious infections in hospital patients and which are b…

Kategori:
Amino Acids, Peptides, and Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Frovatriptan Approved DB00998
small molecule | CAS: 158747-02-5

Frovatriptan is a triptan drug developed by Vernalis for the treatment of migraine headaches, in particular those associated with menstruation. Frovatriptan causes vasoconstriction of arteries and veins that supply blood to the head.

Kategori:
Agents that produce hypertensionAminesAnalgesics +23
Target Protein:
5-hydroxytryptamine receptor 1D5-hydroxytryptamine receptor 1B
Gen Terkait:
GNB3
Waktu Paruh26 hours
Vol. Distribusi* 4.2 L/kg [males] …
Klirens* 220 mL/min [male …
Genetik 1 Varian
Frovocimab DB15089
biotech | CAS: 1643672-70-1

Frovocimab is under investigation in clinical trial NCT01671085 (A Study of LY3015014 in Healthy Participants With High Cholesterol).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 643-13-0

Deskripsi belum tersedia.

Kategori:
CarbohydratesHexosephosphatesSugar Phosphates
Target Protein:
Fructose-1,6-bisphosphatase 1Fructose-1,6-bisphosphatase isozyme 26-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 1 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fruquintinib Approved DB11679
small molecule | CAS: 1194506-26-7

Fruquintinib is a novel small-molecule anti-VEGFR that targets VEGFR-1,-2, and -3 to inhibit angiogenesis. Tumor angiogenesis is one of the most critical biological processes for increasing oxygen and nutrient supply to cancer cells, and the VEGF/VEGFR pathwa…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsCytochrome P-450 CYP2C19 Substrates +10
Target Protein:
Vascular endothelial growth factor receptor 1Vascular endothelial growth factor receptor 2Vascular endothelial growth factor receptor 3
Waktu ParuhThe fruquintinib's …
Vol. DistribusiThe mean (SD) appar…
KlirensThe apparent cleara…
Genetik -
FT-1101 DB17553
small molecule | CAS: 1776060-36-6

FT-1101 is a novel Bromodomain and Extra-Terminal motif (BET) inhibitor.[A257301] FT-1101 is under investigation in clinical trial NCT02543879 (Study of a Novel BET Inhibitor FT-1101 in Patients With Relapsed or Refractory Hematologic Malignancies).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fucitol DB03815
small molecule | CAS: 13074-06-1

Deskripsi belum tersedia.

Kategori:
AlcoholsCarbohydrates
Target Protein:
L-fucose isomerase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fucose DB15236
small molecule | CAS: 2438-80-4

Fucose is under investigation in clinical trial NCT03354533 (Study of ORL-1F (L-fucose) in Patients With Leukocyte Adhesion Deficiency Type II).

Kategori:
CarbohydratesDeoxy Sugars
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fucoxanthin DB15462
small molecule | CAS: 3351-86-8

Fucoxanthin is under investigation in clinical trial NCT03613740 (Effect of Fucoxanthin on the Components of the Metabolic Syndrome, Insulin Sensitivity and Insulin Secretion). Fucoxanthin isis a marine carotenoid mainly found in brown algae, giving them a br…

Kategori:
AlkenesBiological FactorsCarotenoids +7
Target Protein:
NF-kappa-B inhibitor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fulacimstat DB15085
small molecule | CAS: 1488354-15-9

Fulacimstat is under investigation in clinical trial NCT02452515 (A Single-blind Pilot Study to Investigate Safety and Tolerability of the Chymase Inhibitor BAY1142524 in Clinically Stable Patients With Left-ventricular Dysfunction).

Kategori:
Enzyme Inhibitors
Target Protein:
Chymase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fumaric acid DB01677
small molecule | CAS: 110-17-8

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAntipsoriaticsAntipsoriatics for Topical Use +2
Target Protein:
Interferon gammaMalate dehydrogenaseFumarate reductase flavoprotein subunit +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furaprofen DB06499
small molecule | CAS: 67700-30-5

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furfural DB16856
small molecule | CAS: 98-01-1

Deskripsi belum tersedia.

Kategori:
AldehydesFurans
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furosemide Approved DB00695
small molecule | CAS: 54-31-9

Furosemide is a potent loop diuretic that acts on the kidneys to ultimately increase water loss from the body. It is an anthranilic acid derivative.[L7958] Furosemide is used for edema secondary to various clinical conditions, such as congestive heart failure…

Kategori:
Acids, CarbocyclicAmidesAmines +30
Target Protein:
Solute carrier family 12 member 1Carbonic anhydrase 2G-protein coupled receptor 35
Waktu ParuhThe half-life from …
Vol. DistribusiThe volume of distr…
KlirensFollowing intraveno…
Genetik -
Furoyl-Leucine DB02215
small molecule

Deskripsi belum tersedia.

Target Protein:
Disintegrin and metalloproteinase domain-containing protein 28
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fursultiamine Approved DB08966
small molecule | CAS: 804-30-8

Compound used for therapy of thiamine deficiency. It has also been suggested for several non-deficiency disorders but has not yet proven useful. Fursultiamine is a vitamin B1 derivative.

Kategori:
MicronutrientsPyrimidinesSulfur Compounds +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furvina DB16547
small molecule | CAS: 189935-72-6

Furvina (G1) is an antimicrobial agent active against Gram-positive and Gram-negative bacteria, yeasts, and filamentous fungi. Furvina is marketed in Cuba as Dermofural®, an ointment containing G1 as the only active principle ingredient. It is used to treat d…

Kategori:
AlkenesAnti-Infective AgentsHydrocarbons, Acyclic
Target Protein:
30S ribosomal protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fusicoccin DB01780
small molecule | CAS: 20108-30-9

Deskripsi belum tersedia.

Kategori:
CarbohydratesMycotoxins
Target Protein:
14-3-3 protein epsilon
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fusidic acid Approved DB02703
small molecule | CAS: 6990-06-3

An antibiotic isolated from the fermentation broth of Fusidium coccineum. (From Merck Index, 11th ed) It acts by inhibiting translocation during protein synthesis. It is often used topically in creams and eyedrops but is available in systemic formulations inc…

Kategori:
Agents Causing Muscle ToxicityAnti-Bacterial AgentsAnti-Infective Agents +35
Target Protein:
Elongation factor GChloramphenicol acetyltransferaseChloramphenicol acetyltransferase 3
Waktu ParuhApproximately 5 to …
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 2851–2900 dari 6694
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