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11793

Total database: 17430
Struktur (SMILES)
8607 (73.0%)
Target
6418 (54.4%)
Genomik
102 (0.9%)
Referensi
11793 (100.0%)

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Hasil Pencarian (11793)

Halaman 58 / 236
BMS-986278 DB18011
small molecule | CAS: 2170126-74-4

Deskripsi belum tersedia.

Target Protein:
Lysophosphatidic acid receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BMS184394 DB03466
small molecule

Deskripsi belum tersedia.

Target Protein:
Retinoic acid receptor gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BMSC-0013 DB02474
small molecule

Deskripsi belum tersedia.

Target Protein:
Cholera enterotoxin subunit B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1379866-50-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
BN-201 DB18295
small molecule | CAS: 1361200-34-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BN-82451 DB16950
small molecule | CAS: 335242-75-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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BN104 DB18172
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BNC-210 DB19048
small molecule | CAS: 1020634-41-6

BNC-210 is under investigation in clinical trial NCT04951076 (A Phase 2b Study of BNC210 Tablet Formulation in Adults With Post-traumatic Stress Disorder (PTSD)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BNC105 DB06313
small molecule | CAS: 945772-45-2

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesEthersHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BNT-162A1 DB16402
biotech | CAS: 2417899-74-0

BNT-162A1 is under investigation in clinical trial NCT04380701 (A Trial Investigating the Safety and Effects of Four BNT162 Vaccines Against COVID-2019 in Healthy Adults).

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBiological Factors +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

BNT162a1 is one of four advanced mRNA-based vaccines being developed through "Project Lightspeed," a joint program between Pfizer and BioNTech.[L15002, L15007] BNT162a1 is a uridine mRNA (uRNA) vaccine formulated in lipid nanoparticles for delivery via intram…

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

BNT162b1 is one of four advanced mRNA-based vaccines being developed through "Project Lightspeed," a joint program between Pfizer and BioNTech.[L15002, L15007] BNT162b1 is a nucleoside modified mRNA (modRNA) vaccine encoding the receptor-binding domain (RBD) …

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBiological Factors +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BNT162b2 Omicron (KP.2) Approved DB19415
biotech

BNT162b2 Omicron (KP.2) is COVID-19 mRNA vaccine encoding the viral spike (S) glycoprotein of SARS-CoV-2 Omicron variant lineage KP.2. It is the active ingredient in the 2024-2025 formulation of Pfizer-BioNTech's Comirnaty vaccine.[L36030]

Waktu Paruh-
Vol. Distribusi-
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BNT162b3 DB16442
biotech

The BNT162b3 vaccine is the latest addition to BioNTech and partner Pfizer’s mRNA COVID-19 vaccine program. Similar to [BNT162b2], BNT162b3 uses a nucleoside-modified RNA (modRNA) technology. Pfizer and BioNTech deemed this compound as promising in preclinica…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

BNT162c2 is one of four advanced mRNA-based vaccines being developed through "Project Lightspeed," a joint program between Pfizer and BioNTech.[L15002, L15007] BNT162c2 is a self-amplifying mRNA (saRNA) vaccine formulated in lipid nanoparticles for delivery v…

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BO-653 DB19216
small molecule | CAS: 157360-23-1

BO-653 is under investigation in clinical trial NCT00055510 (A Blinded Study Conducted at Multiple Centers Evaluating Various Doses of an Investigational Agent (BO-653) Against Placebo, for Safety and Effectiveness in Preventing Post-angioplasty Blood Vessel …

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
D-alanyl-D-alanine carboxypeptidase DacAD-alanyl-D-alanine carboxypeptidase DacA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Boceprevir Approved DB08873
small molecule | CAS: 394730-60-0

Boceprevir is a direct acting antiviral medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized into nine…

Kategori:
Amino AcidsAmino Acids, CyclicAmino Acids, Peptides, and Proteins +21
Target Protein:
Genome polyproteinGenome polyprotein
Waktu ParuhBoceprevir has a me…
Vol. DistribusiThe mean apparent v…
KlirensBoceprevir has a me…
Genetik -
Bocidelpar DB16906
small molecule | CAS: 2095128-20-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 2356354-82-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
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Bococizumab DB12456
biotech | CAS: 1407495-02-6

Bococizumab has been used in trials studying the treatment and prevention of Dyslipidemia, Hyperlipidemia, Hypercholesterolemia, Cardiovascular Disease, and Heterozygous Familial Hypercholesterolemia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bolasterone DB01471
small molecule | CAS: 1605-89-6

Deskripsi belum tersedia.

Kategori:
Anabolic AgentsAndrostanesAndrostenes +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Boldenone DB01541
small molecule | CAS: 846-48-0

Boldenone is an anabolic steroid developed for veterinary use, mostly for treatment of horses. It is not indicated for use in humans in the US and is only available through veterinary clinics.

Kategori:
Anabolic AgentsAndrostanesAndrostenes +9
Target Protein:
Androgen receptor
Waktu Paruh14 days
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 13103-34-9

Deskripsi belum tersedia.

Kategori:
AndrostanesAndrostenesAndrostenols +6
Target Protein:
Androgen receptor
Waktu Paruh14 days
Vol. Distribusi-
Klirens-
Genetik -
Boldione DB07373
small molecule | CAS: 897-06-3

Deskripsi belum tersedia.

Kategori:
AndrostanesAndrostenesFused-Ring Compounds +1
Target Protein:
AromatasePentaerythritol tetranitrate reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bombesin DB11724
small molecule | CAS: 31362-50-2

Bombesin is under investigation in clinical trial NCT01205321 (PET/CT Imaging for Radiation Dosimetry, Plasma Pharmacokinetics, Biodistribution, Safety and Tolerability and Diagnostic Performance of BAY86-7548 in Patients With Prostate Cancer and Healthy Volu…

Kategori:
Amino Acids, Peptides, and ProteinsAmphibian VenomsBiological Factors +12
Target Protein:
Gastrin-releasing peptide receptorBombesin receptor subtype-3Neuromedin-B receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bombyx mori fiber Approved DB10609
biotech

Bombyx mori fiber is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2364477-20-1

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bopindolol DB08807
small molecule | CAS: 62658-63-3

Bopindolol (INN) is an ester prodrug for the beta blocker [pindolol].

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +12
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptorBeta-3 adrenergic receptor +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Borate ion DB14553
small molecule | CAS: 12258-53-6

Deskripsi belum tersedia.

Kategori:
AnionsBoric AcidsBoron Compounds +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Boric acid Approved DB11326
small molecule | CAS: 10043-35-3

Boric acid, also known as hydrogen borate, is a weak monobasic Lewis acid of boron with the chemical formula H3BO3. Boric acid is typically utilized in industrial processing and manufacturing, but is also used as an additive in pharmaceutical products, cosmet…

Kategori:
AcidsAcids, NoncarboxylicAgrochemicals +12
Waktu ParuhAccording to human …
Vol. DistribusiVolume of distribut…
KlirensA case report of ac…
Genetik -
Bornaprine DB13619
small molecule | CAS: 20448-86-6

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAnti-Parkinson DrugsAnticholinergic Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bornyl acetate DB14665
small molecule | CAS: 76-49-3

Deskripsi belum tersedia.

Kategori:
Bicyclic MonoterpenesBridged-Ring CompoundsMonoterpenes +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bortezomib Approved DB00188
small molecule | CAS: 179324-69-7

Bortezomib is a dipeptide boronic acid derivative and proteasome inhibitor used to treat multiple myeloma and mantle cell lymphoma.[A204083] The 26S proteasome is a protein complex that degrades ubiquitinated proteins in the ubiquitin-proteasome pathway: reve…

Kategori:
AcidsAcids, NoncarboxylicAntineoplastic Agents +36
Target Protein:
Proteasome subunit beta type-5Serine protease 1Proteasome subunit beta type-1
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe mean distributi…
KlirensFollowing the admin…
Genetik -
Bortezomib D-mannitol Approved DB16741
small molecule | CAS: 444576-08-3

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsProteasome Inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bos taurus hair Approved DB10856
biotech

Bos taurus hair is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bos taurus skin Approved DB10406
biotech

Bos taurus skin or pelt is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bosakitug DB19101
biotech | CAS: 2762183-23-1

Bosakitug (BSI-045B) is under investigation in clinical trial NCT05932654 (POC Study to Evaluate BSI-045B Monotherapy and BSI-045B Add-on Therapy With Dupilumab in Atopic Dermatitis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Boscalid Approved DB12792
small molecule | CAS: 188425-85-6

Boscalid has been investigated for the treatment of OSDI, Glaucoma, Staining, Schirmers, and Disease Severity, among others.

Kategori:
Benzene DerivativesNicotinic AcidsPyridines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bosentan Approved DB00559
small molecule | CAS: 147536-97-8

Bosentan is a dual endothelin receptor antagonist marketed under the trade name Tracleer by Actelion Pharmaceuticals. Bosentan is used to treat pulmonary hypertension by blocking the action of endothelin molecules that would otherwise promote narrowing of the…

Kategori:
AmidesAntihypertensive AgentsAntihypertensives for Pulmonary Arterial Hypertension +24
Target Protein:
Endothelin receptor type BEndothelin-1 receptor
Waktu ParuhTerminal eliminatio…
Vol. Distribusi* 18 L
Klirens* 4 L/h [patients w…
Genetik -
Bosutinib Approved DB06616
small molecule | CAS: 380843-75-4

Bosutinib is a 7-alkoxy-3-quinolinecarbonitrile that functions as a potent, dual SRC and ABL tyrosine kinase inhibitor indicated for chronic myelogenous leukemia (CML), specifically Philadelphia chromosome-positive (Ph+) CML. Philadelphia chromosome is a hall…

Kategori:
AminesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +22
Target Protein:
Tyrosine-protein kinase ABL1Tyrosine-protein kinase LynProto-oncogene tyrosine-protein kinase Src +8
Waktu ParuhThe mean (SD) bosut…
Vol. DistribusiThe mean (SD) appar…
KlirensThe mean (SD) appar…
Genetik -
biotech | CAS: 2417551-39-2

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Botensilimab DB16651
biotech | CAS: 2408310-37-0

Botensilimab is under investigation in clinical trial NCT03860272 (Fc-engineered Anti-ctla-4 Monoclonal Antibody in Advanced Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Botulinum toxin type A Approved DB00083
biotech | CAS: 93384-43-1

In 2002, botulinum toxin A, also known as onabotulinumtoxinA or Botox, was the first type A botulism toxin to be introduced into the market for cosmetic use.[A231824] With a wide variety of applications and favourable safety profile, Botulinum toxin A injecti…

Kategori:
Acetylcholine Release InhibitorsAgents that produce neuromuscular block (indirect)Amino Acids, Peptides, and Proteins +29
Target Protein:
Synaptosomal-associated protein 25Rho-related GTP-binding protein RhoB
Waktu ParuhThere is no readily…
Vol. DistribusiThere are extremely…
KlirensClearance informati…
Genetik -
biotech

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBacterial ProteinsBacterial Toxins +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1383710-57-3

Bovhyaluronidase azoximer is under investigation in clinical trial NCT06458543 (Optimization of Bacterial Vaginosis Treatment in Women of Reproductive Age).

Waktu Paruh-
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Genetik -
Bovine type I collagen Approved DB10771
biotech | CAS: 9050-08-2

Bovine collagen alpha-1 is a naturally occurring extracellular matrix protein which is found in tendons and other connective tissues. It plays a vital role in cell growth, differentiation, attachment, and migration [L2481]. Often combined with other ingredie…

Kategori:
Allogeneic Cultured Cell Scaffold
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BP-14979 DB16302
small molecule | CAS: 1000036-77-0

BP-14979 is under investigation in clinical trial NCT01785147 (Efficacy and Safety of BP1.4979 in Smoking Cessation).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BPC-157 DB11882
small molecule | CAS: 137525-51-0

Bepecin is under investigation in clinical trial NCT02637284 (PCO-02 - Safety and Pharmacokinetics Trial).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Ulcer AgentsGastrointestinal Agents +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BPH-608 DB07404
small molecule

Deskripsi belum tersedia.

Target Protein:
Farnesyl pyrophosphate synthaseDitrans,polycis-undecaprenyl-diphosphate synthase ((2E,6E)-farnesyl-diphosphate specific)
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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