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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 57 / 236
Bethanidine Approved DB00217
small molecule | CAS: 55-73-2

A guanidinium antihypertensive agent that acts by blocking adrenergic transmission.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +13
Target Protein:
Beta-1 adrenergic receptorATP-sensitive inward rectifier potassium channel 1Alpha-2 adrenergic receptors +1
Waktu Paruh9 hours (range 7 to…
Vol. Distribusi-
Klirens-
Genetik -
Betiatide Approved DB14082
small molecule | CAS: 103725-47-9

Deskripsi belum tersedia.

Waktu Paruh-
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Betibeglogene autotemcel Approved DB16900
biotech

Betibeglogene autotemcel is an autologous gene therapy that adds functional copies of the ?-globin gene (?<sup>A-T87Q</sup>-globin) to hematopoietic stem cells in order to treat ?-thalassemia.[L42940] ?-thalassemia is a condition caused by mutations in the ?-…

Kategori:
Autologous Cultured CellAutologous Hematopoietic Stem Cell-Based Gene TherapyBlood and Blood Forming Organs +2
Target Protein:
Alpha globin
Waktu Paruh-
Vol. DistribusiThe nature of betib…
Klirens-
Genetik -
Betrixaban Approved DB12364
small molecule | CAS: 330942-05-7

Betrixaban is a non-vitamin K oral anticoagulant whose action is driven by the competitive and reversible inhibition of the factor Xa [A7708]. It was selected among all lead compounds due to its low hERG channel affinity while sustaining its factor Xa inhibit…

Kategori:
Acids, CarbocyclicAmidesAnticoagulants +11
Target Protein:
Coagulation factor X
Waktu ParuhBetrixaban presents…
Vol. DistribusiThe apparent volume…
KlirensBetrixaban presents…
Genetik -
small molecule | CAS: 8001-88-5

Betula pendula tar oil is an essential oil found in the buds of the plant with the same name. The origin plant, also known as the European white or silver birch, grows mainly in the northern hemisphere. This oil is usually obtained by using both hydrodistilla…

Waktu ParuhThis pharmacokineti…
Vol. DistribusiThis pharmacokineti…
KlirensThis pharmacokineti…
Genetik -
Betula populifolia pollen Approved DB10724
biotech

Betula populifolia pollen is the pollen of the Betula populifolia plant. Betula populifolia pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
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Betulin DB16890
small molecule | CAS: 473-98-3

Deskripsi belum tersedia.

Kategori:
BetulaLupanesPentacyclic Triterpenes +2
Target Protein:
Glycogen phosphorylase, muscle form
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Betulinic Acid Approved DB12480
small molecule | CAS: 472-15-1

Betulinic Acid has been used in trials studying the treatment of Dysplastic Nevus Syndrome.

Kategori:
Agents that produce hypertensionAnalgesicsAnalgesics, Non-Narcotic +22
Target Protein:
DNA polymerase catalytic subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bevacizumab Approved DB00112
biotech | CAS: 216974-75-3

There is a great deal of evidence indicating that vascular endothelial growth factor (VEGF) is important for the survival and proliferation of cancer cells.[A192939,A192837,A192891,A193275] VEGF plays an important role in angiogenesis, lymphangiogenesis, and …

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +27
Target Protein:
Vascular endothelial growth factor A, long formComplement C1q subcomponent subunit AComplement C1q subcomponent subunit B +6
Waktu ParuhThe half-life of be…
Vol. DistribusiThe volume of distr…
KlirensThe clearance (CL) …
Genetik -
biotech

Bevacizumab zirconium Zr-89 is under investigation in clinical trial NCT01338090 (89Zr-bevacizumab PET Imaging in Patients With Neuroendocrine Tumors).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +17
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Bevantolol DB01295
small molecule | CAS: 59170-23-9

Bevantolol is a beta-1 adrenoceptor antagonist that has been shown to be as effective as other beta blockers for the treatment of angina pectoris and hypertension. Mechanism of Action Animal experiments confirm both agonist and antagonist effects on alpha-rec…

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +16
Target Protein:
D(2) dopamine receptorBeta-1 adrenergic receptorBeta-2 adrenergic receptor +1
Waktu Paruh-
Vol. Distribusi-
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Bevasiranib DB06642
biotech | CAS: 959961-96-7

Bevasiranib is a small interfering RNA (siRNA) targeting vascular endothelial growth factor A (VEGF-A).

Kategori:
Antisense Elements (Genetics)Compounds used in a research, industrial, or household settingMolecular Probes +6
Target Protein:
Vascular endothelial growth factor A, long form
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bevenopran DB12464
small molecule | CAS: 676500-67-7

Bevenopran has been used in trials studying the treatment of Renal Impairment and Opioid-Induced Constipation.

Waktu Paruh-
Vol. Distribusi-
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Bevifimod DB15301
biotech | CAS: 2223113-32-2

Bevifimod is under investigation in clinical trial NCT01749787 (Safety Study of PRTX-100 With Methotrexate or Leflunomide to Treat Active Rheumatoid Arthritis).

Kategori:
Amino Acids, Peptides, and ProteinsAntigensAntigens, Bacterial +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bevirimat DB06581
small molecule | CAS: 174022-42-5

Bevirimat, also known as PA-457 or YK-FH312, is investigated in clinical trials for treating HIV infection. Bevirimat is a solid. This compound belongs to the androgens and derivatives, which are hydroxylated C19 steroid hormones. They are known to favour the…

Kategori:
Acids, AcyclicAnti-HIV AgentsDicarboxylic Acids +2
Target Protein:
Gag-Pol polyprotein
Waktu Paruh56.3 to 69.5 hours
Vol. Distribusi-
Klirens-
Genetik -
Bevonescein DB19021
biotech | CAS: 2276787-79-0

Bevonescein is under investigation in clinical trial NCT06227585 (Feasibility Study- REVEAL 475 for Bevonescein-assisted Nerve Visualization in Head & Neck Surgery).

Waktu Paruh-
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Bevonium DB13542
small molecule | CAS: 33371-53-8

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAgents producing tachycardiaAlimentary Tract and Metabolism +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2374772-30-0

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
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Bexagliflozin Approved DB12236
small molecule | CAS: 1118567-05-7

Bexagliflozin is a highly specific and potent sodium-glucose co-transporter 2 (SGLT2) inhibitor.[A256408,A256413,L44758] Similar to other SGLT2 inhibitors, bexagliflozin contains three basic moieties: glucose, two benzene rings and a methylene bridge.[A256413…

Kategori:
Alimentary Tract and MetabolismBenzene DerivativesBlood Glucose Lowering Agents +16
Target Protein:
Sodium/glucose cotransporter 2
Waktu ParuhBexagliflozin has a…
Vol. DistribusiBexagliflozin has a…
KlirensPopulation pharmaco…
Genetik -
Bexarotene Approved DB00307
small molecule | CAS: 153559-49-0

Bexarotene (Targretin) is an antineoplastic agent indicated by the FDA for Cutaneous T cell lymphoma. It has been used off-label for lung cancer, breast cancer, and Kaposi's sarcoma.

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsCompounds used in a research, industrial, or household setting +18
Target Protein:
Retinoic acid receptor RXR-alphaRetinoic acid receptor RXR-betaRetinoic acid receptor RXR-gamma
Waktu Paruh7 hours
Vol. Distribusi-
Klirens-
Genetik -
Bexicaserin DB18885
small molecule | CAS: 2035818-24-5

Bexicaserin is under investigation in clinical trial NCT05626634 (Open-label, Long-term Safety Study of LP352 in Subjects With Developmental and Epileptic Encephalopathy).

Waktu Paruh-
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Bexmarilimab DB16383
biotech | CAS: 2259301-27-2

Bexmarilimab is under investigation in clinical trial NCT03733990 (A Study to Evaluate Safety, Tolerability and Preliminary Efficacy of FP-1305 in Cancer Patients).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bexotegrast DB18444
small molecule | CAS: 2376257-44-0

Deskripsi belum tersedia.

Waktu Paruh-
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Bezafibrate Approved DB01393
small molecule | CAS: 41859-67-0

Antilipemic agent that lowers cholesterol and triglycerides. It decreases low density lipoproteins and increases high density lipoproteins.

Kategori:
Acids, AcyclicAcids, CarbocyclicAgents Causing Muscle Toxicity +26
Target Protein:
Peroxisome proliferator-activated receptor deltaPeroxisome proliferator-activated receptor gammaPeroxisome proliferator-activated receptor alpha +4
Waktu Paruh1-2 hours
Vol. Distribusi-
Klirens-
Genetik -
Bezitramide DB01459
small molecule | CAS: 15301-48-1

Bezitramide is a narcotic analgesic which was discovered in 1961, clinically tested around the 1970's [A14383], and marketed under the name Burgodin. After cases of fatal overdose in the Netherlands in 2004 the drug was withdrawn from the market. Bezitram…

Kategori:
AnalgesicsCentral Nervous System AgentsDiphenylpropylamine Derivatives +6
Waktu Paruh11-24h. [A14383]
Vol. Distribusi-
Klirens-
Genetik -
Bezlotoxumab Approved DB13140
biotech | CAS: 1246264-45-8

Bezlotoxumab is a fully humanized ImmunoglobulinG1 (IgG1) kappa monoclonal antibody that binds to _Clostridium difficile_ toxin B and neutralizes its effects.[L46976] First approved by the FDA on October 21, 2016,[A260106] bezlotoxumab is used to reduce the r…

Kategori:
Amino Acids, Peptides, and ProteinsAntibacterial monoclonal antibodiesAntibodies +11
Target Protein:
Toxin B
Waktu ParuhBased on a populati…
Vol. DistribusiBased on a populati…
KlirensBased on a populati…
Genetik -
BF-37 DB05755
small molecule

BF-37 for the treatment of atopic dermatitis and/or psoriasis. The active ingredient in BF-37 is Riluzole, applied in a topical formulation, which is believed to correct the imbalances of the immune system that cause atopic dermatitis or psoriasis.

Waktu Paruh-
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BF-844 DB17801
small molecule | CAS: 1404506-35-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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BFH772 DB16035
small molecule | CAS: 890128-81-1

BFH772 is under investigation in clinical trial NCT01449591 (Safety, Tolerability and Efficacy of BFH772 in Rosacea Patients).

Waktu Paruh-
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BG-777 DB05839
small molecule

BG-777 is an immunomodulator with proven efficacy against viral and bacterial infections in preclinical studies.

Waktu Paruh-
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Genetik -
BG-P-TAT DB18105
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
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BG-P400-TAT DB17104
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
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BG1805 DB18667
biotech

BG1805 is an investigational anti-CLL1 chimeric antigen receptor (CAR) T-cell therapy.

Waktu Paruh-
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BGA002 DB17125
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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BGB-DXP593 DB16357
biotech

BGB-DXP593 is a SARS-CoV-2 neutralizing antibody.[L27401] It is currently being investigated against COVID-19 in the clinical trial NCT04551898 (Severe Acute Respiratory Syndrome Coronavirus 2 (SARS-CoV-2) Neutralizing Antibody BGB-DXP593 in Participants With…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
BHV-5000 DB17817
small molecule

BHV-5000 is an orally bioavailable, low-trapping, potent N-methyl-D-aspartate (NMDA) receptor antagonist. The active metabolite of BHV-5000 is [lanicemine].[L46446]

Waktu Paruh-
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BI 2536 DB16107
small molecule | CAS: 755038-02-9

BI 2536 is under investigation in clinical trial NCT00376623 (Efficacy and Safety of BI 2536 in Advanced or Metastatic Non Small Cell Lung Cancer).

Kategori:
Antimitotic AgentsHeterocyclic Compounds, Fused-Ring
Target Protein:
Serine/threonine-protein kinase PLK1
Waktu Paruh-
Vol. Distribusi-
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BI 44370 TA DB16037
small molecule | CAS: 866086-05-7

BI 44370 TA is under investigation in clinical trial NCT00751803 (BI 44370 TA in Acute Migraine Attack).

Waktu Paruh-
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BI-1206 DB17429
biotech

BI-1206 is a fully human immunoglobulin G1 monoclonal antibody that targets CD32b.

Waktu Paruh-
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BI-187004 DB18897
small molecule | CAS: 1303515-32-3

Deskripsi belum tersedia.

Waktu Paruh-
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BI-671800 DB12524
small molecule | CAS: 1093108-50-9

Bi 671800 has been used in trials studying the treatment of Asthma and Rhinitis, Allergic, Perennial.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Target Protein:
Prostaglandin D2 receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BI-765063 DB17482
biotech

BI-765063 is a humanized IgG4 monoclonal antibody antagonist of signal regulatory protein ? (SIRP?).

Waktu Paruh-
Vol. Distribusi-
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BI-836826 DB17322
biotech

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BI-836858 DB17267
biotech | CAS: 2206770-25-2

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Waktu Paruh-
Vol. Distribusi-
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BI-836880 DB17484
biotech

BI-836880 is a humanized bispecific nanobody that targets VEGF and Ang2.

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BI-K0376 DB05858
biotech

BI-K0376 is investigated for use/treatment in acne. BI-K0376 is a solid. It is under investigation by Pfizer and has gone through phase I of the clinical trails.

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Bi104 DB18743
biotech

Bi104 is being investigated for the treatment of Angelman syndrome.

Waktu Paruh-
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Bibenzonium DB13630
small molecule | CAS: 59866-76-1

Deskripsi belum tersedia.

Kategori:
Cough and Cold Preparations
Waktu Paruh-
Vol. Distribusi-
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Bibrocathol DB13818
small molecule | CAS: 6915-57-7

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsBenzene DerivativesOphthalmologicals +2
Waktu Paruh-
Vol. Distribusi-
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Bicalutamide Approved DB01128
small molecule | CAS: 90357-06-5

Bicalutamide is an oral non-steroidal anti-androgen for prostate cancer. It is comprised of a racemic mixture that is a 50:50 composition of the (R)-bicalutamide and (S)-bicalutamide enantionmers. Bicalutamide binds to the androgen receptor.

Kategori:
AmidesAminesAndrogen Receptor Antagonists +31
Target Protein:
Androgen receptor
Waktu Paruh5.9 days
Vol. Distribusi-
Klirens* Apparent oral cl=…
Genetik -
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