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13591

Total database: 17430
Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
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13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 57 / 272
Anisomycin DB07374
small molecule | CAS: 22862-76-6

Anisomycin (sometimes known as flagecidin), is an antibiotic retrieved from the bacteria _Streptomyces griseolus_. This drug acts to inhibit bacterial protein and DNA synthesis.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntiparasitic Agents +5
Target Protein:
Ribosomal protein uL16-likeLarge ribosomal subunit protein uL13Large ribosomal subunit protein uL14 +10
Waktu Paruh-
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Anisotropine methylbromide Approved DB00517
small molecule | CAS: 80-50-2

Anisotropine methylbromide is a quaternary ammonium compound. Its use as treatment adjunct in peptic ulcer has been replaced by the use of more effective agents. Depending on the dose, anisotropine methylbromide may reduce the motility and secretory activity …

Kategori:
Agents producing tachycardiaAlkaloidsAnticholinergic Agents +5
Target Protein:
Muscarinic acetylcholine receptor M5Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2 +1
Waktu ParuhNot Known
Vol. Distribusi-
Klirens-
Genetik -
Anlotinib DB11885
small molecule | CAS: 1058156-90-3

Anlotinib has been investigated for the treatment of Non-small Cell Lung Cancer and Metastatic Colorectal Cancer.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Proto-oncogene tyrosine-protein kinase Src
Waktu Paruh-
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Annamycin DB06420
small molecule | CAS: 92689-49-1

Deskripsi belum tersedia.

Kategori:
AnthracyclinesAntibiotics, AntineoplasticAntineoplastic Agents +4
Target Protein:
DNA topoisomerase 2-alphaDNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anrukinzumab DB12294
biotech | CAS: 910649-32-0

Anrukinzumab has been used in trials studying the diagnostic of Asthma.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
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Anselamimab DB17492
biotech | CAS: 2414866-63-8

Deskripsi belum tersedia.

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Ansofaxine DB15052
small molecule | CAS: 916918-80-4

Ansofaxine is under investigation in clinical trial NCT02271412 (Multiple Ascending Dose Study in Healthy Subjects to Evaluate the Safety, Tolerability, and Pharmacokinetics of LY03005).

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Ansuvimab Approved DB16385
biotech | CAS: 2375952-29-5

Infection with pathogenic filoviruses, such as _Zaire ebolavirus_ (Ebola virus, EBOV), can cause severe hemorrhagic fever in humans, resulting in frequent outbreaks with case fatality rates as high as 90%.[A225933, A225938] Virtually all steps of the EBOV lif…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +13
Target Protein:
Envelope glycoprotein
Waktu ParuhThe half-life of an…
Vol. DistribusiThe steady-state vo…
KlirensThe clearance of an…
Genetik -
Anthoxanthum odoratum Approved DB14163
biotech

Anthoxanthum odoratum allergenic extract is used in allergenic testing.

Kategori:
Allergenic ExtractsNon-Standardized Food Allergenic Extract
Waktu Paruh-
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Anthralin Approved DB11157
small molecule | CAS: 1143-38-0

Anthralin (1,8?dihydroxy?9anthrone, dithranol) is an older anti-psoriatic agent that was first synthesized as a derivative of chrysarobin, obtained from the araroba tree in Brazil over 100 years ago. Adverse effects of anthralin include irritation and discolo…

Kategori:
AnthracenesAntipsoriaticsAntipsoriatics for Topical Use +2
Target Protein:
Keratin, type II cytoskeletal 2 epidermalKeratin, type I cytoskeletal 12C-Jun-amino-terminal kinase-interacting protein 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 118-92-3

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAminobenzoatesBenzene Derivatives +2
Target Protein:
L-amino-acid oxidaseD-amino-acid oxidase
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Anthrax vaccine Approved DB11003
biotech

Anthrax vaccine is a vaccine used for the pre- or post-exposure prophylaxis of disease in those at high risk of, suspected or confirmed exposure to *Bacillus anthracis*. It is subcutaneously or intramuscularly administered. It is derived from cell-free filtra…

Kategori:
Actively Acquired ImmunityAnthrax VaccinesBacterial Vaccines +6
Waktu ParuhLimited information…
Vol. DistribusiLimited information…
KlirensLimited information…
Genetik -
biotech

Anti-GD2 monoclonal antibody 3F8 is under investigation in clinical trial NCT00089258 (Biological Therapy in Treating Patients With Neuroblastoma That Has Not Responded to Previous Treatment).

Waktu Paruh-
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biotech

Anti-inhibitor coagulant complex, also known as FEIBA (factor eight inhibitor bypassing activity), contains several proteins involved in the prothrombinase complex. It is used to control bleeding in hemophilia A and B patients with inhibitors.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +7
Target Protein:
Coagulation factor XProthrombinFibrinogen alpha chain +5
Waktu ParuhPlasma half lives o…
Vol. Distribusi-
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Genetik -
biotech

A macrocyclic peptide (BMS-986189) with activity in binding and functional assays comparable to a PD-L1 antibody.

Kategori:
Immune Checkpoint Inhibitors
Target Protein:
Programmed cell death 1 ligand 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Anti-SARS-CoV-2 equine immunoglobulin fragments, also known as INOSARS, is a polyvalent passive immunization being tested in the clinical trial NCT04514302 (Safety and Efficacy of Anti-SARS-CoV-2 Equine Antibody Fragments (INOSARS) for Hospitalized Patients W…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Anti-SARS-CoV-2 IgY are chicken egg antibodies to SARS-CoV-2 which have the potential to provide temporary protection against the virus when administered as intranasal drops.[L27381] To create these antibodies, chickens are injected in the chest with the spik…

Waktu Paruh-
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biotech

Hyperimmune immunoglobulin to SARS-CoV-2 (hIVIG) is obtained from the plasma of patients who recover from COVID-19 and develop neutralizing antibodies.[L27521] Anti-coronavirus immunoglobulin is derived from [COVID-19 convalescent plasma](https://go.drugbank.…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +8
Waktu Paruh-
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biotech

Anti-SARS-COV-2 REGN-COV2 is a combination of novel antibodies designed by Regeneron for both the prevention and treatment of SARS-COV-2, the virus that causes COVID-19. This drug is a combination of the antibodies REGN10933 and REGN10987, derived from human…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +10
Target Protein:
Spike glycoprotein
Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech | CAS: 1628187-15-4

Antihemophilic Factor (Recombinant), PEGylated, was approved by the FDA in December 2016 as the product _Adynovate_ [FDA label]. Antihemophilic Factor (Recombinant), PEGylated, is a recombinant full-length human coagulation factor VIII (2,332 amino acids w…

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsBiological Factors +14
Target Protein:
von Willebrand factor
Waktu Paruh14.69 ± 3.79h for a…
Vol. DistribusiAt steady state: 0.…
Klirens2.27 ± 0.84 for adu…
Genetik -
Antihemophilic factor human Approved DB13192
biotech

Antihemophilic factor human, also known as Coagulation Factor VIII or Anti-Hemophilic Factor (AHF), is a non-recombinant, lyophilized concentrate of coagulation factor VIII, an endogenous protein and essential component of the coagulation cascade. Antihemophi…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +11
Target Protein:
Coagulation factor IXCoagulation factor X
Waktu ParuhThe mean half-life …
Vol. DistribusiThe pharmacokinetic…
KlirensThe reported cleara…
Genetik -
biotech | CAS: 139076-62-3

Human recombinant antihemophilic factor (AHF) or Factor VIII, 2332 residues, glycosylated, produced by CHO cells

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +12
Target Protein:
Coagulation factor XCoagulation factor IXvon Willebrand factor +8
Waktu Paruh8.4-19.3 hrs
Vol. Distribusi-
Klirens* 4.1 mL/h•kg [Prev…
Genetik -
biotech

Equine anti-thymocyte globulin is composed of purified gamma globulin containing primarily IgG against human thymus lymphocytes. It is formed by inoculating a horse with an antigen (human thymoyctes) which then induces the horse immune system's B-lymphocytes …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibody-Surface Protein Interactions +22
Waktu ParuhThe half-life of eq…
Vol. DistribusiDuring infusion of …
Klirens-
Genetik -
Antimonous acid DB02453
small molecule

Deskripsi belum tersedia.

Target Protein:
Arsenical pump-driving ATPase
Waktu Paruh-
Vol. Distribusi-
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Antimony DB13110
small molecule | CAS: 7440-36-0

Antimony has been used in trials studying the treatment of Cutaneous Leishmaniasis.

Kategori:
ElementsMetalloidsMetals +1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 1315-04-4

Deskripsi belum tersedia.

Kategori:
Air PollutantsAnionsCough and Cold Preparations +9
Waktu Paruh-
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small molecule | CAS: 28300-74-5

Antimony potassium tartrate is a schistosomicide possibly useful against other parasites. It has irritant emetic properties and may cause lethal cardiac toxicity among other adverse effects.

Kategori:
AnthelminticsAnti-Infective AgentsAntiparasitic Agents +2
Waktu Paruh-
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Genetik -
small molecule | CAS: 91531-30-5

Antineoplaston A10 has been used in trials studying the treatment of Sarcoma, Lymphoma, Lung Cancer, Liver Cancer, and Kidney Cancer, among others.

Kategori:
AcetamidesAmidesBenzene Derivatives +1
Waktu Paruh-
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Antipain DB15251
small molecule | CAS: 37691-11-5

Antipain is a serine/cysteine protease inhibitor originally isolated from various strains of actinomycetes.[A214481] Early studies investigated the potential for antipain to alter DNA damage and chromosomal aberrations in irradiated cells or those treated wit…

Kategori:
Amino Acids, Peptides, and ProteinsEnzyme InhibitorsOligopeptides +2
Waktu Paruh-
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Genetik -
Antipyrine Approved DB01435
small molecule | CAS: 60-80-0

An analgesic and antipyretic that has been given by mouth and as ear drops. Antipyrine is often used in testing the effects of other drugs or diseases on drug-metabolizing enzymes in the liver. (From Martindale, The Extra Pharmacopoeia, 30th ed, p29)

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +30
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech | CAS: 1311281-25-0

Antithrombin gamma is under investigation in clinical trial NCT04182373 (KW-3357 Study in Patients With Early Onset Severe Preeclampsia).

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biotech | CAS: 308067-60-9

Rabbit anti-thymocyte globulin. Thymoglobulin is a polyclonal antibody that suppresses certain types of immune cells responsible for acute organ rejection in transplant patients. Thymoglobulin is a mixture of antibodies intended to bind to various cell surfac…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibody-Surface Protein Interactions +22
Target Protein:
Major histocompatibility complex class I-related gene proteinIntegrin alpha-LT-lymphocyte activation antigen CD86 +6
Waktu Paruh2-3 days, may incre…
Vol. Distribusi-
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Genetik -
Antrafenine Approved DB01419
small molecule | CAS: 55300-29-3

Antrafenine is a piperazine derivative drug that acts as an analgesic and anti-inflammatory drug with similar efficacy to naproxen. It is not widely used as it has largely been replaced by newer drugs.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnti-Inflammatory Agents +4
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Antroquinonol DB12326
small molecule | CAS: 1010081-09-0

Antroquinonol has been used in trials studying the treatment of Hyperlipidemias, Non-small Cell Lung Cancer, and Non-small Cell Lung Cancer Stage IV.

Kategori:
BenzoquinonesCoenzymesEnzymes and Coenzymes +1
Target Protein:
DNA (cytosine-5)-methyltransferase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2636710-07-9

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ANX-510 DB05308
small molecule

ANX-510 (CoFactor) is a folate-based biomodulator drug being developed to enhance the activity and reduce associated toxicity of the widely used cancer chemotherapy, 5-fluorouracil (5-FU). CoFactor use with 5-FU is being evaluated in clinical trials in first …

Target Protein:
Thymidylate synthase
Waktu Paruh-
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Anzurstobart DB17547
biotech | CAS: 2543693-10-1

Anzurstobart is a monoclonal antibody directed against signal-regulatory protein alpha (SIRP?) on monocytes and macrophages to potently block the CD47-SIRP? interaction. It is being investigated for cancers.

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AOC 1001 DB18620
biotech | CAS: 2653183-66-3

Delpacibart (AOC 1001) is being investigated in a global study for the treatment of Myotonic Dystrophy type 1 (DM1) in clinical trial NCT06411288

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AOD9604 DB06388
small molecule | CAS: 221231-10-3

AOD9604 is a synthetic analogue of the lipolytic domain of human growth hormone, being investigated for the treatment of obesity.

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +8
Waktu Paruh-
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AP-001 DB18511
small molecule | CAS: 660430-03-5

Deskripsi belum tersedia.

Kategori:
Dietary FatsDietary Fats, UnsaturatedFats +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
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AP-102 DB18206
small molecule | CAS: 846569-60-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +8
Waktu Paruh-
Vol. Distribusi-
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AP-22408 DB01830
small molecule | CAS: 268741-43-1

Deskripsi belum tersedia.

Target Protein:
Proto-oncogene tyrosine-protein kinase SrcTyrosine-protein kinase Lck
Waktu Paruh-
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Genetik -
AP103 DB18234
biotech

AP103 is a non-viral gene therapy that uses a delivery vector, HPAE (Highly Branched Poly ?-Amino Ester), to deliver the correct collagen VII gene into skin cells.

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AP1081 DB05233
small molecule

A transdermal gel containing ethinyl estradiol and norelgestromin being investigated by Antares Pharma for use as a female contraceptive.

Target Protein:
Estrogen receptor
Waktu Paruh-
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AP5346 DB04992
small molecule

AP5346 is designed to target a diaminocyclohexane platinum (Pt) moiety to tumors through pH-sensitive linkage to a 25 kDa hydroxypropylmethacrylamide polymer. It is being pursued by Access Pharmaceuticals, Inc.

Kategori:
Organometallic Compounds
Target Protein:
DNA
Waktu Paruh-
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Genetik -
Apabetalone DB12000
small molecule | CAS: 1044870-39-4

Apabetalone has been investigated for the treatment of Diabetes, Atherosclerosis, and Coronary Artery Disease.

Kategori:
Heterocyclic Compounds, Fused-RingQuinazolines
Waktu Paruh-
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Apadamtase alfa Approved DB15164
biotech | CAS: 2086325-24-6

Thrombotic thrombocytopenic purpura (TTP) is a rare blood clotting disorder characterized by thrombocytopenia, microangiopathic hemolytic anemia, and various degrees of organ damage.[A262076] It may be inherited (congenital TTP; cTTP) or acquired due to autoa…

Kategori:
ADAM ProteinsADAMTS ProteinsAmino Acids, Peptides, and Proteins +12
Target Protein:
von Willebrand factor
Waktu ParuhFollowing the intra…
Vol. Distribusi-
Klirens-
Genetik -
Apadenoson DB05009
small molecule | CAS: 250386-15-3

Apadenoson is a selective A2a adenosine receptor agonist designed for use as a pharmacologic stress agent in cardiac perfusion imaging studies. It is developed by Bristol-Myers Squibb and is in phase II of clinical trials.

Kategori:
Acids, CarbocyclicAdenosine A receptor agonistsAdenosine A2 Receptor Agonists +7
Target Protein:
Adenosine receptor A2a
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apalutamide Approved DB11901
small molecule | CAS: 956104-40-8

Apalutamide is a potent androgen receptor (AR) antagonist that selectively binds to the ligand-binding domain of AR and blocks AR nuclear translocation or binding to androgen response elements [A31846]. It has been used in trials studying the treatment of Pro…

Kategori:
Androgen Receptor InhibitorsAntiandrogensAntineoplastic Agents +28
Target Protein:
Androgen receptorGABA(A) Receptor
Waktu ParuhThe mean effective …
Vol. DistribusiThe mean apparent v…
KlirensThe CL/F of apaluta…
Genetik -
biotech | CAS: 2097132-02-8

Deskripsi belum tersedia.

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