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6694

Total database: 17430
Struktur (SMILES)
4518 (67.5%)
Target
3751 (56.0%)
Genomik
81 (1.2%)
Referensi
6694 (100.0%)

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Hasil Pencarian (6694)

Halaman 56 / 134
small molecule | CAS: 54063-42-2

Deskripsi belum tersedia.

Kategori:
Diagnostic RadiopharmaceuticalsVarious Diagnostic Radiopharmaceuticals
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Ferric ammonium citrate Approved DB09501
small molecule | CAS: 1185-57-5

Deskripsi belum tersedia.

Kategori:
AminesAmmonium CompoundsContrast Media +5
Waktu Paruh-
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Genetik -
Ferric cation Approved DB13949
small molecule | CAS: 20074-52-6

Iron is a transition metal with a symbol Fe and atomic number 26. By mass, it is the most common element on Earth. Iron is an essential element involved in various metabolic processes, including oxygen transport, deoxyribonucleic acid (DNA) synthesis, and ene…

Kategori:
Iron CompoundsParenteral Iron ReplacementPhosphate Binder +2
Target Protein:
Transferrin receptor protein 1Iron(3+)-hydroxamate-binding protein FhuD
Waktu ParuhThe pharmacokinetic…
Vol. DistribusiLess than 65% of ir…
KlirensThe rate of iron lo…
Genetik -
Ferric derisomaltose Approved DB15617
small molecule | CAS: 1345510-43-1

Iron deficiency is an extremely common condition and is the most frequent cause of anemia worldwide. Iron deficiency results when iron intake, iron stores, and loss of iron from the body do not adequately support production of erythrocytes, also known as red …

Kategori:
Anemia, Iron-DeficiencyAntianemia DrugsAntianemic Preparations +6
Target Protein:
Hemoglobin subunit alphaTransferrin receptor
Waktu ParuhThe plasma-half liv…
Vol. DistribusiFerric derisomaltos…
KlirensIntravenous iron is…
Genetik -
Ferric maltol Approved DB15598
small molecule | CAS: 33725-54-1

Ferric maltol is an iron(III) atom complexed with 3 maltol molecules to increase the bioavailability compared to iron(II), without depositing it in the duodenum as insoluble ferric hydroxide and phosphate.[A189288] Ferric maltol has been described in literatu…

Kategori:
Antianemic PreparationsBlood and Blood Forming OrgansHematinics +8
Target Protein:
Integrin beta-3Natural resistance-associated macrophage protein 2
Waktu ParuhMaltol has a half l…
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik -
Ferric pyrophosphate citrate Approved DB13995
small molecule | CAS: 1802359-96-1

Ferric pyrophosphate citrate is a soluble iron replacement product. Free iron presents several side effects as it can catalyze free radical formation and lipid peroxidation as well as the presence of interactions of iron in plasma. The ferric ion is strongly …

Kategori:
EnzymesEnzymes and CoenzymesHydrolases +3
Target Protein:
Ferritin light chainFerritin heavy chainHemoglobin subunit alpha +1
Waktu ParuhThe half-life of fe…
Vol. DistribusiThe apparent volume…
KlirensThe mean clearance …
Genetik -
small molecule | CAS: 52031-09-1

Deskripsi belum tersedia.

Kategori:
Antianemic PreparationsBlood and Blood Forming OrgansIron Preparations +1
Waktu Paruh-
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Ferric subsulfate Approved DB13885
small molecule | CAS: 1310-45-8

Ferric subsulfate is a stypic or hemostatic agent that causes agglutination of surface proteins resulting in local hemostasis. It has the chemical formula Fe4(OH)2(SO4)5. It is used after superficial skin biopsies.

Kategori:
AnionsCoagulantsElectrolytes +7
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Ferric sulfate Approved DB11171
small molecule | CAS: 10028-22-5

Ferric sulfate has the molecular formula of Fe2SO4, and it is a dark brown or yellow chemical agent with acidic properties. It is produced by the reaction of sulfuric acid and an oxidizing agent. It is used in different fields such as dermatology, dentistry a…

Kategori:
HematinicsIron Compounds
Waktu ParuhPharmacokinetic stu…
Vol. DistribusiPharmacokinetic stu…
KlirensPharmacokinetic stu…
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Ferrichrome-iron receptor
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Ferrous ascorbate Approved DB14490
small molecule | CAS: 24808-52-4

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAntianemic PreparationsAntioxidants +15
Target Protein:
Transferrin receptor protein 1Egl nine homolog 1Histone deacetylase 8 +10
Waktu Paruh-
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Ferrous asparto glycinate Approved DB11169
small molecule

Ferrous asparto glycinate is an iron-amino acid chelate. It is available as a dietary supplement used in the treatment of iron deficiency and iron deficiency anemia.

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Ferrous bisglycinate Approved DB11210
small molecule | CAS: 20150-34-9

Ferrous bisglycinate is a chelate that is used as a source of dietary iron. Forming a ring structure when reacting with glycine, ferrous bisglycinate acts as both a chelate and a nutritionally functional [A27250]. It is found in foods for food enrichment or i…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsIron Compounds
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Ferrous cysteine glycinate Approved DB11197
small molecule

Deskripsi belum tersedia.

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Ferrous fumarate Approved DB14491
small molecule | CAS: 141-01-5

Used in treatment of iron deficiency anemia.

Kategori:
Antianemic PreparationsBlood and Blood Forming OrgansDiet, Food, and Nutrition +9
Target Protein:
Transferrin receptor protein 1Egl nine homolog 1Histone deacetylase 8 +10
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Ferrous gluconate Approved DB14488
small molecule | CAS: 299-29-6

Deskripsi belum tersedia.

Kategori:
Anemia, Iron-DeficiencyAntianemia DrugsAntianemic Preparations +8
Target Protein:
Transferrin receptor protein 1Egl nine homolog 1Histone deacetylase 8 +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ferrous glycine sulfate Approved DB14501
small molecule | CAS: 14729-84-1

Deskripsi belum tersedia.

Kategori:
Antianemic PreparationsBlood and Blood Forming OrgansIron Bivalent, Oral Preparations +1
Target Protein:
Transferrin receptor protein 1Egl nine homolog 1Histone deacetylase 8 +10
Waktu Paruh-
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Genetik -
Ferrous succinate Approved DB14489
small molecule | CAS: 10030-90-7

Deskripsi belum tersedia.

Kategori:
Antianemic PreparationsBlood and Blood Forming OrgansHematinics +4
Target Protein:
Transferrin receptor protein 1Egl nine homolog 1Histone deacetylase 8 +10
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Ferrous sulfate anhydrous Approved DB13257
small molecule | CAS: 7720-78-7

Iron deficiency anemia is a large public health concern worldwide, especially in young children, infants, and women of childbearing age.[A190804] This type of anemia occurs when iron intake, iron stores, and iron loss do not adequately support the formation o…

Kategori:
Anemia, Iron-DeficiencyDelayed-Action PreparationsHematinics +6
Target Protein:
Hemoglobin subunit alphaTransferrin receptor
Waktu ParuhThe half-life of or…
Vol. DistribusiAbout 60% of iron i…
Klirens-
Genetik -
Ferulic acid DB07767
small molecule | CAS: 1135-24-6

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAnalgesicsAnalgesics, Non-Narcotic +17
Target Protein:
Carbonic anhydrase 12Carbonic anhydrase 2Carbonic anhydrase 14 +9
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Ferumoxytol Approved DB06215
small molecule | CAS: 722492-56-0

Ferumoxytol is an intravenously administered iron preparation indicated in the EU and the US for the treatment of iron deficiency anemia in adult patients with chronic kidney disease (CKD) [A32478]. It is comprised of superparamagnetic iron oxide nanoparti…

Kategori:
Compounds used in a research, industrial, or household settingFerric CompoundsFerrous Compounds +11
Waktu ParuhThe pharmacokinetic…
Vol. DistribusiThe population mean…
KlirensSince there is no r…
Genetik -
Fexinidazole Approved DB12265
small molecule | CAS: 59729-37-2

Human African trypanosomiasis (HAT, also colloquially referred to as sleeping sickness), caused by _T. brucei gambiense_ and _T. brucei rhodesiense_, remains a moderate risk (>1/10,000 inhabitants per year in endemic areas) despite focussed control efforts. T…

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAntiparasitic Products, Insecticides and RepellentsAntiprotozoals +43
Waktu ParuhFexinidazole, M1, a…
Vol. DistribusiFexinidazole has an…
KlirensFexinidazole has a …
Genetik -
Fexofenadine Approved DB00950
small molecule | CAS: 83799-24-0

Fexofenadine is an over-the-counter second-generation antihistamine used in the treatment of various allergic symptoms.[L4269] It is selective for the H<sub>1</sub> receptor, carries little-to-no activity at off-targets, and does not cross the blood-brain bar…

Kategori:
Anti-Allergic AgentsAntihistamines for Systemic UseBenzene Derivatives +12
Target Protein:
Histamine H1 receptor
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe volume of distr…
KlirensThe oral clearance …
Genetik -
FF-10501-01 DB17554
small molecule

FF-10501-01 is a novel, selective inosine monophosphate dehydrogenase (IMPDH) inhibitor with anticancer activity.[A257306] FF-10501-01 is under investigation in clinical trial NCT03486353 (A Study of FF-10501-01 in Combination With Azacitidine in Patients Wit…

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FG-2216 DB08687
small molecule | CAS: 223387-75-5

A orally active prolyl-hydroxylase inhibitor which can stabilize hypoxia-inducible transcription factor independent of oxygen availability. [A14422]

Target Protein:
Egl nine homolog 1Hypoxia-inducible factor 1-alpha
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Genetik -
Fiacitabine DB12901
small molecule | CAS: 69123-90-6

Fiacitabine has been used in trials studying the treatment of HIV Infections and Cytomegalovirus Infections.

Kategori:
Anti-Infective AgentsAntineoplastic AgentsAntiviral Agents +5
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Fianlimab DB18858
biotech | CAS: 2126132-98-5

Fianlimab is under investigation in clinical trial NCT06190951 (A Trial to Learn if Fianlimab and Cemiplimab Are Safe and Work Better Than Anti-pd1 Alone in Adult Participants With Resectable Stage 3 or 4 Melanoma).

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Fibrinogen human Approved DB09222
biotech | CAS: 9001-32-5

Fibrinogen concentrate (human) is a hematological agent. It works by replacing a specific protein in the blood, fibrinogen (factor I), that helps with blood clotting. It is a soluble plasma glycoprotein with a molecular weight of about 340 kDa and is a physi…

Kategori:
Acute-Phase ProteinsAmino Acids, Peptides, and ProteinsBiological Factors +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 106096-92-8

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsFibroblast Growth Factor 1 +4
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Genetik -
Fidanacogene elaparvovec Approved DB16783
biotech | CAS: 1954659-47-2

Fidanacogene elaparvovec is a liver-specific adeno-associated virus (AAV) vector containing a codon-optimized human coagulation FIX gene that was investigated as a potential treatment for hemophilia B.[L46691] Hemophilia B is a rare X-linked genetic disorder …

Kategori:
Adeno-associated Viral Vector TherapiesHepatotoxic Agents
Target Protein:
Coagulation factor IX (F9)
Waktu Paruh-
Vol. DistribusiIn a monkey biodist…
KlirensClearance of vector…
Genetik -
Fidaxomicin Approved DB08874
small molecule | CAS: 873857-62-6

Fidaxomicin is a novel macrolide antibiotic used in the treatment of diarrhea caused by _Clostridioides_ (formerly _Clostridium_) _difficile_ in adult and pediatric patients over the age of 6 months.[L11575] Fidaxomicin is a naturally-occurring 18-member macr…

Kategori:
Alimentary Tract and MetabolismAnti-Bacterial AgentsAnti-Infective Agents +13
Target Protein:
RNA polymerase sigma factor SigA
Waktu ParuhFollowing oral admi…
Vol. DistribusiFidaxomicin is main…
KlirensThere is limited in…
Genetik -
Fidrisertib DB18064
small molecule | CAS: 2141955-96-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Filgotinib Approved DB14845
small molecule | CAS: 1206161-97-8

Rheumatoid arthritis (RA) is a chronic, autoimmune, systemic, and inflammatory disease that causes synovial joint symptoms and can limit range of motion in severe cases.[A221451,A221456] The disease is associated with extra-articular manifestations, progressi…

Kategori:
Antineoplastic and Immunomodulating AgentsArthritis, Rheumatoid, drug therapyImmunosuppressive Agents +5
Target Protein:
Tyrosine-protein kinase JAK1
Waktu ParuhThe half-life of fi…
Vol. Distribusi-
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Genetik -
Filgrastim Approved DB00099
biotech | CAS: 121181-53-1

Filgrastim is a short-acting recombinant, non-pegylated human granulocyte colony-stimulating factor (G-CSF) analog produced by recombinant DNA technology. It has an amino acid sequence identical to endogenous G-CSF, but it is non-glycosylated unlike the endog…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating AgentsBiological Factors +10
Target Protein:
Granulocyte colony-stimulating factor receptor
Waktu ParuhAfter intravenous a…
Vol. DistribusiAfter intravenous a…
KlirensClearance rates of …
Genetik -
Filociclovir DB12438
small molecule | CAS: 632325-71-4

Filociclovir is under investigation in clinical trial NCT01433835 (Safety and Pharmacokinetics of Single Oral Doses of Filociclovir in Healthy Volunteers).

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Genetik -
Fimaporfin DB17253
small molecule | CAS: 1443547-43-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Fimepinostat DB11891
small molecule | CAS: 1339928-25-4

Fimepinostat (CUDC-907) has been used in trials studying the treatment of lymphoma, solid tumors, breast cancer, multiple myeloma, and NUT midline carcinoma, among others.

Kategori:
Antineoplastic AgentsHistone Deacetylase InhibitorsOxazines +3
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Finafloxacin Approved DB09047
small molecule | CAS: 209342-40-5

Finafloxacin is a fluoroquinolone antibiotic indicated in the treatment of acute otitis externa (swimmer's ear) caused by the bacteria Pseudomonas aeruginosa and Staphylococcus aureus. Finafloxacin is marketed by Novartis under the brand Xtoro™, and was appro…

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Finasteride Approved DB01216
small molecule | CAS: 98319-26-7

Finasteride is a synthetic 4-azasteroid compound [L10565] and specific inhibitor of steroid Type II 5?-reductase, which is an intracellular enzyme that converts the androgen testosterone into 5?-dihydrotestosterone (DHT). It works in a similar fashion as [dut…

Kategori:
5-alpha Reductase InhibitorsAdrenergic alpha-AntagonistsAdrenergic Antagonists +22
Target Protein:
3-oxo-5-alpha-steroid 4-dehydrogenase 2Polyprenal reductase3-oxo-5-alpha-steroid 4-dehydrogenase 1 +1
Waktu ParuhIn healthy young su…
Vol. DistribusiThe volume of distr…
KlirensIn healthy young su…
Genetik -
Finerenone Approved DB16165
small molecule | CAS: 1050477-31-0

Finerenone, or BAY 94-8862, is a mineralocorticoid receptor antagonist indicated to reduce the risk of sustained decline in glomerular filtration rate, end stage kidney disease, cardiovascular death, heart attacks, and hospitalization due to heart failure in …

Kategori:
Agents causing hyperkalemiaCytochrome P-450 CYP2C8 SubstratesCytochrome P-450 CYP3A Substrates +6
Target Protein:
Mineralocorticoid receptor
Waktu ParuhThe half life of a …
Vol. DistribusiThe volume of distr…
KlirensThe systemic cleara…
Genetik -
FINLAY-FR-1 DB16524
biotech

FINLAY-FR-1, also known as Soberana 01, is a vaccine candidate for COVID-19 that is being led developmentally by the Finlay Vaccine Institute[L31373]. It is currently being tested in the clinical trial RPCEC00000332 (Phase I / II, randomized, controlled, adap…

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Genetik -
Finotonlimab DB18859
biotech | CAS: 2350298-85-8

Finotonlimab is under investigation in clinical trial NCT04560894 (SCT-I10A Plus SCT510 Versus Sorafenib as First-line Therapy for Advanced Hepatocellular Carcinoma).

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Fipaxalparant DB18124
small molecule | CAS: 1195941-38-8

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Target Protein:
Lysophosphatidic acid receptor 1Lysophosphatidic acid receptor 3
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Vol. Distribusi-
Klirens-
Genetik -
Firocoxib DB09217
small molecule | CAS: 189954-96-9

Firocoxib is a cycooxygenase-2 (COX-2) selective non-steroidal anti-inflammatory drug. It currently approved for veterinary use in dogs and horses under the brand names Equioxx and Previcox. Firocoxib was the first COX-2 inhibitor approved by the U.S. Food an…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnti-Inflammatory Agents +6
Target Protein:
Prostaglandin G/H synthase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

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Firsocostat DB16166
small molecule | CAS: 1434635-54-7

Firsocostat is under investigation in clinical trial NCT02781584 (Safety, Tolerability, and Efficacy of Selonsertib, Firsocostat, and Cilofexor in Adults With Nonalcoholic Steatohepatitis (NASH)).

Kategori:
Acids, AcyclicButyratesEnzyme Inhibitors +5
Waktu Paruh-
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Genetik -
Fish oil Approved DB13961
biotech

Fish oil is a component of SMOFLIPID, which was FDA approved in July 2016. It is indicated in adults as a source of calories and essential fatty acids for parenteral nutrition when oral or enteral nutrition is not possible, insufficient, or contraindicated. …

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsBradycardia-Causing Agents +8
Target Protein:
Diacylglycerol O-acyltransferase 2Prostaglandin G/H synthase 2Free fatty acid receptor 4 +8
Waktu ParuhThe half-life of EP…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of EP…
Genetik -
Fisogatinib DB16167
small molecule | CAS: 1707289-21-1

Fisogatinib is under investigation in clinical trial NCT04194801 (A Phase Ib/ii Study of Fisogatinib(blu-554) in Subjects With Hepatocellular Carcinoma).

Kategori:
Antineoplastic AgentsHeterocyclic Compounds, Fused-Ring
Target Protein:
Fibroblast growth factor receptor 4
Waktu Paruh-
Vol. Distribusi-
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Genetik -
FK352B DB06484
small molecule | CAS: 143881-08-7

FK352B is a adenosine A1 antagonist that is developed for the treatment of dialysis-induced hypotension.

Target Protein:
Adenosine receptor A1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Flavin adenine dinucleotide Approved DB03147
small molecule | CAS: 146-14-5

A condensation product of riboflavin and adenosine diphosphate. The coenzyme of various aerobic dehydrogenases, e.g., D-amino acid oxidase and L-amino acid oxidase. (Lehninger, Principles of Biochemistry, 1982, p972) Flavin adenine dinucleotide is approved f…

Kategori:
Adenine NucleotidesBiological FactorsCoenzymes +13
Target Protein:
Ribosyldihydronicotinamide dehydrogenase [quinone]Nitric oxide synthase 1Dihydropyrimidine dehydrogenase [NADP(+)] +83
Waktu Paruh-
Vol. Distribusi-
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Genetik -
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