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3253

Total database: 17430
Struktur (SMILES)
2451 (75.3%)
Target
1833 (56.3%)
Genomik
35 (1.1%)
Referensi
3253 (100.0%)

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Hasil Pencarian (3253)

Halaman 56 / 66
Sivelestat DB12863
small molecule | CAS: 127373-66-4

Sivelestat has been used in trials studying the treatment of Acute Lung Injury and Respiratory Distress Syndrome, Adult.

Kategori:
AmidesAmino AcidsAmino Acids, Peptides, and Proteins +5
Target Protein:
Neutrophil elastaseChymotrypsin-like elastase family member 1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Sizofiran DB13128
small molecule | CAS: 9050-67-3

A beta-D-glucan obtained from the Aphyllophoral fungus Schizophyllum commune. It is used as an immunoadjuvant in the treatment of neoplasms, especially tumors found in the stomach. Sizofiran has been used in trials studying the treatment of Cervical Cancer.

Kategori:
Adjuvants, ImmunologicAntineoplastic AgentsAntineoplastic Agents, Phytogenic +6
Waktu Paruh-
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Genetik -
SJ-733 DB12659
small molecule | CAS: 1424799-20-1

SJ-733 has been used in trials studying Malaria.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
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SLN124 DB18646
biotech

SLN124 is a synthetic double-stranded siRNA oligonucleotide directed against TMPRSS6 mRNA and covalently linked to a ligand containing 3 N-acetylgalactosamine residues.

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SM-337 DB17112
small molecule | CAS: 1071992-61-4

Deskripsi belum tersedia.

Target Protein:
E3 ubiquitin-protein ligase XIAP
Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

The New York City Board of Health strain of _Vaccinia_ is a viral strain used as a component of some smallpox vaccinations.[L12747] ACAM2000, a percutaneously administered smallpox vaccine that was approved by the FDA in 2007, contains live antigens of this s…

Kategori:
Actively Acquired ImmunityBiological ProductsComplex Mixtures +4
Waktu Paruh-
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Genetik -
Smilagenin DB05450
small molecule | CAS: 126-18-1

Smilagenin is a novel non-peptide, orally bioavailable neurotrophic factor inducer that readily reverses free radical neurotoxicity produced by 1-ethyl-4- phenylpyridium (MPP+) in dopaminergic neurones and reverses the decrease of neuronal growth factors and …

Kategori:
CholestanesDrugs, Chinese HerbalFused-Ring Compounds +4
Waktu Paruh-
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SN-38 DB05482
small molecule | CAS: 86639-52-3

7-ethyl-10-hydroxycamptothecin (SN 38) is a liposomal formulation of the active metabolite of Irinotecan [DB00762], a chemotherapeutic pro-drug approved for the treatment of advanced colorectal cancer. SN 38 has been used in trials studying the treatment of …

Kategori:
AlkaloidsAntineoplastic AgentsCytochrome P-450 CYP3A Inhibitors +9
Target Protein:
DNA topoisomerase 1
Waktu Paruh-
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Genetik -
small molecule | CAS: 1226795-18-1

Snubh-nm-333 F-18 is under investigation in clinical trial NCT02149017 (Phase 1 and Phase 2 Clinical Trials of SNUBH-NM-333(18F)).

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SNX-2112 DB17055
small molecule | CAS: 908112-43-6

SNX-2112 is a heat shock protein 90 (Hsp90) inhibitor.[A253137]

Kategori:
Heterocyclic Compounds, Fused-RingHSP90 Heat-Shock Proteins, antagonists & inhibitors
Target Protein:
Heat shock protein HSP 90-alpha
Waktu Paruh-
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Soblidotin DB12677
small molecule | CAS: 149606-27-9

Soblidotin has been used in trials studying the treatment of Sarcoma, Lung Cancer, and Unspecified Adult Solid Tumor, Protocol Specific.

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsPeptides
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Sodium acetate Approved DB09395
small molecule | CAS: 127-09-3

Sodium Acetate is chemically designated CH3COONa, a hygroscopic powder very soluble in water. Sodium acetate could be used as additives in food, industry, concrete manufacture, heating pads and in buffer solutions. Medically, sodium acetate is important compo…

Kategori:
AcetatesAcids, AcyclicBlood and Blood Forming Organs +5
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Sodium aurothiomalate Approved DB09276
small molecule | CAS: 12244-57-4

Sodium aurothiomalate is a gold compound that is used for its immunosuppressive anti-rheumatic effects. Gold Sodium Thiomalate is supplied as a solution for intramuscular injection containing 50 mg of Gold Sodium Thiomalate per mL. It is most effective in act…

Kategori:
Acids, AcyclicAntiinflammatory and Antirheumatic ProductsAntirheumatic Agents +13
Waktu Paruh12.5 days
Vol. DistribusiThe apparent volume…
Klirens7.0 ml/ kg/day
Genetik -
small molecule | CAS: 17141-74-1

Sodium zirconium cyclosilicate is approved as the trade product Lokelma developed by AstraZeneca - an insoluble, non-absorbed sodium zirconium silicate, formulated as a powder for oral suspension that acts as a highly selective potassium removing agent.[L2933…

Kategori:
AcidsAcids, NoncarboxylicAnions +13
Target Protein:
Potassium
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Sofinicline DB12527
small molecule | CAS: 799279-80-4

Sofinicline has been used in trials studying the treatment of ADHD, Neuralgia, Diabetic, Diabetic Neuropathies, Diabetic Polyneuropathy, and Diabetic Neuropathic Pain, among others.

Kategori:
Aza Compounds
Target Protein:
Neuronal acetylcholine receptor subunit alpha-4Neuronal acetylcholine receptor subunit beta-2
Waktu Paruh-
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Sofosbuvir Approved DB08934
small molecule | CAS: 1190307-88-0

Sofosbuvir (tradename Sovaldi) is a direct acting antiviral medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is c…

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +18
Target Protein:
Genome polyproteinRNA-dependent RNA-polymerase
Waktu ParuhSofosbuvir has a te…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of so…
Genetik -
Solamargine DB12700
small molecule | CAS: 20311-51-7

Solamargine has been used in trials studying the treatment of Actinic Keratosis.

Kategori:
Alkaloids
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Solasodine DB18813
small molecule | CAS: 126-17-0

Deskripsi belum tersedia.

Kategori:
Alkaloids
Waktu Paruh-
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Solasonine DB17103
small molecule | CAS: 19121-58-5

Deskripsi belum tersedia.

Kategori:
AlkaloidsStereoisomerism
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Solnatide DB12136
biotech | CAS: 259206-53-6

Solnatide has been used in trials studying the treatment of Acute Lung Injury.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
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Somapacitan Approved DB15093
biotech | CAS: 1338578-34-9

Somapacitan, also known as NNC0195-0092,[A219136] is a growth hormone analog indicated to treat adults with growth hormone deficiency.[A219126,L15661] This human growth hormone analog differs by the creation of an albumin binding site, and prolonging the effe…

Kategori:
AlcoholsAmino AcidsAmino Acids, Cyclic +25
Target Protein:
Growth hormone receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe approximate vol…
KlirensThe apparent maximu…
Genetik -
Somatorelin DB12656
biotech | CAS: 83930-13-6

Somatorelin has been used in trials studying the treatment of Aging, Elderly, Sleep Disorders, Hormone Deficiency, and Mild Cognitive Impairment.

Kategori:
Amino Acids, Peptides, and ProteinsDiagnostic AgentsGrowth Hormone-Releasing Hormone, agonists +10
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Genetik -
Somatotropin Approved DB00052
biotech | CAS: 12629-01-5

Human growth hormone (HGH), also known as somatotropin, is a peptide hormone that is synthesized and secreted by the somatotropic cells of the anterior pituitary gland.[A228183] Growth hormone plays an essential role in growth regulation during childhood as w…

Kategori:
Agents Causing Muscle ToxicityAmino Acids, Peptides, and ProteinsAnterior Pituitary Lobe Hormones and Analogues +23
Target Protein:
Growth hormone receptorProlactin receptor
Waktu ParuhWhen somatotropin w…
Vol. DistribusiInformation is unav…
KlirensFollowing intraveno…
Genetik -
biotech | CAS: 1088845-67-3

Somatropin pegol is under investigation in clinical trial NCT00715689 (Dose Study in Growth Hormone Deficient Adults Investigating Safety, Pharmacokinetics and Pharmacodynamics of NNC126-0083).

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsEthylene Glycols +10
Waktu Paruh-
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Somavaratan DB12421
biotech | CAS: 1448335-08-7

Somavaratan has been used in trials studying the treatment of Growth Disorders and Adult Growth Hormone Deficiency.

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Sonedenoson DB12443
small molecule | CAS: 131865-88-8

Sonedenoson has been used in trials studying the treatment of Foot Ulcer, Diabetic and Diabetes Complications.

Kategori:
Heterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and NucleosidesNucleosides +3
Target Protein:
Adenosine receptor A2a
Waktu Paruh-
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Genetik -
Sonolisib DB12601
small molecule | CAS: 502632-66-8

Sonolisib has been used in trials studying the treatment of Glioblastoma, Prostate Cancer, Advanced Solid Tumors, Advanced BRAF-mutant Cancers, and Non Small Cell Lung Cancer (NSCLC), among others.

Kategori:
Fused-Ring CompoundsSteroids
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Waktu Paruh-
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Genetik -
Soraphen A DB02859
small molecule | CAS: 122547-72-2

Deskripsi belum tersedia.

Kategori:
LactonesPolyketides
Target Protein:
Acetyl-CoA carboxylase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sorbinil DB02712
small molecule | CAS: 68367-52-2

Deskripsi belum tersedia.

Kategori:
Aldehyde Reductase, antagonists & inhibitorsImidazoles
Target Protein:
Aldo-keto reductase family 1 member B1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sorbitan DB14474
small molecule | CAS: 12441-09-7

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
Sorbitol Approved DB01638
small molecule | CAS: 50-70-4

A polyhydric alcohol with about half the sweetness of sucrose. Sorbitol occurs naturally and is also produced synthetically from glucose. It was formerly used as a diuretic and may still be used as a laxative and in irrigating solutions for some surgical proc…

Kategori:
AlcoholsAlimentary Tract and MetabolismBlood and Blood Forming Organs +22
Waktu Paruh-
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Genetik -
Sotagliflozin Approved DB12713
small molecule | CAS: 1018899-04-1

Sotagliflozin is a dual inhibitor of SGLT1 and SGLT2, the first of its kind,[A244499] which is approved for use in the EU, in combination with insulin, to improve glycemic control in patients with type 1 diabetes mellitus (T1DM) and a BMI ?27 kg/m<sup>2</sup>…

Kategori:
Alimentary Tract and MetabolismBCRP/ABCG2 InhibitorsBlood Glucose Lowering Agents +24
Target Protein:
Sodium/glucose cotransporter 2Sodium/glucose cotransporter 1
Waktu ParuhThe mean terminal h…
Vol. DistribusiSotagliflozin has a…
KlirensIn healthy voluntee…
Genetik -
Sotatercept Approved DB12118
biotech | CAS: 1001080-50-7

Sotatercept is an activin signalling inhibitor. It is a homodimeric recombinant fusion protein consisting of the extracellular domain of the human activin receptor type IIA (ActRIIA) linked to the human IgG1 Fc domain.[L50351] On March 26, 2024, sotatercep…

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsImmunoglobulin G +5
Target Protein:
Activin receptor type-2AActivin receptor type-1BGrowth/differentiation factor 8 +1
Waktu ParuhThe effective half-…
Vol. DistribusiThe population PK m…
KlirensClearance is approx…
Genetik -
Sotevtamab DB19120
biotech | CAS: 2411526-47-9

Sotevtamab is under investigation in clinical trial NCT06225843 (Sotevtamab (AB-16B5) Combined With FOLFOX as Neoadjuvant Treatment Prior to Resection of Colorectal Cancer Liver Metastasis).

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Sotigalimab DB16413
biotech | CAS: 2305607-45-6

Sotigalimab is under investigation in clinical trial NCT03123783 (CD40 Agonistic Antibody APX005M in Combination With Nivolumab).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
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Klirens-
Genetik -
Sotorasib Approved DB15569
small molecule | CAS: 2252403-56-6

Sotorasib, also known as AMG-510, is an acrylamide-derived KRAS inhibitor developed by Amgen.[A187547,A187556] It is indicated in the treatment of adult patients with KRAS G12C mutant non-small cell lung cancer.[L34288] This mutation makes up >50% of all KRAS…

Kategori:
Antineoplastic AgentsAntineoplastic Agents, ImmunologicalAntineoplastic and Immunomodulating Agents +13
Target Protein:
GTPase KRas
Waktu ParuhSotorasib has a ter…
Vol. DistribusiThe volume of distr…
KlirensSotorasib has an ap…
Genetik -
Sotrastaurin DB12369
small molecule | CAS: 425637-18-9

Sotrastaurin has been used in trials studying the basic science and treatment of Uveal Melanoma, Richter Syndrome, Prolymphocytic Leukemia, Recurrent Mantle Cell Lymphoma, and Recurrent Small Lymphocytic Lymphoma, among others.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Protein kinase C theta typeProtein kinase C beta typeProtein kinase C alpha type
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sovaprevir DB12069
small molecule | CAS: 1001667-23-7

Sovaprevir has been investigated for the treatment of Hepatitis C, Chronic.

Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sovesudil DB18812
small molecule | CAS: 1333400-14-8

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicBenzene Derivatives
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Soy sterol DB11325
biotech | CAS: 129311-52-0

Deskripsi belum tersedia.

Kategori:
Biological FactorsCholestanesFused-Ring Compounds +5
Waktu Paruh-
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SP1049C DB04978
small molecule

SP1049C is a novel anthracycline chemotherapeutic agent containing [doxorubicin] and two nonionic pluronic block copolymers.[A260416] It is designed to overcome drug resistance in a number of cancers. It has successfully completed Phase 1 trials. Phase 2 resu…

Kategori:
AlcoholsAnthracyclinesCarbohydrates +8
Target Protein:
DNA topoisomerase 2-alpha
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Sparfloxacin Approved DB01208
small molecule | CAS: 110871-86-8

Sparfloxacin is a fluoroquinolone antibiotic indicated for bacterial infections. Sparfloxacin exerts its antibacterial activity by inhibiting DNA gyrase, a bacterial topoisomerase. DNA gyrase is an essential enzyme which controls DNA topology and assists in D…

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +16
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +2
Waktu ParuhMean terminal elimi…
Vol. Distribusi-
Klirens-
Genetik -
Sparsentan Approved DB12548
small molecule | CAS: 254740-64-2

Sparsentan is a dual antagonist of the endothelin type A receptor (ET<sub>A</sub>R) and the angiotensin II (Ang II) type 1 receptor (AT<sub>1</sub>R) with a similar affinity for both (9.3 nM for ET<sub>A</sub>R and 0.8 nM for AT<sub>1</sub>R).[A257330,L45300]…

Kategori:
Agents Acting on the Renin-Angiotensin SystemAmidesAngiotensin 2 Receptor Blocker +30
Target Protein:
Endothelin-1 receptorType-1 angiotensin II receptorType-2 angiotensin II receptor
Waktu ParuhSparsentan has an e…
Vol. DistribusiAt the approved rec…
KlirensSparsentan has a ti…
Genetik -
Spebrutinib DB11764
small molecule | CAS: 1202757-89-8

Spebrutinib has been used in trials studying the treatment of Rheumatoid Arthritis, Lymphoma, Large B-Cell, Diffuse, and Leukemia Lymphocytic Chronic B-Cell.

Kategori:
Acids, AcyclicAcrylatesAmides +2
Target Protein:
Tyrosine-protein kinase BTK
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Spermidine DB03566
small molecule | CAS: 124-20-9

Spermidine is a polyamine formed from putrescine. It is found in almost all tissues in association with nucleic acids. It is found as a cation at all pH values, and is thought to help stabilize some membranes and nucleic acid structures. It is a precursor of …

Kategori:
AminesBiogenic AminesBiogenic Polyamines +2
Target Protein:
Thioredoxin reductase 1, cytoplasmicBeta-1 adrenergic receptorBeta-2 adrenergic receptor +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Spermine DB00127
small molecule | CAS: 71-44-3

Spermine is a spermidine-derived biogenic polyamine found as a polycation at all pH values. Found in various tissues and organisms, it often acts as an essential growth factor in some bacterial species. Spermine is associated with nucleic acids, particularly …

Kategori:
AminesBiogenic AminesBiogenic Polyamines +4
Target Protein:
Spermine synthaseCarbonic anhydrase 4Glutamate receptor ionotropic, NMDA 1 +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SPH-3127 DB19108
small molecule | CAS: 1399849-02-5

SPH-3127 is under investigation in clinical trial NCT05359068 (Study to Evaluate the Efficacy and Safety of SPH3127 in Patients With Mild-moderate Essential Hypertension).

Kategori:
Oxazines
Waktu Paruh-
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Sphingosine DB03203
small molecule | CAS: 123-78-4

An amino alcohol with a long unsaturated hydrocarbon chain. Sphingosine and its derivative sphinganine are the major bases of the sphingolipids in mammals. (Dorland, 28th ed)

Kategori:
AlcoholsAminesAmino Alcohols +2
Target Protein:
Choline-phosphate cytidylyltransferase BGenome polyproteinGenome polyprotein +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Spiradoline DB12704
small molecule | CAS: 87151-85-7

Spiradoline has been investigated for the basic science of Bipolar Depression.

Kategori:
AnalgesicsAntiarrhythmic agentsCardiovascular Agents +6
Target Protein:
Kappa-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SPL23-2 DB17866
biotech

SPL23-2 is an antisense oligonucleotide (ASO) targeting the W1282X nonsense mutation associated with a severe form of cystic fibrosis.[L46767]

Waktu Paruh-
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