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6694

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Halaman 55 / 134
biotech

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biotech

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biotech | CAS: 2226647-27-2

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
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Ezatiostat DB05460
small molecule | CAS: 168682-53-9

Ezatiostat is investigated in clinical trials for treating myelodysplastic syndrome. This compound belongs to the peptides. These are compounds containing an amide derived from two or more amino carboxylic acid molecules (the same or different) by formation o…

Kategori:
Amino Acids, Peptides, and ProteinsOligopeptidesPeptides
Target Protein:
Glutathione S-transferase P
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Ezetimibe Approved DB00973
small molecule | CAS: 163222-33-1

Ezetimibe is a lipid-lowering compound that inhibits intestinal cholesterol and phytosterol absorption. The discovery and research of this drug began in the early 1990s, after the intravenous administration of radiolabelled ezetimibe in rats revealed that it …

Kategori:
Anticholesteremic AgentsAzetinesBCRP/ABCG2 Substrates +20
Target Protein:
NPC1-like intracellular cholesterol transporter 1Sterol O-acyltransferase 1Aminopeptidase N
Waktu ParuhBoth ezetimibe and …
Vol. DistribusiThe relative volume…
KlirensThere are no pharma…
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Ezogabine Approved DB04953
small molecule | CAS: 150812-12-7

Ezogabine (D23129) is a close structural analog of the centrally acting analgesic flupitrine. It is a neuronal potassium channel opener being developed as a first-in-class antiepileptic drug (AED) and is currently being studied in Phase 3 trials as an adjunct…

Kategori:
Acids, AcyclicAminesAniline Compounds +15
Target Protein:
Potassium voltage-gated channel subfamily KQT member 3Potassium voltage-gated channel subfamily KQT member 2Potassium voltage-gated channel subfamily KQT member 4 +1
Waktu ParuhTerminal half-life …
Vol. Distribusi8.7 L/kg
Klirens0.58 - 0.76 L/h·kg.…
Genetik -
F6-734 DB17444
biotech

F6-734 is a bispecific monoclonal antibody with affinity for anticarcinoembryonic antigen (CEA) and anti-diethylenetriamine pentaacetic acid (DTPA) (hMN-14 × m734).[A255217,A255222]

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Facinicline DB05586
small molecule | CAS: 677306-35-3

Deskripsi belum tersedia.

Kategori:
Bridged-Ring CompoundsHeterocyclic Compounds, Fused-RingPyrazoles
Target Protein:
Neuronal acetylcholine receptor subunit alpha-7
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Factor IX Complex (Human) Approved DB11330
biotech | CAS: 37224-63-8

Factor IX Complex is a sterile, lyophilized concentrate composed of a number of Vitamin K-dependent clotting factors found in functioning human plasma. Also known as prothrombin complex concentrate, products containing this complex often include Factor IX (an…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +6
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Factor XIII (human) Approved DB12909
biotech | CAS: 9013-56-3

Factor XIII (human) is a heat-treated, lyophilized concentrate of coagulation factor XIII, an endogenous enzyme responsible for the crosslinking of fibrin and an essential component of the coagulation cascade [FDA Label]. For people with congenital deficiency…

Kategori:
AcyltransferasesAmino Acids, Peptides, and ProteinsAminoacyltransferases +14
Waktu Paruh6.6 ±2.29 days [FDA…
Vol. DistribusiVss = 51.1 mL/kg (v…
Klirens0.25 ±0.09 mL/hr/kg…
Genetik -
Falnidamol DB12966
small molecule | CAS: 196612-93-8

Falnidamol has been used in trials studying the treatment of Unspecified Adult Solid Tumor, Protocol Specific.

Target Protein:
Epidermal growth factor receptor
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Famciclovir Approved DB00426
small molecule | CAS: 104227-87-4

Famciclovir, marketed as Famvir by Novartis, is a guanine analogue used to treat herpes virus infections. It is most commonly used to treat herpes zoster (shingles). Famciclovir is a prodrug of penciclovir with higher oral bioavailability.

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +12
Target Protein:
DNA polymerase catalytic subunit
Waktu Paruh10 hours
Vol. Distribusi* 1.08±0.17 L/kg [h…
Klirens* 36.6 +/- 6.3 L/hr…
Genetik -
Famotidine Approved DB00927
small molecule | CAS: 76824-35-6

Famotidine is a competitive histamine-2 (H<sub>2</sub>) receptor antagonist that works to inhibit gastric acid secretion. It is commonly used in gastrointestinal conditions related to acid secretion, such as gastric ulcers and gastroesophageal reflux disease …

Kategori:
Acid ReducersAlimentary Tract and MetabolismAnti-Ulcer Agents +20
Target Protein:
Histamine H2 receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe steady-state vo…
KlirensRenal clearance is …
Genetik -
Famphur DB11408
small molecule | CAS: 52-85-7

Deskripsi belum tersedia.

Kategori:
AgrochemicalsCompounds used in a research, industrial, or household settingInsecticides +8
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Famprofazone DB16702
small molecule | CAS: 22881-35-2

Famprofazone is a nonsteroidal anti-inflammatory agent found in combination products such as ‘Gewodin’ which is marketed in Taiwan.[L34724] It is important to note that the drug is metabolized to [methamphetamine] and [amphetamine] in the body and can lead to…

Kategori:
AminesAmphetaminesAnalgesics +7
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Famtozinameran Approved DB17088
biotech

The Omicron variant of SARS-CoV-2 is a variant of concern that was first reported in November 2021.[L43922] It tends to cause less severe disease but is significantly more virulent than both the original virus and earlier variants (e.g. Delta).[L43917] As of …

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBiological Factors +12
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Faricimab Approved DB15303
biotech | CAS: 1607793-29-2

Retinal vascular diseases (RVDs) such as diabetic macular edema (DME), age-related macular degeneration (AMD), and retinal vein occlusion (RVO) are typically caused by retinal ischemia and subsequent neovascularization (NV).[A225985, A225990, A225995] Vascula…

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +15
Target Protein:
Vascular endothelial growth factor A, long formAngiopoietin-2
Waktu ParuhFaricimab has an es…
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biotech | CAS: 2407465-18-1

Farletuzumab ecteribulin is under investigation in clinical trial NCT04300556 (A Study to Evaluate the Safety, Tolerability, and Efficacy of Morab-202 (Herein Referred to as Farletuzumab Ecteribulin), a Folate Receptor Alpha (Fr?)-targeting Antibody-drug Conj…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
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Farnesol DB02509
small molecule | CAS: 4602-84-0

A colorless liquid extracted from oils of plants such as citronella, neroli, cyclamen, and tuberose. It is an intermediate step in the biological synthesis of cholesterol from mevalonic acid in vertebrates. It has a delicate odor and is used in perfumery. (Fr…

Kategori:
AlcoholsFatty AlcoholsLipids +2
Target Protein:
Amine oxidase [flavin-containing] BBile acid receptor
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Farudodstat DB16049
small molecule | CAS: 1035688-66-4

Farudodstat (ASLAN003) is under investigation in clinical trial NCT03451084 (A Dose Optimisation Study of ASLAN003 in Acute Myeloid Leukemia).

Kategori:
AminesEnzyme InhibitorsPyridines
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Fasinumab DB12157
biotech | CAS: 1190239-42-9

Fasinumab is a human IgG1k monoclonal antibody targeted against nerve growth factor (NGF). It is currently under investigation for the treatment osteoarthritic pain[A241045] and has demonstrated significantly greater pain relief and functional improvement as …

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAnalgesics, Non-Narcotic +11
Target Protein:
Beta-nerve growth factor
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FAV-201 DB06130
biotech

FAV-201 is a patient-specific immunotherapy for the treatment of T-cell lymphoma.

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Favezelimab DB16729
biotech | CAS: 2231068-83-8

Favezelimab is under investigation in clinical trial NCT04626479 (Substudy 03A: A Study of Immune and Targeted Combination Therapies in Participants With First Line (1L) Renal Cell Carcinoma (MK-3475-03A)).

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Fazirsiran DB17891
biotech | CAS: 2175009-08-0

Deskripsi belum tersedia.

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Fazpilodemab DB18924
biotech | CAS: 2517935-02-1

Fazpilodemab is under investigation in clinical trial NCT04171765 (A Study to Evaluate the Efficacy, Safety, and Pharmacokinetics of BFKB8488A Compared With Placebo in Participants With Non-alcoholic Steatohepatitis).

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fb-PMT DB17394
small molecule

Deskripsi belum tersedia.

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FBX-101 DB18340
biotech

FBX-101 is an adeno-associated virus serotype rhesus 10 vector expressing the human galactocerebrosidase (GALC) gene

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FCR001 DB18595
biotech

FCR001 is a somatic cell therapy product containing hematopoietic progenitor cells (HPC), Facilitating Cells (FC), and alpha beta T cells.

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Febuxostat Approved DB04854
small molecule | CAS: 144060-53-7

Febuxostat is a non-purine xanthine oxidase (XO) inhibitor.[A39743] In early 2008, febuxostat was granted marketing authorization by the European Commission for the treatment of chronic hyperuricemia and gout.[A230548] In the following year, the FDA for appro…

Kategori:
Antigout PreparationsAntirheumatic AgentsBCRP/ABCG2 Inhibitors +15
Target Protein:
Xanthine dehydrogenase/oxidase
Waktu ParuhThe apparent mean t…
Vol. DistribusiThe apparent steady…
KlirensFollowing oral admi…
Genetik -
Fecal microbiota Approved DB17743
biotech

Fecal microbiota, given either as a rectal transplant or in an oral formulation of live spores, is an FDA-approved option to prevent the recurrence of _Clostridioides difficile_ infection (CDI) in patients given an antibacterial treatment for recurrent CDI.[A…

Kategori:
Miscellaneous Therapeutic Agents
Waktu ParuhNot available.
Vol. DistribusiNot available.
KlirensNot available.
Genetik -
Feladilimab DB16415
biotech

Feladilimab is under investigation in clinical trial NCT04128696 (Study of GSK3359609 and Pembrolizumab in Programmed Death Receptor 1-ligand 1 Positive Recurrent or Metastatic Head and Neck Squamous Cell Carcinoma).

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Felbamate Approved DB00949
small molecule | CAS: 25451-15-4

Felbamate is an anticonvulsant drug used in the treatment of epilepsy. In particular, in the adult patient population, it can be employed to treat partial seizures (with and without generalization). Alternatively, it is used to treat partial and generalized s…

Kategori:
Acids, AcyclicAlcoholsAnti-epileptic Agent +28
Target Protein:
Glutamate receptor ionotropic, NMDA 2BGlutamate receptor ionotropic, NMDA 2A
Waktu Paruh20-23 hours
Vol. Distribusi* 756±82 mL/kg
Klirens* 26 +/- 3 mL/hr/kg…
Genetik -
Felcisetrag DB12725
small molecule | CAS: 916075-84-8

Felcisetrag (TD-8954) has been used in trials studying the treatment of Enteral Feeding Intolerance and Gastrointestinal Motility Disorder.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsHeterocyclic Compounds, Fused-Ring +4
Target Protein:
5-hydroxytryptamine receptor 4
Waktu Paruh-
Vol. Distribusi-
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Felodipine Approved DB01023
small molecule | CAS: 72509-76-3

Felodipine is a long-acting 1,4-dihydropyridine calcium channel blocker (CCB)b. It acts primarily on vascular smooth muscle cells by stabilizing voltage-gated L-type calcium channels in their inactive conformation. By inhibiting the influx of calcium in smoot…

Kategori:
ACE Inhibitors and Calcium Channel BlockersAgents causing hyperkalemiaAntiarrhythmic agents +31
Target Protein:
Voltage-dependent L-type calcium channel subunit alpha-1CVoltage-dependent calcium channel subunit alpha-2/delta-1Voltage-dependent L-type calcium channel subunit beta-2 +10
Waktu Paruh17.5-31.5 hours in …
Vol. Distribusi* 10 L/kg
Klirens* 0.8 L/min [Young …
Genetik -
Felypressin DB00093
biotech | CAS: 56-59-7

A synthetic nonapeptide comprising cysteinyl, phenylalanyl, phenylalanyl, glutaminyl, asparaginyl, cysteinyl, prolyl, lysyl, and glycinamide residues in sequence, with a disulfide bridge joining the two cysteine residues. Its antidiuretic effects are less tha…

Kategori:
Amino Acids, Peptides, and ProteinsCardiovascular AgentsHormones +12
Target Protein:
Vasopressin V1a receptor
Waktu Paruh-
Vol. Distribusi-
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Fenbendazole DB11410
small molecule | CAS: 43210-67-9

Fenbendazole is a benzimidazole that presents a wide spectrum anthelmintic effect. It is used against a number of gastrointestinal parasites including giardia, roundworms, hookworms, whipworms, the Taenia genus of tapeworms, pinworms, aelurostrongylus, parago…

Kategori:
Acids, AcyclicAnthelminticsAnti-Infective Agents +7
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Fenbufen Approved DB08981
small molecule | CAS: 36330-85-5

Fenbufen is a non-steroidal anti-inflammatory drug used primarily to treat inflammation in osteoarthritis, ankylosing spondylitis, and tendinitis. It can also be used to relieve backaches, sprains, and fractures. Fenbufen is available as a capsule or tablet s…

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +15
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu Paruh-
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Fencamfamin DB01463
small molecule | CAS: 1209-98-9

Fencamfamin (Glucoenergan, Reactivan) is a stimulant which was developed in the 1960s as an appetite suppressant, but was later withdrawn for this application due to problems with dependence and abuse. It is around half the potency of [dexamphetamine], and is…

Kategori:
Bridged-Ring CompoundsCentral Nervous System AgentsCentral Nervous System Depressants +7
Target Protein:
Sodium-dependent dopamine transporterD(2) dopamine receptor
Waktu Paruh-
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Fendiline DB08980
small molecule | CAS: 13042-18-7

Fendiline is a coronary vasodilator which inhibits calcium function in muscle cells in excitation-contraction coupling. It has been proposed as an antiarrhythmic and antianginal agent. Fendiline is non-selective.

Kategori:
Agents causing hyperkalemiaAminesAntiarrhythmic agents +15
Target Protein:
5-hydroxytryptamine receptor 2B
Waktu Paruh-
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Fenfluramine Approved DB00574
small molecule | CAS: 458-24-2

Dravet syndrome is a pediatric encephalopathy that typically manifests within the first year of life following exposure to elevated temperatures. It is characterized by recurrent pharmacoresistant seizures, which increase in frequency and severity with diseas…

Kategori:
Alimentary Tract and MetabolismAminesAnticonvulsants +27
Target Protein:
Sodium-dependent serotonin transporter5-hydroxytryptamine receptor 1D5-hydroxytryptamine receptor 2C +4
Waktu ParuhFenfluramine has an…
Vol. DistribusiFenfluramine has an…
KlirensFenfluramine has a …
Genetik -
Fenofibrate Approved DB01039
small molecule | CAS: 49562-28-9

Fenofibrate is a fibric acid derivative like [clofibrate] and [gemfibrozil].[A185954] Fenofibrate is used to treat primary hypercholesterolemia, mixed dyslipidemia, severe hypertriglyceridemia.[L8588,L8591] Fenofibrate was granted FDA approval on 31 Decemb…

Kategori:
Acids, AcyclicAgents Causing Muscle ToxicityBenzene Derivatives +39
Target Protein:
Peroxisome proliferator-activated receptor alphaNuclear receptor subfamily 1 group I member 2Matrix metalloproteinase-25
Waktu ParuhFenofibric acid, th…
Vol. DistribusiThe volume of distr…
KlirensThe oral clearance …
Genetik -
Fenofibric acid Approved DB13873
small molecule | CAS: 42017-89-0

Fenofibric acid is a lipid-lowering agent that is used in severe hypertriglyceridemia, primary hyperlipidemia, and mixed dyslipidemia. It works to decrease elevated low-density lipoprotein cholesterol, total cholesterol, triglycerides, apolipoprotein B, while…

Kategori:
Acids, AcyclicAgents Causing Muscle ToxicityAnticholesteremic Agents +17
Target Protein:
Peroxisome proliferator-activated receptor alphaFatty acid-binding protein, liverMatrix metalloproteinase-25 +3
Waktu ParuhFollowing once dail…
Vol. DistribusiThe volume of distr…
KlirensIn five elderly vol…
Genetik -
Fenoprofen Approved DB00573
small molecule | CAS: 29679-58-1

An anti-inflammatory analgesic and antipyretic highly bound to plasma proteins. It is pharmacologically similar to aspirin, but causes less gastrointestinal bleeding.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +18
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1Peroxisome proliferator-activated receptor alpha +1
Waktu ParuhPlasma half-life is…
Vol. Distribusi-
Klirens-
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Fenproporex DB01550
small molecule | CAS: 16397-28-7

Fenproporex is an orally active stimulant drug, which was developed in the 1960s. It is used as an appetite suppressant and a treatment for obesity. It is listed as an illicit substance in many countries due to addiction issues and listed as a prohibited subs…

Kategori:
AminesDrugs that are Mainly Renally ExcretedEthylamines +2
Waktu Paruh-
Vol. Distribusi-
KlirensThe amphetamine met…
Genetik -
Fenpyroximate DB16164
small molecule | CAS: 134098-61-6

Fenpyroximate is under investigation in clinical trial NCT02533336 (The Effectiveness of Non-pyrethroid Insecticide-treated Durable Wall Liners as a Method for Malaria Control in Endemic Rural Tanzania).

Kategori:
Acids, CarbocyclicBenzene DerivativesElectron Transport Complex I, antagonists & inhibitors
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Fentanyl Approved DB00813
small molecule | CAS: 437-38-7

Fentanyl, a potent opioid agonist, was developed in the 1950s to fill a need for strong and rapid analgesia.[A179542] Because of these characteristics, fentanyl is commonly used to treat chronic cancer pain or in anesthesia.[Label,L6598,L6601,L6604,L6607,L922…

Kategori:
AdjuvantsAdjuvants, AnesthesiaAgents that produce hypertension +32
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor +1
Waktu ParuhThe half life of fe…
Vol. DistribusiThe intravenous vol…
KlirensTotal plasma cleara…
Genetik -
Fenthion DB11412
small molecule | CAS: 55-38-9

Fenthion is an _organothiophosphate_ drug used as an insecticide, avicide, and acaricide. Its mode of action is explained by cholinesterase enzyme inhibition, which is similar to other organophosphates. Fenthion is listed as a restricted use compound by the U…

Kategori:
AgrochemicalsCholinergic AgentsCholinesterase Inhibitors +13
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Fentiazac DB13217
small molecule | CAS: 18046-21-4

Deskripsi belum tersedia.

Kategori:
Acetic Acid Derivatives and Related SubstancesAcids, AcyclicAgents causing hyperkalemia +19
Waktu Paruh-
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Fenvalerate DB18391
small molecule | CAS: 51630-58-1

Deskripsi belum tersedia.

Kategori:
AgrochemicalsCompounds used in a research, industrial, or household settingCyclopentane Monoterpenes +7
Waktu Paruh-
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Fepixnebart DB19079
biotech | CAS: 1799706-87-8

Fepixnebart is under investigation in clinical trial NCT04456686 (Chronic Pain Master Protocol (CPMP): A Study of LY3016859 in Participants With Osteoarthritis).

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