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15718

Total database: 17430
Struktur (SMILES)
10762 (68.5%)
Target
7957 (50.6%)
Genomik
112 (0.7%)
Referensi
15718 (100.0%)

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Hasil Pencarian (15718)

Halaman 55 / 315
Amoxapine Approved DB00543
small molecule | CAS: 14028-44-5

Amoxapine, the <i>N</i>-demethylated derivative of the antipsychotic agent loxapine, is a dibenzoxazepine-derivative tricyclic antidepressant (TCA). TCAs are structurally similar to phenothiazines. They contain a tricyclic ring system with an alkyl amine subs…

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +49
Target Protein:
Sodium-dependent serotonin transporterSodium-dependent noradrenaline transporterD(2) dopamine receptor +22
Waktu Paruh8 hours
Vol. DistribusiWidely distributed …
Klirens-
Genetik -
Amoxicillin Approved DB01060
small molecule | CAS: 26787-78-0

Amoxicillin, or BRL-2333, is a penicillin G derivative first described in the literature in 1972.[A190648] Amoxicillin has similar activity to [penicillin] and [ampicillin], but leads to higher serum concentrations than ampicillin.[A190648] Amoxicillin was…

Kategori:
Alimentary Tract and MetabolismAmidesAminopenicillins +19
Target Protein:
Penicillin binding protein
Waktu ParuhThe half life of am…
Vol. DistribusiThe central volume …
KlirensThe mean clearance …
Genetik -
AMP-101 DB18253
biotech

AMP-101 is a gene therapy comprising an adeno-associated virus type 9 (AAV9) vector encoding the human Dok-7 protein. It is under investigation for the treatment of Dok-7-associated myasthenia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
AMP-201 DB18663
biotech

AMP-201 comprises an adeno-associated virus type 8 vector (AAV8) encoding the collagen Q gene (COLQ). It is under investigation for the treatment of collagen Q congenital myasthenia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
AMP-224 DB15767
biotech | CAS: 1422184-00-6

Deskripsi belum tersedia.

Kategori:
Immune Checkpoint Inhibitors
Target Protein:
Programmed cell death protein 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AMPCPR DB01975
small molecule

Deskripsi belum tersedia.

Target Protein:
ADP-ribose pyrophosphataseMutT/nudix family protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Amphetamine Approved DB00182
small molecule | CAS: 300-62-9

Amphetamine, a compound discovered over 100 years ago, is one of the more restricted controlled drugs. It was previously used for a large variety of conditions and this changed until this point where its use is highly restricted. Amphetamine, with the chemica…

Kategori:
Adrenergic AgentsAgents producing tachycardiaAgents that produce hypertension +31
Target Protein:
Synaptic vesicular amine transporterSodium-dependent dopamine transporterCocaine- and amphetamine-regulated transcript protein +8
Waktu ParuhThe half-life of am…
Vol. DistribusiAmphetamine is repo…
KlirensThe reported normal…
Genetik -
biotech

Amphiachyris dracunculoides pollen is the pollen of the Amphiachyris dracunculoides plant. Amphiachyris dracunculoides pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Amphomycin DB11499
small molecule | CAS: 1402-82-0

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Amphotericin B Approved DB00681
small molecule | CAS: 1397-89-3

Amphotericin B shows a high order of in vitro activity against many species of fungi. Histoplasma capsulatum, Coccidioides immitis, Candida species, Blastomyces dermatitidis, Rhodotorula, Cryptococcus neoformans, Sporothrix schenckii, Mucor mucedo, and Asperg…

Kategori:
Agents Causing Muscle ToxicityAgents that reduce seizure thresholdAlimentary Tract and Metabolism +30
Target Protein:
Ergosterol
Waktu ParuhAn elimination half…
Vol. Distribusi-
Klirens* 39 +/- 22 mL/hr/k…
Genetik -
Ampicillin Approved DB00415
small molecule | CAS: 69-53-4

Ampicillin is a semi-synthetic derivative of penicillin that functions as an orally active broad-spectrum antibiotic.

Kategori:
AmidesAminopenicillinsAnti-Bacterial Agents +14
Target Protein:
Penicillin-binding protein 2aPenicillin-binding protein 1bPenicillin-binding protein 3 +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ampiroxicam DB16877
small molecule | CAS: 99464-64-9

Deskripsi belum tersedia.

Kategori:
Sulfur Compounds
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ampreloxetine DB15348
small molecule | CAS: 1227056-84-9

Ampreloxetine is under investigation in clinical trial NCT03750552 (Clinical Effect of TD-9855 for Treating snOH in Subjects With Primary Autonomic Failure).

Kategori:
Benzene DerivativesEthersPhenols
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Amprenavir Approved DB00701
small molecule | CAS: 161814-49-9

Amprenavir is a protease inhibitor used to treat HIV infection.

Kategori:
Acids, AcyclicAmidesAmprenavir and Prodrugs +37
Target Protein:
Pol polyproteinGag-Pol polyprotein
Waktu Paruh7.1-10.6 hours
Vol. Distribusi-
Klirens-
Genetik -
Amprolium DB11374
small molecule | CAS: 121-25-5

Amprolium is a coccidiostat used in poultry.

Kategori:
Anti-Infective AgentsAntiparasitic AgentsAntiprotozoals +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Amrinone Approved DB01427
small molecule | CAS: 60719-84-8

Amrinone (or inamrinone) is a type 3 pyridine phosphodiesterase inhibitor. It is used in the treatment of congestive heart failure.

Kategori:
AminesAminopyridinesCalcium-Regulating Hormones and Agents +14
Target Protein:
cAMP-specific 3',5'-cyclic phosphodiesterase 4 (PDE4)cGMP-inhibited 3',5'-cyclic phosphodiesterase 3AcGMP-inhibited 3',5'-cyclic phosphodiesterase 3B +1
Waktu Paruh5 to 8 hours
Vol. Distribusi* 1.2 L/kg [normal …
Klirens-
Genetik -
Amrubicin DB06263
small molecule | CAS: 110267-81-7

Amrubicin is a third-generation synthetic anthracycline currently in development for the treatment of small cell lung cancer. Pharmion licensed the rights to Amrubicin in November 2006. In 2002, Amrubicin was approved and launched for sale in Japan based on P…

Kategori:
Anthracyclines and Related SubstancesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +4
Target Protein:
DNA topoisomerase 2-alphaDNA
Waktu Paruh20-30 h [A32143] …
Vol. DistribusiModerate volume of …
KlirensThe plasma pharmaco…
Genetik -
Amsacrine Approved DB00276
small molecule | CAS: 51264-14-3

Aminoacridine derivative that is a potent intercalating antineoplastic agent. It is effective in the treatment of acute leukemias and malignant lymphomas, but has poor activity in the treatment of solid tumors. It is frequently used in combination with other …

Kategori:
AcridinesAminoacridinesAntineoplastic Agents +11
Target Protein:
DNADNA topoisomerase 2-betaDNA topoisomerase 2-alpha +3
Waktu Paruh8-9 hours
Vol. Distribusi-
Klirens-
Genetik -
AMT-080 DB17846
biotech

AMT-080 is an investigational gene therapy being investigated for the treatment of Duchenne muscular dystrophy.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AMT-101 DB18555
biotech

AMT-101 is a recombinant human interleukin-10 fusion protein.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AMT-130 DB16975
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AMT-162 DB17922
biotech

AMT-162 is an adeno-associated virus serotype rh10 encoding artificial anti-SOD1 miRNA.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 87344-05-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Amubarvimab DB16493
biotech | CAS: 2509447-07-6

Amubarvimab (BRII-196) was under investigation in clinical trials (NCT04691180 and NCT04787211) to treat COVID-19, focusing on its safety, tolerability, and efficacy.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Amuvatinib DB12742
small molecule | CAS: 850879-09-3

Amuvatinib has been used in trials studying the treatment of Solid Tumors and Small Cell Lung Carcinoma. Amuvatinib is an oral, selective multi-targeted tyrosine kinase inhibitor that suppresses c-MET, c-RET and the mutant forms of c-KIT, PDGFR and FLT3. Amuv…

Kategori:
AmidesSulfur Compounds
Target Protein:
Platelet-derived growth factor receptor alphaMast/stem cell growth factor receptor KitHepatocyte growth factor receptor +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AMY-101 DB14803
small molecule | CAS: 1427001-89-5

AMY-101, also known as compstatin 40, is a peptidic inhibitor of the central complement component C3. AMY-101 is under investigation in clinical trial NCT03694444 (A Study of the C3 Complement Inhibitor AMY-101 in Adults With Gingivitis).

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Target Protein:
Complement C3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Amyl acetate DB15927
small molecule | CAS: 628-63-7

Deskripsi belum tersedia.

Kategori:
AlcoholsFatty AlcoholsLipids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Amyl Nitrite Approved DB01612
small molecule | CAS: 8017-89-8

Amyl Nitrite is an antihypertensive medicine. Amyl nitrite is employed medically to treat heart diseases such as angina and to treat cyanide poisoning. Its use as a prescription medicine comes from its ability to lower blood pressure. As an inhalant, it also …

Kategori:
Antianginal AgentsAntidotesCardiovascular Agents +5
Target Protein:
Atrial natriuretic peptide receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Amylamine DB02045
small molecule | CAS: 110-58-7

Deskripsi belum tersedia.

Target Protein:
Serine protease 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Amylmetacresol Approved DB13908
small molecule | CAS: 1300-94-3

Amylmetacresol is an antiseptic available in Canada over-the-counter in a number of lozenges for the treatment of sore throat and minor mouth infections [L2570], [L2571]. Amylmetacresol is often combined with dichlorobenzyl alcohol and menthol in the commonl…

Kategori:
Anti-Infective Agents, LocalBenzene DerivativesMiscellaneous Anti-infectives +1
Target Protein:
Sodium channel protein type 2 subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Amylocaine Approved DB09088
small molecule | CAS: 644-26-8

Despite the introduction of using cocaine injections for regional anesthesia in 1884, non-addictive substitutes were sought after immediately [L1882]. Finally, in 1903 the world's first synthetic and non-addictive local anesthetic, amylocaine, was synthesized…

Kategori:
Acids, CarbocyclicBenzene Derivatives
Target Protein:
Voltage-gated sodium channel alpha subunit
Waktu ParuhA lack of detailed …
Vol. DistribusiA lack of detailed …
KlirensA lack of detailed …
Genetik -
Amylopectin DB14927
small molecule | CAS: 9037-22-3

Amylopectin is under investigation in clinical trial NCT01708694 (Role of Slowly Digesible Starch on Diabetes Risk Factors).

Kategori:
CarbohydratesDietary CarbohydratesGlucans +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Amylose DB15216
small molecule | CAS: 9005-82-7

Amylose is under investigation in clinical trial NCT01027325 (Resistant Starch Insulin Sensitivity Trial).

Kategori:
CarbohydratesDietary CarbohydratesGlucans +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AMZ002 DB17017
biotech

AMZ002 is a sterile injectable hormone developed as a purified synthetic polypeptide alternative to current FDA-approved epileptic seizure treatments.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AN-2718 DB12810
small molecule | CAS: 174672-06-1

An2718 has been used in trials studying Tinea Pedis.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AN-9 DB05103
small molecule | CAS: 122110-53-6

Pivaloyloxymethyl butyrate (AN-9), an acyloxyalkyl ester prodrug of butyric acid (BA), exhibited low toxicity and significant anticancer activity in vitro and in vivo. It shows greater potency than BA at inducing malignant cell differentiation and tumor growt…

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +1
Target Protein:
Histone deacetylase 1Apoptosis regulator Bcl-2Caspase-8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AN0128 DB05054
small molecule

AN0128 is a novel compound that contains a boron atom within a borinic acid complex. AN0128 has broad spectrum activity against a wide variety of Gram positive bacteria, including many that are known skin colonizers. Of particular importance is P. acnes and …

Kategori:
Boron Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AN2898 DB16039
small molecule | CAS: 906673-33-4

AN2898 is under investigation in clinical trial NCT01301508 (Efficacy and Safety of AN2898 and AN2728 Topical Ointments to Treat Mild-to-moderate Atopic Dermatitis).

Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4D3',5'-cyclic-AMP phosphodiesterase 4B3',5'-cyclic-AMP phosphodiesterase 4A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ANA971 DB05127
small molecule

ANA971, an orally administered prodrug of isatoribine. Isatoribine is a nucleoside analog in development for the treatment of chronic hepatitis C virus (HCV) infection. ANA971 is a prodrug designed to improve the oral bioavailability of isatoribine. ANA971 re…

Target Protein:
Toll-like receptor 7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anacaulase Approved DB17449
biotech

Anacaulase (anacaulase-bcdb) is a mixture of proteolytic enzymes extracted from the stems of pineapple plants (_Ananas comosus_ [L.] Merr.). It is mostly composed (80-95% w/w) of proteins such as stem bromelain, ananain, jacalin-like lectin, bromelain inhibit…

Kategori:
Administration, TopicalCysteine EndopeptidasesCytochrome P-450 CYP2C8 Inhibitors +9
Target Protein:
Alpha-1-antichymotrypsinAlpha-2-macroglobulin
Waktu ParuhThe mean eliminatio…
Vol. Distribusi-
Klirens-
Genetik -
Anagliptin DB12417
small molecule | CAS: 739366-20-2

Anagliptin is under investigation for the treatment of LDL Cholesterol, Coronary Disease, Diabetes Mellitus, Glycosylated Hemoglobin, and Dipeptidyl-Peptidase 4 Inhibitors.

Kategori:
Agents causing angioedemaBlood Glucose Lowering AgentsDPP-IV Inhibitors +2
Target Protein:
Dipeptidyl peptidase 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anagrelide Approved DB00261
small molecule | CAS: 68475-42-3

Anagrelide is a platelet-reducing agent used to lower dangerously elevated platelet levels (i.e. to treat thrombocythemia) in patients with myeloproliferative neoplasms.[L14153] It is an oral imidazoquinazoline that was first approved for use in the US in 199…

Kategori:
Agents producing tachycardiaAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +18
Target Protein:
cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A
Waktu ParuhThe t<sub>1/2</sub>…
Vol. Distribusi-
Klirens-
Genetik -
Anakinra Approved DB00026
biotech | CAS: 143090-92-0

Anakinra is a recombinant human interleukin-1 (IL-1) receptor antagonist (IL-1Ra) composed of 153 amino acid residues. Unlike native human IL-1Ra, anakinra has an additional methionine residue at the amino terminus. This drug binds to the IL-1 receptor, compe…

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating Agents +12
Target Protein:
Interleukin-1 receptor type 1
Waktu ParuhIn patients with rh…
Vol. DistribusiIn adult subjects w…
KlirensIn patients with rh…
Genetik -
Anamorelin DB06645
small molecule | CAS: 249921-19-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +2
Target Protein:
Growth hormone secretagogue receptor type 1Lysosomal alpha-glucosidaseNeutral alpha-glucosidase AB +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ananain DB18353
biotech | CAS: 119129-70-3

Deskripsi belum tersedia.

Kategori:
Cysteine ProteasesEndopeptidasesEnzymes +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anaritide DB17613
biotech | CAS: 95896-08-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsDiureticsHormones +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anas platyrhynchos feather Approved DB10421
biotech

Anas platyrhynchos feather is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anastrozole Approved DB01217
small molecule | CAS: 120511-73-1

Anastrozole is a non-steroidal aromatase inhibitor (AI), similar to [letrozole], used to decrease circulating estrogen levels in the treatment of postmenopausal women with estrogen-responsive breast cancer.[L8863] Anastrozole is also related to [exemestane], …

Kategori:
Antineoplastic AgentsAntineoplastic Agents, HormonalAntineoplastic and Immunomodulating Agents +30
Target Protein:
Aromatase
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensAnastrozole's clear…
Genetik -
Anbenitamab DB18411
biotech | CAS: 2367012-88-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ANC-501 DB18907
small molecule | CAS: 1370444-22-6

ANC-501 is under investigation in clinical trial NCT05439603 (ANC-501 in the Treatment of Adults With Major Depressive Disorder).

Kategori:
AcetatesAcids, AcyclicAmides +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 2701–2750 dari 15718
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