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14494

Total database: 17430
Struktur (SMILES)
9687 (66.8%)
Target
7525 (51.9%)
Genomik
112 (0.8%)
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14494 (100.0%)

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Hasil Pencarian (14494)

Halaman 54 / 290
small molecule

Deskripsi belum tersedia.

Target Protein:
(S)-2-haloacid dehalogenase
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small molecule | CAS: 110954-19-3

Aspartyl-alanyl-diketopiperazine is under investigation in clinical trial NCT03349645 (An Open Label Extension Study to Assess the Safety of Long-Term Treatment With Ampion for Severe OA of the Knee).

Kategori:
Amino Acids, Peptides, and ProteinsOligopeptidesPeptides
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biotech

Deskripsi belum tersedia.

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Aspergillus flavus Approved DB10694
biotech

Aspergillus flavus is a fungus which can provoke allergic reactions. Aspergillus flavus extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Fungal Allergenic Extract
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Aspergillus fumigatus Approved DB10425
biotech

Aspergillus fumigatus is a fungus which can provoke allergic reactions. Aspergillus fumigatus extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Fungal Allergenic Extract
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Aspergillus nidulans Approved DB11022
biotech

Aspergillus nidulans is a fungus which can provoke allergic reactions. Aspergillus nidulans extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Aspergillus niger var. niger Approved DB10426
biotech

Aspergillus niger var. niger is a fungus which can provoke allergic reactions. Aspergillus niger var. niger extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Aspergillus oryzae Approved DB10448
biotech

Aspergillus oryzae allergenic extract is used in allergenic testing.

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Aspergillus repens Approved DB10449
biotech

Aspergillus repens is a fungus which can provoke allergic reactions. Aspergillus repens extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Aspergillus terreus Approved DB10450
biotech

Aspergillus terreus is a fungus which can provoke allergic reactions. Aspergillus terreus extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Aspoxicillin DB13816
small molecule | CAS: 63358-49-6

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAntibacterials for Systemic Use +9
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Astaxanthin DB06543
small molecule | CAS: 472-61-7

Astaxanthin is a keto-carotenoid in the terpenes class of chemical compounds. It is classified as a xanthophyll but it is a carotenoid with no vitamin A activity. It is found in the majority of aquatic organisms with red pigment. Astaxanthin has shown to medi…

Kategori:
AlkenesAnticoagulantsBiological Factors +9
Target Protein:
NF-kappa-B inhibitor alpha
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Astegolimab DB16386
biotech | CAS: 2173054-79-8

Astegolimab is under investigation in clinical trial NCT04386616 (A Study to Evaluate the Safety and Efficacy of MSTT1041A (Astegolimab) or UTTR1147A in Patients With Severe COVID-19 Pneumonia).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAnti-Inflammatory Agents +10
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Astemizole Approved DB00637
small molecule | CAS: 68844-77-9

Astemizole is a long-acting, non-sedating second generation antihistamine used in the treatment of allergy symptoms. It was withdrawn from market by the manufacturer in 1999 due to the potential to cause arrhythmias at high doses, especially when when taken …

Kategori:
Anti-Allergic AgentsAntihistamines for Systemic UseBenzimidazoles +27
Target Protein:
Histamine H1 receptorVoltage-gated inwardly rectifying potassium channel KCNH2Voltage-gated delayed rectifier potassium channel KCNH1 +1
Waktu Paruh1 day
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Astodrimer DB11854
biotech | CAS: 1379746-42-5

Astodrimer has been used in trials studying the treatment and prevention of Bacterial Vaginosis. It is a lysine-based dendrimer with naphthalene disulfonic acid surface groups.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +10
Target Protein:
Envelope glycoprotein gp160
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small molecule

Deskripsi belum tersedia.

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AstraZeneca COVID-19 Vaccine Approved DB15656
biotech | CAS: 2420395-83-9

The AstraZeneca COVID-19 Vaccine (previously known as ChAdOx1 nCoV-19 or AZD1222) is one of several vaccines developed in 2020 for the prevention of COVID-19 caused by SARS-CoV-2.[L12669,L32649] The ChAdOx1 viral vector was developed at the University of Oxfo…

Kategori:
Biological ProductsComplex MixturesCOVID-19 Vaccines +6
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ASTX-029 DB18900
small molecule | CAS: 2095719-92-7

ASTX-029 is under investigation in clinical trial NCT03520075 (Study of ASTX029 in Subjects With Advanced Solid Tumors).

Kategori:
Heterocyclic Compounds, Fused-Ring
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Asunaprevir Approved DB11586
small molecule | CAS: 630420-16-5

Asunaprevir, also named BMS-650032, is a potent hepatitis C virus (HCV) NS3 protease inhibitor. It has been shown to have a very high efficacy in dual-combination regimens with daclatasvir in patients chronically infected with HCV genotype 1b.[A32528] It was …

Kategori:
AmidesAntiinfectives for Systemic UseAntiviral Agents +35
Target Protein:
Gag-Pol polyproteinGenome polyprotein
Waktu ParuhClinical pharmacoki…
Vol. DistribusiThe registered volu…
KlirensClinical pharmacoki…
Genetik -
Asundexian DB19088
small molecule | CAS: 2064121-65-7

Asundexian is under investigation in clinical trial NCT05686070 (A Study to Test Asundexian for Preventing a Stroke Caused by a Clot in Participants After an Acute Ischemic Stroke or After a High-risk Transient Ischemic Attack, a So-called Mini Stroke).

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +2
Target Protein:
Coagulation factor XI
Waktu Paruh-
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Asunercept DB15160
biotech | CAS: 1450882-18-4

Asunercept is under investigation in clinical trial NCT02853565 (A Study of CAN008 for Newly Diagnosed Glioblastoma Multiforme).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +10
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Asvasiran DB05638
biotech | CAS: 870094-26-1

Asvasiran is an siRNA that targets the respiratory syncytial virus (RSV) N gene and inhibits viral replication. It has the potential to treat or prevent RSV infection.

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AT-001 DB15121
small molecule | CAS: 1355612-71-3

AT-001 is under investigation in clinical trial NCT03062384 (AT-001 for Long-term Preservation of Brain Health in Aging).

Kategori:
Heterocyclic Compounds, Fused-RingPyridinesThiazoles
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AT-301 DB16507
biotech

AT-301 was under investigation in clinical trial NCT01675284 to evaluate the safety, reactogenicity, and humoral immune responses to an inactivated H5N1 influenza vaccine

Kategori:
Experimental Unapproved Treatments for COVID-19
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AT-7519 DB08142
small molecule | CAS: 844442-38-2

AT7519 is a selective inhibitor of certain Cyclin Dependent Kinases (CDKs) leading to tumour regression. It is developed by Astex for the treatment of solid tumours and haematological malignancies.

Kategori:
Cyclin-Dependent Kinases, antagonists & inhibitors
Target Protein:
Cyclin-dependent kinase 2Cyclin-dependent kinase 1
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AT-GTX-502 DB17001
biotech

AT-GTX-502 is an experimental, one-time gene therapy that uses AAV9 to deliver a functional copy of CLN3.

Kategori:
Non-Replicating Recombinant, Self-Complementary Adeno-Associated Virus Serotype 9 Containing the Human CLN3 Gene
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AT1022 DB04995
small molecule

AT1022 is a hydromorphone skin patch designed to provide rapid and sustained delivery of a potent opiate for the management of severe pain. AT1022 incorporates PassPort(TM) system, developed to deliver protein and peptide drugs, small-molecule drugs, genes a…

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AT1391 DB05120
small molecule

AT1391 is a daily insulin skin patch designed to provide continuous basal levels of insulin for patients with diabetes.

Target Protein:
Insulin receptor
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AT2220 DB05200
small molecule

AT2220 is an experimental, oral therapy for the treatment of Pompe disease and belongs to a class of molecules known as pharmacological chaperones. It is a small molecule designed to act as a pharmacological chaperone that specifically binds, stabilizes, and …

Target Protein:
Lysosomal alpha-glucosidase
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AT3022 DB05172
small molecule

AT3022, the Altea Therapeutics’s fentanyl citrate transdermal patch designed to provide safe and rapid management of moderate to severe chronic pain.

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AT9283 DB05169
small molecule | CAS: 896466-04-9

AT9283 is an aurora Kinase inhibitor developed by Astex Therapeutics for the treatment of cancer. It was discovered and developed internally using Astex’s fragment-based drug discovery platform, Pyramid.

Kategori:
AmidesHeterocyclic Compounds, Fused-RingProtein Kinase Inhibitors
Target Protein:
Aurora kinase BAurora kinase A
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ATA-100 DB18329
biotech

ATA-100 is an adeno-associated virus serotype 9 carrying the human Fukutin-Related protein gene and target sequence of the miR-208a

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Atabecestat DB15307
small molecule | CAS: 1200493-78-2

Atabecestat is under investigation in clinical trial NCT02211079 (A Study to Assess Effect of JNJ-54861911 on Pharmacokinetics of Cocktail Representatives for Cytochrome P450 (CYP) 3A4, CYP2B6, CYP2C9, and CYP1A2 Substrates).

Kategori:
Sulfur Compounds
Waktu Paruh-
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Atacicept DB06399
biotech | CAS: 845264-92-8

Atacicept is a recombinant fusion protein combined with the extracellular ligand binding portion of TACI.

Kategori:
Amino Acids, Peptides, and ProteinsProteinsRecombinant Proteins
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Ataciguat DB12805
small molecule | CAS: 254877-67-3

Ataciguat has been investigated for the basic science of Aortic Valve Stenosis.

Kategori:
Acids, CarbocyclicAmidesAminobenzoates +5
Target Protein:
Atrial natriuretic peptide receptor 1
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Ataluren Approved DB05016
small molecule | CAS: 775304-57-9

Ataluren is a novel, orally administered drug that targets nonsense mutations. Ataluren is approved for use by the European Medicines Agency to treat Duchenne Muscular Dystrophy in patients aged 5 years and older who are able to walk. More specifically, atalu…

Kategori:
Musculo-Skeletal SystemOAT1/SLC22A6 inhibitorsOAT3/SLC22A8 Inhibitors +3
Target Protein:
Dystrophin
Waktu ParuhAtaluren plasma hal…
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Atamestane DB12194
small molecule | CAS: 96301-34-7

Atamestane has been used in trials studying the treatment of Breast Cancer, Breast Neoplasms, and Neoplasms, Hormone-Dependent.

Kategori:
17-KetosteroidsAdrenal Cortex HormonesAndrostanes +10
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Atamparib DB19028
small molecule | CAS: 2381037-82-5

Atamparib is under investigation in clinical trial NCT05127590 (RBN-2397 in Combination With Pembrolizumab in Patients With SCCL).

Target Protein:
Protein mono-ADP-ribosyltransferase TIPARP
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Atazanavir Approved DB01072
small molecule | CAS: 198904-31-3

Atazanavir (formerly known as BMS-232632) is an antiretroviral drug of the protease inhibitor (PI) class. Like other antiretrovirals, it is used to treat infection of human immunodeficiency virus (HIV). Atazanavir is distinguished from other PIs in that it ca…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-HIV AgentsAnti-Infective Agents +45
Target Protein:
Pol polyproteinGag-Pol polyprotein
Gen Terkait:
UGT1A1 UGT1A1 UGT1A1
Waktu ParuhThe mean eliminatio…
Vol. DistribusiIn patients with HI…
KlirensIn patients with HI…
Genetik 3 Varian
ATB-346 DB15377
small molecule | CAS: 1226895-20-0

ATB-346 is under investigation in clinical trial NCT03220633 (Study To Assess Safety, Tolerability And PK Of ATB-346 In Healthy Subjects).

Kategori:
Naphthaleneacetic AcidsNaphthalenes
Waktu Paruh-
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small molecule | CAS: 433937-93-0

Atecegatran metoxil has been used in trials studying the basic science and prevention of Nonvalvular Atrial Fibrillation, Persistent or Permanent Nonvalvular Atrial Fibrillation, and Persistent or Permanent Non-valvular Atrial Fibrillation.

Kategori:
Azetines
Target Protein:
Prothrombin
Waktu Paruh-
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Atelocollagen DB18450
biotech

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBiopolymersDrug Carriers +5
Waktu Paruh-
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Atenolol Approved DB00335
small molecule | CAS: 29122-68-7

Atenolol is a cardioselective beta-blocker used in a variety of cardiovascular conditions. Sir James Black, a Scottish pharmacologist, pioneered the use of beta-blockers for the management of angina pectoris in 1958 for which he received the Nobel Prize.[…

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-1 Receptor Antagonists +23
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptor
Gen Terkait:
ADRB1
Waktu Paruh6-7 hrs.[label]
Vol. DistribusiTotal Vd of 63.8-11…
KlirensTotal clearance is …
Genetik 1 Varian
Atevirdine DB12264
small molecule | CAS: 136816-75-6

Atevirdine has been used in trials studying the treatment of HIV Infections.

Kategori:
Anti-Infective AgentsAnti-Retroviral AgentsAntiviral Agents +3
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
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Atexakin alfa DB19234
biotech | CAS: 143631-61-2

Atexakin alfa is under investigation in clinical trial NCT05435742 (SON-080 in Patients With Persistent Chemotherapy-induced Peripheral Neuropathy (CIPN)).

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Atezolizumab Approved DB11595
biotech | CAS: 1380723-44-3

Atezolizumab is a humanized monoclonal antibody used to prevent the interaction of PD-L1 and PD-1, removing inhibition of immune responses seen in some cancers.[A18493,L7489] This medication is reserved for patients whose tumors express PD-L1, cannot receive …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +19
Target Protein:
Programmed cell death 1 ligand 1Programmed cell death protein 1
Waktu ParuhThe half life of at…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of at…
Genetik -
ATG-101 DB17162
biotech

ATG-101 is a novel PD-L1/4-1BB bispecific antibody that was designed to block the binding of immunosuppressive PD-1/PD-L1 and conditionally induce 4-1BB stimulation, thus activating anti-tumor immune effectors, while delivering enhanced anti-tumor activity, w…

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ATG-Fresenius S DB05320
small molecule

ATG-Fresenius S is a concentrated anti-human T-lymphocyte immunoglobulin preparation derived from rabbits after immunization with a T-lympoblast cell line. ATG-Fresenius S is an immunosuppressive product for the prevention and treatment of acute rejection fol…

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ATG002 DB05068
small molecule

ATG002 is a completely new approach to treating chronic wounds such as diabetic foot ulcers, which is based upon stimulation of angiogenesis in the wound bed to help drive the wound-healing process. Unlike protein-derived growth factors, ATG002 is a small mol…

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ATG003 DB05069
small molecule

ATG003, a novel anti-angiogenic drug candidate and a formulation of mecamylamine, is currently in clinical development for neovascular age-related macular degeneration.

Target Protein:
Neuronal acetylcholine receptor subunit alpha-10Neuronal acetylcholine receptor subunit alpha-9
Waktu Paruh-
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