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2677

Total database: 17430
Struktur (SMILES)
1588 (59.3%)
Target
1494 (55.8%)
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51 (1.9%)
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2677 (100.0%)

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Halaman 54 / 54
Zalcitabine Approved DB00943
small molecule | CAS: 7481-89-2

A dideoxynucleoside compound in which the 3'-hydroxyl group on the sugar moiety has been replaced by a hydrogen. This modification prevents the formation of 5' to 3' phosphodiester linkages, which are needed for the elongation of DNA chains, thus resulting in…

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +20
Target Protein:
Gag-Pol polyproteinReverse transcriptase/RNaseH
Waktu Paruh2 hours
Vol. Distribusi* 0.304 to 0.734 L/…
Klirens* 285 mL/min [HIV-i…
Genetik -
Zanidatamab Approved DB15471
biotech | CAS: 2169946-15-8

Zanidatamab is a bispecific antibody that binds two non-overlapping sites of HER2 (ERBB2).[A264718] It has been investigated for the treatment of HER2-positive solid tumors, including gastroesophageal, colorectal, and biliary tract cancers.[A264718] In No…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Target Protein:
Receptor tyrosine-protein kinase erbB-2
Waktu ParuhBased on population…
Vol. DistribusiBased on population…
KlirensBased on population…
Genetik -
Zanubrutinib Approved DB15035
small molecule | CAS: 1691249-45-2

Zanubrutinib is a novel Bruton's tyrosine kinase (BTK) inhibitor used for the treatment of adult patients with mantle cell lymphoma (MCL) who have received at least one prior therapy.[L10163] Mantle cell lymphoma is an aggressive mature B-cell non-Hodgkin lym…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBruton's tyrosine kinase (BTK) inhibitors +19
Target Protein:
Tyrosine-protein kinase BTKEpidermal growth factor receptorReceptor tyrosine-protein kinase erbB-2 +12
Waktu ParuhFollowing administr…
Vol. DistribusiThe geometric mean …
KlirensThe mean (%CV) appa…
Genetik -
Zavegepant Approved DB15688
small molecule | CAS: 1337918-83-8

Zavegepant (BHV-3500) is a calcitonin gene-related peptide (CGRP) receptor antagonist.[L45505] CGRP is released from sensory nerves and acts as a strong vasodilator, and thanks to these properties, it is involved in pain pathways. CGRP receptors are expressed…

Kategori:
Antimigraine PreparationsCalcitonin Gene-Related Peptide (CGRP) AntagonistsCalcitonin Gene-Related Peptide Receptor Antagonists +14
Target Protein:
Calcitonin gene-related peptide type 1 receptor
Waktu ParuhFollowing a 10 mg d…
Vol. DistribusiIntranasal zavegepa…
KlirensIntranasal zavegepa…
Genetik -
Zeaxanthin Approved DB11176
small molecule | CAS: 144-68-3

Zeaxanthin is a most common carotenoid alcohols found in nature that is involved in the xanthophyll cycle. As a coexistent isomer of lutein, zeaxanthin is synthesized in plants and some micro-organisms. It gives the distinct yellow color to many vegetables an…

Kategori:
AlkenesBiological FactorsCarotenoids +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zebularine DB03068
small molecule | CAS: 3690-10-6

A chemically stable, cytidine analog that displays anti-tumor properties. It acts as a transition state analog inhibitor of cytidine deaminase by binding to the active site as covalent hydrates. Also shown to inhibit DNA methylation and tumor growth both in v…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleosidesPyrimidine Nucleosides +2
Target Protein:
Cytidine deaminase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zelavespib DB12638
small molecule | CAS: 873436-91-0

Zelavespib (PU-H71) has been used in trials studying the treatment of LYMPHOMA, Solid Tumors, Metastatic Solid Tumor, and Myeloproliferative Neoplasms (MPN).

Kategori:
Antineoplastic AgentsDioxolesHeterocyclic Compounds, Fused-Ring
Target Protein:
Heat shock protein HSP 90-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zeluvalimab DB18868
biotech | CAS: 2315361-37-4

Zeluvalimab is under investigation in clinical trial NCT04631601 (Safety and Efficacy of Therapies for Metastatic Castration-resistant Prostate Cancer (Mcrpc)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zifibancimig DB19332
biotech | CAS: 2517939-46-5

Zifibancimig is under investigation in clinical trial NCT04567303, focusing on participants with neovascular age-related macular degeneration.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zileuton Approved DB00744
small molecule | CAS: 111406-87-2

Leukotrienes are substances that induce numerous biological effects including augmentation of neutrophil and eosinophil migration, neutrophil and monocyte aggregation, leukocyte adhesion, increased capillary permeability, and smooth muscle contraction. These …

Kategori:
Agents to Treat Airway DiseaseAmidesAnalgesics +19
Target Protein:
Polyunsaturated fatty acid 5-lipoxygenase
Waktu Paruh2.5 hours
Vol. Distribusi* 1.2 L/kg
Klirens* Apparent oral cl=…
Genetik -
Zinc Approved DB01593
small molecule | CAS: 7440-66-6

A metallic element of atomic number 30 and atomic weight 65.38. It is a necessary trace element in the diet, forming an essential part of many enzymes, and playing an important role in protein synthesis and in cell division. Zinc deficiency is associated with…

Kategori:
Agents for Treatment of Hemorrhoids and Anal Fissures for Topical UseDiet, Food, and NutritionElements +12
Target Protein:
B1 bradykinin receptorMethylated-DNA--protein-cysteine methyltransferaseFructose-bisphosphate aldolase A +121
Waktu ParuhThe half-life of zi…
Vol. DistribusiA pharmacokinetic s…
KlirensIn one study of hea…
Genetik -
Zinc citrate DB11154
small molecule | CAS: 546-46-3

Zinc citrate is a zinc salt of citric acid. It is available as dietary supplements as a treatment of zinc deficiency and source of zinc, which is an essential trace element. Zinc citrate demonstrates effective absorption following oral administration [A27280].

Kategori:
Metal cationsMetal divalent cationsZinc Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zinc gluconate Approved DB11248
small molecule | CAS: 4468-02-4

Zinc gluconate is a zinc salt of gluconic acid comprised of two gluconic acid molecules for each zinc cation (2+). Zinc gluconate is a generally recognized as safe (GRAS) substance by FDA [L2081]. It is available as a trace mineral supplement and over the cou…

Kategori:
Acids, AcyclicAgents for Treatment of Hemorrhoids and Anal Fissures for Topical UseAlimentary Tract and Metabolism +8
Waktu Paruh280 days [L2091]
Vol. DistribusiStored primarily in…
KlirensPlease refer to Dru…
Genetik -
small molecule | CAS: 955009-96-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 62008-21-3

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicDermatologicalsDicarboxylic Acids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zinc picolinate DB11175
small molecule | CAS: 17949-65-4

Zinc picolinate is a zinc salt of picolinic acid. It is available as OTC dietary supplements as a source of zinc to treat and prevent zinc deficiency. The absorption of zinc after oral administration of zinc picolinate is shown to be effective.

Kategori:
Compounds used in a research, industrial, or household settingMetal cationsMetal divalent cations +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Zinc sulfate is a common zinc supplement in parenteral nutrition.[A216916,L12888]

Kategori:
Agents for Treatment of Hemorrhoids and Anal Fissures for Topical UseMetal cationsMetal divalent cations +2
Target Protein:
B1 bradykinin receptorMethylated-DNA--protein-cysteine methyltransferaseFructose-bisphosphate aldolase A +94
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ziprasidone Approved DB00246
small molecule | CAS: 146939-27-7

Disorders such as schizophrenia and bipolar disorder can significantly impair mood, cognition, and behavior.[A190525] These mental illnesses can often be accompanied by comorbidities such as depression and substance abuse, and can significantly impact the qua…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +45
Target Protein:
D(2) dopamine receptorNeuronal acetylcholine receptor subunit alpha-75-hydroxytryptamine receptor 2A +24
Waktu ParuhThe half life of zi…
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent s…
Genetik -
Zirconium chloride hydroxide Approved DB15479
small molecule | CAS: 10119-31-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1323976-37-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zoledronic acid Approved DB00399
small molecule | CAS: 118072-93-8

Zoledronic acid, or CGP 42'446,[A203120] is a third generation, nitrogen containing bisphosphonate similar to [ibandronic acid], [minodronic acid], and [risedronic acid].[A203111] Zoledronic acid is used to treat and prevent multiple forms of osteoporosis, hy…

Kategori:
BisphosphonatesBone Density Conservation AgentsDrugs Affecting Bone Structure and Mineralization +5
Target Protein:
Geranylgeranyl pyrophosphate synthaseHydroxylapatiteFarnesyl pyrophosphate synthase
Waktu ParuhZoledronic acid has…
Vol. Distribusi-
KlirensZoledronic acid has…
Genetik -
Zolmitriptan Approved DB00315
small molecule | CAS: 139264-17-8

Zolmitriptan is a member of the triptan class of 5-hydroxytryptamine(5-HT)<sub>1B/1D/(1F)</sub> receptor agonists used to treat acute migraine.[A462, L12978] [Sumatriptan] was the first triptan to be developed, but had poor oral bioavailability and lipophilic…

Kategori:
Agents that produce hypertensionAminesAnalgesics +24
Target Protein:
5-hydroxytryptamine receptor 1B5-hydroxytryptamine receptor 1D5-hydroxytryptamine receptor 1F +5
Gen Terkait:
GNB3
Waktu ParuhZolmitriptan has a …
Vol. DistribusiZolmitriptan has a …
KlirensZolmitriptan has a …
Genetik 1 Varian
Zolpidem Approved DB00425
small molecule | CAS: 82626-48-0

Zolpidem, also known as _Ambien_, is a hypnotic drug that was initially approved by the FDA in 1992 [FDA label]. Zolpidem improves sleep in patients with insomnia. It is aimed for use in patients with difficulties initiating sleep. This drug decreases the ti…

Kategori:
Benzodiazepine hypnotics and sedativesCentral Nervous System AgentsCentral Nervous System Depressants +21
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Gamma-aminobutyric acid receptor subunit gamma-3Gamma-aminobutyric acid receptor subunit alpha-2 +2
Waktu ParuhThe average zolpide…
Vol. Distribusi0.54 to 0.68 L/kg (…
KlirensIn a clinical trial…
Genetik -
Zopiclone Approved DB01198
small molecule | CAS: 43200-80-2

Zopiclone is a novel hypnotic agent used in the treatment of insomnia. Its mechanism of action is based on modulating benzodiazepine receptors. In addition to zopiclone's benzodiazepine pharmacological properties it also has some barbiturate-like properties.

Kategori:
Aza CompoundsBenzodiazepine hypnotics and sedativesCentral Nervous System Agents +16
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Gamma-aminobutyric acid receptor subunit alpha-2Gamma-aminobutyric acid receptor subunit alpha-3 +2
Waktu ParuhElimination half li…
Vol. Distribusi-
Klirens-
Genetik -
Zorubicin DB11618
small molecule | CAS: 54083-22-6

Zorubicin is a drug of the anthracycline class - a class of medications that have historically demonstrated effective chemotherapy for a variety of cancer types.

Kategori:
AnthracyclinesAnthracyclines and Related SubstancesAntibiotics, Antineoplastic +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zunsemetinib DB16502
small molecule | CAS: 1640282-42-3

ATI-450 was under investigation in clinical trials (NCT05279417 and NCT05216224) for treating patients with rheumatoid arthritis and hidradenitis suppurativa, respectively. Additionally, ATI-450 was studied in a terminated trial (NCT05511519) to treat patient…

Kategori:
Experimental Unapproved Treatments for COVID-19
Target Protein:
MAP kinase-activated protein kinase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ZYCOV-D DB15892
biotech

The ZYCOV-D vaccine candidate was developed by Cadila Healthcare Ltd. based in India[A219758]. The vaccine was developed using a DNA vaccine platform with a non-replicating and non-integrating plasmid carrying the gene of interest[L16503]. Once the plasmid D…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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