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16749

Total database: 17430
Struktur (SMILES)
11810 (70.5%)
Target
9015 (53.8%)
Genomik
112 (0.7%)
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16749 (100.0%)

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Hasil Pencarian (16749)

Halaman 53 / 335
Abaloparatide Approved DB05084
biotech | CAS: 247062-33-5

Abaloparatide is an N-terminal analog of parathyroid hormone-related protein (PTHrP) [A256778] and an agonist at the parathyroid hormone type 1 (PTH1) receptor.[L740] It is a synthetic 34 amino acid peptide with 41% homology to human parathyroid hormone 1-34 …

Kategori:
Amino Acids, Peptides, and ProteinsAnalogs/DerivativesBiological Factors +13
Target Protein:
Parathyroid hormone/parathyroid hormone-related peptide receptor
Waktu ParuhThe mean half-life …
Vol. DistribusiThe volume of distr…
KlirensThe mean apparent t…
Genetik -
Abametapir Approved DB11932
small molecule | CAS: 1762-34-1

Abametapir is a novel pediculicidal metalloproteinase inhibitor used to treat infestations of head lice.[L15153] The life cycle of head lice (_Pediculus capitis_) is approximately 30 days, seven to twelve of which are spent as eggs laid on hair shafts near th…

Kategori:
Antiparasitic Products, Insecticides and RepellentsCytochrome P-450 CYP1A2 InhibitorsCytochrome P-450 CYP1A2 Inhibitors (strength unknown) +13
Waktu ParuhThe elimination hal…
Vol. DistribusiData regarding the …
KlirensThe clearance and e…
Genetik -
Abarelix Approved DB00106
small molecule | CAS: 183552-38-7

Synthetic decapeptide antagonist to gonadotropin releasing hormone (GnRH). It is marketed by Praecis Pharmaceuticals as Plenaxis. Praecis announced in June 2006 that it was voluntarily withdrawing the drug from the market.

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating AgentsEndocrine Therapy +4
Target Protein:
Gonadotropin-releasing hormone receptor
Waktu Paruh13.2 ± 3.2 d…
Vol. Distribusi-
Klirens-
Genetik -
Abatacept Approved DB01281
biotech | CAS: 332348-12-6

Abatacept is a soluble fusion protein, which links the extracellular domain of human cytotoxic T-lymphocyte-associated antigen 4 (CTLA-4) to the modified Fc (hinge, CH2, and CH3 domains) portion of human immunoglobulin G1 (IgG1).[L20504,L42715] Structurally, …

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAntibodies +18
Target Protein:
T-lymphocyte activation antigen CD80T-lymphocyte activation antigen CD86Cytotoxic T-lymphocyte protein 4
Waktu Paruh16.7 (12-23) days i…
Vol. Distribusi* 0.07 L/kg [RA Pat…
Klirens* 0.23 mL/h/kg [Hea…
Genetik -
ABBV-011 DB18622
biotech

ABBV-011 is an antibody-drug conjugate of humanized, cysteine-engineered IgG1 monoclonal antibody targeting seizure-related 6 homolog conjugated to N-acetyl-gamma-calicheamicin.

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ABBV-514 DB17586
biotech

ABBV-514 is in development for the treatment of non-small cell lung cancer (NSCLC) and head and neck squamous cell carcinoma (HNSCC) as a single agent and in combination with a PD-1 inhibitor.[L45464]

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ABBV-706 DB18710
biotech

ABBV-706 is an antibody-drug conjugate that is anti-SEZ6.[L49156,L49161]

Waktu Paruh-
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ABBV-744 DB19199
small molecule | CAS: 2138861-99-9

Deskripsi belum tersedia.

Target Protein:
Bromodomain-containing protein 3Bromodomain-containing protein 2Bromodomain-containing protein 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ABBV-CLS-7262 DB18407
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
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Abciximab Approved DB00054
biotech | CAS: 143653-53-6

Abciximab is a Fab fragment of the chimeric human-murine monoclonal antibody 7E3. Abciximab binds to the glycoprotein (GP) IIb/IIIa receptor of human platelets and inhibits platelet aggregation by preventing the binding of fibrinogen, von Willebrand factor, a…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +18
Target Protein:
Integrin beta-3Integrin alpha-IIbLow affinity immunoglobulin gamma Fc region receptor II-a +2
Waktu ParuhFollowing intraveno…
Vol. Distribusi-
Klirens-
Genetik -
Abediterol DB12100
small molecule | CAS: 915133-65-2

Abediterol has been used in trials studying the treatment of Asthma, Chronic Obstructive Pulmonary Disease (COPD), and Chronic Obstructive Pulmonary Disease (COPD) and Asthma.

Kategori:
Adrenergic AgonistsAdrenergic beta-2 Receptor AgonistsAdrenergic beta-Agonists +4
Target Protein:
Beta-2 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Abelacimab DB16682
biotech | CAS: 2098724-83-3

Abelacimab is under investigation in clinical trial NCT04755283 (Safety and Tolerability of Abelacimab (MAA868) vs. Rivaroxaban in Patients With Atrial Fibrillation).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Abemaciclib Approved DB12001
small molecule | CAS: 1231929-97-7

Abemaciclib is an antitumor agent and dual inhibitor of cyclin-dependent kinases 4 (CDK4) and 6 (CDK6) that are involved in the cell cycle and promotion of cancer cell growth in case of unregulated activity. On September 28, 2017, FDA granted approval of abem…

Kategori:
AminesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +36
Target Protein:
Cyclin-dependent kinase 4Cyclin-dependent kinase 6
Waktu ParuhThe mean plasma eli…
Vol. DistribusiThe geometric mean …
KlirensThe geometric mean …
Genetik -
Abeprazan DB16078
small molecule | CAS: 1902954-60-2

Abeprazan is under investigation in clinical trial NCT04341454 (Study to Evaluate the Efficacy and Safety of DWP14012 in Patients With Acute or Chronic Gastritis).

Kategori:
Gastrointestinal Agents
Waktu Paruh-
Vol. Distribusi-
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Abequolixron DB17146
small molecule | CAS: 610318-54-2

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicBenzene Derivatives
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Abequose DB02590
small molecule | CAS: 56816-60-5

Deskripsi belum tersedia.

Kategori:
CarbohydratesMonosaccharides
Target Protein:
Tail fiber protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Abetimus DB06662
biotech | CAS: 167362-48-3

Abetimus was developed by La Jolla Pharmaceuticals as an immunosuppressant but was never marketed in American or Europe despite application for marketing authorization in the mid-2000s.

Kategori:
Antineoplastic and Immunomodulating AgentsImmunologic FactorsImmunosuppressive Agents +4
Waktu Paruh-
Vol. Distribusi-
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Abexinostat DB12565
small molecule | CAS: 783355-60-2

Abexinostat has been used in trials studying the treatment of Sarcoma, Lymphoma, Leukemia, Lymphocytic, and Hodgkin Disease, among others. It is a novel, broad-spectrum hydroxamic acid-based inhibitor of histone deacetylase (HDAC) with potential antineoplasti…

Kategori:
AminesAntineoplastic AgentsEnzyme Inhibitors +6
Target Protein:
Histone deacetylase 1Histone deacetylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ABG-023 DB18829
biotech

ABG-023 is a glucagon analog which is soluble and solution-stable.[L50778]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ABH001 DB16177
small molecule | CAS: 502-97-6

ABH001 is under investigation in clinical trial NCT01749306 (A Study of the Efficacy and Safety of ABH001 in the Treatment of Patients With Epidermolysis Bullosa Who Have Wounds That Are Not Healing).

Waktu Paruh-
Vol. Distribusi-
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Abicipar Pegol DB12258
biotech | CAS: 1327278-94-3

Abicipar Pegol has been used in trials studying the treatment of Macular Edema and Macular Degeneration.

Kategori:
Amino Acids, Peptides, and ProteinsAntineovascularisation AgentsOcular Vascular Disorder Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Abiprubart DB19333
biotech | CAS: 2765071-95-0

Abiprubart is being evaluated for its efficacy and safety in participants with Sjögren's Disease in clinical trial NCT06531395

Waktu Paruh-
Vol. Distribusi-
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Abiraterone Approved DB05812
small molecule | CAS: 154229-19-3

Abiraterone is a potent, irreversible, and selective inhibitor of 17 ?hydroxylase/C17,20-lyase (CYP17), an enzyme expressed in testicular, adrenal, and prostatic tumour tissues, to regulate androgen biosynthesis.[A3811, A260880, L40968] Abiraterone was first …

Kategori:
AndrostanesAndrostenesAntineoplastic Agents +32
Target Protein:
Steroid 17-alpha-hydroxylase/17,20 lyase
Waktu ParuhIn patients with mC…
Vol. DistribusiThe mean (± SD) app…
Klirens-
Genetik -
small molecule | CAS: 2486052-18-8

Abiraterone decanoate is under investigation in clinical trial NCT04729114 (Open-label, Multicenter Study of Intramuscular PRL-02 Depot in Patients With Advanced Prostate Cancer).

Kategori:
Cytochrome P450 17A1 Inhibitors
Waktu Paruh-
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Abituzumab DB12775
biotech | CAS: 1105038-73-0

Abituzumab has been used in trials studying the treatment of Prostate Cancer Metastatic.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Abivertinib DB15327
small molecule | CAS: 1557267-42-1

Abivertinib is a tyrosine kinase inhibitor targeted against mutant forms of both human epidermal growth factor receptor (EGFR) and Bruton's tyrosine kinase (BTK).[L17383] It has been investigated for use in the treatment of non-small cell lung cancer (NSCLC) …

Kategori:
Acids, AcyclicAcrylatesAmides +4
Target Protein:
Epidermal growth factor receptorTyrosine-protein kinase BTK
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ABO-201 DB17951
biotech

Deskripsi belum tersedia.

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ABP-700 DB15411
small molecule | CAS: 1446482-29-6

ABP-700 is under investigation in clinical trial NCT02800590 (Study to Investigate the Safety and Efficacy of 3 Dosing Regimens of ABP-700 for Procedural Sedation in Adult Participants Undergoing Colonoscopy).

Kategori:
GABA AgentsGABA AgonistsGABA-A Receptor Agonists +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Abrilumab DB15076
biotech | CAS: 1342290-43-0

Abrilumab is under investigation in clinical trial NCT01290042 (Study to Evaluate Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of AMG 181.).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Abrocitinib Approved DB14973
small molecule | CAS: 1622902-68-4

Abrocitinib is an oral small-molecule inhibitor of Janus kinase 1 (JAK1). Janus kinases are intracellular enzymes involved in transduction pathways that regulate hematopoiesis and immune cell function.[L39774] The Janus kinase (JAK)–signal transducer and acti…

Kategori:
Agents for Dermatitis, Excluding CorticosteroidsAmidesCytochrome P-450 CYP2B6 Substrates +17
Target Protein:
Tyrosine-protein kinase JAK1Tyrosine-protein kinase JAK2Tyrosine-protein kinase JAK3 +1
Waktu ParuhThe mean eliminatio…
Vol. DistribusiAfter intravenous a…
KlirensThere is no informa…
Genetik -
Abscisic Acid DB16829
small molecule | CAS: 21293-29-8

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAlkenesCarotenoids +11
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Absidia capillata Approved DB10972
biotech

Absidia capillata allergenic extract is used in allergenic testing.

Waktu Paruh-
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Genetik -
ABSK-012 DB18035
small molecule | CAS: 2271209-99-3

Deskripsi belum tersedia.

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ABSK-091 DB18442
small molecule | CAS: 1035270-39-3

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesAntineoplastic Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ABT-072 DB15156
small molecule | CAS: 1132936-00-5

ABT-072 is under investigation in clinical trial NCT00890318 (A Study in Healthy Adult Subjects to Evaluate the Safety, Tolerability, and Pharmacokinetic Profiles of Multiple Doses of ABT-072 Used to Treat Hepatitis C).

Kategori:
AmidesPyrimidinesPyrimidinones +2
Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
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Genetik -
ABT-288 DB15192
small molecule | CAS: 948845-91-8

ABT-288 is under investigation in clinical trial NCT01018875 (Efficacy and Safety Study of ABT-288 in Subjects With Mild-to-Moderate Alzheimer's Disease).

Kategori:
Histamine Antagonists
Target Protein:
Histamine H3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ABT-341 DB08044
small molecule | CAS: 913623-69-5

ABT-341 is a potent and selective DPP-4 inhibitor with a structure very similar to sitagliptin (in 2D; the 3D structure is significantly different). [A39406]

Kategori:
Benzene DerivativesEnzyme InhibitorsProtease Inhibitors
Target Protein:
Dipeptidyl peptidase 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ABT-384 DB12501
small molecule | CAS: 868623-40-9

ABT-384 has been used in trials studying the treatment of Alzheimer's Disease.

Kategori:
11-beta-Hydroxysteroid Dehydrogenase Type 1, antagonists & inhibitorsBridged-Ring CompoundsCycloparaffins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ABT-510 DB05434
small molecule | CAS: 251579-55-2

ABT-510 is a peptide mimetic of thrombospondin-1 (TSP-1), blocks angiogenesis in vitro and in vivo, and slows tumor growth. It is developed by Abbott Laboratories for the treatment of Solid Tumors, Lymphoma and Melanoma.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Target Protein:
Thrombospondin-1Fibroblast growth factor 2Hepatocyte growth factor +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ABT-560 DB06093
small molecule

ABT-560 is a neuronal nicotinic receptor (NNR) modulator, which has shown promise in preclinical models relevant for the treatment of cognitive deficits.

Waktu Paruh-
Vol. Distribusi-
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ABT-639 DB15055
small molecule | CAS: 1235560-28-7

ABT-639 is under investigation in clinical trial NCT01345045 (A Multicenter Study Comparing the Analgesic Effects and Safety of ABT-639 Compared to Placebo in Subjects With Diabetic Neuropathic Pain).

Kategori:
AmidesBenzene DerivativesHeterocyclic Compounds, Fused-Ring +3
Target Protein:
Voltage-dependent T-type calcium channel subunit alpha-1H
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ABT-737 DB17023
small molecule | CAS: 852808-04-9

An inhibitor of members of the Bcl?2 family of apoptosis regulators.[A252977]

Kategori:
AmidesBenzene DerivativesNitro Compounds +4
Target Protein:
Apoptosis regulator Bcl-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ABT-751 DB12254
small molecule | CAS: 141430-65-1

ABT-751 has been investigated for the treatment of Lung Cancer, Non-Small Cell Lung Cancer, and Non-Small-Cell Lung Cancer.

Kategori:
AmidesAminesAniline Compounds +5
Waktu Paruh-
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Genetik -
ABX-002 DB18157
small molecule | CAS: 2156649-32-8

Deskripsi belum tersedia.

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ABX-1431 DB16036
small molecule | CAS: 1446817-84-0

ABX-1431 is under investigation in clinical trial NCT03625453 (Study of ABX-1431 in Adult Patients With Tourette Syndrome or Chronic Motor Tic Disorder).

Target Protein:
Monoglyceride lipase
Waktu Paruh-
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ABX-196 DB16339
small molecule | CAS: 1161877-58-2

ABX-196 is under investigation in clinical trial NCT03897543 (ABX196 in Combination With Nivolumab in Patients With Hepatocellular Carcinoma).

Kategori:
AmidesCarbohydratesCeramides +8
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Genetik -
ABX-464 DB14828
small molecule | CAS: 1258453-75-6

ABX-464 is under investigation in clinical trial NCT03905109 (Safety Evaluation of ABX464 in Patients With Moderate to Severe Active Crohn's Disease).

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
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ABX-PTH DB05883
biotech

ABX-PTH is a fully human monoclonal antibody generated by Abgenix's technology platform. This drug targets and neutralizes the action of parathyroid hormone (PTH) for the treatment of a secondary hyperparathyroidism.

Target Protein:
Parathyroid hormone
Waktu Paruh-
Vol. Distribusi-
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Genetik -
ABX1100 DB17655
biotech

ABX1100 is an investigational Centyrin-siRNA conjugate that targets the Gys1 gene, which encodes glycogen synthase 1 (Gys1), an enzyme that is responsible for glycogen synthesis in the muscle. It was first developed by Aro Biotherapeutics and is being investi…

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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Prothrombin
Waktu Paruh-
Vol. Distribusi-
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Genetik -
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