Hasil Filter

11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (11778)

Halaman 53 / 236
Barasertib DB11747
small molecule | CAS: 722543-31-9

Barasertib has been used in trials studying the treatment of Tumors, Lymphoma, Solid Tumors, Solid Tumours, and Myeloid Leukemia, among others.

Kategori:
Heterocyclic Compounds, Fused-RingOrganophosphorus CompoundsProtein Kinase Inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Barbexaclone DB09001
small molecule | CAS: 4388-82-3

Barbexaclone, a salt compound of propylhexedrine and phenobarbital, is a potent antiepileptic. By weight, barbexaclone is 40% propylhexedrine and 60% phenobarbital. While barbexaclone has sedative properties, propylhexedrine has psychostimulant properties in…

Kategori:
AnticonvulsantsBarbituratesBarbiturates and Derivatives +8
Waktu ParuhAfter IV administra…
Vol. DistribusiIn mice, the volume…
Klirens-
Genetik -
Barbital DB01483
small molecule | CAS: 57-44-3

A long-acting barbiturate that depresses most metabolic processes at high doses. It is used as a hypnotic and sedative and may induce dependence. Barbital is also used in veterinary practice for central nervous system depression. Barbital is a schedule IV con…

Kategori:
Anticholinergic AgentsAnticonvulsantsBarbiturates +20
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Gamma-aminobutyric acid receptor subunit alpha-2Gamma-aminobutyric acid receptor subunit alpha-3 +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Barecetamab DB17479
biotech | CAS: 2275727-74-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Baricitinib Approved DB11817
small molecule | CAS: 1187594-09-7

Baricitinib is a Janus kinase (JAK) inhibitor. JAKs are tyrosine protein kinases that play an important role in pro-inflammatory signaling pathways. Overactive JAKs have been implicated in autoimmune disorders, such as rheumatoid arthritis. By inhibiting the …

Kategori:
AmidesAntineoplastic and Immunomodulating AgentsAntirheumatic Agents +31
Target Protein:
Tyrosine-protein kinase JAK1Tyrosine-protein kinase JAK2Tyrosine-protein kinase JAK3 +1
Waktu ParuhThe elimination hal…
Vol. DistribusiFollowing intraveno…
KlirensThe total body clea…
Genetik -
Barium DB12481
small molecule | CAS: 7440-39-3

Barium is under investigation for the diagnostic of Known or Suspected Abdominal Disease.

Kategori:
ElementsMetalsMetals, Alkaline Earth +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Barium sulfate Approved DB11150
small molecule | CAS: 7727-43-7

Barium sulfate is an inorganic compound with the chemical formula BaSO4 [L1957]. Barium sulfate occurs in nature as the mineral _barite_. It is also used in various manufacturing applications and mixed into heavy concrete to serve as a radiation shield [L1…

Kategori:
Barium CompoundsBarium Sulfate Containing X-Ray Contrast MediaCompounds used in a research, industrial, or household setting +9
Waktu Paruh-
Vol. Distribusi-
KlirensThe rate of excreti…
Genetik -
Barnidipine DB09227
small molecule | CAS: 104713-75-9

Barnidipine is a long-acting novel calcium antagonist that belongs to the dihydropyridine (DHP) group of calcium channel blockers. Used in the treatment of hypertension, barnidipine displays high affinity for the calcium channels of the smooth muscle cells in…

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsBradycardia-Causing Agents +17
Target Protein:
Voltage-dependent L-type calcium channel subunit alpha-1CVoltage-dependent T-type calcium channel subunit alpha-1GVoltage-dependent T-type calcium channel subunit alpha-1H
Waktu ParuhIn a two-compartmen…
Vol. DistribusiAfter administratio…
Klirens-
Genetik -
Barusiban DB12292
small molecule | CAS: 285571-64-4

Barusiban has been used in trials studying the treatment of Infertility and In Vitro Fertilisation (IVF) Treatment.

Kategori:
Amino Acids, Peptides, and ProteinsPeptidesReceptors, Oxytocin, antagonists & inhibitors
Target Protein:
Oxytocin receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Basifungin DB14058
small molecule | CAS: 127785-64-2

Basifungin, also known as _aureuobacidin A_, is a phosphorylceramide synthase inhibitor [L2960], [A33381].

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntifungal Agents +3
Target Protein:
Inositol phosphorylceramide synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Basiliximab Approved DB00074
biotech | CAS: 179045-86-4

A recombinant chimeric (murine/human) monoclonal antibody (IgG1k) that functions as an immunosuppressive agent, specifically binding to and blocking the interleukin-2 receptor a-chain (IL-2R alpha, also known as CD25 antigen) on the surface of activated T-lym…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +14
Target Protein:
Interleukin-2 receptor subunit alphaInterleukin-2 receptor subunit beta
Waktu Paruh7.2 +/- 3.2 days (a…
Vol. Distribusi* 7.8 ± 5.1 L [Pedi…
Klirens* 41 +/- 19 mL/h [A…
Genetik -
Basimglurant DB11833
small molecule | CAS: 802906-73-6

Basimglurant has been used in trials studying the diagnostic and treatment of Depression, Fragile X Syndrome, and Major Depressive Disorder.

Target Protein:
Metabotropic glutamate receptor 5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Basmisanil DB11877
small molecule | CAS: 1159600-41-5

Basmisanil has been used in trials studying the treatment and basic science of Down Syndrome.

Kategori:
Oxazines
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Batabulin DB16103
small molecule | CAS: 195533-53-0

Batabulin is under investigation in clinical trial NCT00057382 (T138067 Versus Doxorubicin in Chemotherapy-naive, Unresectable, Hepatocellular Carcinoma Patients).

Kategori:
AmidesBenzene DerivativesHydrocarbons, Fluorinated +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Batefenterol DB12526
small molecule | CAS: 743461-65-6

Batefenterol has been used in trials studying the treatment of Pulmonary Disease, Chronic Obstructive.

Kategori:
Acids, AcyclicAdrenergic AgonistsAdrenergic beta-2 Receptor Agonists +5
Target Protein:
Beta-2 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Batimastat DB03880
small molecule | CAS: 130370-60-4

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +6
Target Protein:
Stromelysin-1Disintegrin and metalloproteinase domain-containing protein 28A disintegrin and metalloproteinase with thrombospondin motifs 5 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Batiraxcept DB17522
biotech | CAS: 2268717-61-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Batoclimab DB16104
biotech | CAS: 2187430-05-1

Batoclimab is under investigation in clinical trial NCT04428255 (A Clinical Study on the Efficacy and Safety of HBM9161 in Patients With ITP).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Batoprotafib DB19137
small molecule | CAS: 1801765-04-7

Batoprotafib is under investigation in clinical trial NCT04330664 (Adagrasib in Combination With TNO155 in Patients With Cancer (KRYSTAL 2)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Batroxobin DB09005
biotech | CAS: 9039-61-6

Batroxobin is a defibrinogenating hemostatic agent derived from the venom of a pit viper, Bothrops atrox moojeni. In addition to batroxobin, the venom of Bothrops atrox has a composition of 10.2% neutral carbohydrate. Batroxobin is a serine protease, which cl…

Kategori:
Biological FactorsBlood and Blood Forming OrgansCardiovascular Agents +18
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bavdegalutamide DB19032
small molecule | CAS: 2222112-77-6

Bavdegalutamide is under investigation in clinical trial NCT03888612 (Trial of ARV-110 in Patients With Metastatic Castration Resistant Prostate Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BAX 335 DB17845
biotech

BAX 335 is an adeno-associated virus vector 8 (AAV8)–based FIX gene therapy being investigated for the treatment of hemophilia B.[A259791]

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Baxdrostat DB19090
small molecule | CAS: 1428652-17-8

Baxdrostat is under investigation in clinical trial NCT06344104 (A Phase III Study to Investigate the Efficacy and Safety of Baxdrostat in Asian Participants With Uncontrolled Hypertension on Two or More Medications Including Participants With Resistant Hyper…

Target Protein:
Cytochrome P450 11B2, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BAY-876 DB16758
small molecule | CAS: 1799753-84-6

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bazlitoran DB14990
biotech | CAS: 1378549-07-5

Bazlitoran is under investigation in clinical trial NCT02092909 (Phase 1/2 Dose Escalation Study in Patients With Relapsed or Refractory Waldenstrom's Macroglobulinemia).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BB 21217 DB17373
biotech

BB 21217 is an anti-BCMA CAR T cell therapy that uses the same CAR molecule as [idecabtagene vicleucel] (bb2121), but adds the PI3K inhibitor bb007 during ex vivo culture to enrich the drug product (DP) for memory-like T cells.[L44291]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BB-1701 DB17443
biotech

BB-1701 is a humanized IgG1 kappa monoclonal antibody (anti-HER2 antibody) conjugated to eribulin developed by Bliss Biopharmaceutical.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BB-301 DB17011
biotech

BB-301 is a modified AAV serotype 9 (AAV9) capsid expressing a unique, single bifunctional construct promoting co-expression of both codon-optimized Poly-A Binding Protein Nuclear-1 (PABPN1) and two small inhibitory RNAs (siRNAs) against mutant PABPN1.[A26011…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bb-3497 DB04368
small molecule | CAS: 235784-88-0

Deskripsi belum tersedia.

Kategori:
AminesHydroxy AcidsHydroxylamines
Target Protein:
Peptide deformylasePeptide deformylasePeptide deformylase, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BBIBP-CorV DB15807
biotech

BBIBP-CorV vaccine contains a SARS-CoV-2 strain inactivated inside Vero Cells. Investigation shows this vaccine induces neutralizing antibodies in several mammalian species while also showing protective efficacy with SARS-CoV-2 challenge in rhesus macaques[A2…

Kategori:
Biological ProductsComplex MixturesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BBM-H803 DB17700
biotech

BBM-H803 is a recombinant adeno-associated virus (AAV) based gene therapy drug for hemophilia A developed and manufactured by Belief BioMed. It consists of an adeno-associated virus vector containing an expression cassette of the human Factor VIII transgene.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BBM-H901 DB17704
biotech

BBM-H901 is a liver-tropic adeno-associated viral (AAV) vector carrying cassette coding hyperactive Padua factor IX (FIX) protein. It is being investigated for the treatment of hemophilia B.[A259048]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BBP-671 DB18498
small molecule

BBP-671 is a small molecule activator of pantothenate kinases.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BBP-711 DB18199
small molecule

BBP-711 is a glycolate oxidase inhibitor.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BBT-877 DB18668
small molecule

BBT-877 is an autotaxin enzyme inhibitor being investigated for the treatment of fibrotic diseases, such as idiopathic pulmonary fibrosis.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BBV152 DB15847
biotech

BBV152 is a vaccine candidate created by the Indian Council of Medical Research (ICMR). The candidate, a whole virion inactivated SARS-CoV-2 vaccine, was developed from a well-known SARS-CoV-2 strain and a vero cell platform (CCL-81) with adjuncts of either a…

Kategori:
Biological ProductsComplex MixturesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BC9KBY85WY DB17820
small molecule | CAS: 1259013-14-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BCG vaccine Approved DB12768
biotech

BCG vaccine has been investigated for the treatment of Neoplasms, Bladder Cancer, Neoplasms by Site, Urologic Diseases, and Urologic Neoplasms, among others.

Kategori:
Adjuvants, ImmunologicAntineoplastic and Immunomodulating AgentsBacterial Vaccines +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BCL-005 DB17242
biotech

BCL-005 is a product formed by fused (hybrid) melanoma-dendritic cells.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BD-111 DB18247
biotech

BD-111 is an HSV-1-erasing lentivirus-like particle delivering gRNA-expressing cassette and SpCas9 mRNA.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BDB-001 DB16480
biotech

BDB-001, was under investigation in multiple clinical trials to evaluate its safety, tolerability, and efficacy across various conditions. In NCT05075304 and NCT04449588, BDB-001 was studied in mild to severe COVID-19 patients. It was also explored for solid …

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BDBM249432 DB17119
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BEA-17 DB18574
small molecule

BEA-17 is a small molecule targeted degrader of the epigenetic enzyme LSD1 and its co-factor CoREST.[L48330] It is under investigation for the treatment of glioblastoma.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bean Approved DB14709
biotech

Bean allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bebtelovimab DB16755
biotech | CAS: 2578319-11-4

Bebtelovimab (LY-COV1404, LY-3853113) is a human monoclonal antibody approved for emergency use in the treatment of COVID-19. It binds to a portion of the SARS-CoV-2 spike (S) protein's receptor-binding domain, thereby preventing spike protein interaction wit…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesApproved Treatments for COVID-19 +6
Target Protein:
Spike glycoprotein
Waktu ParuhFollowing a single …
Vol. DistribusiAt steady-state, th…
KlirensFollowing a single …
Genetik -
Becatecarin DB06362
small molecule | CAS: 119673-08-4

Becatecarin is a derivative of [rebeccamycin].

Kategori:
CarbohydratesGlycosidesHeterocyclic Compounds, Fused-Ring +1
Target Protein:
DNA topoisomerase 1DNA topoisomerase 2-alphaDNA topoisomerase 2-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Beclanorsen DB05606
small molecule | CAS: 1072859-54-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 5534-18-9

An ester of beclomethasone.

Kategori:
Adrenal Cortex HormonesCorticosteroidsFused-Ring Compounds +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Beclomethasone dipropionate Approved DB00394
small molecule | CAS: 5534-09-8

Beclomethasone dipropionate is a second-generation[A179842] synthetic corticosteroid and diester of beclomethasone, which is structurally similar to [dexamethasone].[L6871] It is a prodrug of an active metabolite beclomethasone 17-monopropionate (17-BMP)[A179…

Kategori:
Adrenal Cortex HormonesAdrenalsAgents to Treat Airway Disease +40
Target Protein:
Glucocorticoid receptor
Waktu ParuhFollowing intraveno…
Vol. DistribusiFollowing intraveno…
KlirensFollowing intraveno…
Genetik -
Becocalcidiol DB04891
small molecule | CAS: 524067-21-8

Becocalcidiol is a vitamin D(3) analogue which has not caused hypercalcaemia or significant irritation in preclinical trials.

Kategori:
CholestanesCholestenesFused-Ring Compounds +8
Target Protein:
Mediator of RNA polymerase II transcription subunit 1Vitamin D3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 2601–2650 dari 11778
Sebelumnya Halaman 53 / 236 Berikutnya