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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
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14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 53 / 282
Alcloxa Approved DB11205
small molecule | CAS: 1317-25-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Alcuronium DB13648
small molecule | CAS: 23214-96-2

A non-depolarizing skeletal muscle relaxant similar to [tubocurarine]. It is used as an anesthesia adjuvant.

Kategori:
Adjuvants, AnesthesiaAlkaloidsAmines +21
Target Protein:
Neuronal acetylcholine receptor subunit alpha-7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aldafermin DB16086
biotech | CAS: 1616639-03-2

Aldafermin is under investigation in clinical trial NCT03912532 (Evaluation of Efficacy, Safety and Tolerability of Aldafermin in a Phase 2b, Randomized, Double-blind, Placebo-controlled, Multi-center Study in Subjects With Nonalcoholic Steatohepatitis and St…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsIntercellular Signaling Peptides and Proteins +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aldesleukin Approved DB00041
biotech | CAS: 110942-02-4

Aldesleukin, a lymphokine, is produced by recombinant DNA technology using a genetically engineered E. coli strain containing an analog of the human interleukin-2 gene. Genetic engineering techniques were used to modify the human IL-2 gene, and the resulting …

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAnti-HIV Agents +26
Target Protein:
Interleukin-2 receptor subunit betaInterleukin-2 receptor subunit alphaCytokine receptor common subunit gamma
Waktu Paruh13 min-85 min
Vol. Distribusi0.18 l/kg
Klirens-
Genetik -
Aldosterone DB04630
small molecule | CAS: 52-39-1

A hormone secreted by the adrenal cortex that regulates electrolyte and water balance by increasing the renal retention of sodium and the excretion of potassium.

Kategori:
11-HydroxycorticosteroidsAdrenal Cortex HormonesCorticosteroids +18
Target Protein:
Solute carrier family 12 member 1Mineralocorticoid receptorGlucocorticoid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aldoxorubicin DB06013
small molecule | CAS: 1361644-26-9

Aldoxorubicin, an antineoplastic agents, is an albumin-binding prodrug of doxorubicin.

Kategori:
AnthracyclinesAntineoplastic AgentsCarbohydrates +4
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aldumastat DB18824
small molecule | CAS: 1957278-93-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alectinib Approved DB11363
small molecule | CAS: 1256580-46-7

Alectinib is a second generation oral drug that selectively inhibits the activity of anaplastic lymphoma kinase (ALK) tyrosine kinase. It is specifically used in the treatment of non-small cell lung cancer (NSCLC) expressing the ALK-EML4 (echinoderm microtubu…

Kategori:
Anaplastic lymphoma kinase (ALK) inhibitorsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +14
Target Protein:
ALK tyrosine kinase receptor
Waktu ParuhThe mean eliminatio…
Vol. Distribusi4016 L
KlirensThe apparent cleara…
Genetik -
Alefacept Approved DB00092
biotech | CAS: 222535-22-0

Immunosuppressive dimeric fusion protein that consists of the extracellular CD2-binding portion of the human leukocyte function antigen-3 (LFA-3) linked to the Fc (hinge, CH2 and CH3 domains) portion of human IgG1. Produced by CHO cells, mW is 91.4 kD.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntineoplastic and Immunomodulating Agents +20
Target Protein:
T-cell surface antigen CD2Low affinity immunoglobulin gamma Fc region receptor III-ALow affinity immunoglobulin gamma Fc region receptor III-B
Waktu Paruh~270 hours
Vol. Distribusi-
Klirens-
Genetik -
Alemtuzumab Approved DB00087
biotech | CAS: 216503-57-0

Alemtuzumab is a humanized monoclonal antibody specific to lymphocyte antigens. It is a recombinant DNA-derived humanized monoclonal antibody (Campath-1H) that is directed against the 21-28 kD cell surface glycoprotein, CD52. The Campath-1H antibody is an IgG…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +18
Target Protein:
CAMPATH-1 antigenLow affinity immunoglobulin gamma Fc region receptor III-BLow affinity immunoglobulin gamma Fc region receptor III-A +4
Waktu ParuhThe elimination hal…
Vol. DistribusiAlemtuzumab is larg…
KlirensClearance of alemtu…
Genetik -
Alendronic acid Approved DB00630
small molecule | CAS: 66376-36-1

Alendronic acid is a second generation bisphosphonate that is used for the treatment of some forms of osteoperosis and Paget's disease[FDA Label][A959,A203111]. It functions by preventing resorption of bone[FDA Label][A959].

Kategori:
Agents Causing Muscle ToxicityBisphosphonatesBone Density Conservation Agents +5
Target Protein:
Farnesyl pyrophosphate synthaseHydroxylapatiteTyrosine-protein phosphatase non-receptor type 4 +3
Waktu ParuhDue to alendronic a…
Vol. Distribusi28L[FDA Label].
Klirens71mL/min[FDA Label].
Genetik -
Aleplasinin DB12635
small molecule | CAS: 481629-87-2

Aleplasinin has been investigated in Alzheimer Disease.

Target Protein:
Plasminogen activator inhibitor 1Plasminogen activator inhibitor 2Plasma serine protease inhibitor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alethine DB05800
small molecule | CAS: 646-08-2

Alethine is studied in the treatment of cancer. It belongs to a family of chemicals called disulfides. It is a low molecular weight disulfide that has been shown to exhibit in vivo antitumor activity in murine myeloma and melanoma models.

Kategori:
AminesEthylaminesMercaptoethylamines +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alexitol sodium DB15908
small molecule | CAS: 66813-51-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alfacalcidol Approved DB01436
small molecule | CAS: 41294-56-8

Alfacalcidol, or 1-alpha-hydroxycholecalciferol or 1-alpha-hydroxyvitamin D3, is a non-endogenous analogue of [vitamin D].[A234044] It plays an essential function in calcium homeostasis and bone metabolism. Alfacaldisol is activated by the enzyme 25-hydroxyla…

Kategori:
Alimentary Tract and MetabolismBone Density Conservation AgentsCholestanes +13
Target Protein:
Vitamin D3 receptor25-hydroxyvitamin D-1 alpha hydroxylase, mitochondrialRetinoic acid receptor RXR-alpha
Waktu ParuhThe half-life of al…
Vol. Distribusi-
Klirens-
Genetik -
Alfaxalone DB11371
small molecule | CAS: 23930-19-0

Alfaxalone, also known as alphaxalone or alphaxolone, is a neuroactive steroid and general anaesthetic. It is used in veterinary practice under the trade name Alfaxan, and is licensed for use in both dogs and cats. Along with alfadolone, it is also one of the…

Kategori:
AnestheticsAnesthetics, GeneralCentral Nervous System Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alfentanil Approved DB00802
small molecule | CAS: 71195-58-9

A short-acting opioid anesthetic and analgesic derivative of fentanyl. It produces an early peak analgesic effect and fast recovery of consciousness. Alfentanil is effective as an anesthetic during surgery, for supplementation of analgesia during surgical pro…

Kategori:
Agents that produce hypertensionAnalgesicsAnesthetics +25
Target Protein:
Mu-type opioid receptor
Waktu Paruh90-111 minutes
Vol. Distribusi* 0.4 to 1 L/kg
Klirens* 5 mL/kg/min
Genetik -
Alfimeprase DB04919
biotech | CAS: 259074-76-5

Alfimeprase is a recombinant analog of fibrolase. Fibrolase is a zinc-containing metalloproteinase isolated from the venom of the southern copperhead snake (<i>Agkistrodon contortrix contortrix</i>). It is a small protein that contains 203 residues (Randolph …

Kategori:
EndopeptidasesEnzymesEnzymes and Coenzymes +3
Target Protein:
Fibrinogen alpha chainFibrinogen beta chain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alflorex Approved DB18507
biotech

Alflorex is a probiotic with 35624 cultures, part of the Bifidobacterium longum.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alflutinib DB16087
small molecule | CAS: 1869057-83-9

Alflutinib is under investigation in clinical trial NCT03452592 (Efficacy and Safety of Alflutinib in Locally Advanced or Metastatic Non-small Cell Lung Cancer Patients With T790M).

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingProtein Kinase Inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alfuzosin Approved DB00346
small molecule | CAS: 81403-80-7

Benign prostatic hyperplasia (BPH) refers to a benign growth or hyperplasia of the prostate and leads to lower urinary tract symptoms in men, such as urgency, frequency and changes to urine flow. The prevalence of BPH is as high as 50%-60% for males in their …

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +17
Target Protein:
Alpha-1 adrenergic receptorsAlpha-1A adrenergic receptorAlpha-1B adrenergic receptor +1
Waktu ParuhThe apparent elimin…
Vol. DistribusiThe volume of distr…
KlirensExercise caution if…
Genetik -
Algestone DB18000
small molecule | CAS: 595-77-7

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesContraceptive Agents, FemaleContraceptive Agents, Hormonal +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 24356-94-3

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesAlgestoneAnti-Inflammatory Agents +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alginic acid Approved DB13518
small molecule | CAS: 9005-32-7

Alginic acid, also referred to as algin or alginate, is a hydrophilic or anionic polysaccharide isolated from certain brown seaweed (_Phacophycae_) via alkaline extraction. It is present in cell walls of brown algae where it forms a viscous gel when binding w…

Kategori:
Acids, AcyclicAcids, AldehydicAlginates +11
Waktu ParuhThis pharmacokineti…
Vol. DistribusiThis pharmacokineti…
KlirensThis pharmacokineti…
Genetik -
Alglucerase Approved DB00088
biotech | CAS: 143003-46-7

Human Beta-glucocerebrosidase or Beta-D-glucosyl-N-acylsphingosine glucohydrolase E.C. 3.2.1.45. 497 residue protein with N-linked carbohydrates, MW=59.3 kD. Alglucerase is prepared by modification of the oligosaccharide chains of human Beta-glucocerebrosidas…

Kategori:
Alimentary Tract and MetabolismEnzyme Replacement TherapyEnzymes +6
Target Protein:
Glucocerebroside
Waktu Paruh3.6-10.4 min
Vol. Distribusi* 49.4 to 282.1 mL/…
Klirens-
Genetik -
Alglucosidase alfa Approved DB01272
biotech | CAS: 420784-05-0

Aglucosidase alfa consists of the human enzyme acid alpha-glucosidase (GAA) which is essential for the degradation of glygogen to glucose in lysosomes. It is encoded by the most predominant of nine observed haplotypes of this gene. Aglucosidase alfa is produc…

Kategori:
Alimentary Tract and MetabolismEnzymesEnzymes and Coenzymes +5
Target Protein:
Cation-dependent mannose-6-phosphate receptorGlycogen
Waktu Paruh2.3 &plusmn; 0.4 ho…
Vol. Distribusi* 96 ± 16 mL/kg [20…
Klirens* 25+/- 4 mL/hr/kg …
Genetik -
ALGRX 1207 DB06482
small molecule

ALGRX 1207 is a topical local anesthetic that acts by binding to the fast sodium channel. ALGRX 1207 entered clinical trials for cutaneous neuropathic pain, such as chemotherapy-induced neuropathy, in 2006. It was being developed by Anesiva, but trials have h…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alicaforsen DB06224
small molecule | CAS: 185229-68-9

Deskripsi belum tersedia.

Kategori:
Gastrointestinal AgentsImmunologic FactorsNucleic Acids, Nucleotides, and Nucleosides +3
Target Protein:
Intercellular adhesion molecule 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alidornase alfa DB18144
biotech | CAS: 1788036-49-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alimemazine Approved DB01246
small molecule | CAS: 84-96-8

A phenothiazine derivative that is used as an antipruritic.

Kategori:
Antihistamines for Systemic UseAntipruriticsAntipsychotic Agents +13
Target Protein:
Histamine H1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alintegimod DB18879
small molecule | CAS: 1378535-08-0

Alintegimod is under investigation in clinical trial NCT06362369 (A Study of Oral 7HP349 (Alintegimod) in Combination With Ipilimumab Followed by Nivolumab Monotherapy).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alipogene tiparvovec Approved DB13521
biotech | CAS: 929881-05-0

Alipogene tiparvovec is an adeno-associated viral vector of serotype 1-based gene therapy that delivers the Ser(447)X variant of the human lipoprotein lipase (LPL) gene. It is being investigated for the treatment of lipoprotein lipase (LPL) deficiency.[A25979…

Kategori:
Adeno-associated Viral Vector TherapiesLipid Modifying AgentsLipid Modifying Agents, Plain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alirinetide DB17007
biotech | CAS: 725715-18-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alirocumab Approved DB09302
biotech | CAS: 1245916-14-6

Alirocumab is a biopharmaceutical that obtained FDA approval in July 2015 as a second line treatment for high cholesterol in adults whose LDL-cholesterol (LDL-C) is not controlled by the combination of diet and statin treatment. It is a human monoclonal antib…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +20
Target Protein:
Proprotein convertase subtilisin/kexin type 9
Waktu ParuhIn monotherapy, the…
Vol. DistribusiAlirocumab is mainl…
Klirens-
Genetik -
Alisertib DB05220
small molecule | CAS: 1028486-01-2

Alisertib is a novel aurora A kinase inhibitor under investigation for the treatment of various forms of cancer.

Kategori:
Protein Kinase Inhibitors
Target Protein:
Aurora kinase A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aliskiren Approved DB09026
small molecule | CAS: 173334-57-1

Aliskiren is the first drug in the renin inhibitor drug class and is used for the treatment of hypertension.[A203624] It was developed by Speedel and Novartis and initially approved by the FDA in early 2007.[L14018] Aliskiren has been proven to efficacious in…

Kategori:
Acids, AcyclicAgents Acting on the Renin-Angiotensin SystemAgents causing hyperkalemia +14
Target Protein:
Renin
Waktu ParuhPlasma half-life fo…
Vol. DistribusiUnchanged aliskiren…
KlirensAliskiren is partia…
Genetik -
Alisporivir DB12139
small molecule | CAS: 254435-95-5

Alisporivir has been used in trials studying the treatment of Hepatitis C and Chronic Hepatitis C.

Kategori:
Amino Acids, Peptides, and ProteinsCyclosporin DerivativesPeptides +1
Target Protein:
Guided entry of tail-anchored proteins factor CAMLG
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alitretinoin Approved DB00523
small molecule | CAS: 5300-03-8

An important regulator of gene expression during growth and development, and in neoplasms. Tretinoin, also known as retinoic acid and derived from maternal vitamin A, is essential for normal growth; and embryonic development. An excess of tretinoin can be ter…

Kategori:
Agents for Dermatitis, Excluding CorticosteroidsAlkenesAntineoplastic Agents +19
Target Protein:
Retinoic acid receptor alphaRetinoic acid receptor RXR-alphaRetinoic acid receptor beta +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alizapride DB01425
small molecule | CAS: 59338-93-1

Alizapride is a dopamine antagonist that is capable of demonstrating both prokinetic and antiemetic effects. This kind of pharmacological activity makes it effective for use in the treatment of various kinds of nausea and vomiting, including that which may oc…

Kategori:
Alimentary Tract and MetabolismAntiemeticsAutonomic Agents +7
Target Protein:
D(2) dopamine receptor
Waktu Paruh3 hours
Vol. Distribusi-
Klirens-
Genetik -
ALK-4290 DB15269
small molecule | CAS: 1251528-23-0

ALK-4290 is under investigation in clinical trial NCT03558061 (Evaluate the Effects and Safety of ALK4290 in Patients With Newly Diagnosed Wet Age-Related Macular Degeneration).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ALKS 27 DB05752
small molecule

ALKS 27 is an inhaled formulation of trospium chloride for the treatment of chronic obstructive pulmonary disease (COPD). Study showed that ALKS 27 was well-tolerated over a wide dose range, with no dose-limited effects observed.

Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ALKS 29 DB05723
small molecule

ALKS 29 is a new product candidate for the treatment of alcohol dependence. It is being developed by Alkermes, Inc.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Allantoin Approved DB11100
small molecule | CAS: 97-59-6

Allantoin is a substance that is endogenous to the human body and also found as a normal component of human diets [FDA Label]. In healthy human volunteers, the mean plasma concentration of allantoin is about 2-3 mg/l. During exercise, the plasma allantoin con…

Kategori:
AmidesBasic Ointments and ProtectantsDermatologicals +5
Waktu ParuhWhen studied in cat…
Vol. Distribusi-
KlirensSome studies sugges…
Genetik -
small molecule | CAS: 947331-05-7

Allisartan isoproxil is under investigation in clinical trial NCT03264352 (Intervention for High-normal Blood Pressure in Adults With Type 2 Diabetes).

Kategori:
Agents Acting on the Renin-Angiotensin SystemAngiotensin II receptor antagonistsAngiotensin II Type 1 Receptor Blockers +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Allitinib DB18840
small molecule | CAS: 897383-62-9

Allitinib is under investigation in clinical trial NCT04671303 (To Evaluate the Efficacy and Safety of Anlotinib Combined With Allitinib in Lung Cancer).

Kategori:
Acids, AcyclicAcrylatesAmides +2
Target Protein:
Epidermal growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Allobarbital DB13577
small molecule | CAS: 52-43-7

Deskripsi belum tersedia.

Kategori:
Barbiturates, PlainCentral Nervous System DepressantsHypnotics and Sedatives +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Allocetra DB16424
biotech

Allocetra is a novel therapy where billions of early apoptotic cells are infused into the bloodstream of a patient, using the body's own natural regulation mechanisms to rebalance an unbalanced immune system without immune system suppression. With infusion, t…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Stratagraft (allogeneic cultured keratinocytes and dermal fibroblasts in murine collagen-dsat) is an allogeneic cellularized scaffold product used for the treatment of adults with thermal burns containing intact dermal elements for which surgical intervention…

Kategori:
FibroblastsKeratinocytes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Allogeneic processed thymus tissue is used for immune reconstitution in immune disorders where the patients are severely immunocompromised due to the absence of a functional thymus, such as congenital athymia. As part of the immune system, the thymus is an or…

Waktu ParuhThe pharmacokinetic…
Vol. DistribusiThe pharmacokinetic…
KlirensThe pharmacokinetic…
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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