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3253

Total database: 17430
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2451 (75.3%)
Target
1833 (56.3%)
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35 (1.1%)
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3253 (100.0%)

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Halaman 53 / 66
biotech | CAS: 2253753-17-0

Rocakinogene sifuplasmid is under investigation in clinical trial NCT03491683 (INO-5401 and INO-9012 Delivered by Electroporation (EP) in Combination With Cemiplimab (REGN2810) in Newly-diagnosed Glioblastoma (GBM)).

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBiological Factors +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rofecoxib Approved DB00533
small molecule | CAS: 162011-90-7

Rofecoxib is used for the treatment of osteoarthritis, rheumatoid arthritis, acute pain in adults, and primary dysmenorrhea, as well as acute treatment of migraine attacks with or without auras. Rofecoxib is a solid. This compound belongs to the stilbenes. Th…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +29
Target Protein:
Prostaglandin G/H synthase 2Elastin
Waktu Paruh17 hours
Vol. Distribusi-
Klirens-
Genetik -
Rogaratinib DB15078
small molecule | CAS: 1443530-05-9

Rogaratinib is under investigation in clinical trial NCT03762122 (Rogaratinib in Patients With Advanced Pretreated Squamous-cell Non-small Cell Lung Cancer (SQCLC)).

Kategori:
Sulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rolapitant Approved DB09291
small molecule | CAS: 552292-08-7

Rolapitant is a potent, highly selective, long-acting Neurokinin-1 (NK-1) receptor antagonist approved for the prevention of delayed chemotherapy-induced nausea and vomiting (CINV) in adults. Delayed-phase CINV typically occurs >24 hours after chemotherapy tr…

Kategori:
Alimentary Tract and MetabolismAntiemetics and AntinauseantsBCRP/ABCG2 Inhibitors +11
Target Protein:
Substance-P receptor
Waktu ParuhMean terminal half …
Vol. Distribusi460 L
Klirens0.96 L/hour
Genetik -
Rolofylline DB12670
small molecule | CAS: 136199-02-5

Rolofylline is under clinical development by pharmaceutical company NovaCardia for the treatment of congestive heart failure.

Kategori:
AlkaloidsDiureticsHeterocyclic Compounds, Fused-Ring +3
Target Protein:
Adenosine receptor A1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Romidepsin Approved DB06176
small molecule | CAS: 128517-07-7

Romidepsin is a selective inhibitor of histone deacetylase, approved in the US in 2009 for the treatment of cutaneous T-cell lymphoma (CTCL) in patients who have received at least one prior systemic therapy.

Kategori:
Amino Acids, Peptides, and ProteinsAntibiotics, AntineoplasticAntineoplastic Agents +30
Target Protein:
Histone deacetylase 1Histone deacetylase 2Histone deacetylase 4 +3
Waktu ParuhApproximately 3 hou…
Vol. Distribusi44.5L
Klirens8.4L/h
Genetik -
Romosozumab Approved DB11866
biotech | CAS: 909395-70-6

Romosozumab is a humanized monoclonal antibody indicated for the treatment of osteoperosis in postmenopausal women at high risk of fracture and patients who have failed in other treatments or are intolerant to other osteoperosis therapies[L9554]. Romosozumab …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +12
Target Protein:
Sclerostin
Waktu Paruh12.8 days[L9554].
Vol. Distribusi3.92L[L9554].
Klirens0.38mL/hr/kg[L9554].
Genetik -
Roniciclib DB12974
small molecule | CAS: 1223498-69-8

Roniciclib has been investigated for the treatment of Small Cell Lung Carcinoma.

Kategori:
Sulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ronopterin DB12575
small molecule | CAS: 185243-78-1

Ronopterin has been used in trials studying the treatment of Traumatic Brain Injury.

Kategori:
CoenzymesEnzymes and CoenzymesHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rontalizumab DB12844
biotech | CAS: 948570-30-7

Rontalizumab has been used in trials studying the treatment of Systemic Lupus Erythematosus.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ropanicant DB19134
small molecule | CAS: 2414674-70-5

Ropanicant is under investigation in clinical trial NCT06126497 (Study Evaluating Safety and Efficacy of Ropanicant in MDD Patients).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ropeginterferon alfa-2b Approved DB15119
biotech | CAS: 1335098-50-4

Polycythemia vera (PV) is the most common Philadelphia chromosome-negative myeloproliferative neoplasm (MPN), characterized by increased hematocrit and platelet/leukocyte counts, an increased risk for hemorrhage and thromboembolic events, and a long-term prop…

Kategori:
Adjuvants, ImmunologicAlfa InterferonsAntineoplastic and Immunomodulating Agents +12
Target Protein:
Interferon alpha/beta receptor (IFNAR)
Waktu ParuhRopeginterferon alf…
Vol. DistribusiRopeginterferon alf…
KlirensRopeginterferon alf…
Genetik -
Ropivacaine Approved DB00296
small molecule | CAS: 84057-95-4

Ropivacaine is an aminoamide local anesthetic drug marketed by AstraZeneca under the trade name Naropin. It exists as a racemate of its S- and R-enantiomers, although the marketed form is supplied only as the purified S-enantiomer.[L42140]

Kategori:
AmidesAminesAnesthetics +19
Target Protein:
Sodium channel protein type 10 subunit alpha
Waktu ParuhThe mean terminal h…
Vol. DistribusiFollowing intravasc…
KlirensFollowing intraveno…
Genetik -
Ropsacitinib DB18709
small molecule | CAS: 2127109-84-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rosiglitazone Approved DB00412
small molecule | CAS: 122320-73-4

Rosiglitazone is an anti-diabetic drug in the thiazolidinedione class of drugs. It is marketed by the pharmaceutical company GlaxoSmithKline as a stand-alone drug (Avandia) and in combination with metformin (Avandamet) or with glimepiride (Avandaryl). Like ot…

Kategori:
Alimentary Tract and MetabolismBlood Glucose Lowering AgentsBSEP/ABCB11 Substrates +33
Target Protein:
Peroxisome proliferator-activated receptor gammaLong-chain-fatty-acid--CoA ligase 4Peroxisome proliferator-activated receptor alpha +4
Waktu Paruh3-4 hours (single o…
Vol. Distribusi* 17.6 L [oral volu…
Klirens* Oral clearance (C…
Genetik -
Rosnilimab DB18851
biotech | CAS: 2412764-40-8

Rosnilimab is under investigation in clinical trial NCT06041269 (A Study of Efficacy and Safety of Rosnilimab in Subjects With Moderate to Severe Rheumatoid Arthritis (RENOIR)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rostafuroxin DB12350
small molecule | CAS: 156722-18-8

Rostafuroxin has been used in trials studying the treatment of Essential Hypertension.

Kategori:
AndrostanesFused-Ring CompoundsSteroids
Target Protein:
Sodium/potassium-transporting ATPase subunit beta-1Sodium/potassium-transporting ATPase subunit beta-2Sodium/potassium-transporting ATPase subunit beta-3 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rotavirus vaccine Approved DB10276
biotech

Rotavirus commonly infects children and infants causing severe diarrhea and vomiting leading to potentially fatal dehydration.[L1117] Two rotavirus vaccines are available for the prevention of rotavirus gastroenteritis, Rotateq and Rotarix. Rotateq is a live …

Kategori:
Actively Acquired ImmunityAntiinfectives for Systemic UseBiological Products +6
Waktu ParuhThe median duration…
Vol. Distribusi-
Klirens-
Genetik -
Rotenone DB11457
small molecule | CAS: 83-79-4

Rotenone is an isoflavone compound that naturally occurs in the jicama vine plant as well as many Fabaceae plants. It has broad spectrum insecticide and pesticide activity and is also toxic to fish.

Kategori:
AgrochemicalsBenzopyransChromones +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rotigaptide DB13067
small molecule | CAS: 355151-12-1

Rotigaptide is under investigation for the basic science of Heart Disease and Vascular Disease.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 912809-27-9

Rovafovir etalafenamide is under investigation in clinical trial NCT03472326 (Efficacy of GS-9131 Functional Monotherapy in HIV-1-Infected Adults Failing a Nucleos(t)Ide Reverse Transcriptase Inhibitor-Containing Regimen).

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Roxarsone DB11458
small molecule | CAS: 121-19-7

Roxarsone is an organoarsenic molecule added to poultry feed. The addition of this compound to poultry feed improves weight gain and feed efficiency as well as prevent the growth of coccidian parasites. The drug is also approved in the United States for use i…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntiparasitic Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rozanolixizumab Approved DB14919
biotech | CAS: 1584645-37-3

Rozanolixizumab is a humanized high-affinity anti-human neonatal Fc receptor (FcRn) monoclonal antibody (IgG4P) targeting the immunoglobulin G (IgG). Rozonolixizumab itself is an IgG4P, an inactive isotype, to reduce the likelihood of unwanted chain exchange.…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
IgG receptor FcRn large subunit p51
Waktu Paruh-
Vol. DistribusiThe apparent volume…
KlirensThe apparent cleara…
Genetik -
RPR128515 DB04424
small molecule

Deskripsi belum tersedia.

Target Protein:
Serine protease 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RPR131247 DB02744
small molecule

Deskripsi belum tersedia.

Target Protein:
Serine protease 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RRx-001 DB12060
small molecule | CAS: 925206-65-1

RRx-001 has been used in trials studying the treatment of Lymphomas, Brain Metastases, Cholangiocarcinoma, Colorectal Neoplasms, and Malignant Solid Tumor, among others.

Kategori:
AzetinesCarbon Radioisotopes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RS-39604 DB17050
small molecule | CAS: 161362-65-8

RS-39604 is a selective 5-HT4 receptor antagonist.[A253112]

Kategori:
AlkanesHydrocarbons, Acyclic
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
rsPSMA Vaccine Approved DB06361
biotech

Prostate-specific membrane antigen (PSMA) is an ?100 kDa transmembrane glycoprotein that is abundantly and preferentially expressed in prostate cancer, including recurrent and hormone-refractory cases. rsPSMA Vaccine is a subunit vaccine based on a novel rsPS…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RSV-604 DB15197
small molecule | CAS: 676128-63-5

RSV-604 is under investigation in clinical trial NCT00416442 (Safety, Tolerability and Pharmacokinetic Study of Single and Multiple Intravenous Doses of RSV604 in Healthy Subjects.).

Kategori:
AmidesBenzazepinesBenzene Derivatives +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RU85053 DB03712
small molecule

Deskripsi belum tersedia.

Target Protein:
Proto-oncogene tyrosine-protein kinase Src
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rubitecan DB06159
small molecule | CAS: 91421-42-0

Deskripsi belum tersedia.

Kategori:
AlkaloidsAntineoplastic AgentsEnzyme Inhibitors +2
Target Protein:
DNA topoisomerase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rucaparib Approved DB12332
small molecule | CAS: 283173-50-2

Rucaparib is an anticancer drug and poly (ADP-ribose) polymerase (PARP) inhibitor. PARP is an enzyme that plays an essential role in DNA repair.[A18745] Rucaparib is proposed to work in several PARP-dependent and PARP-independent mechanisms of action; however…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +47
Target Protein:
Poly [ADP-ribose] polymerase 1Poly [ADP-ribose] polymerase 2Protein mono-ADP-ribosyltransferase PARP3
Waktu ParuhThe mean (coefficie…
Vol. DistribusiThe mean (coefficie…
KlirensThe mean (coefficie…
Genetik -
Rulonilimab DB18922
biotech | CAS: 2417124-95-7

Rulonilimab is under investigation in clinical trial NCT05408221 (The Efficacy and Safety of Rulonilimab in Combination With Lenvatinib in Hepatocellular Carcinoma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rurioctocog alfa pegol Approved DB16007
biotech | CAS: 1417412-83-9

Rurioctocog alfa pegol is a pegylated recombinant human coagulation factor VIII or antihemophilic factor. Factor VIII is an essential protein involved in normal blood clotting; thus, a deficient level of functional factor VIII is associated with an elevated r…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +9
Target Protein:
von Willebrand factorCoagulation factor VIII
Waktu ParuhFollowing intraveno…
Vol. DistribusiFollowing intraveno…
KlirensFollowing intraveno…
Genetik -
Ruxolitinib Approved DB08877
small molecule | CAS: 941678-49-5

Ruxolitinib, formerly known as INCB018424 or INC424, is an anticancer drug and a Janus kinase (JAK) inhibitor. It is a potent and selective inhibitor of JAK1 and JAK2,[A229698] which are tyrosine kinases involved in cytokine signalling and hematopoiesis.[A745…

Kategori:
Agents for Dermatitis, Excluding CorticosteroidsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +18
Target Protein:
Urokinase plasminogen activator surface receptorTyrosine-protein kinase JAK2Tyrosine-protein kinase JAK1 +2
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe mean volume of …
KlirensRuxolitinib clearan…
Genetik -
RWJ-56423 DB02812
small molecule

Deskripsi belum tersedia.

Target Protein:
Serine protease 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
S-3304 DB12149
small molecule | CAS: 203640-27-1

S-3304 has been used in trials studying the treatment of Lung Cancer, Solid Tumors, Non Small Cell Lung Cancer, Stage IIIB Non Small Cell Lung Cancer, and Stage IIIA Non Small Cell Lung Cancer, among others.

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingMatrix Metalloproteinase Inhibitors +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
S-49076 DB16821
small molecule | CAS: 1265965-22-7

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsHeterocyclic Compounds, Fused-RingSulfur Compounds +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
S-55746 DB18365
small molecule | CAS: 1448584-12-0

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingOxazines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sabarubicin DB12410
small molecule | CAS: 211100-13-9

Sabarubicin has been used in trials studying the treatment of Prostate Cancer, Testicular Germ Cell Tumor, and Unspecified Adult Solid Tumor, Protocol Specific.

Kategori:
AnthracyclinesCarbohydratesGlycosides +3
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sabestomig DB19326
biotech | CAS: 2648346-74-9

Sabestomig is under investigation in clinical trial NCT05216835 (Safety and Preliminary Efficacy Assessment of AZD7789 in Patients With Relapsed or Refractory Classical Hodgkin Lymphoma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Saccharide isomerate Approved DB11232
small molecule | CAS: 100843-69-4

Deskripsi belum tersedia.

Kategori:
BiopolymersCarbohydratesMacromolecular Substances +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Saccharin DB12418
small molecule | CAS: 81-07-2

Saccharin has been investigated for the treatment of Hypertension and Hyperglycemia.

Kategori:
BenzothiazolesCompounds used in a research, industrial, or household settingDiet, Food, and Nutrition +9
Target Protein:
Carbonic anhydrase 1Carbonic anhydrase 9Carbonic anhydrase 12 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sacituzumab govitecan Approved DB12893
biotech | CAS: 1491917-83-9

Metastatic triple-negative breast cancer (mTNBC) is an aggressive form of breast cancer with limited treatment options involving cytotoxic chemotherapy agents.[A193653] Targeted chemotherapy through the application of antibody-conjugated agents (ADCs) is a re…

Kategori:
AlkaloidsAmino Acids, Peptides, and ProteinsAntibodies +20
Target Protein:
Tumor-associated calcium signal transducer 2DNA topoisomerase 1Far upstream element-binding protein 1
Waktu ParuhSacituzumab govitec…
Vol. DistribusiSacituzumab govitec…
KlirensSacituzumab govitec…
Genetik -
Sacubitrilat DB14127
small molecule | CAS: 149709-44-4

A metabolite of LCZ696 with neprilysin inhibitory activity.

Kategori:
Acids, AcyclicAmino AcidsAmino Acids, Peptides, and Proteins +4
Target Protein:
Neprilysin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Safflower oil Approved DB09446
biotech | CAS: 8001-23-8

Safflower (_Carthamus tinctorius_ L) is a herbaceous plant in the Asteraceae family. Extracted from the seeds of safflowers, safflower oil is a rich source of various saturated fatty acids, monounsaturated fatty acid (oleic acid) or essential n-6 polyunsatura…

Kategori:
Biological ProductsComplex MixturesDiet, Food, and Nutrition +10
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Sagopilone DB12391
small molecule | CAS: 305841-29-6

Sagopilone has been used in trials studying the treatment of Melanoma, Neoplasms, CNS Disease, Breast Cancer, and Breast Neoplasms, among others. It is a so-called fully synthetic epothilone and is the first such compound to be in clinical development to comb…

Kategori:
Anti-Bacterial AgentsAntineoplastic AgentsCytochrome P-450 CYP3A Inhibitors +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sakuranetin DB08517
small molecule | CAS: 2957-21-3

Deskripsi belum tersedia.

Kategori:
BenzopyransBiological FactorsChromones +3
Target Protein:
Adenosine receptor A2bAdenosine receptor A1Adenosine receptor A3 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Salirasib DB12681
small molecule | CAS: 162520-00-5

Salirasib has been used in trials studying the diagnostic of Carcinoma, Non-Small-Cell Lung.

Kategori:
Acids, CarbocyclicAlcoholsAntineoplastic Agents +11
Target Protein:
Serine/threonine-protein kinase mTORGTPase NRas
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 121521-90-2

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAldehyde ReductaseAldehyde Reductase, antagonists & inhibitors +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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