Hasil Filter

17430

Total database: 17430
Struktur (SMILES)
12313 (70.6%)
Target
9368 (53.7%)
Genomik
112 (0.6%)
Referensi
17430 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (17430)

Halaman 53 / 1743
small molecule

Deskripsi belum tersedia.

Target Protein:
Carbonic anhydrase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 124192-87-6

Deskripsi belum tersedia.

Target Protein:
Amine oxidase [flavin-containing] B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 57452-98-9

(R)-Praziquantel is under investigation in clinical trial NCT02271984 (Relative Bioavailability Trial of L-Praziquantel in Healthy Volunteers).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
(R)-Propafenone DB19162
small molecule | CAS: 107381-31-7

Propafenone, (r)- is under investigation in clinical trial NCT02710669 (New Formulations of Propafenone to Treat Atrial Fibrillation).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 4254-14-2

A clear, colorless, viscous organic solvent and diluent used in pharmaceutical preparations.

Target Protein:
Isocitrate dehydrogenase [NADP]Lysozyme C
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Leukotriene A-4 hydrolase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
(R)-Rolipram DB04149
small molecule | CAS: 85416-75-7

The (R)-enantiomer of rolipram, it is a phosphodiesterase inhibitor with antidepressant properties.

Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4A3',5'-cyclic-AMP phosphodiesterase 4B3',5'-cyclic-AMP phosphodiesterase 4D
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 20780-53-4

Deskripsi belum tersedia.

Target Protein:
Halohydrin dehalogenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Acetylcholinesterase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
(R)-warfarin DB08496
small molecule | CAS: 40281-89-8

Warfarin consists of a racemic mixture of two active enantiomers—R- and S- forms—each of which is cleared by different pathways. S-warfarin is 2-5 times more potent than the R-isomer in producing an anticoagulant response.[A1038]

Kategori:
AnticoagulantsCytochrome P-450 CYP1A2 SubstratesCytochrome P-450 CYP2C18 Substrates +7
Waktu Paruh-
Vol. DistribusiThe volume of distr…
Klirens0.125L/h, (95% conf…
Genetik -
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