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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
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12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 52 / 252
AT-7519 DB08142
small molecule | CAS: 844442-38-2

AT7519 is a selective inhibitor of certain Cyclin Dependent Kinases (CDKs) leading to tumour regression. It is developed by Astex for the treatment of solid tumours and haematological malignancies.

Kategori:
Cyclin-Dependent Kinases, antagonists & inhibitors
Target Protein:
Cyclin-dependent kinase 2Cyclin-dependent kinase 1
Waktu Paruh-
Vol. Distribusi-
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AT-GTX-502 DB17001
biotech

AT-GTX-502 is an experimental, one-time gene therapy that uses AAV9 to deliver a functional copy of CLN3.

Kategori:
Non-Replicating Recombinant, Self-Complementary Adeno-Associated Virus Serotype 9 Containing the Human CLN3 Gene
Waktu Paruh-
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AT1022 DB04995
small molecule

AT1022 is a hydromorphone skin patch designed to provide rapid and sustained delivery of a potent opiate for the management of severe pain. AT1022 incorporates PassPort(TM) system, developed to deliver protein and peptide drugs, small-molecule drugs, genes a…

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AT1391 DB05120
small molecule

AT1391 is a daily insulin skin patch designed to provide continuous basal levels of insulin for patients with diabetes.

Target Protein:
Insulin receptor
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AT2220 DB05200
small molecule

AT2220 is an experimental, oral therapy for the treatment of Pompe disease and belongs to a class of molecules known as pharmacological chaperones. It is a small molecule designed to act as a pharmacological chaperone that specifically binds, stabilizes, and …

Target Protein:
Lysosomal alpha-glucosidase
Waktu Paruh-
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AT3022 DB05172
small molecule

AT3022, the Altea Therapeutics’s fentanyl citrate transdermal patch designed to provide safe and rapid management of moderate to severe chronic pain.

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AT845 DB17638
biotech

Deskripsi belum tersedia.

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AT9283 DB05169
small molecule | CAS: 896466-04-9

AT9283 is an aurora Kinase inhibitor developed by Astex Therapeutics for the treatment of cancer. It was discovered and developed internally using Astex’s fragment-based drug discovery platform, Pyramid.

Kategori:
AmidesHeterocyclic Compounds, Fused-RingProtein Kinase Inhibitors
Target Protein:
Aurora kinase BAurora kinase A
Waktu Paruh-
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Atabecestat DB15307
small molecule | CAS: 1200493-78-2

Atabecestat is under investigation in clinical trial NCT02211079 (A Study to Assess Effect of JNJ-54861911 on Pharmacokinetics of Cocktail Representatives for Cytochrome P450 (CYP) 3A4, CYP2B6, CYP2C9, and CYP1A2 Substrates).

Kategori:
Sulfur Compounds
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Atacicept DB06399
biotech | CAS: 845264-92-8

Atacicept is a recombinant fusion protein combined with the extracellular ligand binding portion of TACI.

Kategori:
Amino Acids, Peptides, and ProteinsProteinsRecombinant Proteins
Waktu Paruh-
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Ataciguat DB12805
small molecule | CAS: 254877-67-3

Ataciguat has been investigated for the basic science of Aortic Valve Stenosis.

Kategori:
Acids, CarbocyclicAmidesAminobenzoates +5
Target Protein:
Atrial natriuretic peptide receptor 1
Waktu Paruh-
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Atagabalin DB12032
small molecule | CAS: 223445-75-8

Atagabalin has been used in trials studying the treatment of Insomnia, Primary Insomnia, and Nonrestorative Sleep.

Kategori:
Acids, AcyclicCycloparaffinsFatty Acids +2
Target Protein:
Voltage-dependent calcium channel subunit alpha-2/delta-1
Waktu Paruh-
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Ataluren Approved DB05016
small molecule | CAS: 775304-57-9

Ataluren is a novel, orally administered drug that targets nonsense mutations. Ataluren is approved for use by the European Medicines Agency to treat Duchenne Muscular Dystrophy in patients aged 5 years and older who are able to walk. More specifically, atalu…

Kategori:
Musculo-Skeletal SystemOAT1/SLC22A6 inhibitorsOAT3/SLC22A8 Inhibitors +3
Target Protein:
Dystrophin
Waktu ParuhAtaluren plasma hal…
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Atamparib DB19028
small molecule | CAS: 2381037-82-5

Atamparib is under investigation in clinical trial NCT05127590 (RBN-2397 in Combination With Pembrolizumab in Patients With SCCL).

Target Protein:
Protein mono-ADP-ribosyltransferase TIPARP
Waktu Paruh-
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ATB-346 DB15377
small molecule | CAS: 1226895-20-0

ATB-346 is under investigation in clinical trial NCT03220633 (Study To Assess Safety, Tolerability And PK Of ATB-346 In Healthy Subjects).

Kategori:
Naphthaleneacetic AcidsNaphthalenes
Waktu Paruh-
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small molecule | CAS: 433937-93-0

Atecegatran metoxil has been used in trials studying the basic science and prevention of Nonvalvular Atrial Fibrillation, Persistent or Permanent Nonvalvular Atrial Fibrillation, and Persistent or Permanent Non-valvular Atrial Fibrillation.

Kategori:
Azetines
Target Protein:
Prothrombin
Waktu Paruh-
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Atelocollagen DB18450
biotech

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBiopolymersDrug Carriers +5
Waktu Paruh-
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Atenolol Approved DB00335
small molecule | CAS: 29122-68-7

Atenolol is a cardioselective beta-blocker used in a variety of cardiovascular conditions. Sir James Black, a Scottish pharmacologist, pioneered the use of beta-blockers for the management of angina pectoris in 1958 for which he received the Nobel Prize.[…

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-1 Receptor Antagonists +23
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptor
Gen Terkait:
ADRB1
Waktu Paruh6-7 hrs.[label]
Vol. DistribusiTotal Vd of 63.8-11…
KlirensTotal clearance is …
Genetik 1 Varian
Atesidorsen DB18159
biotech | CAS: 872063-57-5

Deskripsi belum tersedia.

Kategori:
Antisense OligonucleotidesNucleic Acids, Nucleotides, and NucleosidesNucleotides +1
Waktu Paruh-
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Atevirdine DB12264
small molecule | CAS: 136816-75-6

Atevirdine has been used in trials studying the treatment of HIV Infections.

Kategori:
Anti-Infective AgentsAnti-Retroviral AgentsAntiviral Agents +3
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
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Atexakin alfa DB19234
biotech | CAS: 143631-61-2

Atexakin alfa is under investigation in clinical trial NCT05435742 (SON-080 in Patients With Persistent Chemotherapy-induced Peripheral Neuropathy (CIPN)).

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Atezolizumab Approved DB11595
biotech | CAS: 1380723-44-3

Atezolizumab is a humanized monoclonal antibody used to prevent the interaction of PD-L1 and PD-1, removing inhibition of immune responses seen in some cancers.[A18493,L7489] This medication is reserved for patients whose tumors express PD-L1, cannot receive …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +19
Target Protein:
Programmed cell death 1 ligand 1Programmed cell death protein 1
Waktu ParuhThe half life of at…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of at…
Genetik -
ATG-Fresenius S DB05320
small molecule

ATG-Fresenius S is a concentrated anti-human T-lymphocyte immunoglobulin preparation derived from rabbits after immunization with a T-lympoblast cell line. ATG-Fresenius S is an immunosuppressive product for the prevention and treatment of acute rejection fol…

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ATG002 DB05068
small molecule

ATG002 is a completely new approach to treating chronic wounds such as diabetic foot ulcers, which is based upon stimulation of angiogenesis in the wound bed to help drive the wound-healing process. Unlike protein-derived growth factors, ATG002 is a small mol…

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ATG003 DB05069
small molecule

ATG003, a novel anti-angiogenic drug candidate and a formulation of mecamylamine, is currently in clinical development for neovascular age-related macular degeneration.

Target Protein:
Neuronal acetylcholine receptor subunit alpha-10Neuronal acetylcholine receptor subunit alpha-9
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ATHX-105 DB06008
small molecule

ATHX-105 is an investigational selective 5HT2c receptor agonist developed by Athersys Inc. for the treatment of Obesity.

Target Protein:
5-hydroxytryptamine receptor 2C
Waktu Paruh-
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ATI-1013 DB18185
biotech

ATI-1013 is a fully human nicotine-specific monoclonal antibody.

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ATI-355 DB17923
biotech

ATI-355 is a humanized anti-Nogo-A antibody developed by Novartis.

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Atibuclimab DB06546
biotech | CAS: 2417175-94-9

Atibuclimab (IC14) is a chimeric CD14 antibody investigated for the treatment of patients with severe sepsis.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Target Protein:
Monocyte differentiation antigen CD14
Waktu Paruh-
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Aticaprant DB12341
small molecule | CAS: 1174130-61-0

Aticaprant has been used in trials studying the health services research and basic science of Anxiety Disorders and Alcohol Dependence.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +5
Target Protein:
Kappa-type opioid receptor
Waktu Paruh-
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Atidarsagene autotemcel Approved DB17538
biotech

Atidarsagene autotemcel, sold under the brand name Libmeldy, is a gene therapy comprising genetically modified autologous CD34+ enriched hematopoietic stem and progenitor cells transduced _ex vivo_ using a lentiviral vector encoding the human arylsulfatase A …

Kategori:
Alimentary Tract and MetabolismAutologous Cultured CellAutologous Hematopoietic Stem Cell-Based Gene Therapy +2
Target Protein:
Human Arylsulfatase A mRNA
Waktu Paruh-
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Atilotrelvir DB19439
small molecule | CAS: 2850365-55-6

Atilotrelvir is under investigation in clinical trial NCT05041907 (Finding Treatments for COVID-19: A Trial of Antiviral Pharmacodynamics in Early Symptomatic COVID-19 (PLATCOV)).

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Atipamezole DB11481
small molecule | CAS: 104054-27-5

Atipamezole is a synthetic ?2 adrenoceptor antagonistused to reverse the sedative and analgesic effects of dexmedetomidine and medetomidine in dogs. It has also been undergone research as a potential anti-Parkinsonian drug for humans.

Kategori:
Adrenergic AgentsAdrenergic alpha-2 Receptor AntagonistsAdrenergic alpha-Antagonists +3
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Atiprimod DB05513
small molecule | CAS: 123018-47-3

Deskripsi belum tersedia.

Target Protein:
Signal transducer and activator of transcription 3Interleukin-6Tumor necrosis factor
Waktu Paruh-
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ATIR101 DB18650
biotech

ATIR101 is a haploidentical, naïve cell-enriched T-cell therapy.

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Atisnolerbart DB19418
biotech | CAS: 2456308-79-3

Atisnolerbart is under investigation in clinical trial NCT06602739 (A Study to Demonstrate the Effect of REGN5713-5715 on Reducing Ocular Allergy Signs and Symptoms in Adult Participants With Birch Pollen Allergy).

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ATL-104 DB05670
biotech

ATL-104 is a potent mitogen for epithelial cells of the gastrointestinal tract. In animal models, ATL-104 aids regeneration of the gastrointestinal tract after treatment with chemotherapeutic agents.

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ATL-2502 DB05340
small molecule

ATL-2502(Colal-Pred) is an old drug (prednisolone metasulphobenzoate, a steroid) with a new delivery system that releases the medication only in the colon. Releasing the drug directly into the colon reduces the potential for significant side effects often exp…

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ATL1101 DB05023
small molecule

ATL1101 is a second-generation antisense drug designed to block the synthesis of the IGF-1 receptor, a protein involved in the regulation of cell overgrowth in psoriasis. ATL1101 is being developed as a cream for the topical treatment of mild to moderate case…

Target Protein:
Insulin-like growth factor 1 receptor
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Atl146e DB05191
small molecule

ATL146e is an anti-inflammatory compounds which is an agonist of A2A adenosine receptors.

Kategori:
Acids, CarbocyclicAdenosine A receptor agonistsAdenosine A2 Receptor Agonists +3
Target Protein:
Adenosine receptor A2a
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Atlantic halibut Approved DB15549
biotech

Atlantic halibut allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
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Atlantic mackerel Approved DB15542
biotech

Atlantic mackerel allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
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ATM-3507 DB17198
small molecule | CAS: 1861449-70-8

Deskripsi belum tersedia.

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ATN-161 DB05491
small molecule | CAS: 262438-43-7

ATN-161 is a non-RGD based integrin binding peptide targeting alpha-5 beta-1 and alpha-v beta-3. It inhibits the migration and adhesion of particular integrins on activated endothelial cells that play a critical role in tumor angiogenesis. This approach targe…

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
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Atoltivimab Approved DB15898
biotech | CAS: 2135632-29-8

Ebola virus (EBOV) remains an important human pathogen within the _Ebolavirus_ genus, having been responsible for at least 17 known outbreaks with an average case fatality rate of 43.92%.[A221825] Immune therapy using monoclonal antibodies (mAbs) is becoming …

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +10
Target Protein:
Envelope glycoprotein
Waktu ParuhAtoltivimab adminis…
Vol. DistribusiAtoltivimab adminis…
KlirensAtoltivimab adminis…
Genetik -
Atomoxetine Approved DB00289
small molecule | CAS: 83015-26-3

Atomoxetine is a selective norepinephrine (NE) reuptake inhibitor used for the treatment of attention deficit hyperactivity disorder (ADHD). Also known as the marketed product Strattera, atomoxetine is used with other treatment modalities (psychological, educ…

Kategori:
Adrenergic AgentsAgents producing tachycardiaAgents that produce hypertension +17
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporterNMDA receptor +2
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +3
Waktu ParuhThe reported half-l…
Vol. DistribusiThe reported volume…
KlirensThe clearance rate …
Genetik 6 Varian
Atopaxar DB12046
small molecule | CAS: 751475-53-3

Atopaxar has been investigated for the treatment of Coronary Artery Disease and Acute Coronary Syndrome.

Kategori:
Receptors, Thrombin, antagonists & inhibitors
Target Protein:
Proteinase-activated receptor 1
Waktu Paruh-
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Atorvastatin Approved DB01076
small molecule | CAS: 134523-00-5

Atorvastatin (Lipitor®), is a lipid-lowering drug included in the statin class of medications. By inhibiting the endogenous production of cholesterol in the liver, statins lower abnormal cholesterol and lipid levels, and ultimately reduce the risk of cardiova…

Kategori:
Agents Causing Muscle ToxicityAnticholesteremic AgentsBSEP/ABCB11 Substrates +37
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductaseDipeptidyl peptidase 4Aryl hydrocarbon receptor +2
Gen Terkait:
KIF6 HMGCR CYP3A4
Waktu ParuhThe half-life of at…
Vol. DistribusiThe reported volume…
KlirensThe registered tota…
Genetik 3 Varian
Atosiban Approved DB09059
small molecule | CAS: 90779-69-4

Atosiban is an inhibitor of the hormones oxytocin and vasopressin. It is used intravenously to halt premature labor. Although initial studies suggested it could be used as a nasal spray and hence would not require hospital admission, it is not used in that fo…

Kategori:
Amino Acids, Peptides, and ProteinsGenito Urinary System and Sex HormonesHormone Antagonists +8
Target Protein:
Oxytocin receptorVasopressin V1a receptorVasopressin V1b receptor +1
Waktu ParuhAtosiban does not c…
Vol. DistribusiAtosiban has a mean…
KlirensAtosiban has a mean…
Genetik -
Atovaquone Approved DB01117
small molecule | CAS: 95233-18-4

Atovaquone is a hydroxynaphthoquinone, or an analog of ubiquinone, that has antimicrobial and antipneumocystis activity. It is being used in antimalarial protocols.

Kategori:
Anti-Infective AgentsAntibiotics for Pneumocystis PneumoniaAntimalarials +16
Target Protein:
Cytochrome bDihydroorotate dehydrogenase (quinone), mitochondrialDihydroorotate dehydrogenase (quinone), mitochondrial
Waktu Paruh2.2 to 3.2 days
Vol. Distribusi* 0.60 ± 0.17 L/kg
Klirens* 10.4 +/- 5.5 ml/m…
Genetik -
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