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3253

Total database: 17430
Struktur (SMILES)
2451 (75.3%)
Target
1833 (56.3%)
Genomik
35 (1.1%)
Referensi
3253 (100.0%)

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Hasil Pencarian (3253)

Halaman 52 / 66
Remtolumab DB15128
biotech | CAS: 1791410-27-9

Remtolumab is under investigation in clinical trial NCT02433340 (Phase 2, Multicenter, Open-Label Extension (OLE) Study With ABT-122 in Rheumatoid Arthritis Subjects Who Have Completed the Preceding M12-963 Study).

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsGlobulins +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
REN-850 DB05912
small molecule

REN-850 is an oral drug for multiple sclerosis which is in Phase I of clinical trials.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Renzapride DB04917
small molecule | CAS: 112727-80-7

Renzapride is currently in Phase III clinical development in the United States for the treatment of constipation-predominant irritable bowel syndrome (IBS-C). It has been suggested that renzapride is effective in the treatment of irritable bowel syndrome with…

Kategori:
Acids, CarbocyclicAmidesAntidepressive Agents +8
Target Protein:
5-hydroxytryptamine receptor 45-hydroxytryptamine receptor 3A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Repaglinide Approved DB00912
small molecule | CAS: 135062-02-1

Repaglinide is an oral antihyperglycemic agent used for the treatment of non-insulin-dependent diabetes mellitus (NIDDM). It belongs to the meglitinide class of short-acting insulin secretagogues, which act by binding to ? cells of the pancreas to stimulate i…

Kategori:
Acids, AcyclicAlimentary Tract and MetabolismBlood Glucose Lowering Agents +14
Target Protein:
ATP-binding cassette sub-family C member 9ATP-binding cassette sub-family C member 8Histamine H1 receptor +1
Waktu Paruh1 hour
Vol. Distribusi31 L following IV a…
Klirens33-38 L/hour follow…
Genetik -
Reparixin DB12614
small molecule | CAS: 266359-83-5

Reparixin has been used in trials studying the treatment and prevention of Breast Cancer, Metastatic Breast Cancer, Pancreatectomy for Chronic Pancreatitis, Islet Transplantation in Diabetes Mellitus Type 1, and Pancreatic Islet Transplantation in Type 1 Diab…

Kategori:
AmidesSulfonesSulfur Compounds
Target Protein:
C-X-C chemokine receptor type 2C-X-C chemokine receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Reproterol DB12846
small molecule | CAS: 54063-54-6

Reproterol has been used in trials studying the treatment of Asthma, Exercise-Induced.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-Agonists +25
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Reserpine Approved DB00206
small molecule | CAS: 50-55-5

An alkaloid found in the roots of Rauwolfia serpentina and R. vomitoria. Reserpine inhibits the uptake of norepinephrine into storage vesicles resulting in depletion of catecholamines and serotonin from central and peripheral axon terminals. It has been used …

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAlkaloids +37
Target Protein:
Synaptic vesicular amine transporterChromaffin granule amine transporterBaculoviral IAP repeat-containing protein 5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Resmetirom Approved DB12914
small molecule | CAS: 920509-32-6

Resmetirom is a thyroid hormone receptor-beta (THR-beta) agonist. On March 14, 2024, it was approved by the FDA as the first treatment of liver fibrosis due to noncirrhotic non-alcoholic steatohepatitis (NASH), which is a form of non-alcoholic fatty liver dis…

Kategori:
BCRP/ABCG2 InhibitorsBCRP/ABCG2 SubstratesBSEP/ABCB11 Inhibitors +15
Target Protein:
Thyroid hormone receptor beta
Waktu ParuhThe median terminal…
Vol. DistribusiResmetirom apparent…
KlirensThe steady state ap…
Genetik -
Resminostat DB12392
small molecule | CAS: 864814-88-0

Resminostat has been used in trials studying the treatment of Sezary Syndrome, Mycosis fungoides, Hodgkin's Lymphoma, Hepatocellular Carcinoma, and Lymphoma, T-Cell, Cutaneous, among others.

Kategori:
AmidesAminesHydroxy Acids +3
Target Protein:
Histone deacetylase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Resolvin E1 DB13105
small molecule | CAS: 552830-51-0

Resolvin E1 (RX 10001) is under investigation in clinical trial NCT00941018 (Single and Multiple Ascending Oral Dose Study of Resolvin E1 in Healthy Volunteers).

Kategori:
Dietary FatsDietary Fats, UnsaturatedEicosanoids +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Retagliptin DB14898
small molecule | CAS: 1174122-54-3

Retagliptin is under investigation in clinical trial NCT02822534 (The Pharmacokinetics and Pharmacodynamics Study of Single and Multiple Dose of SP2086 in Type 2 Diabetes Patients).

Target Protein:
Dipeptidyl peptidase 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Retapamulin Approved DB01256
small molecule | CAS: 224452-66-8

Retapamulin, marketed by GlaxoSmithKline as the ointment Altabax, is an antibiotic for skin infections like impetigo. It was approved by the FDA in April 2007.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibiotics for Topical Use +6
Target Protein:
50S ribosomal protein L3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Retifanlimab Approved DB15766
biotech | CAS: 2079108-44-2

Retifanlimab is a humanized IgG4 kappa monoclonal antibody that binds to the programmed death receptor-1 (PD-1), blocking PD-1 interaction with its ligands, programmed death-ligand 1 (PD-L1) and programmed death-ligand 2 (PD-L2). By blocking the PD-1/PD-L1/2 …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +11
Target Protein:
Programmed cell death protein 1
Waktu ParuhAt steady-state, re…
Vol. DistribusiAt steady-state, re…
KlirensFollowing the first…
Genetik -
Reversin 121 DB14072
small molecule | CAS: 174630-04-7

Reversin 121 is a hydrophobic peptide chemosensitizer that can reverse P-glycoprotein-mediated multidrug resistance.

Kategori:
Amino Acids, Peptides, and ProteinsDrug Resistance, MultipleP-glycoprotein inhibitors +1
Target Protein:
ATP-dependent translocase ABCB1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rezatomidine DB12143
small molecule | CAS: 847829-38-3

Rezatomidine has been used in trials studying the treatment of Fibromyalgia, Cystitis, Interstitial, Irritable Bowel Syndrome, and Diabetic Neuropathy, Painful.

Target Protein:
Alpha-2C adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RG-2833 DB16955
small molecule | CAS: 1215493-56-3

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAcids, CarbocyclicAmides +5
Target Protein:
Histone deacetylase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RGLS-8429 DB18127
biotech

RGLS-8429 is an investigational anti-miR-17 oligonucleotide.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RGX-121 DB17681
biotech

RGX-121 is designed to use the NAV AAV9 vector to deliver the human iduronate-2-sulfatase gene to the central nervous system.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 104114-27-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
rhThrombin Approved DB04923
biotech | CAS: 1270043-60-1

rhThrombin (recombinant human thrombin) is being developed by ZymoGenetics, Inc. as a general aid to achieving hemostasis during surgery. ZymoGenetics is developing rhThrombin, a recombinant form of human thrombin that is not derived from animal or human bloo…

Waktu ParuhApproximately 15 ho…
Vol. Distribusi-
Klirens-
Genetik -
Ribavirin Approved DB00811
small molecule | CAS: 36791-04-5

Producing a broad-spectrum activity against several RNA and DNA viruses, Ribavirin is a synthetic guanosine nucleoside and antiviral agent that interferes with the synthesis of viral mRNA. It is primarily indicated for use in treating hepatitis C and viral he…

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntimetabolites +13
Target Protein:
Inosine-5'-monophosphate dehydrogenase 1RNA-directed RNA polymerase LGenome polyprotein +2
Gen Terkait:
IFNL3
Waktu ParuhThe terminal half-l…
Vol. DistribusiRibavirin displays …
KlirensThe total apparent …
Genetik 1 Varian
Ribociclib Approved DB11730
small molecule | CAS: 1211441-98-3

Ribociclib is a selective cyclin-dependent kinase inhibitor, a class of drugs that help slow the progression of cancer by inhibiting two proteins called cyclin-dependent kinase 4 and 6 (CDK4/6). These proteins, when over-activated, can enable cancer cells to …

Kategori:
AminesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +17
Target Protein:
Cyclin-dependent kinase 4Cyclin-dependent kinase 6
Waktu ParuhAt steady-state in …
Vol. DistribusiAt steady-state, th…
KlirensAt steady-state in …
Genetik -
Rice bran oil Approved DB11293
biotech

Rice bran oil is extracted from the hard outer brown layer of rice after chaff (rice husk) used for high-temperature cooking methods such as deep frying and stir frying. It contains monosaturated fatty acids, polyunsaturated fatty acids, and saturated fatty a…

Kategori:
Biological ProductsComplex MixturesDietary Fats +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ricinoleic acid DB02955
small molecule | CAS: 141-22-0

Deskripsi belum tersedia.

Kategori:
Biological ProductsFatsFats, Unsaturated +6
Target Protein:
Cannabinoid receptor 1Cannabinoid receptor 2Transient receptor potential cation channel subfamily V member 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ricolinostat DB12376
small molecule | CAS: 1316214-52-4

Ricolinostat is under investigation for the treatment of Breast Carcinoma and Metastatic Breast Cancer.

Kategori:
AminesAntineoplastic AgentsEnzyme Inhibitors +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ridogrel DB01207
small molecule | CAS: 110140-89-1

Ridogrel is a dual action drug useful for the prevention of systemic thrombo-embolism and as an adjunctive agent to thrombolytic therapy in acute myocardial infarction. However, there currently are no clinical indications for preferential use of ridogrel over…

Kategori:
Acids, AcyclicAntiplatelet agentsEnzyme Inhibitors +7
Target Protein:
Thromboxane-A synthaseThromboxane A2 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rifalazil DB04934
small molecule | CAS: 129791-92-0

Rifalazil is a derivative of the antibiotic rifamycin. It is being investigated by ActivBiotics for the treatment of various bacterial infections.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibiotics, Antitubercular +7
Target Protein:
DNA-directed RNA polymerase subunit beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rifampin Approved DB01045
small molecule | CAS: 13292-46-1

Rifampin, also known as rifampicin, is a broad-spectrum antimicrobial [A263748] that was first discovered in 1965 [A263753] and clinically used in 1968.[A263768] Rifampin is used to treat tuberculosis and works by inhibiting the microbial DNA-dependent RNA po…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +55
Target Protein:
DNA-directed RNA polymerase subunit betaNuclear receptor subfamily 1 group I member 2
Waktu ParuhIn healthy adults, …
Vol. DistribusiFollowing intraveno…
KlirensFollowing intraveno…
Genetik -
Rifapentine Approved DB01201
small molecule | CAS: 61379-65-5

Rifapentine is an antibiotic drug used in the treatment of tuberculosis. It inhibits DNA-dependent RNA polymerase activity in susceptible cells. Specifically, it interacts with bacterial RNA polymerase but does not inhibit the mammalian enzyme.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibiotics, Antitubercular +24
Target Protein:
DNA-directed RNA polymerase subunit beta'
Waktu Paruh-
Vol. Distribusi* 70.2 ± 9.1 L
Klirens* Apparent Oral cl=…
Genetik -
Rifaximin Approved DB01220
small molecule | CAS: 80621-81-4

Rifaximin is a semisynthetic, rifamycin-based non-systemic antibiotic, meaning that the drug will not pass the gastrointestinal wall into the circulation as is common for other types of orally administered antibiotics. It has multiple indications and is used …

Kategori:
Alimentary Tract and MetabolismAnti-Bacterial AgentsAnti-Infective Agents +22
Target Protein:
DNA-directed RNA polymerase subunit betaNuclear receptor subfamily 1 group I member 2
Waktu ParuhApproximately 6 hou…
Vol. Distribusi-
Klirens-
Genetik -
Rigosertib DB12146
small molecule | CAS: 592542-59-1

Rigosertib has been used in trials studying the treatment and basic science of MDS, RAEB, Cancer, Hepatoma, and Neoplasms, among others.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAntineoplastic Agents +3
Target Protein:
Serine/threonine-protein kinase PLK1Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rilapladib DB05119
small molecule | CAS: 412950-08-4

Rilapladib is the third genomics-derived small molecule drug arising from the Human Genome Sciences-GlaxoSmithKline collaboration to enter clinical development. It is a lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitor. Lp-PLA2 is an enzyme associat…

Kategori:
AcetatesAcids, AcyclicAmides +2
Target Protein:
Thymidine kinase, cytosolicPhospholipase A2Platelet-activating factor acetylhydrolase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rilonacept Approved DB06372
biotech | CAS: 501081-76-1

Rilonacept is a dimeric fusion protein consisting of portions of IL-1R and the IL-1R accessory protein linked to the Fc portion of immunoglobulin G1. Rilonacept functions as an interleukin 1 inhibitor and is used in the treatment of CAPS, also known as cryopy…

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAnti-Inflammatory Agents +9
Target Protein:
Interleukin-1 betaInterleukin-1 alphaInterleukin-1 receptor antagonist protein
Waktu Paruh8.6 days
Vol. Distribusi-
Klirens-
Genetik -
Rimacalib DB12571
small molecule | CAS: 215174-50-8

Rimacalib has been used in trials studying the treatment of Rheumatoid Arthritis (RA).

Kategori:
Enzyme InhibitorsOxazinesProtein Kinase Inhibitors
Target Protein:
Calcium/calmodulin-dependent protein kinase type II subunit alphaCalcium/calmodulin-dependent protein kinase type II subunit betaCalcium/calmodulin-dependent protein kinase type II subunit delta +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rimegepant Approved DB12457
small molecule | CAS: 1289023-67-1

Rimegepant is an oral antagonist of the CGRP receptor developed by Biohaven Pharmaceuticals.[L11028] It received FDA approval on February 27, 2020 for the acute treatment migraine headache,[L11974] and was subsequently approved by the European Commission in A…

Kategori:
AnalgesicsAntimigraine PreparationsBCRP/ABCG2 Substrates +19
Target Protein:
Calcitonin gene-related peptide type 1 receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiAt steady state, th…
Klirens-
Genetik -
Rimeporide DB12861
small molecule | CAS: 187870-78-6

Rimeporide has been used in trials studying the treatment of Muscular Dystrophy, Duchenne.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rintatolimod DB16425
biotech | CAS: 38640-92-5

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntiviral AgentsBase Pair Mismatch +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Risankizumab Approved DB14762
biotech | CAS: 1612838-76-2

Risankizumab is a fully humanized IgG1 monoclonal antibody (mAb) directed against interleukin 23 (IL-23).[L39885] It gained its first global approval in Japan in March 2019, followed by approval in Canada, the US, and Europe in April 2019.[A254716] Risankizum…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +15
Target Protein:
Interleukin-23
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe estimated stead…
KlirensThe estimated syste…
Genetik -
Risdiplam Approved DB15305
small molecule | CAS: 1825352-65-5

Risdiplam is an orally bioavailable mRNA splicing modifier used for the treatment of spinal muscular atrophy (SMA).[L12615] It increases systemic SMN protein concentrations by improving the efficiency of _SMN2_ gene transcription. This mechanism of action is …

Kategori:
BCRP/ABCG2 SubstratesCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +11
Waktu ParuhThe terminal elimin…
Vol. DistribusiFollowing oral admi…
KlirensFor a 14.9kg patien…
Genetik -
Risperidone Approved DB00734
small molecule | CAS: 106266-06-2

Risperidone is a second-generation antipsychotic (SGA) medication used in the treatment of a number of mood and mental health conditions including schizophrenia and bipolar disorder.[L12885] It is one of the most widely used SGAs. [Paliperidone], another comm…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +42
Target Protein:
5-hydroxytryptamine receptor 2AD(2) dopamine receptorAlpha-1B adrenergic receptor +9
Waktu Paruh3 hours in extensiv…
Vol. DistribusiThe volume of distr…
KlirensRisperidone is clea…
Genetik -
Ritanserin DB12693
small molecule | CAS: 87051-43-2

Ritanserin has been used in trials studying the treatment of Cocaine-Related Disorders.

Kategori:
Anti-Anxiety AgentsAntidepressive AgentsAntidepressive Agents, Second-Generation +21
Target Protein:
5-hydroxytryptamine receptor 2B5-hydroxytryptamine receptor 2CVoltage-dependent N-type calcium channel subunit alpha-1B +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ritlecitinib Approved DB14924
small molecule | CAS: 1792180-81-4

Ritlecitinib (PF-06651600) is a highly selective inhibitor of Janus kinase 3 (JAK3) and the tyrosine kinase expressed in hepatocellular carcinoma (TEC) kinase family. In June 2023, it was approved by the FDA for the treatment of severe alopecia areata in adul…

Kategori:
Antineoplastic and Immunomodulating AgentsCytochrome P-450 CYP1A2 InhibitorsCytochrome P-450 CYP1A2 Inhibitors (strength unknown) +16
Target Protein:
Tyrosine-protein kinase JAK3Tyrosine-protein kinase TecTyrosine-protein kinase ITK/TSK +3
Waktu ParuhRitlecitinib has a …
Vol. DistribusiRitlecitinib is pre…
KlirensRitlecitinib is pre…
Genetik -
Ritobegron DB12080
small molecule | CAS: 255734-04-4

Ritobegron is under investigation in clinical trial NCT02256735 (Study to Investigate the Effect of KUC 7483 CL on the QT/QTc Interval of the ECG in Comparison to Placebo and Moxifloxacin in Healthy Male and Female Volunteers).

Kategori:
Acids, AcyclicAdrenergic AgentsAdrenergic Agonists +15
Target Protein:
Beta-3 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rivastigmine Approved DB00989
small molecule | CAS: 123441-03-2

Rivastigmine is a parasympathomimetic or cholinergic agent for the treatment of mild to moderate dementia of the Alzheimer's type. Rivastigmine is a cholinesterase inhibitor that inhibits both butyrylcholinesterase and acetylcholinesterase.

Kategori:
Acids, AcyclicAnti-Dementia DrugsBradycardia-Causing Agents +13
Target Protein:
AcetylcholinesteraseCholinesterase
Waktu Paruh1.5 hours
Vol. Distribusi* 1.8 to 2.7 L/kg
Klirens* renal cl=2.1-2.8 …
Genetik -
Rivipansel DB12778
small molecule | CAS: 927881-99-0

Rivipansel has been used in trials studying the other, basic science, and treatment of Pain Crisis, Renal impairment, Anemia, Sickle Cell, Sickle Cell Disease, and Sickle Cell Disorders, among others.

Kategori:
CarbohydratesGlycoconjugatesLipids
Target Protein:
E-selectinL-selectinP-selectin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RLYB212 DB17727
biotech

RLYB212 is a human monoclonal antibody against Antigen-1A Immunoglobulin (HPA-1A). It is currently being developed by Rallybio for the prevention of fetal and neonatal alloimmune thrombocytopenia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ro 12-7310 DB08455
small molecule | CAS: 65316-65-6

Deskripsi belum tersedia.

Kategori:
AlkenesBiological FactorsCarotenoids +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RO-4987655 DB12933
small molecule | CAS: 874101-00-5

RO4987655 has been used in trials studying the treatment of Neoplasms.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RO-5028442 DB12721
small molecule | CAS: 920022-47-5

RO5028442 has been used in trials studying Autistic Disorder.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Robatumumab DB12976
biotech | CAS: 934235-44-6

Robatumumab has been used in trials studying the treatment of Osteosarcoma, Sarcoma, Ewing's, and Peripheral Neuroectodermal Tumor.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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