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6694

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Halaman 51 / 134
Elivaldogene autotemcel Approved DB16746
biotech

Elivaldogene autotemcel is a gene therapy consisting of genetically modified autologous cells. It is used to provide functional copies of human adrenoleukodystrophy protein (ALDP) in patients with adrenoleukodystrophy,[L39491] an X-linked genetic disorder cha…

Kategori:
Alimentary Tract and MetabolismCellular and Gene TherapyVarious Alimentary Tract and Metabolism Products
Waktu ParuhAs elivaldogene aut…
Vol. DistribusiAs elivaldogene aut…
KlirensAs elivaldogene aut…
Genetik -
biotech | CAS: 1905397-73-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ellagic acid DB08846
small molecule | CAS: 476-66-4

Ellagic acid is present in several fruits such as cranberries, strawberries, raspberries, and pomegranates. In pomegranates, there are several therapeutic compounds but ellagic acid is the most active and abundant. Ellagic acid is also present in vegetables. …

Kategori:
BenzopyransCytochrome P-450 CYP2E1 InhibitorsCytochrome P-450 CYP2E1 Inhibitors (strength unknown) +6
Target Protein:
Heat shock 70 kDa protein 1AHeat shock 70 kDa protein 1BGlycogen synthase kinase-3 beta +17
Waktu Paruh-
Vol. Distribusi-
KlirensEllagic acid is eli…
Genetik -
Ellipticine DB17026
small molecule | CAS: 519-23-3

Ellipticine is a potent antineoplastic agent.[A252992]

Kategori:
AlkaloidsAntineoplastic AgentsCarbazoles +8
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elobixibat DB12486
small molecule | CAS: 439087-18-0

Elobixibat has been used in trials studying the treatment and basic science of Dyslipidemia, Constipation, Chronic Constipation, Functional Constipation, and Chronic Idiopathic Constipation.

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsAzepines +5
Target Protein:
Ileal sodium/bile acid cotransporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elocalcitol DB06194
small molecule | CAS: 199798-84-0

Elocalcitol is a calcitriol analog for inhibition of prostate cell growth; in phase II clinical trial in patients with benign prostate hyperplasia (4/2004).

Kategori:
CholestanesCholestenesFused-Ring Compounds +8
Target Protein:
Vitamin D3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elotuzumab Approved DB06317
biotech | CAS: 915296-00-3

Elotuzumab is a humanized IgG1 (Immunoglobulin G) monoclonal antibody indicated in combination with lenalidomide and dexamethasone for the treatment of patients with multiple myeloma who have received one to three prior therapies. Elotuzumab targets SLAMF7, a…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +15
Target Protein:
SLAM family member 7
Waktu Paruh-
Vol. Distribusi-
KlirensThe clearance of el…
Genetik -
Elranatamab Approved DB15395
biotech | CAS: 2408850-14-4

Elranatamab is a bispecific B-cell maturation antigen (BCMA)-directed CD3 T-cell engager. It is a humanized immunoglobulin 2-alanine kappa antibody derived from two monoclonal antibodies (mAbs), an anti-BCMA mAb and an anti-CD3 mAb,[A261060] each of which con…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalBispecific B-cell maturation antigen (BCMA)-directed CD3 T-cell engager +5
Target Protein:
Tumor necrosis factor receptor superfamily member 17T-cell surface glycoprotein CD3
Waktu ParuhThe mean (CV%) half…
Vol. DistribusiThe mean (CV%) stea…
KlirensThe mean (CV%) clea…
Genetik -
Elsamitrucin DB05129
small molecule | CAS: 97068-30-9

The cytostatic agent Elsamitrucin is a new fermentation product active in a variety of in vivo tumor models of murine and human origin. (PMID: 8150873)

Kategori:
Antibiotics, AntineoplasticAntineoplastic AgentsCarbohydrates +1
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-betaDNA +1
Waktu Paruh36–60 h
Vol. Distribusi-
Klirens-
Genetik -
Elsubrutinib DB18850
small molecule | CAS: 1643570-24-4

Elsubrutinib is under investigation in clinical trial NCT04451772 (A Study of the Safety of Oral Elsubrutinib Capsules and Oral Upadacitinib Tablets Given Alone or in Combination (ABBV-599) for Adult Participants With Moderately to Severely Active Systemic Lu…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eltanolone DB12308
small molecule | CAS: 128-20-1

Eltanolone is under investigation in clinical trial NCT02603926 (Treatment of Fragile-X Associated Tremor/Ataxia Syndrome (FXTAS) With Allopregnanolone).

Kategori:
AnestheticsCentral Nervous System AgentsCentral Nervous System Depressants +3
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Gamma-aminobutyric acid receptor subunit beta-2Gamma-aminobutyric acid receptor subunit gamma-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eltrekibart DB19017
biotech | CAS: 2484883-56-7

Eltrekibart is under investigation in clinical trial NCT06046729 (A Study of Eltrekibart (LY3041658) in Adult Participants With Moderate to Severe Hidradenitis Suppurativa).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eltrombopag Approved DB06210
small molecule | CAS: 496775-61-2

Eltrombopag is used to treat low blood platelet counts in adults with chronic immune (idiopathic) thrombocytopenia (ITP), when certain other medicines, or surgery to remove the spleen, have not worked well enough. ITP is a condition that may cause unusual bru…

Kategori:
Acids, CarbocyclicBCRP/ABCG2 InhibitorsBenzene Derivatives +25
Target Protein:
Thrombopoietin receptor
Gen Terkait:
F5 SERPINC1
Waktu ParuhAbout 21-32 hours i…
Vol. DistribusiBased on a radiolab…
Klirens-
Genetik 2 Varian
Eluvixtamab DB17252
biotech | CAS: 1679391-73-1

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eluxadoline Approved DB09272
small molecule | CAS: 864821-90-9

Eluxadoline is a mixed mu-opioid receptor agonist, kappa-opioid receptor agonist, and a-delta opioid receptor antagonist indicated for use in diarrhea-predominant irritable bowel syndrome (IBS-D). The mu-, kappa-, and delta-opioid receptors mediate endogenous…

Kategori:
Alimentary Tract and MetabolismAmino AcidsAmino Acids, Aromatic +15
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor
Waktu ParuhThe mean plasma eli…
Vol. Distribusi-
Klirens-
Genetik -
Elvitegravir Approved DB09101
small molecule | CAS: 697761-98-1

Elvitegravir is a human immunodeficiency virus type 1 (HIV-1) integrase strand transfer inhibitor (INSTI) used for the treatment of HIV-1 infection in antiretroviral treatment-experienced adults. Because integrase is necessary for viral replication, inhibitio…

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +22
Target Protein:
IntegraseGag-Pol polyprotein
Waktu ParuhThe median terminal…
Vol. Distribusi-
Klirens-
Genetik -
Elvucitabine DB06236
small molecule | CAS: 181785-84-2

Deskripsi belum tersedia.

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +13
Target Protein:
Gag-Pol polyproteinReverse transcriptase/RNaseH
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elzovantinib DB18918
small molecule | CAS: 2271119-26-5

Elzovantinib is under investigation in clinical trial NCT03993873 (Study of TPX-0022 in Patients With Advanced NSCLC, Gastric Cancer or Solid Tumors Harboring Genetic Alterations in MET).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Emactuzumab DB14905
biotech | CAS: 1448221-67-7

Emactuzumab is under investigation in clinical trial NCT01494688 (A Study of RO5509554 as Monotherapy and in Combination With Paclitaxel in Participants With Advanced Solid Tumors).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Emapunil DB12666
small molecule | CAS: 226954-04-7

Emapunil has been used in trials studying the basic science and diagnostic of Baseline, Blocking Receptor Binding, and Neurodegenerative Disorders.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Translocator protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EMB-01 DB16091
biotech

EMB-01 is under investigation in clinical trial NCT03797391 (A Dose Escalation Study of EMB-01 in Participants With Advanced/metastatic Solid Tumors).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Emerfetamab DB18474
biotech | CAS: 2250261-27-7

Emerfetamab is a bispecific T cell engager antibody construct with a half-life extension Fc moiety capable of binding to the neonatal Fc receptor.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Emibetuzumab DB11849
biotech | CAS: 1365287-97-3

Emibetuzumab has been used in trials studying the treatment of Advanced Cancer, Renal Cell Carcinoma, Hepatocellular Cancer, Gastric Adenocarcinoma, and Non-Small Cell Lung Cancer, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Emicerfont DB12910
small molecule | CAS: 786701-13-1

Emicerfont has been used in trials studying the diagnostic and treatment of Social Anxiety Disorder and Irritable Bowel Syndrome (IBS).

Kategori:
Corticotropin-Releasing Hormone, antagonists & inhibitors
Target Protein:
Corticotropin-releasing factor receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Emicizumab Approved DB13923
biotech | CAS: 1610943-06-0

Emicizumab is a humanized recombinant monoclonal antibody that mimics the function of the coagulation Factor VIII and it has the capacity to bind simultaneously to activated Factor IX and Factor X. The ability of Emicizumab to bind to all these three differen…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Target Protein:
Coagulation factor IXCoagulation factor X
Waktu ParuhEmcicizumab present…
Vol. DistribusiThe apparent volume…
KlirensThe apparent cleara…
Genetik -
Emivirine DB08188
small molecule | CAS: 149950-60-7

Emivirine has been used in trials studying the treatment of HIV Infections.

Kategori:
Anti-Infective AgentsAnti-Retroviral AgentsAntiviral Agents +5
Target Protein:
Gag-Pol polyproteinGag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Empagliflozin Approved DB09038
small molecule | CAS: 864070-44-0

Empagliflozin is an inhibitor of sodium-glucose co-transporter-2 (SGLT2), the transporters primarily responsible for the reabsorption of glucose in the kidney.[A203453] It is used clinically as an adjunct to diet and exercise, often in combination with other …

Kategori:
Alimentary Tract and MetabolismBCRP/ABCG2 SubstratesBenzene Derivatives +16
Target Protein:
Sodium/glucose cotransporter 2
Waktu ParuhThe apparent termin…
Vol. DistribusiThe estimated appar…
KlirensApparent oral clear…
Genetik -
Emrusolmin DB13927
small molecule | CAS: 882697-00-9

Emrusolmin restores hippocampal synaptic and transcriptional plasticity as well as spatial memory in a mouse model for Alzheimer's disease, when given orally before or after the onset of pathology. [A31409]

Kategori:
DioxolesHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Emtricitabine Approved DB00879
small molecule | CAS: 143491-57-0

Emtricitabine is a nucleoside reverse transcriptase inhibitor (NRTI) indicated for the treatment of HIV infection in adults[L9019] or combined with [tenofovir alafenamide] for the prevention of HIV-1 infection in high risk adolescents and adults.[L9010] Emtri…

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +23
Target Protein:
Reverse transcriptase/RNaseHGag-Pol polyprotein
Waktu ParuhThe half life of em…
Vol. DistribusiThe apparent centra…
KlirensEmtricitabine has a…
Genetik -
Enadenotucirev DB14873
biotech | CAS: 1402042-02-7

Enadenotucirev is under investigation in clinical trial NCT02636036 (Phase I Study of Enadenotucirev and PD-1 Inhibitor in Subjects With Metastatic or Advanced Epithelial Tumors).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enalapril Approved DB00584
small molecule | CAS: 75847-73-3

Enalapril is a prodrug belonging to the angiotensin-converting enzyme (ACE) inhibitor drug class that works on the renin-angiotensin-aldosterone system, which is responsible for the regulation of blood pressure and fluid and electrolyte homeostasis. Enalapril…

Kategori:
ACE Inhibitors and Calcium Channel BlockersACE Inhibitors and DiureticsAgents Acting on the Renin-Angiotensin System +21
Target Protein:
Angiotensin-converting enzyme
Waktu ParuhThe average termina…
Vol. DistribusiThe volume of distr…
KlirensFollowing oral admi…
Genetik -
Enasidenib Approved DB13874
small molecule | CAS: 1446502-11-9

Enasidenib is an orally available treatment for the treatment of adult patients with relapsed or refractory acute myeloid leukemia (AML) with specific mutations in the isocitrate dehydrogenase 2 (IDH2) gene, which is a recurrent mutation detected in 12-20% of…

Kategori:
AminesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +62
Target Protein:
Isocitrate dehydrogenase [NADP] cytoplasmicIsocitrate dehydrogenase [NAD] subunit alpha, mitochondrialIsocitrate dehydrogenase [NAD] subunit beta, mitochondrial +2
Waktu ParuhEnasidenib has a te…
Vol. DistribusiThe mean volume of …
KlirensEnasidenib has a me…
Genetik -
Enavogliflozin DB18970
small molecule | CAS: 1415472-28-4

Enavogliflozin is under investigation in clinical trial NCT06399835 (Enavogliflozin vs. Pioglitazone on Glucose and Atherosclerosis).

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Encainide Approved DB01228
small molecule | CAS: 66778-36-7

All drug products containing encainide hydrochloride. Encainide hydrochloride, formerly marketed as Enkaid capsules, was associated with increased death rates in patients who had asymptomatic heart rhythm abnormalities after a recent heart attack. The manufac…

Kategori:
AmidesAminesAnilides +13
Target Protein:
Sodium channel protein type 5 subunit alpha
Waktu Paruh1-2 hours
Vol. Distribusi-
Klirens-
Genetik -
Encaleret DB18096
small molecule | CAS: 787583-71-5

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAlcoholsAmines +3
Target Protein:
Extracellular calcium-sensing receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Encorafenib Approved DB11718
small molecule | CAS: 1269440-17-6

Encorafenib, also known as _BRAFTOVI_, is a kinase inhibitor. Encorafenib inhibits BRAF gene, which encodes for B-raf protein, which is a proto-oncogene involved in various genetic mutations.[L12216] This protein plays a role in regulating the MAP kinase/E…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +47
Target Protein:
Serine/threonine-protein kinase B-rafG1/S-specific cyclin-D1RAF proto-oncogene serine/threonine-protein kinase +7
Waktu ParuhThe mean (CV%) term…
Vol. DistribusiThe blood-to-plasma…
KlirensThe apparent cleara…
Genetik -
Endostar DB11727
biotech

Endostar is under investigation for the treatment of Nasopharyngeal Carcinoma. Endostar has been investigated for the treatment of Non-small Cell Lung Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +15
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Endothelin-1 DB12652
biotech | CAS: 117399-94-7

Endothelin 1 is under investigation in clinical trial NCT00745693 (The Effects of Diesel Exhaust Inhalation on Vascular Function - the Role of Endothelin).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsEndothelin-1, antagonists & inhibitors +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enfuvirtide Approved DB00109
biotech | CAS: 159519-65-0

Enfuvirtide is a 36 amino acid biomimetic peptide that is structurally similar to the HIV proteins that are responsible for the fusion of the virus to cell membranes and subsequent intracellular uptake. The first agent in the novel class of antiretroviral dru…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-HIV AgentsAnti-Infective Agents +31
Target Protein:
Envelope glycoprotein
Waktu Paruh3.8 +/- 0.6 hrs
Vol. Distribusi* 5.5 ± 1.1 L
Klirens* 24.8 +/- 4.1 mL/h…
Genetik -
biotech | CAS: 2567881-77-8

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2417199-08-5

Englumafusp alfa is under investigation in clinical trial NCT04077723 (A Study to Evaluate the Safety, Pharmacokinetics and Preliminary Anti-tumor Activity of Englumafusp Alfa in Combination With Obinutuzumab and in Combination With Glofitamab Following a Pre…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enibarcimab DB16730
biotech | CAS: 2305638-98-4

Enibarcimab is under investigation in clinical trial NCT03989531 (Adrecizumab in Cardiogenic Shock).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eniluracil DB03516
small molecule | CAS: 59989-18-3

Eniluracil, which was previously under development by GlaxoSmithKline (GSK), is being developed by Adherex to enhance the therapeutic value and effectiveness of 5-fluorouracil (5-FU), one of the world’s most widely-used oncology agents. 5-FU is widely used i…

Kategori:
Enzyme InhibitorsPyrimidinesPyrimidinones
Target Protein:
Dihydropyrimidine dehydrogenase [NADP(+)]Aldehyde oxidaseXanthine dehydrogenase/oxidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enisoprost DB19319
small molecule | CAS: 81026-63-3

Deskripsi belum tersedia.

Kategori:
Anti-Ulcer AgentsAutacoidsBiological Factors +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enitociclib DB17297
small molecule | CAS: 1610408-97-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enmetazobactam Approved DB18716
small molecule | CAS: 1001404-83-6

Enmetazobactam is a penicillanic acid sulfone extended-spectrum beta (?)-lactamase (ESBL) inhibitor.[A263266] Because ESBL enzymes can hydrolyze important antibiotics such as penicillins, broad-spectrum cephalosporins and monobactams, ESBL-producing bacteria …

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAza Compounds +7
Target Protein:
Extended-spectrum beta-lactamase PER-1Beta-lactamase
Waktu ParuhThe mean (SD) half-…
Vol. DistribusiMean (SD) steady st…
KlirensThe mean (SD) clear…
Genetik -
Enoxacin Approved DB00467
small molecule | CAS: 74011-58-8

A broad-spectrum 6-fluoronaphthyridinone antibacterial agent (fluoroquinolones) structurally related to nalidixic acid.

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +14
Target Protein:
DNA topoisomerase 2-betaDNA gyrase subunit ADNA topoisomerase 4 subunit A +1
Waktu ParuhPlasma half-life is…
Vol. Distribusi-
Klirens-
Genetik -
Enoxaparin Approved DB01225
small molecule | CAS: 9005-49-6

Enoxaparin is a common low-molecular-weight heparin (LMWH) used in the prevention and management of various thromboembolic disorders. Initially approved by the FDA in 1993, it is administered by a subcutaneous or intravenous injection and marketed by several …

Kategori:
Agents causing hyperkalemiaAnticoagulantsBlood and Blood Forming Organs +7
Target Protein:
Antithrombin-IIICoagulation factor XProthrombin
Waktu ParuhThe half-life of en…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik -
Enoxolone DB13089
small molecule | CAS: 471-53-4

Enoxolone (glycyrrhetic acid) has been investigated for the basic science of Apparent Mineralocorticoid Excess (AME).

Kategori:
Anti-Inflammatory AgentsCicatrizantsDermatologicals +4
Target Protein:
Tyrosine-protein phosphatase non-receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enpatoran DB16501
small molecule | CAS: 2101938-42-3

Enpatoran (M5049) was under investigation in clinical trials for various conditions. It was investigated for systemic lupus erythematosus and cutaneous lupus erythematosus in completed trials (NCT04647708 and NCT05162586) and in a recruiting trial (NCT0554032…

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 2501–2550 dari 6694
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