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11793

Total database: 17430
Struktur (SMILES)
8607 (73.0%)
Target
6418 (54.4%)
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102 (0.9%)
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11793 (100.0%)

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Halaman 51 / 236
Batoclimab DB16104
biotech | CAS: 2187430-05-1

Batoclimab is under investigation in clinical trial NCT04428255 (A Clinical Study on the Efficacy and Safety of HBM9161 in Patients With ITP).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
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Batoprotafib DB19137
small molecule | CAS: 1801765-04-7

Batoprotafib is under investigation in clinical trial NCT04330664 (Adagrasib in Combination With TNO155 in Patients With Cancer (KRYSTAL 2)).

Waktu Paruh-
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Batroxobin DB09005
biotech | CAS: 9039-61-6

Batroxobin is a defibrinogenating hemostatic agent derived from the venom of a pit viper, Bothrops atrox moojeni. In addition to batroxobin, the venom of Bothrops atrox has a composition of 10.2% neutral carbohydrate. Batroxobin is a serine protease, which cl…

Kategori:
Biological FactorsBlood and Blood Forming OrgansCardiovascular Agents +18
Waktu Paruh-
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Bavdegalutamide DB19032
small molecule | CAS: 2222112-77-6

Bavdegalutamide is under investigation in clinical trial NCT03888612 (Trial of ARV-110 in Patients With Metastatic Castration Resistant Prostate Cancer).

Waktu Paruh-
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Bavisant DB12299
small molecule | CAS: 929622-08-2

Bavisant has been used in trials studying the basic science and treatment of Alcoholism, Pharmacokinetics, Drug Interactions, Attention Deficit Hyperactivity Disorder, and Attention Deficit Disorders With Hyperactivity.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +2
Target Protein:
Histamine H3 receptor
Waktu Paruh-
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Bavituximab DB05136
biotech | CAS: 648904-28-3

Bavituximab is a chimeric Anti-PS monoclonal antibody analog which is used to potentially treat cancers and viral infections. It binds to phosphatidylserine and other exposed host cell lipids when induced by cellular stress. Additional analogs in the class in…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntineoplastic Agents +7
Waktu Paruh30 Hrs
Vol. Distribusi-
Klirens-
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Baxdrostat DB19090
small molecule | CAS: 1428652-17-8

Baxdrostat is under investigation in clinical trial NCT06344104 (A Phase III Study to Investigate the Efficacy and Safety of Baxdrostat in Asian Participants With Uncontrolled Hypertension on Two or More Medications Including Participants With Resistant Hyper…

Target Protein:
Cytochrome P450 11B2, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BAY-876 DB16758
small molecule | CAS: 1799753-84-6

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bazedoxifene Approved DB06401
small molecule | CAS: 198481-32-2

Bazedoxifene is a third generation selective estrogen receptor modulator (SERM), developed by Pfizer following the completion of their takeover of Wyeth Pharmaceuticals. In late 2013, Pfizer received approval for bazedoxifene as part of the combination drug D…

Kategori:
Bone Density Conservation AgentsEstrogen Agonist/AntagonistEstrogen Receptor Modulators +8
Target Protein:
Estrogen receptorEstrogen receptor beta
Waktu Paruh~30 hours.
Vol. DistribusiFollowing intraveno…
KlirensThe apparent oral c…
Genetik -
BB-301 DB17011
biotech

BB-301 is a modified AAV serotype 9 (AAV9) capsid expressing a unique, single bifunctional construct promoting co-expression of both codon-optimized Poly-A Binding Protein Nuclear-1 (PABPN1) and two small inhibitory RNAs (siRNAs) against mutant PABPN1.[A26011…

Waktu Paruh-
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Bb-3497 DB04368
small molecule | CAS: 235784-88-0

Deskripsi belum tersedia.

Kategori:
AminesHydroxy AcidsHydroxylamines
Target Protein:
Peptide deformylasePeptide deformylasePeptide deformylase, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BBIBP-CorV DB15807
biotech

BBIBP-CorV vaccine contains a SARS-CoV-2 strain inactivated inside Vero Cells. Investigation shows this vaccine induces neutralizing antibodies in several mammalian species while also showing protective efficacy with SARS-CoV-2 challenge in rhesus macaques[A2…

Kategori:
Biological ProductsComplex MixturesVaccines +1
Waktu Paruh-
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BBP-671 DB18498
small molecule

BBP-671 is a small molecule activator of pantothenate kinases.

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BBP-812 DB16983
biotech

Deskripsi belum tersedia.

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BBT-877 DB18668
small molecule

BBT-877 is an autotaxin enzyme inhibitor being investigated for the treatment of fibrotic diseases, such as idiopathic pulmonary fibrosis.

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BC9KBY85WY DB17820
small molecule | CAS: 1259013-14-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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BCc1 DB16504
small molecule

BCc1 is a nanomedicine that demonstrated potent anticancer effects in both in vitro and in vivo studies.

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
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BCG vaccine Approved DB12768
biotech

BCG vaccine has been investigated for the treatment of Neoplasms, Bladder Cancer, Neoplasms by Site, Urologic Diseases, and Urologic Neoplasms, among others.

Kategori:
Adjuvants, ImmunologicAntineoplastic and Immunomodulating AgentsBacterial Vaccines +9
Waktu Paruh-
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BCX10013 DB18496
small molecule

BCX10013 is a small molecule inhibitor of human complement factor D.

Waktu Paruh-
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BCX9250 DB18069
small molecule

Deskripsi belum tersedia.

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BDB-001 DB16480
biotech

BDB-001, was under investigation in multiple clinical trials to evaluate its safety, tolerability, and efficacy across various conditions. In NCT05075304 and NCT04449588, BDB-001 was studied in mild to severe COVID-19 patients. It was also explored for solid …

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
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Bebtelovimab DB16755
biotech | CAS: 2578319-11-4

Bebtelovimab (LY-COV1404, LY-3853113) is a human monoclonal antibody approved for emergency use in the treatment of COVID-19. It binds to a portion of the SARS-CoV-2 spike (S) protein's receptor-binding domain, thereby preventing spike protein interaction wit…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesApproved Treatments for COVID-19 +6
Target Protein:
Spike glycoprotein
Waktu ParuhFollowing a single …
Vol. DistribusiAt steady-state, th…
KlirensFollowing a single …
Genetik -
Becaplermin Approved DB00102
biotech | CAS: 165101-51-9

Becaplermin is produced by recombinant DNA technology by insertion of the gene for the B chain of platelet derived growth factor (PDGF) into the yeast, Saccharomyces cerevisiae. Becaplermin has a molecular weight of approximately 25 KD and is a homodimer comp…

Kategori:
AcidsAcids, NoncarboxylicAlimentary Tract and Metabolism +24
Target Protein:
Platelet-derived growth factor receptor betaPlatelet-derived growth factor receptor alphaAlpha-2-macroglobulin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Becatecarin DB06362
small molecule | CAS: 119673-08-4

Becatecarin is a derivative of [rebeccamycin].

Kategori:
CarbohydratesGlycosidesHeterocyclic Compounds, Fused-Ring +1
Target Protein:
DNA topoisomerase 1DNA topoisomerase 2-alphaDNA topoisomerase 2-beta
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Beclamide DB09011
small molecule | CAS: 501-68-8

Beclamide (N-benzyl-B-chloropropionamide) is a no longer used drug that possesses anticonvulsant and sedative activity. It was studied in the 1950s for generalised tonic-clonic seizures but was not effective for absence seizures.

Kategori:
Acids, AcyclicAnticonvulsantsCentral Nervous System Depressants +4
Waktu Paruh-
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Beclanorsen DB05606
small molecule | CAS: 1072859-54-1

Deskripsi belum tersedia.

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Beclomethasone dipropionate Approved DB00394
small molecule | CAS: 5534-09-8

Beclomethasone dipropionate is a second-generation[A179842] synthetic corticosteroid and diester of beclomethasone, which is structurally similar to [dexamethasone].[L6871] It is a prodrug of an active metabolite beclomethasone 17-monopropionate (17-BMP)[A179…

Kategori:
Adrenal Cortex HormonesAdrenalsAgents to Treat Airway Disease +40
Target Protein:
Glucocorticoid receptor
Waktu ParuhFollowing intraveno…
Vol. DistribusiFollowing intraveno…
KlirensFollowing intraveno…
Genetik -
Becocalcidiol DB04891
small molecule | CAS: 524067-21-8

Becocalcidiol is a vitamin D(3) analogue which has not caused hypercalcaemia or significant irritation in preclinical trials.

Kategori:
CholestanesCholestenesFused-Ring Compounds +8
Target Protein:
Mediator of RNA polymerase II transcription subunit 1Vitamin D3 receptor
Waktu Paruh-
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Becotatug DB19069
biotech | CAS: 2648260-93-7

Becotatug is under investigation in clinical trial NCT06380348 (JMT101 in Combination With Osimertinib, Versus Cisplatin-pemetrexed in Participants With Locally Advanced or Metastatic Non-small Cell Lung Cancer (NSCLC) Characterized by Epithermal Growth Facto…

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Bectumomab DB04962
biotech | CAS: 158318-63-9

Bectumomab (marketed under the trade name LymphoScan®) is a mouse monoclonal antibody and which it's used to treat non-Hodgkin's lymphoma. It has a radioisotope, technetium (99m TC) which it's added.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bedaquiline Approved DB08903
small molecule | CAS: 843663-66-1

Bedaquiline is a bactericidal antimycobacterial drug belonging to the class of diarylquinoline. The quinolinic central heterocyclic nucleus with alcohol and amine side chains is responsible for bedaquiline-mediated antimycobacterial activity.[A261866] Althoug…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntiinfectives for Systemic Use +10
Target Protein:
ATP synthase subunit c
Waktu ParuhThe mean terminal e…
Vol. DistribusiThe volume of distr…
KlirensBedaquiline has a l…
Genetik -
Bee pollen DB16612
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Beef liver Approved DB14694
biotech

Beef liver allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
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Beeswax Approved DB11600
biotech | CAS: 8012-89-3

The wax obtained from the honeycomb of the bee. It consists primarily of myricyl palmitate, cerotic acid esters and some high-carbon paraffins. Beeswax is used as a stiffening agent in ointments and creams, and enables water to be incorporated to produce wate…

Kategori:
BeesLipids
Waktu Paruh-
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Beet Approved DB10640
biotech

Beet allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Befiradol DB19033
small molecule | CAS: 208110-64-9

Befiradol is under investigation in clinical trial NCT05148884 (Study to Assess the Safety, Tolerability and Preliminary Efficacy of NLX-112 Versus Placebo in L-dopa-induced Dyskinesia).

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsNeurotransmitter Agents +3
Target Protein:
5-hydroxytryptamine receptor 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Befotertinib DB18844
small molecule | CAS: 1835667-63-4

Befotertinib is under investigation in clinical trial NCT05007938 (Befotertinib and Icotinib in Treatment-naive Patients With Advanced Egfr-mutant Lung Cancer).

Waktu Paruh-
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Befovacimab DB16188
biotech | CAS: 2156634-62-5

Deskripsi belum tersedia.

Waktu Paruh-
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Begacestat DB12263
small molecule | CAS: 769169-27-9

Begacestat has been used in trials studying the treatment and basic science of Alzheimer Disease.

Kategori:
AmidesAmyloid Precursor Protein SecretasesEnzyme Inhibitors +3
Target Protein:
Gamma-secretase subunit APH-1BNicastrinGamma-secretase subunit APH-1A +2
Waktu Paruh-
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Begelomab DB13241
biotech | CAS: 1403744-56-8

Begelomab is a murine monoclonal antibody against CD26.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntineoplastic and Immunomodulating Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Bekanamycin DB13673
small molecule | CAS: 4696-76-8

Deskripsi belum tersedia.

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +9
Waktu Paruh-
Vol. Distribusi-
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Belantamab mafodotin Approved DB15719
biotech | CAS: 2050232-20-5

Belantamab mafodotin, or GSK2857916, is an afucosylated monoclonal antibody that targets B cell maturation antigen conjugated to the microtubule disrupter monomethyl auristatin-F (MMAF).[A216756] Belantamab mafodotin was granted FDA accelerated approval on…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +18
Target Protein:
Tumor necrosis factor receptor superfamily member 17
Waktu ParuhThe terminal half l…
Vol. DistribusiThe mean steady sta…
KlirensThe clearance of be…
Genetik -
Belatacept Approved DB06681
biotech | CAS: 706808-37-9

Belatacept is a soluble fusion protein, which links the extracellular domain of human cytotoxic T-lymphocyte-associated antigen 4 (CTLA-4) to the modified Fc (hinge, CH2, and CH3 domains) portion of human immunoglobulin G1 (IgG1). Structurally, abatacept is a…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntineoplastic Agents, Immunological +15
Target Protein:
T-lymphocyte activation antigen CD86T-lymphocyte activation antigen CD80
Waktu ParuhMean terminal elimi…
Vol. DistribusiVd, steady state, t…
KlirensIncreased body weig…
Genetik -
Belcesiran DB18226
biotech | CAS: 2375562-54-0

Deskripsi belum tersedia.

Waktu Paruh-
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Belimumab Approved DB08879
biotech | CAS: 356547-88-1

Belimumab is a fully human recombinant IgG1? monoclonal antibody that inhibits soluble human B lymphocyte stimulator protein (BLyS, also referred to as BAFF and TNFSF13B), a B cell survival factor.[L42630] BLyS levels are often elevated in immunodeficient and…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +13
Target Protein:
Tumor necrosis factor ligand superfamily member 13B
Waktu ParuhFollowing administr…
Vol. DistribusiFollowing administr…
KlirensFollowing administr…
Genetik -
Belinostat Approved DB05015
small molecule | CAS: 866323-14-0

Belinostat is a novel agent that inhibits the enzyme histone deacetylase (HDAC) with a sulfonamide-hydroxamide structure. It was developed as an orphan drug to target hematological malignancies and solid tumors by TopoTarget. The safety and efficacy of belino…

Kategori:
AmidesAminesAntineoplastic Agents +31
Target Protein:
Histone deacetylase
Gen Terkait:
UGT1A1 UGT1A1
Waktu ParuhDisplays a three-co…
Vol. DistribusiThe volume of distr…
Klirens1240 mL/min
Genetik 2 Varian
Beloranib DB12671
small molecule | CAS: 251111-30-5

Beloranib has been used in trials studying the treatment of Obesity, Over-weight, Type 2 Diabetes, Craniopharyngioma, and Hypothalamic Injury, among others.

Kategori:
Acids, CarbocyclicAngiogenesis InhibitorsAngiogenesis Modulating Agents +7
Target Protein:
Methionine aminopeptidase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Belotecan DB12459
small molecule | CAS: 256411-32-2

Belotecan has been investigated for the treatment of Epithelial Ovarian Cancer.

Kategori:
AlkaloidsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +4
Target Protein:
DNA topoisomerase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Belrestotug DB19066
biotech | CAS: 2574438-65-4

Belrestotug is under investigation in clinical trial NCT05565378 (A Platform Study of Novel Immunotherapy Combinations in Participants With Previously Untreated, Advanced/metastatic Non-small-cell Lung Cancer).

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Beludavimab DB18952
biotech | CAS: 2423016-74-2

Beludavimab is under investigation in clinical trial NCT04746183 (AGILE (Early Phase Platform Trial for COVID-19)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
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Genetik -
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