Hasil Filter

12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (12560)

Halaman 51 / 252
Arylacenamide DB05792
small molecule | CAS: 132173-07-0

Arylacenamide (SR31747) is a peripheral [sigma] ligand that binds four proteins in human cells, i.e. SRBP-1, [sigma]-2, HSI and its relative SRBP-2. It is a dual agent with both immunomodulatory and antiproliferative activities.

Kategori:
CycloparaffinsEnzyme InhibitorsImmunologic Factors +1
Target Protein:
3-beta-hydroxysteroid-Delta(8),Delta(7)-isomeraseHCG20471, isoform CRA_c
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arzoxifene Approved DB06249
small molecule | CAS: 182133-25-1

Deskripsi belum tersedia.

Kategori:
Sulfur Compounds
Target Protein:
Estrogen receptorEstrogen receptor beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AS-8112 DB09207
small molecule

AS-8112 is a synthetic compound that acts as a selective antagonist at the dopamine receptor subtypes D2 and D3, and the serotonin receptor 5-HT3. It has been shown to exert potent antiemetic effects in animal studies and has been investigated for potential m…

Kategori:
Dopamine AgentsDopamine AntagonistsDopamine D2 Receptor Antagonists +1
Target Protein:
D(2) dopamine receptorD(3) dopamine receptor5HT3 serotonin receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AS1409 DB05182
small molecule

AS1409 is a genetically engineered fusion protein made up of two distinct components. One is the cytokine IL12, which has anti-cancer activity. The other is an antibody that targets tumours. It is developed by Antisoma is in a phase I of clinical trial for th…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Asafoetida DB15928
biotech | CAS: 9000-04-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ASC-JM-17 DB16931
small molecule | CAS: 1039760-91-2

Deskripsi belum tersedia.

Kategori:
AlkanesBenzene DerivativesCatechols +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Asciminib Approved DB12597
small molecule | CAS: 1492952-76-7

Asciminib is a tyrosine kinase inhibitor (TKI) used in the treatment of chronic-phase Philadelphia chromosome-positive chronic myeloid leukemia (Ph+ CML). More specifically, it is an inhibitor of the ABL1 kinase activity of the BCR-ABL1 fusion protein[L38995]…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBcr-Abl Tyrosine Kinase Inhibitors +26
Target Protein:
Tyrosine-protein kinase ABL1
Waktu ParuhThe terminal elimin…
Vol. DistribusiAt steady-state, th…
KlirensThe total apparent …
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ascorbic acid Approved DB00126
small molecule | CAS: 50-81-7

A six carbon compound related to glucose. It is found naturally in citrus fruits and many vegetables. Ascorbic acid is an essential nutrient in human diets, and necessary to maintain connective tissue and bone. Its biologically active form, vitamin C, functio…

Kategori:
Acids, AcyclicAlimentary Tract and MetabolismAntioxidants +20
Target Protein:
Solute carrier family 23 member 2Solute carrier family 23 member 1Hyaluronate lyase +23
Waktu Paruh16 days (3.4 hours …
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 129499-78-1

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicCarbohydratesHydroxy Acids +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ascorbyl phosphate Approved DB11352
small molecule

Ascorbyl phosphate is a synthetic form of Vitamin C and is found in different salt forms such as magnesium ascorbyl phosphate and sodium ascorbyl phosphate. These salts are present in cosmetic products at concentrations ranging from 0.001 % to 3% [A27211]. As…

Kategori:
Acids, AcyclicCarbohydratesHydroxy Acids +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ascrinvacumab DB12261
biotech | CAS: 1463459-96-2

Ascrinvacumab has been used in trials studying the treatment and basic science of Neoplasms, Advanced Solid Tumors, Carcinoma, Hepatocellular, and Malignant Pleural Mesothelioma.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Asenapine Approved DB06216
small molecule | CAS: 65576-45-6

Developed by Schering-Plough after its merger with Organon International, asenapine is a sublingually administered, atypical antipsychotic for treatment of schizophrenia and acute mania associated with bipolar disorder. Asenapine also belongs to the dibenzo-o…

Kategori:
Acid ReducersAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +41
Target Protein:
5-hydroxytryptamine receptor 2AD(2) dopamine receptor5-hydroxytryptamine receptor 1A +17
Waktu Paruh24 hours (range of …
Vol. Distribusi20-25 L/kg
Klirens-
Genetik -
ASF-1075 DB05727
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Asfotase alfa Approved DB09105
biotech | CAS: 1174277-80-5

Asfotase alfa is a first-in-class bone-targeted enzyme replacement therapy designed to address the underlying cause of hypophosphatasia (HPP)—deficient alkaline phosphatase (ALP). Hypophosphatasia is almost always fatal when severe skeletal disease is obvious…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsAntibodies +16
Target Protein:
Pyrophosphate
Waktu ParuhApproximately 5 day…
Vol. Distribusi-
Klirens-
Genetik -
ASI402 DB06373
biotech | CAS: 372075-37-1

ASI402 is a monoclonal antibody that targets an aberrantly glycosylated antigen Mucin 1. It is being investigated in cancers.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Mucin-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Asiatic acid DB14054
small molecule | CAS: 464-92-6

From Centella asiatica and other plants; shows a variety of bioactivities.

Kategori:
TerpenesTriterpenes
Target Protein:
Glycogen phosphorylase, muscle form
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Asiaticoside DB14081
small molecule | CAS: 16830-15-2

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsTerpenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Asimadoline DB05104
small molecule | CAS: 153205-46-0

Asimadoline is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, Germany. Asimadoline was originally developed to treat peripheral pain such as arthritis. Asimadoline is an orally administered agent that acts as a kap…

Kategori:
AcetatesAcids, AcyclicAmides
Target Protein:
Kappa-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Asm-024 cation DB19385
small molecule | CAS: 1609534-88-4

Asm-024 cation is under investigation in clinical trial NCT01855230 (Safety, Tolerability, and Clinical Activity of ASM-024 Administered to Patients With GOLD 2 or GOLD 3 Chronic Obstructive Pulmonary Disease (COPD)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ASN120290 DB16988
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ASP-3026 DB12729
small molecule | CAS: 1097917-15-1

ASP3026 has been used in trials studying the treatment of Solid Tumor, B-Cell Lymphoma, Advanced Malignancies, Positive for Anaplastic Lymphoma Kinase, and Positive for Proto-Oncogene Tyrosine-Protein Kinase ROS.

Kategori:
Sulfur Compounds
Target Protein:
ALK tyrosine kinase receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ASP-4058 DB11819
small molecule | CAS: 952565-91-2

ASP4058 has been used in trials studying Food Effect of ASP4058 and Pharmacokinetics of ASP4058.

Kategori:
Heterocyclic Compounds, Fused-RingOxazoles
Target Protein:
Sphingosine 1-phosphate receptor 1Sphingosine 1-phosphate receptor 5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ASP-7317 DB18549
biotech

ASP-7317 consists of human embryonic stem cell-derived retinal pigment epithelium cells.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ASP-8731 DB17696
small molecule | CAS: 2488255-42-9

ASP-8731 is a novel BACH1 inhibitor that potentially induces fetal hemoglobin (HbF). Developed by Mitobridge, it is being investigated for the treatment of sickle cell disease.[L46093]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aspacytarabine DB17226
small molecule | CAS: 2098942-53-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1349719-22-7

Asparaginase _Erwinia chrysanthemi_ is an asparaginase-specific enzyme derived from _Erwinia_ _chrysanthemi_ used as an anticancer agent. It works by depleting the stores of an important amino acid called asparagine, which is involved in DNA synthesis and cel…

Kategori:
AmidohydrolasesAntineoplastic AgentsAsparaginase +7
Waktu ParuhThe apparent half-l…
Vol. DistribusiThe volume of distr…
KlirensThe geometric mean …
Genetik -
biotech | CAS: 9015-68-3

Asparaginase derived from _Escherichia coli_ (L-asparagine amidohydrolase, EC 3.5.1.1) is an enzyme responsible for the metabolism of L-asparagine, by catalyzing L-asparagine into L-aspartic acid and ammonia. It also facilitates the production of oxaloacetate…

Kategori:
AmidohydrolasesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +7
Target Protein:
L-asparagine
Waktu ParuhPlasma half life of…
Vol. DistribusiApparent volume of …
Klirens-
Genetik -
Asparagus Approved DB10503
biotech

Asparagus allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1Sugar phosphatase YbiVChemotaxis protein CheY
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aspartic acid Approved DB00128
small molecule | CAS: 56-84-8

One of the non-essential amino acids commonly occurring in the L-form. It is found in animals and plants, especially in sugar cane and sugar beets. It may be a neurotransmitter.

Kategori:
Amino AcidsAmino Acids, AcidicAmino Acids, Dicarboxylic +5
Target Protein:
Glutamate receptor ionotropic, NMDA 2AGlutamate receptor ionotropic, NMDA 2BGlutamate receptor ionotropic, NMDA 1 +18
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
(S)-2-haloacid dehalogenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Aspartate--tRNA(Asp) ligase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 110954-19-3

Aspartyl-alanyl-diketopiperazine is under investigation in clinical trial NCT03349645 (An Open Label Extension Study to Assess the Safety of Long-Term Treatment With Ampion for Severe OA of the Knee).

Kategori:
Amino Acids, Peptides, and ProteinsOligopeptidesPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aspergillus fumigatus Approved DB10425
biotech

Aspergillus fumigatus is a fungus which can provoke allergic reactions. Aspergillus fumigatus extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Fungal Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aspergillus terreus Approved DB10450
biotech

Aspergillus terreus is a fungus which can provoke allergic reactions. Aspergillus terreus extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aspoxicillin DB13816
small molecule | CAS: 63358-49-6

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAntibacterials for Systemic Use +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Astaxanthin DB06543
small molecule | CAS: 472-61-7

Astaxanthin is a keto-carotenoid in the terpenes class of chemical compounds. It is classified as a xanthophyll but it is a carotenoid with no vitamin A activity. It is found in the majority of aquatic organisms with red pigment. Astaxanthin has shown to medi…

Kategori:
AlkenesAnticoagulantsBiological Factors +9
Target Protein:
NF-kappa-B inhibitor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Astegolimab DB16386
biotech | CAS: 2173054-79-8

Astegolimab is under investigation in clinical trial NCT04386616 (A Study to Evaluate the Safety and Efficacy of MSTT1041A (Astegolimab) or UTTR1147A in Patients With Severe COVID-19 Pneumonia).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAnti-Inflammatory Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Astodrimer DB11854
biotech | CAS: 1379746-42-5

Astodrimer has been used in trials studying the treatment and prevention of Bacterial Vaginosis. It is a lysine-based dendrimer with naphthalene disulfonic acid surface groups.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +10
Target Protein:
Envelope glycoprotein gp160
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AstraZeneca COVID-19 Vaccine Approved DB15656
biotech | CAS: 2420395-83-9

The AstraZeneca COVID-19 Vaccine (previously known as ChAdOx1 nCoV-19 or AZD1222) is one of several vaccines developed in 2020 for the prevention of COVID-19 caused by SARS-CoV-2.[L12669,L32649] The ChAdOx1 viral vector was developed at the University of Oxfo…

Kategori:
Biological ProductsComplex MixturesCOVID-19 Vaccines +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ASTX-029 DB18900
small molecule | CAS: 2095719-92-7

ASTX-029 is under investigation in clinical trial NCT03520075 (Study of ASTX029 in Subjects With Advanced Solid Tumors).

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Asunaprevir Approved DB11586
small molecule | CAS: 630420-16-5

Asunaprevir, also named BMS-650032, is a potent hepatitis C virus (HCV) NS3 protease inhibitor. It has been shown to have a very high efficacy in dual-combination regimens with daclatasvir in patients chronically infected with HCV genotype 1b.[A32528] It was …

Kategori:
AmidesAntiinfectives for Systemic UseAntiviral Agents +35
Target Protein:
Gag-Pol polyproteinGenome polyprotein
Waktu ParuhClinical pharmacoki…
Vol. DistribusiThe registered volu…
KlirensClinical pharmacoki…
Genetik -
Asundexian DB19088
small molecule | CAS: 2064121-65-7

Asundexian is under investigation in clinical trial NCT05686070 (A Study to Test Asundexian for Preventing a Stroke Caused by a Clot in Participants After an Acute Ischemic Stroke or After a High-risk Transient Ischemic Attack, a So-called Mini Stroke).

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +2
Target Protein:
Coagulation factor XI
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Asunercept DB15160
biotech | CAS: 1450882-18-4

Asunercept is under investigation in clinical trial NCT02853565 (A Study of CAN008 for Newly Diagnosed Glioblastoma Multiforme).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Asvasiran DB05638
biotech | CAS: 870094-26-1

Asvasiran is an siRNA that targets the respiratory syncytial virus (RSV) N gene and inhibits viral replication. It has the potential to treat or prevent RSV infection.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AT-001 DB15121
small molecule | CAS: 1355612-71-3

AT-001 is under investigation in clinical trial NCT03062384 (AT-001 for Long-term Preservation of Brain Health in Aging).

Kategori:
Heterocyclic Compounds, Fused-RingPyridinesThiazoles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AT-301 DB16507
biotech

AT-301 was under investigation in clinical trial NCT01675284 to evaluate the safety, reactogenicity, and humoral immune responses to an inactivated H5N1 influenza vaccine

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AT-527 DB16451
small molecule | CAS: 2241337-84-6

Deskripsi belum tersedia.

Kategori:
AcidsAcids, NoncarboxylicExperimental Unapproved Treatments for COVID-19 +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 2501–2550 dari 12560
Sebelumnya Halaman 51 / 252 Berikutnya