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14494

Total database: 17430
Struktur (SMILES)
9687 (66.8%)
Target
7525 (51.9%)
Genomik
112 (0.8%)
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14494 (100.0%)

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Hasil Pencarian (14494)

Halaman 50 / 290
biotech | CAS: 139076-62-3

Human recombinant antihemophilic factor (AHF) or Factor VIII, 2332 residues, glycosylated, produced by CHO cells

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +12
Target Protein:
Coagulation factor XCoagulation factor IXvon Willebrand factor +8
Waktu Paruh8.4-19.3 hrs
Vol. Distribusi-
Klirens* 4.1 mL/h•kg [Prev…
Genetik -
biotech

Equine anti-thymocyte globulin is composed of purified gamma globulin containing primarily IgG against human thymus lymphocytes. It is formed by inoculating a horse with an antigen (human thymoyctes) which then induces the horse immune system's B-lymphocytes …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibody-Surface Protein Interactions +22
Waktu ParuhThe half-life of eq…
Vol. DistribusiDuring infusion of …
Klirens-
Genetik -
Antimonous acid DB02453
small molecule

Deskripsi belum tersedia.

Target Protein:
Arsenical pump-driving ATPase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Antimony DB13110
small molecule | CAS: 7440-36-0

Antimony has been used in trials studying the treatment of Cutaneous Leishmaniasis.

Kategori:
ElementsMetalloidsMetals +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 28300-74-5

Antimony potassium tartrate is a schistosomicide possibly useful against other parasites. It has irritant emetic properties and may cause lethal cardiac toxicity among other adverse effects.

Kategori:
AnthelminticsAnti-Infective AgentsAntiparasitic Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 91531-30-5

Antineoplaston A10 has been used in trials studying the treatment of Sarcoma, Lymphoma, Lung Cancer, Liver Cancer, and Kidney Cancer, among others.

Kategori:
AcetamidesAmidesBenzene Derivatives +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Antipain DB15251
small molecule | CAS: 37691-11-5

Antipain is a serine/cysteine protease inhibitor originally isolated from various strains of actinomycetes.[A214481] Early studies investigated the potential for antipain to alter DNA damage and chromosomal aberrations in irradiated cells or those treated wit…

Kategori:
Amino Acids, Peptides, and ProteinsEnzyme InhibitorsOligopeptides +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Antipyrine Approved DB01435
small molecule | CAS: 60-80-0

An analgesic and antipyretic that has been given by mouth and as ear drops. Antipyrine is often used in testing the effects of other drugs or diseases on drug-metabolizing enzymes in the liver. (From Martindale, The Extra Pharmacopoeia, 30th ed, p29)

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +30
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Antithrombin Alfa Approved DB11166
biotech | CAS: 84720-88-7

Antithrombin Alfa is a recombinant antithrombin , an anticoagulant, that is used for the prevention of thromboembolic events in patients that have hereditary deficiency of antithrombin in high risk situations.

Kategori:
AnticoagulantsDecreased Coagulation Factor ActivityFactor Xa Inhibitors +2
Target Protein:
ProthrombinCoagulation factor X
Waktu ParuhDose of: 50IU/kg: …
Vol. DistribusiDose of: 50IU/kg: …
KlirensDose of: 50IU/kg: …
Genetik -
biotech | CAS: 1311281-25-0

Antithrombin gamma is under investigation in clinical trial NCT04182373 (KW-3357 Study in Patients With Early Onset Severe Preeclampsia).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Antithrombin III human Approved DB11598
biotech | CAS: 9000-94-6

A plasma alpha 2 glycoprotein that accounts for the major antithrombin activity of normal plasma and also inhibits several other enzymes. It is a member of the serpin superfamily.

Kategori:
Alpha-GlobulinsAmino Acids, Peptides, and ProteinsAnticoagulants +18
Target Protein:
Antithrombin-III
Waktu Paruh2.5 - 3.8 hs
Vol. DistribusiDistributed into pl…
Klirens-
Genetik -
biotech | CAS: 308067-60-9

Rabbit anti-thymocyte globulin. Thymoglobulin is a polyclonal antibody that suppresses certain types of immune cells responsible for acute organ rejection in transplant patients. Thymoglobulin is a mixture of antibodies intended to bind to various cell surfac…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibody-Surface Protein Interactions +22
Target Protein:
Major histocompatibility complex class I-related gene proteinIntegrin alpha-LT-lymphocyte activation antigen CD86 +6
Waktu Paruh2-3 days, may incre…
Vol. Distribusi-
Klirens-
Genetik -
Antrafenine Approved DB01419
small molecule | CAS: 55300-29-3

Antrafenine is a piperazine derivative drug that acts as an analgesic and anti-inflammatory drug with similar efficacy to naproxen. It is not widely used as it has largely been replaced by newer drugs.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnti-Inflammatory Agents +4
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Antroquinonol DB12326
small molecule | CAS: 1010081-09-0

Antroquinonol has been used in trials studying the treatment of Hyperlipidemias, Non-small Cell Lung Cancer, and Non-small Cell Lung Cancer Stage IV.

Kategori:
BenzoquinonesCoenzymesEnzymes and Coenzymes +1
Target Protein:
DNA (cytosine-5)-methyltransferase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2636710-07-9

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ANX-005 DB16977
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ANX-510 DB05308
small molecule

ANX-510 (CoFactor) is a folate-based biomodulator drug being developed to enhance the activity and reduce associated toxicity of the widely used cancer chemotherapy, 5-fluorouracil (5-FU). CoFactor use with 5-FU is being evaluated in clinical trials in first …

Target Protein:
Thymidylate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anzurstobart DB17547
biotech | CAS: 2543693-10-1

Anzurstobart is a monoclonal antibody directed against signal-regulatory protein alpha (SIRP?) on monocytes and macrophages to potently block the CD47-SIRP? interaction. It is being investigated for cancers.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AOC 1001 DB18620
biotech | CAS: 2653183-66-3

Delpacibart (AOC 1001) is being investigated in a global study for the treatment of Myotonic Dystrophy type 1 (DM1) in clinical trial NCT06411288

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AOC-1020 DB18621
biotech

AOC-1020 is an antibody oligonucleotide conjugate, comprised of a human transferrin receptor 1 targeting, effector function null, humanized IgG1 antibody, a MCC maleimide linker, and a double-stranded siRNA oligonucleotide targeting DUX4.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AOD9604 DB06388
small molecule | CAS: 221231-10-3

AOD9604 is a synthetic analogue of the lipolytic domain of human growth hormone, being investigated for the treatment of obesity.

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AP-001 DB18511
small molecule | CAS: 660430-03-5

Deskripsi belum tersedia.

Kategori:
Dietary FatsDietary Fats, UnsaturatedFats +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AP-101 DB17947
biotech

AP-101 is a recombinant human antibody directed against human misfolded superoxide dismutase 1.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AP-102 DB18206
small molecule | CAS: 846569-60-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AP103 DB18234
biotech

AP103 is a non-viral gene therapy that uses a delivery vector, HPAE (Highly Branched Poly ?-Amino Ester), to deliver the correct collagen VII gene into skin cells.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AP1081 DB05233
small molecule

A transdermal gel containing ethinyl estradiol and norelgestromin being investigated by Antares Pharma for use as a female contraceptive.

Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AP5280 DB05112
small molecule

AP5280 is a novel N-(2-hydroxypropyl)methacrylamide (HPMA) copolymer-bound platinum (Pt) therapeutic designed to increase the therapeutic index relative to conventional, small-molecule platinum agents.

Kategori:
Acids, AcyclicAcrylatesAmides +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AP5346 DB04992
small molecule

AP5346 is designed to target a diaminocyclohexane platinum (Pt) moiety to tumors through pH-sensitive linkage to a 25 kDa hydroxypropylmethacrylamide polymer. It is being pursued by Access Pharmaceuticals, Inc.

Kategori:
Organometallic Compounds
Target Protein:
DNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apabetalone DB12000
small molecule | CAS: 1044870-39-4

Apabetalone has been investigated for the treatment of Diabetes, Atherosclerosis, and Coronary Artery Disease.

Kategori:
Heterocyclic Compounds, Fused-RingQuinazolines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apadamtase alfa Approved DB15164
biotech | CAS: 2086325-24-6

Thrombotic thrombocytopenic purpura (TTP) is a rare blood clotting disorder characterized by thrombocytopenia, microangiopathic hemolytic anemia, and various degrees of organ damage.[A262076] It may be inherited (congenital TTP; cTTP) or acquired due to autoa…

Kategori:
ADAM ProteinsADAMTS ProteinsAmino Acids, Peptides, and Proteins +12
Target Protein:
von Willebrand factor
Waktu ParuhFollowing the intra…
Vol. Distribusi-
Klirens-
Genetik -
Apadenoson DB05009
small molecule | CAS: 250386-15-3

Apadenoson is a selective A2a adenosine receptor agonist designed for use as a pharmacologic stress agent in cardiac perfusion imaging studies. It is developed by Bristol-Myers Squibb and is in phase II of clinical trials.

Kategori:
Acids, CarbocyclicAdenosine A receptor agonistsAdenosine A2 Receptor Agonists +7
Target Protein:
Adenosine receptor A2a
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apalutamide Approved DB11901
small molecule | CAS: 956104-40-8

Apalutamide is a potent androgen receptor (AR) antagonist that selectively binds to the ligand-binding domain of AR and blocks AR nuclear translocation or binding to androgen response elements [A31846]. It has been used in trials studying the treatment of Pro…

Kategori:
Androgen Receptor InhibitorsAntiandrogensAntineoplastic Agents +28
Target Protein:
Androgen receptorGABA(A) Receptor
Waktu ParuhThe mean effective …
Vol. DistribusiThe mean apparent v…
KlirensThe CL/F of apaluta…
Genetik -
biotech | CAS: 2097132-02-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apararenone DB15024
small molecule | CAS: 945966-46-1

Apararenone is under investigation in clinical trial NCT02531568 (Drug Interaction Study of Warfarin and MT-3995).

Kategori:
AmidesSulfonesSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apatorsen DB06094
biotech | CAS: 1002331-21-6

Apatorsen is a second generation antisense drug which in preclinical experiments, inhibits production of Heat Shock Protein 27 (Hsp27) a cell survival protein found at elevated levels in many human cancers including prostate, lung, breast, ovarian, bladder, r…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Target Protein:
Heat shock protein beta-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apaziquone DB12593
small molecule | CAS: 114560-48-4

Apaziquone has been investigated for the treatment of Bladder Cancer and Bladder Neoplasms.

Kategori:
Antineoplastic AgentsAzirinesHeterocyclic Compounds, Fused-Ring +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apc001 DB17819
biotech

Apc001 is an aptamer developed for the treatment of osteogenesis imperfecta.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apc001PE DB17902
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
APC8020 DB17228
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
APD-209 DB18759
small molecule | CAS: 1261156-82-4

Deskripsi belum tersedia.

Target Protein:
Beta-2 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
APD668 DB05166
small molecule

APD668 is a novel, highly potent and orally active glucose-dependent insulinotropic receptor (GDIR) agonist intended to more efficiently stimulate insulin release by beta cells in response to elevated blood glucose levels, and to also avoid hypoglycemia.

Target Protein:
Glucose-dependent insulinotropic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
APD791 DB05227
small molecule

APD791 is an oral anti-thrombotic drug candidate being evaluated in a Phase 1 clinical trial by Arena. APD791 is intended to lower the risk of arterial thrombosis by reducing the amplification of platelet aggregation, arterial constriction and intimal hyperpl…

Kategori:
Acids, CarbocyclicAmidesAntidepressive Agents +8
Target Protein:
5-hydroxytryptamine receptor 2A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apelin DB18909
biotech | CAS: 372170-33-7

Apelin is under investigation in clinical trial NCT03449251 (A Series of Pilot Studies to Evaluate the Haemodynamic and Metabolic Effects of Apelin and Relaxin).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsIntercellular Signaling Peptides and Proteins +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
APG-1387 DB16095
small molecule | CAS: 1570231-89-8

APG-1387 is under investigation in clinical trial NCT04568265 (A Clinical Study of APG-1387 in Combination With Entecavir in Patients With Chronic Hepatitis B).

Kategori:
AmidesSulfonesSulfur Compounds
Target Protein:
E3 ubiquitin-protein ligase XIAPBaculoviral IAP repeat-containing protein 2Baculoviral IAP repeat-containing protein 3 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
APG-157 DB18683
small molecule

APG-157 consists of zinflavonoids being investigated for the treatment of cancers.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aphidicolin DB17742
small molecule | CAS: 38966-21-1

Aphidicolin is an antimitotic and antiviral metabolite of the mould _Cephalosporium aphidicola_. It inhibits DNA polymerase alpha and blocks DNA replication.[A259157, A259162]

Kategori:
Anti-Infective AgentsAntiviral AgentsDiterpenes +2
Target Protein:
DNA polymerase catalytic subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apinocaltamide DB16241
small molecule | CAS: 1838651-58-3

Apinocaltamide is under investigation in clinical trial NCT03239691 (A Study to Evaluate the Effect of ACT-709478 in Photosensitive Epilepsy Patients).

Kategori:
AcetatesAcids, AcyclicAmides +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apiospora montagnei Approved DB10844
biotech

Apiospora montagnei is a fungus which can provoke allergic reactions. Apiospora montagnei extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Fungal Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apis mellifera venom Approved DB10955
biotech

Apis mellifera venom is an extract of Apis mellifera venom. Apis mellifera venom is used in allergenic testing.

Kategori:
Allergenic ExtractsBee and Wasp VenomCell-mediated Immunity +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apitegromab DB16096
biotech | CAS: 2278276-46-1

Apitegromab is under investigation in clinical trial NCT03921528 (An Active Treatment Study of SRK-015 in Patients With Type 2 or Type 3 Spinal Muscular Atrophy).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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