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11778

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8554 (72.6%)
Target
6383 (54.2%)
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96 (0.8%)
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11778 (100.0%)

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Halaman 50 / 236
AVI-014 DB17086
biotech

AVI-014 is a glycosylated, recombinant human granulocyte colony-stimulating factor (G-CSF).

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AVI-4020 DB05873
small molecule

AVI-4020 is a neugene antisense drug candidate for the treatment of patients with acute West Nile virus disease who have serious neurological impairment (WNV neuroinvasive disease).

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AVI-4065 DB05620
small molecule

AVI-4065, a phosphorodiamidate Morpholino oligomer (PMO), is an investigational antisense HCV drug. It was developed by Sarepta Therapeutics, Inc. After phase II trials it was cancelled due to lack of potency. [L2917]

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AVI-4557 DB05447
small molecule

AVI-4557 is an oral antisense compound that selectively inhibits the metabolic enzyme cytochrome P450 3A4 (CYP), a liver enzyme responsible for the metabolism or breakdown of approximately half of currently marketed drugs. Studies indicate that AVI-4557 can s…

Target Protein:
Hepatocyte nuclear factor 4-alpha
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AVI-5126 DB05726
small molecule

AVI-526 is an improved formulation of [AVI-4557], developed for use on Vein Grafts before use in Heart by-Pass Graft Surgery. AVI-526 works by silencing a gene known as c-myc, a key regulatory gene involved in cardiovascular restenosis. The drug was under inv…

Kategori:
MorpholinesNucleic Acids, Nucleotides, and NucleosidesNucleotides +3
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AVI-7287 DB17799
biotech

Deskripsi belum tersedia.

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AVI-7288 DB17800
biotech

Deskripsi belum tersedia.

Kategori:
MorpholinesNucleic Acids, Nucleotides, and NucleosidesNucleotides +3
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AVI-7537 DB15433
biotech

AVI-7537 is an antisense molecule that binds to the Ebola virus mRNA to prevent the viral replication.[L46207] AVI-7537 is under investigation in clinical trial NCT01593072 (A Study to Assess the Safety, Tolerability and Pharmacokinetics of AVI-7537 in Health…

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Avicin D DB17240
small molecule | CAS: 197787-20-5

Deskripsi belum tersedia.

Kategori:
CarbohydratesGlycosides
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Avidin DB15228
biotech | CAS: 110539-97-4

Avidin is under investigation in clinical trial NCT00345618 (Clinical Study Assessing Idrabiotaparinux Sodium Injections Once-weekly in Pulmonary Embolism Therapeutic Approach).

Kategori:
AlbuminsAmino Acids, Peptides, and ProteinsAnimal Proteins, Dietary +10
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Avilamycin DB11375
small molecule | CAS: 11051-71-1

Deskripsi belum tersedia.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsCarbohydrates +2
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Aviptadil DB06260
small molecule | CAS: 40077-57-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsErectile DysfunctionGastrointestinal Hormones +9
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Aviscumine DB12684
biotech | CAS: 223577-45-5

Cy 503 is under investigation in clinical trial NCT00658437 (Aviscumine for the Treatment of Malignant Melanoma Stage IV After Failure of Prior Therapy).

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsBiological Factors +12
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Avizakimab DB18842
biotech | CAS: 2229685-51-0

Avizakimab is under investigation in clinical trial NCT03371251 (Study of BOS161721 in Systemic Lupus Erythematosus (SLE) Patients on a Background of Limited Standard of Care).

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AVL-3288 DB18707
small molecule | CAS: 917837-54-8

Deskripsi belum tersedia.

Target Protein:
Neuronal acetylcholine receptor subunit alpha-7
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Avobenzone Approved DB09495
small molecule | CAS: 70356-09-1

Avobenzone is dibenzoyl methane derivative. It is oil soluble ingredient. Avobenzone has the ability to absorb ultraviolet light over wider range of wavelengths. It is included in many commercially available sunscreens which are used as wide spectrum sunscree…

Kategori:
Compounds used in a research, industrial, or household settingCosmeticsDermatologicals +4
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Avoplacel DB18659
biotech

Avoplacel (PLX-R18) is an allogeneic cell therapy under investigation for the treatment of acute radiation syndrome.[L48370]

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Avoralstat DB12120
small molecule | CAS: 918407-35-9

Avoralstat has been used in trials studying the prevention of HAE and Hereditary Angioedema.

Kategori:
Acids, CarbocyclicAlkenesAmides +6
Target Protein:
Kallikrein-2Kininogen-1
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Avotaciclib DB16652
small molecule | CAS: 1983983-41-0

Avotaciclib is under investigation in clinical trial NCT03579836 (Evaluation of Safety and Efficacy in BEY1107 in Monotherapy Gemcitabine Combination in Patient With Pancreatic Cancer).

Target Protein:
Cyclin-dependent kinase 1
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AVP-21D9 DB17798
biotech

AVP-21D9 is a fully human anthrax monoclonal antibody that is being investigated as an anthrax antitoxin.[A259522]

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
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AVR-RD-01 DB17651
biotech

AVR-RD-01 is an investigational _ex vivo_ lentiviral gene therapy developed by AVROBIO Inc. It consists of autologous CD34+ cells that transduced with Lentiviral Vector/alpha-galactosidase A (AGA) encoding for the human AGA complementary deoxyribonucleic acid…

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AVR-RD-02 DB17650
biotech

AVR-RD-02 is an investigational _ex vivo_ lentiviral gene therapy developed by AVROBIO Inc. It consists of autologous CD34+ enriched hematopoietic stem cells (HSCs) that have been genetically modified _ex vivo_ with a lentiviral vector (LV) to contain a ribon…

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AVR118 DB04979
biotech

AVR118 represents a new type of biopolymer chemistry that also possesses novel immunomodulator activity. This non-toxic peptide-nucleic acid, which to date has shown no indication of human toxicity, appears to stimulate the proinflammatory responses required …

Kategori:
HIVNucleic Acids, Nucleotides, and NucleosidesNucleotides +2
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AVS-100 DB18068
small molecule | CAS: 2245942-72-5

Deskripsi belum tersedia.

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Avutometinib DB15254
small molecule | CAS: 946128-88-7

Avutometinib (RO-5126766 free base) is under investigation in clinical trial NCT03875820 (Phase I Trial of VS-6063 and RO5126766.).

Kategori:
BenzopyransHeterocyclic Compounds, Fused-RingProtein Kinase Inhibitors +1
Target Protein:
Serine/threonine-protein kinase A-RafSerine/threonine-protein kinase B-rafRAF proto-oncogene serine/threonine-protein kinase
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AVX-470 DB18455
biotech

AVX-470 is an anti-tumor necrosis factor (TNF) polyclonal antibody (bovine).

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsGlobulins +4
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AVXS-201 DB16997
biotech

Deskripsi belum tersedia.

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AVXS-301 DB17943
biotech

AVXS-301 consists of an adeno-associated virus serotype 9 (AAV9) designed to express the superoxide dismutase 1 (SOD1) gene. It is being investigated for the treatment of Amyotrophic Lateral Sclerosis (ALS).[L47077]

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biotech

Axalimogene filolisbac is under investigation in clinical trial NCT02853604 (Study of ADXS11-001 in Subjects With High Risk Locally Advanced Cervical Cancer).

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Axelopran DB12013
small molecule | CAS: 949904-48-7

Axelopran has been used in trials studying the treatment of OIC and Opioid-induced Constipation.

Kategori:
Acids, CarbocyclicAlkaloidsAmides +5
Target Protein:
Mu-type opioid receptor
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Axicabtagene ciloleucel Approved DB13915
biotech

Axicabtagene ciloleucel is an anti-CD19 chimeric antigen receptor (CAR) T-cell therapy. The drug has a unique mechanism of action, as it utilizes the patient's own T cells, which play a central role in immune response to cancer.[A216163] Once T-cells are coll…

Kategori:
AntigensAntigens, CDAntigens, Differentiation +16
Target Protein:
B-lymphocyte antigen CD19
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Axitinib Approved DB06626
small molecule | CAS: 319460-85-0

Axitinib is a second generation tyrosine kinase inhibitor that works by selectively inhibiting vascular endothelial growth factor receptors (VEGFR-1, VEGFR-2, VEGFR-3).[L6676] Through this mechanism of action, axitinib blocks angiogenesis, tumour growth and m…

Kategori:
Acids, CarbocyclicAmidesAntineoplastic Agents +31
Target Protein:
Tyrosine-protein kinase ABL1Vascular endothelial growth factor receptor 1Vascular endothelial growth factor receptor 2 +1
Waktu ParuhAxitinib has a half…
Vol. DistribusiThe volume of distr…
KlirensThe average clearan…
Genetik -
Axomadol DB16100
small molecule | CAS: 187219-99-4

Axomadol is under investigation in clinical trial NCT01043263 (Efficacy and Safety of EN3324 (Axomadol) in Subjects With Chronic Low Back Pain).

Kategori:
AlcoholsCyclohexanesCycloparaffins +3
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Azacitidine Approved DB00928
small molecule | CAS: 320-67-2

Azacitidine is a pyrimidine nucleoside analogue with anti-neoplastic activity. It differs from cytosine by the presence of nitrogen in the C5-position, key in its hypomethylating activity.[A1406,A1413,A1415] Two main mechanisms of action have been proposed fo…

Kategori:
AntimetabolitesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +17
Target Protein:
DNA (cytosine-5)-methyltransferase 1RNADNA
Waktu ParuhThe mean half-life …
Vol. DistribusiIn patients given a…
KlirensAzacitidine has an …
Genetik -
Azadirachtin DB19419
small molecule | CAS: 11141-17-6

Azadirachtin is under investigation in clinical trial NCT06617026 (Short-term Outcome of Medical vs. Surgical Management of Chronic Anal Fissure).

Kategori:
AgrochemicalsAzadirachtaCompounds used in a research, industrial, or household setting +5
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Azafenidin DB19031
small molecule | CAS: 68049-83-2

Azafenidin is under investigation in clinical trial NCT01726582 (Pancreas Cancer: Molecular Profiling as a Guide to Therapy Before and After Surgery ("Personalized Medicine")).

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Azanidazole DB13350
small molecule | CAS: 62973-76-6

Deskripsi belum tersedia.

Kategori:
Antiparasitic Products, Insecticides and RepellentsAntiprotozoalsGenito Urinary System and Sex Hormones +5
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Azapentacene DB15951
small molecule | CAS: 3863-80-7

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
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Azaperone DB11376
small molecule | CAS: 1649-18-9

Azaperone is a pyridinylpiperazine and butyrophenone agent that is capable of eliciting neuroleptic sedative and antiemetic effects. It is subsequently employed predominantly as a veterinary tranquilizer and mainly for pigs and elephants. At the same time, th…

Kategori:
Antipsychotic AgentsAntipsychotic Agents (First Generation [Typical])Butyrophenones +11
Target Protein:
D(3) dopamine receptorD(2) dopamine receptor
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Azapetine DB13727
small molecule | CAS: 146-36-1

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingPeripheral Vasodilators
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Azapropazone DB07402
small molecule | CAS: 13539-59-8

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +13
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Azasetron DB16837
small molecule | CAS: 123040-69-7

Deskripsi belum tersedia.

Kategori:
Antidepressive AgentsAntiemeticsAutonomic Agents +7
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Azatadine Approved DB00719
small molecule | CAS: 3964-81-6

Antihistamines such as azatadine appear to compete with histamine for histamine H1- receptor sites on effector cells. The antihistamines antagonize those pharmacological effects of histamine which are mediated through activation of H1- receptor sites and ther…

Kategori:
Agents that reduce seizure thresholdAnticholinergic AgentsAntihistamines for Systemic Use +10
Target Protein:
Histamine H1 receptor
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Azathioprine Approved DB00993
small molecule | CAS: 446-86-6

Azathioprine is a prodrug of 6-mercaptopurine, first synthesized in 1956 by Gertrude Elion, William Lange, and George Hitchings in an attempt to produce a derivative of 6-mercaptopurine with a better therapeutic index.[A189678,A189687,A189690] Azathioprine is…

Kategori:
AntimetabolitesAntineoplastic and Immunomodulating AgentsAntirheumatic Agents +21
Target Protein:
AmidophosphoribosyltransferaseRas-related C3 botulinum toxin substrate 1
Gen Terkait:
TPMT TPMT TPMT
Waktu ParuhThe half life of az…
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik 3 Varian
AZD-1305 DB11766
small molecule | CAS: 872045-91-5

AZD1305 has been used in trials studying the treatment and basic science of Atrial Flutter, Atrial Fibrillation, and Left Ventricle Function.

Kategori:
Acids, AcyclicAza Compounds
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AZD-1386 DB15333
small molecule | CAS: 942937-80-6

AZD-1386 is under investigation in clinical trial NCT00945178 (Double-blind Placebo-controlled 2-part Study Assessing the Safety, Tolerability and PK of AZD1386 in Healthy Volunteers).

Kategori:
Heterocyclic Compounds, Fused-Ring
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AZD-1656 DB14810
small molecule | CAS: 919783-22-5

AZD-1656 is under investigation in clinical trial NCT00747175 (A Study to Evaluate Safety, Tolerability and P-Glucose After Multiple Ascending Oral Doses of AZD1656 in Type 2 Diabetes).

Kategori:
AzetinesGlucokinase
Target Protein:
Hexokinase-4
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AZD-1940 DB17077
small molecule | CAS: 881413-29-2

Deskripsi belum tersedia.

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AZD-3043 DB12576
small molecule | CAS: 579494-66-9

AZD3043 has been used in trials studying the treatment and basic science of Safety, Sedation, Tolerability, and Pharmacokinetics.

Kategori:
Acids, CarbocyclicCentral Nervous System DepressantsHypnotics and Sedatives
Target Protein:
Gamma-aminobutyric acid receptor subunit gamma-3
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AZD-3759 DB14795
small molecule | CAS: 1626387-80-1

AZD-3759 is under investigation in clinical trial NCT03360929 (Evaluate Safety, Tolerability, Pharmacokinetics and Anti-tumor Activity of AZD3759).

Kategori:
Heterocyclic Compounds, Fused-Ring
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