Hasil Filter

12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (12560)

Halaman 50 / 252
small molecule | CAS: 506-32-1

An unsaturated, essential fatty acid. It is found in animal and human fat as well as in the liver, brain, and glandular organs, and is a constituent of animal phosphatides. It is formed by the synthesis from dietary linoleic acid and is a precursor in the bio…

Kategori:
Arachidonic AcidsCytochrome P-450 CYP2C9 SubstratesCytochrome P-450 Substrates +5
Target Protein:
Prostaglandin G/H synthase 1Peroxisome proliferator-activated receptor alphaBile acid receptor +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 149301-79-1

Specific inhibitor of phospholipase A2.[A252972]

Kategori:
EicosanoidsEnzyme InhibitorsFatty Acids +3
Target Protein:
Cytosolic phospholipase A2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 7075-11-8

Deskripsi belum tersedia.

Target Protein:
Cytidylate kinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aramchol DB11860
small molecule | CAS: 246529-22-6

Aramchol has been used in trials studying the treatment of HIV, Gallstones, Fatty Liver, Metabolic Syndrome, and Nonalcoholic Steatohepatitis, among others.

Kategori:
Bile Acids and SaltsCholanesFused-Ring Compounds +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aranidipine DB09229
small molecule | CAS: 86780-90-7

Aranidipine is a novel dihydropyridine derivative that gives rise to two active metabolites (M-1? and M-1?) that exhibit hypotensive activity. It is a calcium antagonist with the formula methyl 2-oxopropyl 1,4-dihydro-2,6-dimethyl-4-(2-nitrophenyl)-3,5-pyridi…

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsBradycardia-Causing Agents +8
Target Protein:
Voltage-dependent L-type calcium channel subunit alpha-1CVoltage-dependent L-type calcium channel subunit alpha-1DVoltage-dependent L-type calcium channel subunit alpha-1F +3
Waktu ParuhThe elimination hal…
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 583057-48-1

Arasertaconazole is under investigation in clinical trial NCT01144286 (Arasertaconazole Nitrate Pessaries - Dose Finding Study for the Vulvovaginal Candidiasis (VVC) Treatment).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arazasetron DB19237
small molecule | CAS: 2025360-90-9

Arazasetron is currently under investigation in clinical trial NCT05258773 (Evaluation of the Presence of SENS-401 in the Perilymph).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 847353-30-4

Arbaclofen Placerbil is a prodrug of Arbaclofen, which is a selective gamma-amino-butyric acid type B receptor agonist and the R-enantiomer of baclofen. It was discovered, and has been patented by XenoPort as a new chemical entity with an improved pharmacokin…

Kategori:
Acids, AcyclicAminobutyratesButyrates +10
Target Protein:
Gamma-aminobutyric acid type B receptor subunit 1Gamma-aminobutyric acid receptor subunit gamma-3Gamma-aminobutyric acid type B receptor subunit 2
Waktu ParuhIV bolus administra…
Vol. DistribusiRadioactive labelin…
KlirensBlood clearance of …
Genetik -
Arbekacin DB06696
small molecule | CAS: 51025-85-5

An semisynthetic aminoglycoside antibiotic. Often used for treatment of multi-resistant bacterial infection such as methicillin-resistant _Staphylococcus aureus_ (MRSA).

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +9
Target Protein:
30S ribosomal protein S12
Waktu Paruh3 hours
Vol. Distribusi-
Klirens-
Genetik -
Arbutin Approved DB11217
small molecule | CAS: 497-76-7

Extracted from the dried leaves of bearberry plant in the genus _Arctostaphylos_ and other plants commonly in the _Ericaceae_ family, arbutin is a beta-D-glucopyranoside of [DB09526]. It is found in foods, over-the-counter drugs, and herbal dietary supplement…

Kategori:
CarbohydratesGlucosidesGlycosides
Target Protein:
Tyrosinase
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
ARC-19499 DB15285
biotech | CAS: 1350667-54-7

ARC-19499 is under investigation in clinical trial NCT01191372 (First-in-Human and Proof-of-Mechanism Study of ARC19499 Administered to Hemophilia Patients).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ARC183 DB05124
biotech

ARC183 is a DNA aptamer, which is a single-stranded DNA molecule consisting of 15 deoxynucleotides that forms well-defined three-dimensional configuration, allowing it to bind to thrombin with high affinity and specificity. The key advantage of ARC183 compar…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Archexin DB05971
small molecule

Deskripsi belum tersedia.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Target Protein:
RAC-alpha serine/threonine-protein kinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arcitumomab DB17201
biotech | CAS: 154361-48-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ardeparin Approved DB00407
small molecule | CAS: 9005-49-6

Ardeparin, marketed under the US trade name Normiflo, is a low molecular weight heparin (LMWH) anticoagulant used for the prevention of postoperative venous thrombosis. Ardeparin is derived via peroxide degradation of heparin extracted from porcine intestinal…

Kategori:
Agents causing hyperkalemiaAnticoagulantsCarbohydrates +7
Target Protein:
Antithrombin-IIIHeparin cofactor 2
Waktu ParuhElimination half-li…
Vol. Distribusi-
Klirens-
Genetik -
Arecoline DB04365
small molecule | CAS: 63-75-2

An alkaloid obtained from the betel nut (Areca catechu), fruit of a palm tree. It is an agonist at both muscarinic and nicotinic acetylcholine receptors. It is used in the form of various salts as a ganglionic stimulant, a parasympathomimetic, and a vermifuge…

Kategori:
AlkaloidsCholinergic AgentsCholinergic Agonists +3
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ARG201 DB06621
biotech

ARG201, a bovine-derived Type I collagen, aims to induce immune tolerance in patients with Diffuse Systemic Scleroderma (dcSSc). This drug was investigated in the completed clinical trial NCT0000567 (Multicenter Phase II Trial of Oral Type I Bovine Collagen i…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Argadin DB04350
small molecule | CAS: 289665-92-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Target Protein:
Chitotriosidase-1Endochitinase B1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Argifin DB03632
small molecule | CAS: 243975-37-3

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsChitinases, antagonists & inhibitorsPeptides
Target Protein:
Chitotriosidase-1Endochitinase B1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arginine DB00125
small molecule | CAS: 74-79-3

An essential amino acid that is physiologically active in the L-form.

Kategori:
Acids, AcyclicAmino AcidsAmino Acids, Basic +14
Target Protein:
Cationic amino acid transporter 3Antizyme inhibitor 2Argininosuccinate lyase +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 7675-83-4

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, AcidicAmino Acids, Basic +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 4320-30-3

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBile and Liver Therapy +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arginine PCA DB16025
small molecule | CAS: 56265-06-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arimoclomol Approved DB05025
small molecule | CAS: 289893-25-0

Arimoclomol is a hydroxylamine derivative [A264414] and a heat-shock protein-70 (HSP70) co-inducer.[L51384] Arimoclomol was approved by the FDA on September 20, 2024, making it the first treatment for Niemann-Pick disease, type C (NPC).[L51389] It is also bei…

Kategori:
AminesMATE 1 SubstratesMATE 2 Substrates +3
Waktu ParuhThe elimination hal…
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent c…
Genetik -
Aripiprazole Approved DB01238
small molecule | CAS: 129722-12-9

Aripiprazole is an atypical antipsychotic orally indicated for the treatment of schizophrenia, bipolar I, major depressive disorder, irritability associated with autism, and Tourette's.[L45859] It is also indicated as an injection for agitation associated wit…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +48
Target Protein:
D(2) dopamine receptor5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 1A +35
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe steady-state vo…
KlirensThe clearance of ar…
Genetik -
Aripiprazole lauroxil Approved DB14185
small molecule | CAS: 1259305-29-7

Aripiprazole lauroxil is a long-acting injectable atypical antipsychotic drug used in the treatment of schizophrenia in adult patients. It is a prodrug of [aripiprazole], which acts as a partial agonist at the D2 and 5-HT1A receptors, and as an antagonist at …

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +29
Target Protein:
D(2) dopamine receptor5-hydroxytryptamine receptor 1A5-hydroxytryptamine receptor 2A +22
Waktu ParuhThe mean aripiprazo…
Vol. DistribusiBased on population…
KlirensIn rats, the cleara…
Genetik -
Arketamine DB19150
small molecule | CAS: 33643-49-1

Arketamine is under investigation in clinical trial NCT05414422 (A Randomized, Placebo-controlled, Double-blind Study to Assess Safety and Efficacy of PCN-101 in TRD).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ARM-210 DB16944
small molecule | CAS: 1467605-57-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arnica montana DB14297
biotech | CAS: 8057-65-6

Arnica montana is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
AngiospermsAsteraceaeBiological Products +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ARO-ANG3 DB17626
biotech

ARO-ANG3 is a subcutaneously administered RNA interference (RNAi)-based investigational medicine targeting angiopoietin-like protein 3 (ANGPTL3). It was granted an orphan drug designation for the treatment of homozygous familial hypercholesterolemia (HoFH).[L…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ARO-APOC3 DB17625
biotech

ARO-APOC3 is an investigational RNAi therapeutic targeting apolipoprotein C-III (APOC3). It received an Orphan Drug designation by the FDA for the treatment of familial chylomicronemia syndrome.[L45864]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arotinoid acid DB02877
small molecule | CAS: 71441-28-6

Arotinoid acid is a retinoic acid analog which acts as a selective RAR agonist.

Kategori:
Acids, CarbocyclicAlkenesBenzene Derivatives +9
Target Protein:
Retinoic acid receptor beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ARRY-502 DB16053
small molecule | CAS: 1202891-16-4

ARRY-502 is under investigation in clinical trial NCT01561690 (A Study of ARRY-502 in Patients With Persistent Asthma).

Target Protein:
Prostaglandin D2 receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arsanilic acid DB03006
small molecule | CAS: 98-50-0

An arsenical which has been used as a feed additive for enteric conditions in pigs and poultry. It causes blindness and is ototoxic and nephrotoxic in animals. [PubChem]

Kategori:
Adjuvants, ImmunologicAlkenesAnti-Infective Agents +10
Target Protein:
Lysozyme C
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arsenic trioxide Approved DB01169
small molecule | CAS: 1327-53-3

Arsenic trioxide is a chemotherapeutic agent of idiopathic function used to treat leukemia that is unresponsive to first line agents. It is suspected that arsenic trisulfide induces cancer cells to undergo apoptosis. In general, arsenic is known to be a natur…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsArsenicals +16
Target Protein:
Inhibitor of nuclear factor kappa-B kinase subunit betaThioredoxin reductase 1, cytoplasmicTranscription factor Jun +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arsenite ion DB18509
small molecule | CAS: 15502-74-6

Deskripsi belum tersedia.

Kategori:
AnionsArsenicalsElectrolytes +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arsenous acid DB04456
small molecule | CAS: 13464-58-9

Deskripsi belum tersedia.

Kategori:
AnionsArsenicalsElectrolytes +1
Target Protein:
Arsenate reductaseArsenical pump-driving ATPase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ART5803 DB18379
biotech

ART5803 is a humanized one-armed monoclonal antibody with a high affinity for the NMDA receptor.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Artemether Approved DB06697
small molecule | CAS: 71963-77-4

Artemether is an antimalarial agent used to treat acute uncomplicated malaria. It is administered in combination with lumefantrine for improved efficacy. This combination therapy exerts its effects against the erythrocytic stages of <i>Plasmodium spp.</i> and…

Kategori:
Anti-Infective AgentsAntimalarialsAntiparasitic Agents +25
Target Protein:
Sodium/potassium-transporting ATPase subunit alpha-1
Waktu ParuhArtemether, 1.6 +/-…
Vol. Distribusi-
Klirens-
Genetik -
Artemin DB15438
biotech | CAS: 309758-71-2

Artemin is under investigation in clinical trial NCT01842126 (Phase 1 Subcutaneous Single and Multiple Ascending Dose Study of BG00010 (Neublastin)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Artemisia annua pollen Approved DB10582
biotech

Artemisia annua pollen is the pollen of the Artemisia annua plant. Artemisia annua pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Pollen Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Artemisone DB16097
small molecule | CAS: 255730-18-8

Artemisone is under investigation in clinical trial NCT00936767 (Artemisone for the Treatment of Uncomplicated Falciparum Malaria in Western Cambodia).

Kategori:
Free RadicalsPeroxidesReactive Oxygen Species +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Artemotil Approved DB13851
small molecule | CAS: 75887-54-6

Artemotil, also known as ?-arteether, is a semi-synthetic derivative of artemisinin and a fast acting blood schizonticide specifically indicated for the treatment of chloroquine-resistant _Plasmodium falciparum_ malaria and cerebral malaria cases.

Kategori:
AmebicidesAnti-Infective AgentsAntimalarials +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Artenimol Approved DB11638
small molecule | CAS: 71939-50-9

Artenimol is an artemisinin derivative and antimalarial agent used in the treatment of uncomplicated *Plasmodium falciparum* infections [FDA Label]. It was first authorized for market by the European Medicines Agency in October 2011 in combination with [DB139…

Kategori:
Anti-Infective AgentsAntimalarialsAntiparasitic Agents +16
Target Protein:
Actin, cytoplasmic 2Alpha-aminoadipic semialdehyde dehydrogenaseAnnexin A2 +188
Waktu ParuhArtenimol was repor…
Vol. DistribusiArtenimol was obser…
KlirensArtenimol was obser…
Genetik -
Arterolane DB19027
small molecule | CAS: 664338-39-0

Arterolane is under investigation in clinical trial NCT03452475 (Comparison of Arterolane-piperaquine Versus Arterolane-piperaquine+mefloquine Versus Artemether-lumefantrine in Kenyan Children).

Kategori:
AnionsAntimalarialsAntiparasitic Products, Insecticides and Repellents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Artesunate Approved DB09274
small molecule | CAS: 88495-63-0

Artesunate is indicated for the initial treatment of severe malaria.[L14099] The World Health Organization recommends artesunate as first line treatment for severe malaria.[L890] Artesunate was developed out of a need for a more hydrophilic derivative of [art…

Kategori:
Acids, AcyclicAnionsAnthelmintics +28
Target Protein:
Malaria protein EXP-1
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of ar…
Genetik -
Articaine Approved DB09009
small molecule | CAS: 23964-58-1

Articaine is a dental local anesthetic. Articaine is widely used around the world and is the most popular local anesthetic in many European countries.

Kategori:
AmidesAnestheticsAnesthetics, Local +11
Target Protein:
Voltage-gated sodium channel alpha subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arundic acid DB05343
small molecule | CAS: 185517-21-9

Arundic acid has been investigated for the treatment of Amyotrophic Lateral Sclerosis (ALS).

Kategori:
Acids, AcyclicFatty AcidsLipids
Target Protein:
Beta-3 adrenergic receptorProtein S100-B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ARX201 DB05082
small molecule

ARX201 (PEG-ahGH) is a recombinant form of human growth hormone that has been modified using Ambrx’s patented ReCODE™ technology to achieve precise spatial positioning of the site of polyethylene glycol (PEG) attachment to human growth hormone, by biosyntheti…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 2451–2500 dari 12560
Sebelumnya Halaman 50 / 252 Berikutnya