Hasil Filter

2279

Total database: 17430
Struktur (SMILES)
866 (38.0%)
Target
1100 (48.3%)
Genomik
31 (1.4%)
Referensi
2279 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (2279)

Halaman 5 / 46
biotech | CAS: 308067-60-9

Rabbit anti-thymocyte globulin. Thymoglobulin is a polyclonal antibody that suppresses certain types of immune cells responsible for acute organ rejection in transplant patients. Thymoglobulin is a mixture of antibodies intended to bind to various cell surfac…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibody-Surface Protein Interactions +22
Target Protein:
Major histocompatibility complex class I-related gene proteinIntegrin alpha-LT-lymphocyte activation antigen CD86 +6
Waktu Paruh2-3 days, may incre…
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2636710-07-9

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ANX-005 DB16977
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AOC 1001 DB18620
biotech | CAS: 2653183-66-3

Delpacibart (AOC 1001) is being investigated in a global study for the treatment of Myotonic Dystrophy type 1 (DM1) in clinical trial NCT06411288

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AOC-1020 DB18621
biotech

AOC-1020 is an antibody oligonucleotide conjugate, comprised of a human transferrin receptor 1 targeting, effector function null, humanized IgG1 antibody, a MCC maleimide linker, and a double-stranded siRNA oligonucleotide targeting DUX4.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AOD9604 DB06388
small molecule | CAS: 221231-10-3

AOD9604 is a synthetic analogue of the lipolytic domain of human growth hormone, being investigated for the treatment of obesity.

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AP-101 DB17947
biotech

AP-101 is a recombinant human antibody directed against human misfolded superoxide dismutase 1.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apadamtase alfa Approved DB15164
biotech | CAS: 2086325-24-6

Thrombotic thrombocytopenic purpura (TTP) is a rare blood clotting disorder characterized by thrombocytopenia, microangiopathic hemolytic anemia, and various degrees of organ damage.[A262076] It may be inherited (congenital TTP; cTTP) or acquired due to autoa…

Kategori:
ADAM ProteinsADAMTS ProteinsAmino Acids, Peptides, and Proteins +12
Target Protein:
von Willebrand factor
Waktu ParuhFollowing the intra…
Vol. Distribusi-
Klirens-
Genetik -
Apalutamide Approved DB11901
small molecule | CAS: 956104-40-8

Apalutamide is a potent androgen receptor (AR) antagonist that selectively binds to the ligand-binding domain of AR and blocks AR nuclear translocation or binding to androgen response elements [A31846]. It has been used in trials studying the treatment of Pro…

Kategori:
Androgen Receptor InhibitorsAntiandrogensAntineoplastic Agents +28
Target Protein:
Androgen receptorGABA(A) Receptor
Waktu ParuhThe mean effective …
Vol. DistribusiThe mean apparent v…
KlirensThe CL/F of apaluta…
Genetik -
biotech | CAS: 2097132-02-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apatorsen DB06094
biotech | CAS: 1002331-21-6

Apatorsen is a second generation antisense drug which in preclinical experiments, inhibits production of Heat Shock Protein 27 (Hsp27) a cell survival protein found at elevated levels in many human cancers including prostate, lung, breast, ovarian, bladder, r…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Target Protein:
Heat shock protein beta-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apitegromab DB16096
biotech | CAS: 2278276-46-1

Apitegromab is under investigation in clinical trial NCT03921528 (An Active Treatment Study of SRK-015 in Patients With Type 2 or Type 3 Spinal Muscular Atrophy).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
APL-502 DB17473
biotech | CAS: 2303884-58-2

APL 502 is a humanised immunoglobulin G1 (IgG1) monoclonal antibody targeting the programmed cell death-1 ligand-1 (PD-L1).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apolizumab DB06467
biotech | CAS: 267227-08-7

Apolizumab is a humanized monoclonal antibody that is being studied as a treatment for hematologic cancers.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apramycin DB04626
small molecule | CAS: 37321-09-8

Apramycin is an aminoglycoside antibiotic and has a bactericidal action against many gram-negative bacteria. Apramycin is a structurally unique antibiotic that contains a bicyclic sugar moiety and a monosubstituted deoxystreptamine. It is not approved for use…

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +4
Target Protein:
16S ribosomal RNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aprepitant Approved DB00673
small molecule | CAS: 170729-80-3

Aprepitant, an antiemetic, is a substance P/neurokinin 1 (NK1) receptor antagonist which, in combination with other antiemetic agents, is indicated for the prevention of acute and delayed nausea and vomiting associated with initial and repeat courses of highl…

Kategori:
Alimentary Tract and MetabolismAntiemeticsAntiemetics and Antinauseants +36
Target Protein:
Substance-P receptor
Waktu Paruh9-13 hours
Vol. Distribusi* 70 L
Klirens* Apparent plasma c…
Genetik -
Aprocitentan Approved DB15059
small molecule | CAS: 1103522-45-7

Aprocitentan is a dual antagonist of endothelin receptors A and B used for treatment-resistant hypertension. It is the active metabolite of [macitentan]. Approximately 10-15% of patients with hypertension have resistant hypertension, defined as uncontrolle…

Kategori:
AmidesAntihypertensive AgentsBCRP/ABCG2 Inhibitors +26
Target Protein:
Endothelin-1 receptorEndothelin receptor type B
Waktu ParuhThe effective half-…
Vol. DistribusiThe apparent volume…
KlirensThe apparent cleara…
Genetik -
Apronalide Approved DB13221
small molecule | CAS: 528-92-7

Apronalide is approved in Japan. Apronalide has been withdrawn from the market in many other countries due to patient development of thrombocytopenic purpura [A174814].

Kategori:
AmidesCentral Nervous System DepressantsHypnotics and Sedatives +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 506-32-1

An unsaturated, essential fatty acid. It is found in animal and human fat as well as in the liver, brain, and glandular organs, and is a constituent of animal phosphatides. It is formed by the synthesis from dietary linoleic acid and is a precursor in the bio…

Kategori:
Arachidonic AcidsCytochrome P-450 CYP2C9 SubstratesCytochrome P-450 Substrates +5
Target Protein:
Prostaglandin G/H synthase 1Peroxisome proliferator-activated receptor alphaBile acid receptor +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ARC-19499 DB15285
biotech | CAS: 1350667-54-7

ARC-19499 is under investigation in clinical trial NCT01191372 (First-in-Human and Proof-of-Mechanism Study of ARC19499 Administered to Hemophilia Patients).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arcitumomab DB17201
biotech | CAS: 154361-48-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ARGX-119 DB18133
biotech

ARGX-119 is a monoclonal antibody that targets and activates muscle-specific kinase (MuSK).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arimoclomol Approved DB05025
small molecule | CAS: 289893-25-0

Arimoclomol is a hydroxylamine derivative [A264414] and a heat-shock protein-70 (HSP70) co-inducer.[L51384] Arimoclomol was approved by the FDA on September 20, 2024, making it the first treatment for Niemann-Pick disease, type C (NPC).[L51389] It is also bei…

Kategori:
AminesMATE 1 SubstratesMATE 2 Substrates +3
Waktu ParuhThe elimination hal…
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent c…
Genetik -
Aripiprazole Approved DB01238
small molecule | CAS: 129722-12-9

Aripiprazole is an atypical antipsychotic orally indicated for the treatment of schizophrenia, bipolar I, major depressive disorder, irritability associated with autism, and Tourette's.[L45859] It is also indicated as an injection for agitation associated wit…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +48
Target Protein:
D(2) dopamine receptor5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 1A +35
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe steady-state vo…
KlirensThe clearance of ar…
Genetik -
Armodafinil Approved DB06413
small molecule | CAS: 112111-43-0

Armodafinil is the enantiopure of the wakefulness-promoting agent modafinil (Provigil), and is indicated to improve wakefulness in adult patients with excessive sleepiness associated with obstructive sleep apnea (OSA), narcolepsy, or shift work disorder (SWD)…

Kategori:
Benzene DerivativesBenzhydryl CompoundsCentral Nervous System Agents +21
Target Protein:
Alpha-1D adrenergic receptorSodium-dependent dopamine transporter
Waktu ParuhTerminal half-life …
Vol. DistribusiApparent volume of …
KlirensThe oral clearance …
Genetik -
ART5803 DB18379
biotech

ART5803 is a humanized one-armed monoclonal antibody with a high affinity for the NMDA receptor.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Artemisia vulgaris root Approved DB14170
biotech

Artemisia vulgaris root allergenic extract is used in allergenic testing.

Kategori:
Non-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Articaine Approved DB09009
small molecule | CAS: 23964-58-1

Articaine is a dental local anesthetic. Articaine is widely used around the world and is the most popular local anesthetic in many European countries.

Kategori:
AmidesAnestheticsAnesthetics, Local +11
Target Protein:
Voltage-gated sodium channel alpha subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ARX201 DB05082
small molecule

ARX201 (PEG-ahGH) is a recombinant form of human growth hormone that has been modified using Ambrx’s patented ReCODE™ technology to achieve precise spatial positioning of the site of polyethylene glycol (PEG) attachment to human growth hormone, by biosyntheti…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arylacenamide DB05792
small molecule | CAS: 132173-07-0

Arylacenamide (SR31747) is a peripheral [sigma] ligand that binds four proteins in human cells, i.e. SRBP-1, [sigma]-2, HSI and its relative SRBP-2. It is a dual agent with both immunomodulatory and antiproliferative activities.

Kategori:
CycloparaffinsEnzyme InhibitorsImmunologic Factors +1
Target Protein:
3-beta-hydroxysteroid-Delta(8),Delta(7)-isomeraseHCG20471, isoform CRA_c
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ASC-618 DB18423
biotech

ASC-618 is a recombinant adeno-associated virus serotype 8 (rAAV2/8) vector expressing bioengineered B domain deleted liver-codon-optimized human factor VIII.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ascorbic acid Approved DB00126
small molecule | CAS: 50-81-7

A six carbon compound related to glucose. It is found naturally in citrus fruits and many vegetables. Ascorbic acid is an essential nutrient in human diets, and necessary to maintain connective tissue and bone. Its biologically active form, vitamin C, functio…

Kategori:
Acids, AcyclicAlimentary Tract and MetabolismAntioxidants +20
Target Protein:
Solute carrier family 23 member 2Solute carrier family 23 member 1Hyaluronate lyase +23
Waktu Paruh16 days (3.4 hours …
Vol. Distribusi-
Klirens-
Genetik -
Asenapine Approved DB06216
small molecule | CAS: 65576-45-6

Developed by Schering-Plough after its merger with Organon International, asenapine is a sublingually administered, atypical antipsychotic for treatment of schizophrenia and acute mania associated with bipolar disorder. Asenapine also belongs to the dibenzo-o…

Kategori:
Acid ReducersAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +41
Target Protein:
5-hydroxytryptamine receptor 2AD(2) dopamine receptor5-hydroxytryptamine receptor 1A +17
Waktu Paruh24 hours (range of …
Vol. Distribusi20-25 L/kg
Klirens-
Genetik -
ASI402 DB06373
biotech | CAS: 372075-37-1

ASI402 is a monoclonal antibody that targets an aberrantly glycosylated antigen Mucin 1. It is being investigated in cancers.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Mucin-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Asimadoline DB05104
small molecule | CAS: 153205-46-0

Asimadoline is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, Germany. Asimadoline was originally developed to treat peripheral pain such as arthritis. Asimadoline is an orally administered agent that acts as a kap…

Kategori:
AcetatesAcids, AcyclicAmides
Target Protein:
Kappa-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ASP-7317 DB18549
biotech

ASP-7317 consists of human embryonic stem cell-derived retinal pigment epithelium cells.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Astemizole Approved DB00637
small molecule | CAS: 68844-77-9

Astemizole is a long-acting, non-sedating second generation antihistamine used in the treatment of allergy symptoms. It was withdrawn from market by the manufacturer in 1999 due to the potential to cause arrhythmias at high doses, especially when when taken …

Kategori:
Anti-Allergic AgentsAntihistamines for Systemic UseBenzimidazoles +27
Target Protein:
Histamine H1 receptorVoltage-gated inwardly rectifying potassium channel KCNH2Voltage-gated delayed rectifier potassium channel KCNH1 +1
Waktu Paruh1 day
Vol. Distribusi-
Klirens-
Genetik -
AstraZeneca COVID-19 Vaccine Approved DB15656
biotech | CAS: 2420395-83-9

The AstraZeneca COVID-19 Vaccine (previously known as ChAdOx1 nCoV-19 or AZD1222) is one of several vaccines developed in 2020 for the prevention of COVID-19 caused by SARS-CoV-2.[L12669,L32649] The ChAdOx1 viral vector was developed at the University of Oxfo…

Kategori:
Biological ProductsComplex MixturesCOVID-19 Vaccines +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Asunercept DB15160
biotech | CAS: 1450882-18-4

Asunercept is under investigation in clinical trial NCT02853565 (A Study of CAN008 for Newly Diagnosed Glioblastoma Multiforme).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AT1022 DB04995
small molecule

AT1022 is a hydromorphone skin patch designed to provide rapid and sustained delivery of a potent opiate for the management of severe pain. AT1022 incorporates PassPort(TM) system, developed to deliver protein and peptide drugs, small-molecule drugs, genes a…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AT3022 DB05172
small molecule

AT3022, the Altea Therapeutics’s fentanyl citrate transdermal patch designed to provide safe and rapid management of moderate to severe chronic pain.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ATA-100 DB18329
biotech

ATA-100 is an adeno-associated virus serotype 9 carrying the human Fukutin-Related protein gene and target sequence of the miR-208a

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Atacicept DB06399
biotech | CAS: 845264-92-8

Atacicept is a recombinant fusion protein combined with the extracellular ligand binding portion of TACI.

Kategori:
Amino Acids, Peptides, and ProteinsProteinsRecombinant Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Atazanavir Approved DB01072
small molecule | CAS: 198904-31-3

Atazanavir (formerly known as BMS-232632) is an antiretroviral drug of the protease inhibitor (PI) class. Like other antiretrovirals, it is used to treat infection of human immunodeficiency virus (HIV). Atazanavir is distinguished from other PIs in that it ca…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-HIV AgentsAnti-Infective Agents +45
Target Protein:
Pol polyproteinGag-Pol polyprotein
Gen Terkait:
UGT1A1 UGT1A1 UGT1A1
Waktu ParuhThe mean eliminatio…
Vol. DistribusiIn patients with HI…
KlirensIn patients with HI…
Genetik 3 Varian
small molecule | CAS: 433937-93-0

Atecegatran metoxil has been used in trials studying the basic science and prevention of Nonvalvular Atrial Fibrillation, Persistent or Permanent Nonvalvular Atrial Fibrillation, and Persistent or Permanent Non-valvular Atrial Fibrillation.

Kategori:
Azetines
Target Protein:
Prothrombin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Atenolol Approved DB00335
small molecule | CAS: 29122-68-7

Atenolol is a cardioselective beta-blocker used in a variety of cardiovascular conditions. Sir James Black, a Scottish pharmacologist, pioneered the use of beta-blockers for the management of angina pectoris in 1958 for which he received the Nobel Prize.[…

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-1 Receptor Antagonists +23
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptor
Gen Terkait:
ADRB1
Waktu Paruh6-7 hrs.[label]
Vol. DistribusiTotal Vd of 63.8-11…
KlirensTotal clearance is …
Genetik 1 Varian
Atezolizumab Approved DB11595
biotech | CAS: 1380723-44-3

Atezolizumab is a humanized monoclonal antibody used to prevent the interaction of PD-L1 and PD-1, removing inhibition of immune responses seen in some cancers.[A18493,L7489] This medication is reserved for patients whose tumors express PD-L1, cannot receive …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +19
Target Protein:
Programmed cell death 1 ligand 1Programmed cell death protein 1
Waktu ParuhThe half life of at…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of at…
Genetik -
ATG-Fresenius S DB05320
small molecule

ATG-Fresenius S is a concentrated anti-human T-lymphocyte immunoglobulin preparation derived from rabbits after immunization with a T-lympoblast cell line. ATG-Fresenius S is an immunosuppressive product for the prevention and treatment of acute rejection fol…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ATI-1013 DB18185
biotech

ATI-1013 is a fully human nicotine-specific monoclonal antibody.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ATI-355 DB17923
biotech

ATI-355 is a humanized anti-Nogo-A antibody developed by Novartis.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 201–250 dari 2279
Sebelumnya Halaman 5 / 46 Berikutnya