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3253

Total database: 17430
Struktur (SMILES)
2451 (75.3%)
Target
1833 (56.3%)
Genomik
35 (1.1%)
Referensi
3253 (100.0%)

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Hasil Pencarian (3253)

Halaman 49 / 66
small molecule | CAS: 25322-68-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Polyethylene glycol 400 Approved DB11077
small molecule | CAS: 25322-68-3

Polyethylene glycols (PEGs) are products made of condensed ethylene oxide and water that can contain various derivatives and have various functions. Because many PEG types are hydrophilic, they are favorably used as enhancers of penetration, and used heavily …

Kategori:
AlcoholsArtificial TearsCompounds used in a research, industrial, or household setting +8
Target Protein:
Ectonucleotide pyrophosphatase/phosphodiesterase family member 1Oxidoreductase HTATIP2
Waktu ParuhGreat than 24h [L17…
Vol. Distribusi-
KlirensIn mice, lease than…
Genetik -
Polysilicone-15 Approved DB11271
small molecule | CAS: 207574-74-1

Polysilicone-15 is a silicone based UVB absorber [L2796, L2797, L2799, F87, F88, F89]. The compound is a colorless to pale yellow viscous liquid which is soluble in organic solvents of medium polarity and insoluble in water [L2796, L2797, L2799, F87, F88, F89…

Kategori:
Sunscreen Agents
Waktu ParuhPolysilicone-15 is …
Vol. DistribusiPolysilicone-15 is …
KlirensPolysilicone-15 is …
Genetik -
biotech

Polyvalent antigen-KLH conjugate vaccine is a multivalent cancer vaccine comprised of the five tumor-associated antigens (TAAs) globo H, GM2 ganglioside, Tn-MUC1, TF, and sTn conjugated with the immunoadjuvant keyhole limpet hemocyanin (KLH). It is under inve…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ponatinib Approved DB08901
small molecule | CAS: 943319-70-8

Ponatinib is a novel Bcr-Abl tyrosine kinase inhibitor that is especially effective against the T315I mutation for the treatment of chronic myeloid leukemia. FDA approved on December 14, 2012.

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBcr-Abl Tyrosine Kinase Inhibitors +23
Target Protein:
Tyrosine-protein kinase ABL1Breakpoint cluster region proteinMast/stem cell growth factor receptor Kit +12
Waktu ParuhAfter oral administ…
Vol. DistribusiAfter oral administ…
Klirens-
Genetik -
Ponesimod Approved DB12016
small molecule | CAS: 854107-55-4

Ponesimod is a selective sphingosine 1-phosphate receptor 1 modulator indicated in the treatment of relapsing forms of multiple sclerosis in adults.[A232079,L32709] Ponesimod was developed out of a need for a more selective modulator of sphingosine 1-phosphat…

Kategori:
Antineoplastic and Immunomodulating AgentsCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +13
Target Protein:
Sphingosine 1-phosphate receptor 1
Waktu ParuhPonesimod has an el…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of po…
Genetik -
Poractant alfa Approved DB09113
biotech | CAS: 129069-19-8

Poractant alfa is a pulmonary surfactant marketed as Curosurf in the United States and Canada. It is used to treat Respiratory Distress Syndrome (RDS) in premature infants with an endogenous pulmonary surfactant deficiency. Poractant alfa is an extract of nat…

Kategori:
Alveolar Surface Tension ReductionBradycardia-Causing AgentsComplex Mixtures +6
Waktu ParuhThe half-life of po…
Vol. DistribusiNo studies on the d…
KlirensNo studies on clear…
Genetik -
Porgaviximab DB17773
biotech | CAS: 1792982-55-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Posaconazole Approved DB01263
small molecule | CAS: 171228-49-2

Posaconazole is a triazole antifungal drug that is used to treat invasive infections by Candida species and Aspergillus species in severely immunocompromised patients.

Kategori:
14-alpha Demethylase InhibitorsAnti-Infective AgentsAntifungal Agents +23
Target Protein:
Lanosterol 14-alpha demethylase
Waktu ParuhPosaconazole is eli…
Vol. Distribusi* 1774 L
Klirens* 32 L/hr * 51 L/h…
Genetik -
Potassium acetate Approved DB14498
small molecule | CAS: 127-08-2

Deskripsi belum tersedia.

Kategori:
AcetatesAcids, AcyclicAgents causing hyperkalemia +8
Target Protein:
Sodium/potassium-transporting ATPase subunit alpha-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Potassium alum Approved DB09087
small molecule | CAS: 10043-67-1

Potassium alum is considered by the FDA as a generally recognized as safe (GRAS) substance.[L1070] It is an inorganic salt, also called potassium aluminum sulfate with a formula of AlK(SO4)2 that is predominantly produced in the dodecahydrate form (AlK(SO4)2 …

Kategori:
Adjuvants, ImmunologicAluminium CompoundsImmunologic Factors +7
Waktu ParuhStudies performed w…
Vol. DistribusiThe distribution of…
KlirensRenal clearance of …
Genetik -
small molecule | CAS: 868-14-4

Potassium bitartate, also referred to as potassium acid tartrate or cream of tartar, is the potassium acid salt of l-( + )-tartaric acid. It is obtained as a byproduct of wine manufacture during the fermentation process. Approved by the FDA as a direct food s…

Kategori:
LaxativesPotassium Salt
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Potassium citrate Approved DB09125
small molecule | CAS: 866-84-2

Potassium citrate (also known as tripotassium citrate) is a potassium salt of citric acid. It is a white, hygroscopic crystalline powder. It is odorless with a saline taste. It contains 38.3% potassium by mass. In the monohydrate form it is highly hygroscopic…

Kategori:
Acids, AcyclicAgents causing hyperkalemiaAlimentary Tract and Metabolism +15
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 12298-68-9

Deskripsi belum tersedia.

Kategori:
AnionsCoagulantsColoring Agents +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Povidone Approved DB11061
small molecule | CAS: 9003-39-8

Povidone, also known as polyvinylpyrrolidone (PVP) or polyvidone, is a synthetic water-soluble polymer made from the monomer N-vinylpyrrolidone used as a binder in many pharmaceutical tablets and lubricant in eye drops. It is also used in many technical appli…

Kategori:
AlkenesArtificial TearsBlood Substitutes +13
Waktu ParuhThis pharmacokineti…
Vol. DistribusiThis pharmacokineti…
KlirensThis pharmacokineti…
Genetik -
Povidone-iodine Approved DB06812
small molecule | CAS: 25655-41-8

Povidone-iodine is a stable chemical complex of polyvinylpyrrolidone (povidone, PVP) and elemental iodine. It contains from 9.0% to 12.0% available iodine, calculated on a dry basis. This unique complex was discovered in 1955 at the Industrial Toxicology Labo…

Kategori:
AlkenesAnti-Infective AgentsAnti-Infective Agents, Local +26
Waktu ParuhPovidone-Iodine is …
Vol. DistribusiPovidone-Iodine is …
KlirensPovidone-Iodine is …
Genetik -
Pozelimab Approved DB15218
biotech | CAS: 2096328-94-6

CD55-deficient protein-losing enteropathy (PLE), or CHAPLE disease, is an ultra-rare hereditary disease, with fewer than 100 patients diagnosed worldwide or fewer than 10 patients in the US.[L47880] The pathophysiology of this disease is mainly attributed to …

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsComplement Inactivating Agents +3
Target Protein:
Complement C5
Waktu ParuhIn healthy adult su…
Vol. DistribusiIn healthy adult su…
KlirensThere is limited in…
Genetik -
Poziotinib DB12114
small molecule | CAS: 1092364-38-9

Poziotinib has been used in trials studying the treatment of Breast Cancer, Metastatic Breast Cancer, Increased Drug Resistance, Adenocarcinoma of Lung Stage IV, and Adenocarcinoma of Lung Stage IIIB, among others.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Receptor tyrosine-protein kinase erbB-2Epidermal growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PP-121 DB08052
small molecule | CAS: 1092788-83-4

Deskripsi belum tersedia.

Target Protein:
Epidermal growth factor receptorDNA-dependent protein kinase catalytic subunitVascular endothelial growth factor receptor 2 +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PPL-100 DB05961
small molecule | CAS: 612547-11-2

Deskripsi belum tersedia.

Target Protein:
Gag-Pol polyproteinPlasma protease C1 inhibitorPlasma serine protease inhibitor +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Praconase DB05584
biotech | CAS: 1186547-12-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBacterial ProteinsBacterial Toxins +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Practolol Approved DB01297
small molecule | CAS: 6673-35-4

A beta-adrenergic antagonist that has been used in the emergency treatment of cardiac arrhythmias.

Kategori:
AcetanilidesAdrenergic AgentsAdrenergic Antagonists +20
Target Protein:
Beta-1 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pradigastat DB12866
small molecule | CAS: 956136-95-1

Pradigastat has been used in trials studying the treatment of Non-alcoholic Fatty Liver Disease (NAFLD).

Kategori:
Acids, AcyclicAminesFatty Acids +4
Target Protein:
Diacylglycerol O-acyltransferase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pradofloxacin DB11453
small molecule | CAS: 195532-12-8

Pradofloxacin is a 3rd generation fluoroquinolone antibiotic developed by Bayer HealthCare AG, Animal Health GmBH. It was approved by the European Commission in April 2011 for bacterial infections in dogs and cats.

Kategori:
4-QuinolonesAnti-Bacterial AgentsFluoroquinolone Antibacterial +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pramlintide Approved DB01278
small molecule | CAS: 151126-32-8

Pramlintide is a relatively new adjunct treatment for diabetes (both type 1 and 2), developed by Amylin Pharmaceuticals. It is derived from amylin, a hormone that is released into the bloodstream, in a similar pattern as insulin, after a meal. Like insulin, a…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsAmylin Agonists +12
Target Protein:
Glucagon-like peptide 1 receptorCalcitonin receptorReceptor activity-modifying protein 1 +2
Waktu ParuhApproximately 48 mi…
Vol. Distribusi-
Klirens-
Genetik -
Prasugrel Approved DB06209
small molecule | CAS: 150322-43-3

Prasugrel, a thienopyridine derivative, is a platelet activation and aggregation inhibitor structurally and pharmacologically related to clopidogrel and ticlopidine. Similar to clopidogrel, prasugrel is a prodrug that requires enzymatic transformation in the …

Kategori:
AnticoagulantsAntiplatelet agentsBlood and Blood Forming Organs +15
Target Protein:
P2Y purinoceptor 12
Waktu ParuhThe active metaboli…
Vol. Distribusi44-68L
KlirensApparent clearance …
Genetik -
Prednimustine DB12832
small molecule | CAS: 29069-24-7

Prednimustine has been used in trials studying the treatment of Lymphoma.

Kategori:
Alkylating DrugsAntineoplastic AgentsAntineoplastic Agents, Alkylating +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prednisone acetate Approved DB14646
small molecule | CAS: 125-10-0

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesAnti-Inflammatory AgentsAntineoplastic Agents +17
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prephenic acid DB08427
small molecule | CAS: 126-49-8

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicCyclohexanesCycloparaffins
Target Protein:
Chorismate mutase AroH
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Presatovir DB12165
small molecule | CAS: 1353625-73-6

Presatovir has been used in trials studying the treatment of RSV Infection, Respiratory Syncytial Virus (RSV), Respiratory Syncytial Virus Infections, and Respiratory Syncytial Virus (RSV) Infections.

Kategori:
AmidesHeterocyclic Compounds, Fused-RingPyrazoles +2
Target Protein:
Fusion glycoprotein F0
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prexasertib DB12008
small molecule | CAS: 1234015-52-1

Prexasertib has been used in trials studying the treatment and basic science of mCRPC, Leukemia, Neoplasm, breast cancer, and Ovarian Cancer, among others.

Kategori:
Enzyme InhibitorsProtein Kinase Inhibitors
Target Protein:
Serine/threonine-protein kinase Chk1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prezatide DB11296
small molecule | CAS: 49557-75-7

Prezatide is a tripeptide consisting of glycine, histidine, and lysine which readily forms a complex with copper ions [A19503]. Prezatide is used in cosmetic products for the skin and hair. It is known to aid wound healing and its potential applications in ch…

Kategori:
Amino Acids, Peptides, and ProteinsGrowth SubstancesPeptides
Waktu ParuhPrezatide is rapidl…
Vol. Distribusi-
Klirens-
Genetik -
PRGN-2012 DB18342
biotech

PRGN-2012 is an adenoviral vector expressing human papillomavirus (HPV) 6 and HPV 11 antigens

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Priliximab DB16920
biotech | CAS: 147191-91-1

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Primidone Approved DB00794
small molecule | CAS: 125-33-7

Primidone is an anticonvulsant used to treat essential tremor as well as grand mal, psychomotor, and focal epileptic seizures.[L11112] Primidone was developed by J Yule Bogue and H C Carrington in 1949.[A189522] Primidone was granted FDA Approval on 8 Marc…

Kategori:
Anti-epileptic AgentAnticholinergic AgentsAnticonvulsants +36
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-2Gamma-aminobutyric acid receptor subunit alpha-3Gamma-aminobutyric acid receptor subunit alpha-4 +8
Waktu ParuhThe half life of pr…
Vol. DistribusiThe volume of distr…
KlirensPrimidone is cleare…
Genetik -
Pristimerin DB17049
small molecule | CAS: 1258-84-0

Pristimerin is a quinone methide triterpenoid researched for its anti-cancer potential.[A253107]

Kategori:
TerpenesTriterpenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pritumumab DB17221
biotech | CAS: 499212-74-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Procaine Approved DB00721
small molecule | CAS: 59-46-1

A local anesthetic of the ester type that has a slow onset and a short duration of action. It is mainly used for infiltration anesthesia, peripheral nerve block, and spinal block. (From Martindale, The Extra Pharmacopoeia, 30th ed, p1016). Procaine has also b…

Kategori:
Acids, CarbocyclicAgents for Treatment of Hemorrhoids and Anal Fissures for Topical UseAgents that reduce seizure threshold +25
Target Protein:
Sodium channel protein type 10 subunit alphaGlutamate receptor ionotropic, NMDA 3A5-hydroxytryptamine receptor 3A +8
Waktu Paruh7.7 minutes
Vol. Distribusi-
Klirens-
Genetik -
Procalcitonin DB14812
biotech | CAS: 56645-65-9

Procalcitonin is under investigation in clinical trial NCT03440060 (Procalcitonin-guided Antibiotic Therapy During Severe Exacerbation of COPD).

Kategori:
Amino Acids, Peptides, and ProteinsBone Density Conservation AgentsCalcitonin Preparations +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Profenamine Approved DB00392
small molecule | CAS: 522-00-9

Profenamine (also known as ethopropazine) is a medication derived from phenothiazine. It is primarily used as an antidyskinetic to treat Parkinsonism. It is sold under the trade name Parsitan in Canada.[L46812] In the US, the marketing of profenamine has been…

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAgents producing tachycardia +12
Target Protein:
Histamine H1 receptorMuscarinic acetylcholine receptor M1Glutamate receptor ionotropic, NMDA 3A +1
Waktu Paruh1 to 2 hours
Vol. Distribusi-
Klirens-
Genetik -
Proflavine Approved DB01123
small molecule | CAS: 92-62-6

3,6-Diaminoacridine. Topical antiseptic used mainly in wound dressings.

Kategori:
AcridinesAminoacridinesAnti-Infective Agents +2
Target Protein:
DNAProthrombinHTH-type transcriptional regulator QacR +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Progesterone Approved DB00396
small molecule | CAS: 57-83-0

Progesterone is a hormone that occurs naturally in females, and is essential for endometrial receptivity, embryo implantation, and the successful establishment of pregnancy. A low progesterone concentration or an insufficient response to progesterone can caus…

Kategori:
Adrenal Cortex HormonesBCRP/ABCG2 InducersBCRP/ABCG2 Inhibitors +47
Target Protein:
Progesterone receptorMineralocorticoid receptorEstrogen receptor +7
Waktu ParuhAbsorption half-lif…
Vol. DistribusiWhen administered v…
Klirens**Apparent clearanc…
Genetik -
Prolactin G129R DB18431
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prolectin-M DB16521
small molecule

Prolectin-M is a (1-6)-alpha-D-mannopyranose[L31338] and acts as an antagonist of galectin.[L31343] It is being investigated in the clinical trial NCT04512027 (Prolectin-M in COVID-19 Patients Having Mild to Moderate Symptoms Not Requiring Oxygen Support. (Pr…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Proline DB00172
small molecule | CAS: 147-85-3

Proline is one of the twenty amino acids used in living organisms as the building blocks of proteins. Proline is sometimes called an imino acid, although the IUPAC definition of an imine requires a carbon-nitrogen double bond. Proline is a non-essential amino…

Kategori:
Amino AcidsAmino Acids, CyclicAmino Acids, Peptides, and Proteins +4
Target Protein:
Peptidyl-prolyl cis-trans isomerase BPeptidyl-prolyl cis-trans isomerase APyrroline-5-carboxylate reductase 1, mitochondrial +19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Promestriene DB12487
small molecule | CAS: 39219-28-8

Promestriene (3-propyl ethyl, 17B-methyl estradiol) has been used in trials studying the prevention of Hypospadias. It is a synthetic estrogen analog, which is used in topical estrogen therapy. Promestriene’s potential for treating vaginal atrophy symptoms as…

Kategori:
Estradiol CongenersEstranesEstrenes +10
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propagermanium DB17608
small molecule | CAS: 12758-40-6

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAntineoplastic AgentsElements +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propanoyl-CoA DB02912
small molecule | CAS: 317-66-8

Deskripsi belum tersedia.

Kategori:
Adenine NucleotidesCoenzymesEnzymes and Coenzymes +7
Target Protein:
Propionyl-CoA carboxylase complex B subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propiverine Approved DB12278
small molecule | CAS: 60569-19-9

Propiverine is a widely used antimuscarinic drug with a mixed mode of action in the treatment of symptoms associated with overactive bladder (OAB) [A32576]. Overactive bladder (OAB) is a chronic condition of the lower urinary tract characterized by urinary…

Kategori:
Acids, CarbocyclicAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +22
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3 +4
Waktu ParuhIn three studies in…
Vol. DistribusiIn one study, the v…
KlirensMean total clearanc…
Genetik -
Propyl Gallate DB12450
small molecule | CAS: 121-79-9

Propyl Gallate is under investigation in clinical trial NCT01450098 (A Study of LY2484595 in Healthy Subjects).

Kategori:
Acids, CarbocyclicAntioxidantsBenzene Derivatives +7
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 2401–2450 dari 3253
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