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2677

Total database: 17430
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1588 (59.3%)
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1494 (55.8%)
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51 (1.9%)
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Halaman 48 / 54
Sulforaphane DB12422
small molecule | CAS: 142825-10-3

Sulforaphane is under investigation for the treatment of Autism Spectrum Disorder. It is a naturally occurring isothiocyanate found in high concentration in a variety of broccoli.

Kategori:
Anticarcinogenic AgentsAntineoplastic AgentsCompounds used in a research, industrial, or household setting +3
Waktu Paruh-
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Sulisobenzone DB11185
small molecule | CAS: 4065-45-6

Sulisobenzone is approved by the FDA in concentrations of up to 10% and in Canada, is approved by Health Canada at the same concentrations [F38]. It works to filter out both UVA and UVB rays, protecting the skin from sun UV damage [L2153]. The UV-filter s…

Kategori:
Benzene DerivativesDrugs that are Mainly Renally ExcretedKetones +1
Target Protein:
Skin epithelial cells
Waktu Paruh-
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Sulpiride Approved DB00391
small molecule | CAS: 15676-16-1

Sulpiride first appeared in published literature in 1967.[A229538] Clinical studies show a greater effect on treating the negative symptoms of schizophrenia rather than positive symptoms at low doses, though the effects are more equal at higher doses.[A229683…

Kategori:
Acids, CarbocyclicAmidesAntidepressive Agents +26
Target Protein:
D(2) dopamine receptorD(3) dopamine receptorCarbonic anhydrase 2 +2
Waktu ParuhReports of the half…
Vol. DistribusiThe average volume …
KlirensThe total systemic …
Genetik -
Suprofen Approved DB00870
small molecule | CAS: 40828-46-4

An ibuprofen-type anti-inflammatory analgesic and antipyretic. It inhibits prostaglandin synthesis and has been proposed as an anti-arthritic. It is no longer approved for use in the United States.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAnalgesics +23
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu Paruh-
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Suptavumab DB12759
biotech | CAS: 1629615-23-1

Suptavumab has been used in trials studying the treatment and basic science of Respiratory Syncytial Virus Infections.

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Suratadenoturev DB18672
biotech | CAS: 1268642-13-2

Suratadenoturev is a gene-modified oncolytic adenovirus expressing the telomerase reverse transcriptase gene.

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Sutilain Approved DB09379
biotech | CAS: 12211-28-8

Sutilain is a member of the keratase family which includes agents such as papain. It is able to dissolve the intercellular matrix which helps with desquamation. Sutilain contains proteolytic enzymes derived from _Bacillus subtilis_ and it is available as a cr…

Kategori:
EndopeptidasesEnzymesEnzymes and Coenzymes +4
Waktu ParuhThis pharmacokineti…
Vol. DistribusiThis pharmacokineti…
KlirensThis pharmacokineti…
Genetik -
Sutimlimab Approved DB14996
biotech | CAS: 2049079-64-1

Cold agglutinin disease (CAD) is a type of autoimmune hemolytic anemia (AIHA) in which autoantibodies directed against red blood cell surface antigens cause hemolysis at low (3-4°C) temperatures.[A245154,L40114] This cold subtype accounts for approximately 15…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Target Protein:
Complement C1s subcomponent
Waktu ParuhAt the approved rec…
Vol. DistribusiAt steady-state, th…
KlirensAt the approved rec…
Genetik -
Suvecaltamide DB19139
small molecule | CAS: 953778-58-0

Suvecaltamide is under investigation in clinical trial NCT05122650 (A Study to Assess the Safety and Efficacy of JZP385 in the Treatment of Adults With Moderate to Severe Essential Tremor (ET)).

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Suvratoxumab DB15172
biotech | CAS: 1629620-18-3

Suvratoxumab is under investigation in clinical trial NCT02296320 (Study of the Efficacy and Safety of MEDI4893).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
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SVV-001 DB06129
biotech

SVV-001 is investigated for use/treatment in cancer/tumors and lung cancer. SVV-001 is a solid. SVV-001 (Seneca Valley Virus) is a novel native picornavirus being developed as a systemically deliverable oncolytic virus for treatment of human cancers with neur…

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SYNB1353 DB17666
biotech

SYNB1353 is a strain of the probiotic bacteria _Escherichia coli_ (_E. coli_) type Nissle and an engineered probiotic drug.[A258833] Developed by Synlogic Operating Company, Inc., SYNB1353 is being investigated for the treatment of homocystinuria. It is desig…

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SynOV1.1 DB17539
biotech

SynOV1.1 is an investigational cancer immunotherapy developed by SyngenTech. It is a recombinant oncolytic adenovirus, controlled by synthetic gene circuit, encoding the human immunostimulating factor cytokine granulocyte-macrophage colony-stimulating factor …

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small molecule

Synthetic conjugated estrogens A are composed of a blend of the following nine synthetic estrogenic substances: estrone sulfate, sodium equilin sulfate, sodium 17?-dihydroequilin sulfate, sodium 17?-estradiol sulfate, sodium 17?­ dihydroequilin sulfate, sodiu…

Kategori:
Cytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 SubstratesCytochrome P-450 Substrates +7
Target Protein:
Estrogen receptor
Waktu ParuhThe half life of ba…
Vol. DistribusiThe distribution of…
Klirens-
Genetik -
small molecule | CAS: 746658-13-9

Synthetic conjugated estrogens, B tablets contain a blend of ten synthetic estrogenic substances. The estrogenic substances are: sodium estrone sulfate, sodium equilin sulfate, sodium 17?-dihydroequilin sulfate, sodium 17?-estradiol sulfate, sodium 17?­ dihyd…

Kategori:
Cytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 SubstratesCytochrome P-450 Substrates +7
Target Protein:
Estrogen receptor
Waktu ParuhThe half life of ba…
Vol. DistribusiThe distribution of…
Klirens-
Genetik -
TA-CIN DB05809
biotech

TA-CIN is a subunit vaccine comprising L2/E6/E7 proteins from Human Papillomavirus (HPV16), designed to generate a strong cellular immune response against HPV-infected cells.

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TA-NIC DB05445
biotech

TA-NIC is a novel and proprietary vaccine in development as an aid to quitting smoking in motivated patients. It is designed to raise anti-nicotine antibodies which bind to nicotine molecules in the patient's blood stream, reducing the rate and quantity of ni…

Kategori:
Biological ProductsComplex Mixtures
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Tabelecleucel Approved DB17072
biotech

Tabelecleucel is an innovative therapy that uses Epstein-Barr virus (EBV)-specific allogeneic cytotoxic T cells (CTLs). It is produced by mixing T-cells with B-cells that have been infected with the Epstein-Barr virus (EBV). Both T-cells and B-cells are obtai…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsAntineoplastic cell and gene therapy
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small molecule | CAS: 2412170-98-8

Tabirafusp tedromer is under investigation in clinical trial NCT06556368 (A Study to Evaluate the Efficacy and Safety of Tarcocimab Tedromer and Tabirafusp Tedromer Compared to Aflibercept in Participants With Neovascular (Wet) Age-related Macular Degeneratio…

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Tacrine Approved DB00382
small molecule | CAS: 321-64-2

A centerally active cholinesterase inhibitor that has been used to counter the effects of muscle relaxants, as a respiratory stimulant, and in the treatment of Alzheimer's disease and other central nervous system disorders. Tacrine has been discontinued for t…

Kategori:
AcridinesAgents Causing Muscle ToxicityAminoacridines +16
Target Protein:
CholinesteraseAcetylcholinesteraseLiver carboxylesterase 1
Waktu Paruh2 to 4 hours
Vol. Distribusi* 349 ± 193 L
Klirens-
Genetik -
Tacrolimus Approved DB00864
small molecule | CAS: 104987-11-3

Tacrolimus (also FK-506 or Fujimycin) is an immunosuppressive drug whose main use is after organ transplant to reduce the activity of the patient's immune system and so the risk of organ rejection. It is also used in a topical preparation in the treatment of …

Kategori:
Agents causing hyperkalemiaAgents Causing Muscle ToxicityAgents for Dermatitis, Excluding Corticosteroids +33
Target Protein:
Protein phosphatase 3 catalytic subunit alphaPeptidyl-prolyl cis-trans isomerase FKBP1A
Gen Terkait:
CYP3A5 ABCB1
Waktu ParuhThe elimination hal…
Vol. Distribusi* 2.6 ± 2.1 L/kg [p…
Klirens* 0.040 L/hr/kg [he…
Genetik 2 Varian
Tafasitamab Approved DB15044
biotech | CAS: 1422527-84-1

Tafasitamab is a humanized, CD19-directed cytolytic monoclonal antibody intended for the treatment of B-cell malignancies.[L15302] It is produced using recombinant DNA technology in Chinese hamster ovary cells, and contains an IgG1/2 hybrid Fc-domain which ha…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +13
Target Protein:
B-lymphocyte antigen CD19
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe total volume of…
KlirensThe clearance of ta…
Genetik -
Tafenoquine Approved DB06608
small molecule | CAS: 106635-80-7

Tafenoquine is an 8-aminoquinoline analogue of primaquine which varies only on the presence of a 5-phenoxy group.[A35671, A35690] It was discovered by the scientists at the Walter Reed Army Institute of Research in 1978 as a substitute for primaquine that wou…

Kategori:
AminoquinolinesAnti-Infective AgentsAntimalarials +11
Waktu ParuhTafenoquine present…
Vol. DistribusiTafenoquine present…
KlirensTafenoquine present…
Genetik -
biotech

Deskripsi belum tersedia.

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TAK-428 DB05499
small molecule

TAK-428 is a drug for treating diabetic neuropathy. It is based on the novel concept that peripheral nervous tissue that was damaged by diabetes can be repaired and regenerated by stimulating an increase in neurotrophic factors.

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biotech | CAS: 308240-58-6

Talactoferrin alfa is a novel immunomodulatory 80 kD protein with demonstrated oral anti-tumor properties. Lactoferrin, a protein found in breast milk is developed by Agennix. It increases body’s immune power and also works as a natural antioxidant, helping t…

Kategori:
Amino Acids, Peptides, and ProteinsAnimal Proteins, DietaryAntineoplastic Agents +21
Waktu Paruh-
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Talbutal Approved DB00306
small molecule | CAS: 115-44-6

Talbutal, also called 5-allyl-5-sec-butylbarbituric acid, is a barbiturate with a short to intermediate duration of action. Talbutal is a schedule III drug in the U.S.

Kategori:
Anticholinergic AgentsBarbiturates, PlainCentral Nervous System Depressants +6
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-2Gamma-aminobutyric acid receptor subunit gamma-3Gamma-aminobutyric acid receptor subunit alpha-3 +9
Waktu Paruh-
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Tallimustine DB15466
small molecule | CAS: 115308-98-0

Tallimustine, a benzoyl mustard derivative of distamycin A, is an alkylating agent that binds to the minor groove of DNA.[A182036,A182039] It's association with severe myelotoxicity lead to the end of its development in favour of ?-halogenoacrylamide derivati…

Kategori:
Alkylating DrugsAmino Acids, Peptides, and ProteinsAntineoplastic Agents +6
Target Protein:
C-X-C chemokine receptor type 2DNA
Waktu Paruh-
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Talmapimod DB05412
small molecule | CAS: 309913-83-5

Talmapimod is the first-generation oral p38 MAP kinase inhibitor developed by Scios. It has shown to be effective to cure inflammatory diseases such as Rheumatoid Arthritis.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Mitogen-activated protein kinase 14Tumor necrosis factorInterleukin-1 beta +1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Talquetamab Approved DB16678
biotech | CAS: 2226212-40-2

Talquetamab is a IgG4-PAA bispecific G protein-coupled receptor class C group 5 member D (GPRC5D)-directed CD3 T-cell engager. It consists of two arms - anti-GPRC5D and anti-CD3 arms - linked by two interchain disulfide bonds, each arm comprising a heavy and …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntineoplastic Agents +7
Target Protein:
T-cell surface glycoprotein CD3G-protein coupled receptor family C group 5 member D
Waktu ParuhThe mean (CV%) term…
Vol. DistribusiThe geometric mean …
KlirensTalquetamab clearan…
Genetik -
Tandutinib DB05465
small molecule | CAS: 387867-13-2

MLN518 is a novel, oral, small molecule designed to inhibit type III receptor tyrosine kinases, including FLT3, (platelet-derived growth-factor receptor) PDGFR and c-KIT. Tyrosine kinases are enzymes involved in several cellular processes and are known to be …

Kategori:
Heterocyclic Compounds, Fused-RingPotential QTc-Prolonging AgentsQTc Prolonging Agents +1
Target Protein:
Receptor-type tyrosine-protein kinase FLT3Platelet-derived growth factor D
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Taniraleucel DB18311
biotech

Deskripsi belum tersedia.

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Tantalum DB12859
small molecule | CAS: 7440-25-7

Tantalum has been investigated for the treatment and prevention of Osteoarthritis, Knee Osteoarthritis, Intraoperative Bleeding, and Adolescent Idiopathic Scoliosis.

Kategori:
ElementsMetalsMetals, Heavy +1
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biotech | CAS: 2411896-53-0

Tarcocimab tedromer is under investigation in clinical trial NCT06270836 (A Study to Evaluate the Efficacy and Safety of Tarcocimab Tedromer Compared With Sham Treatment in Participants With Moderately Severe to Severe Non-proliferative Diabetic Retinopathy (…

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TAS-102 DB08937
small molecule | CAS: 733030-01-8

TAS-102 (Taiho Pharma USA, Inc.) is an anti-cancer drug under development and in stage 3 clinical trials for the treatment of colorectal cancer. It is composed of the thymidine phosphorylase inhibitor (TPI) tipiracil and the cytotoxin trifluridine. Trifluridi…

Kategori:
DeoxyribonucleosidesNucleic Acids, Nucleotides, and NucleosidesNucleosides +4
Waktu Paruh-
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TAS-106 DB06656
small molecule | CAS: 180300-43-0

TAS-106 is a new nucleoside antimetabolite. TAS-106 has demonstrated strong antitumor activity without serious toxicity in nude rat models bearing human tumours [A31693].

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleosidesPyrimidine Nucleosides +2
Target Protein:
DNA-directed RNA polymerase subunit betaDNA-directed RNA polymerase subunit beta'
Waktu Paruh-
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TAS-117 DB15054
small molecule | CAS: 1402602-94-1

TAS-117 is under investigation in clinical trial NCT03017521 (K-BASKET, TAS-117, PI3K/AKT Gene Aberration).

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
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Tasosartan DB01349
small molecule | CAS: 145733-36-4

Tasosartan is a long-acting angiotensin II (AngII) receptor blocker. Its long duration of action has been attributed to its active metabolite enoltasosartan. It is used to treat patients with essential hypertension.

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing hyperkalemiaAngiotensin II receptor blockers (ARBs), plain +4
Target Protein:
Type-1 angiotensin II receptorType-2 angiotensin II receptor
Waktu Paruh-
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Tauroursodeoxycholic acid Approved DB08834
small molecule | CAS: 14605-22-2

Tauroursodeoxycholic acid, also known as ursodoxicoltaurine, is a highly hydrophilic tertiary bile acid [A249070] that is produced in humans at a low concentration.[A249070] It is a taurine conjugate of [ursodeoxycholic acid] [A249065] with comparable therape…

Kategori:
Alimentary Tract and MetabolismBile acids and derivativesBile Acids and Salts +10
Target Protein:
Integrin alpha-5
Waktu Paruh-
Vol. DistribusiThere is evidence t…
Klirens-
Genetik -
biotech | CAS: 1971880-37-1

Tavokinogene telseplasmid consists of a DNA Plasmid Vector Encoding IL-12.

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Tazemetostat Approved DB12887
small molecule | CAS: 1403254-99-8

Tazemetostat is a methyltransferase inhibitor used to treat metastatic or locally advanced epithelioid sarcoma not eligible for complete resection.[L11476] Tazemetostat was first named in literature as EPZ-6438.[A190363] Tazemetaostat was granted FDA appro…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +16
Target Protein:
Histone-lysine N-methyltransferase EZH2Histone-lysine N-methyltransferase EZH1
Waktu ParuhTazemetostat has a …
Vol. DistribusiTazemetostat has a …
KlirensTazemetostat has an…
Genetik -
TBC-3711 DB05407
small molecule | CAS: 349453-49-2

TBC3711 is a next-generation endothelin antagonist that is being studied through oral and intravenous formulations by Encysive Pharmaceuticals.

Kategori:
Endothelin A Receptor AntagonistsEndothelin Receptor AntagonistsSulfur Compounds
Target Protein:
Endothelin-1 receptorEndothelin-1
Waktu Paruh-
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TC-6987 DB14854
small molecule | CAS: 1196701-27-5

TC-6987 is under investigation in clinical trial NCT01296087 (TC-6987 for the Treatment of Mild to Moderate Asthma).

Target Protein:
Neuronal acetylcholine receptor subunit alpha-7
Waktu Paruh-
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Teceleukin DB15389
biotech | CAS: 136279-32-8

Teceleukin is under investigation in clinical trial NCT03610490 (Autologous Tumor Infiltrating Lymphocytes MDA-TIL in Treating Patients With Recurrent or Refractory Ovarian Cancer, Osteosarcoma, or Pancreatic Ductal Adenocarcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAnalgesics, Non-Narcotic +12
Waktu Paruh-
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Technetium Tc-99m disofenin Approved DB09164
small molecule

Technetium Tc-99m disofenin is a radiopharmaceutical agent used in hepatobiliary imaging for diagnostic purposes. It is well suited for both planar and single photon tomographic scintigraphy to quantitatively measure the function of liver, gallbladder and bil…

Kategori:
Amino AcidsAmino Acids, CyclicAmino Acids, Peptides, and Proteins +15
Waktu ParuhTechnetium Tc99m de…
Vol. DistribusiTechnetium Tc99M di…
KlirensTechnetium Tc 99M D…
Genetik -
biotech

Technetium Tc-99m epratuzumab is under investigation in clinical trial NCT00003337 (Radiolabeled Monoclonal Antibody in the Detection and Staging of Patients With Non-Hodgkin's Lymphoma).

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small molecule | CAS: 23288-61-1

Technetium Tc-99m pertechnetate is a radiopharmaceutical diagnostic agent composed of an oxoanion with the chemical formula TcO4-. Pertechnetate has a wide variety of uses within nuclear medicine as it distributes within the body to a similar extent as iodine…

Kategori:
Compounds used in a research, industrial, or household settingDiagnostic RadiopharmaceuticalsDiagnostic Uses of Chemicals +7
Waktu Paruh-
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biotech

Technetium Tc-99m red blood cells is a radiopharmaceutical diagnostic agent that is intravenously administered to be used in blood pool imaging, including cardiac first pass and gated equilibrium imaging and for detection of sites of gastrointestinal bleeding…

Kategori:
Radioactive Diagnostic AgentRadiopharmaceutical Activity
Waktu ParuhTechnetium Tc 99m d…
Vol. DistribusiFollowing intraveno…
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Technetium Tc-99m sestamibi Approved DB09161
small molecule | CAS: 109581-73-9

Technetium Tc-99m sestamibi (commonly sestamibi) is a pharmaceutical agent used in nuclear medicine imaging. The drug is a coordination complex consisting of the radioisotope technetium-99m bound to six methoxyisobutylisonitrile (MIBI) ligands, hence the name…

Kategori:
Compounds used in a research, industrial, or household settingDiagnostic RadiopharmaceuticalsDiagnostic Uses of Chemicals +10
Waktu ParuhTechnetium Tc 99m d…
Vol. Distribusi-
KlirensThe effective half-…
Genetik -
small molecule

Technetium 99m sulfur colloid is a radiopharmaceutical diagnostic agent used in the evaluation of various conditions including lymph node metastases in breast cancer, detection of shunt patency, imaging of reticuloendothelial cells for assessment of liver fun…

Kategori:
Compounds used in a research, industrial, or household settingDiagnostic RadiopharmaceuticalsDiagnostic Uses of Chemicals +9
Waktu ParuhTechnetium Tc 99m d…
Vol. DistribusiFollowing oral inge…
Klirens-
Genetik -
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