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11778

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Halaman 47 / 236
ART5803 DB18379
biotech

ART5803 is a humanized one-armed monoclonal antibody with a high affinity for the NMDA receptor.

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Artemether Approved DB06697
small molecule | CAS: 71963-77-4

Artemether is an antimalarial agent used to treat acute uncomplicated malaria. It is administered in combination with lumefantrine for improved efficacy. This combination therapy exerts its effects against the erythrocytic stages of <i>Plasmodium spp.</i> and…

Kategori:
Anti-Infective AgentsAntimalarialsAntiparasitic Agents +25
Target Protein:
Sodium/potassium-transporting ATPase subunit alpha-1
Waktu ParuhArtemether, 1.6 +/-…
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Artemin DB15438
biotech | CAS: 309758-71-2

Artemin is under investigation in clinical trial NCT01842126 (Phase 1 Subcutaneous Single and Multiple Ascending Dose Study of BG00010 (Neublastin)).

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Artemisia absinthium pollen Approved DB10768
biotech

Artemisia absinthium pollen is the pollen of the Artemisia absinthium plant. Artemisia absinthium pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Pollen Allergenic Extract
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biotech

Deskripsi belum tersedia.

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Artemisia douglasiana pollen Approved DB10761
biotech

Artemisia douglasiana pollen is the pollen of the Artemisia douglasiana plant. Artemisia douglasiana pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Artemisia ludoviciana pollen Approved DB10762
biotech

Artemisia ludoviciana pollen is the pollen of the Artemisia ludoviciana plant. Artemisia ludoviciana pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Pollen Allergenic Extract
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Artemisia vulgaris pollen Approved DB10372
biotech

Artemisia vulgaris pollen is the pollen of the Artemisia vulgaris plant. Artemisia vulgaris pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Pollen Allergenic Extract
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Artemisia vulgaris root Approved DB14170
biotech

Artemisia vulgaris root allergenic extract is used in allergenic testing.

Kategori:
Non-Standardized Food Allergenic Extract
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Artemisone DB16097
small molecule | CAS: 255730-18-8

Artemisone is under investigation in clinical trial NCT00936767 (Artemisone for the Treatment of Uncomplicated Falciparum Malaria in Western Cambodia).

Kategori:
Free RadicalsPeroxidesReactive Oxygen Species +2
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Artemotil Approved DB13851
small molecule | CAS: 75887-54-6

Artemotil, also known as ?-arteether, is a semi-synthetic derivative of artemisinin and a fast acting blood schizonticide specifically indicated for the treatment of chloroquine-resistant _Plasmodium falciparum_ malaria and cerebral malaria cases.

Kategori:
AmebicidesAnti-Infective AgentsAntimalarials +11
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Artenimol Approved DB11638
small molecule | CAS: 71939-50-9

Artenimol is an artemisinin derivative and antimalarial agent used in the treatment of uncomplicated *Plasmodium falciparum* infections [FDA Label]. It was first authorized for market by the European Medicines Agency in October 2011 in combination with [DB139…

Kategori:
Anti-Infective AgentsAntimalarialsAntiparasitic Agents +16
Target Protein:
Actin, cytoplasmic 2Alpha-aminoadipic semialdehyde dehydrogenaseAnnexin A2 +188
Waktu ParuhArtenimol was repor…
Vol. DistribusiArtenimol was obser…
KlirensArtenimol was obser…
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Arterolane DB19027
small molecule | CAS: 664338-39-0

Arterolane is under investigation in clinical trial NCT03452475 (Comparison of Arterolane-piperaquine Versus Arterolane-piperaquine+mefloquine Versus Artemether-lumefantrine in Kenyan Children).

Kategori:
AnionsAntimalarialsAntiparasitic Products, Insecticides and Repellents +7
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Artesunate Approved DB09274
small molecule | CAS: 88495-63-0

Artesunate is indicated for the initial treatment of severe malaria.[L14099] The World Health Organization recommends artesunate as first line treatment for severe malaria.[L890] Artesunate was developed out of a need for a more hydrophilic derivative of [art…

Kategori:
Acids, AcyclicAnionsAnthelmintics +28
Target Protein:
Malaria protein EXP-1
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of ar…
Genetik -
Arundic acid DB05343
small molecule | CAS: 185517-21-9

Arundic acid has been investigated for the treatment of Amyotrophic Lateral Sclerosis (ALS).

Kategori:
Acids, AcyclicFatty AcidsLipids
Target Protein:
Beta-3 adrenergic receptorProtein S100-B
Waktu Paruh-
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Arylacenamide DB05792
small molecule | CAS: 132173-07-0

Arylacenamide (SR31747) is a peripheral [sigma] ligand that binds four proteins in human cells, i.e. SRBP-1, [sigma]-2, HSI and its relative SRBP-2. It is a dual agent with both immunomodulatory and antiproliferative activities.

Kategori:
CycloparaffinsEnzyme InhibitorsImmunologic Factors +1
Target Protein:
3-beta-hydroxysteroid-Delta(8),Delta(7)-isomeraseHCG20471, isoform CRA_c
Waktu Paruh-
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AS-8112 DB09207
small molecule

AS-8112 is a synthetic compound that acts as a selective antagonist at the dopamine receptor subtypes D2 and D3, and the serotonin receptor 5-HT3. It has been shown to exert potent antiemetic effects in animal studies and has been investigated for potential m…

Kategori:
Dopamine AgentsDopamine AntagonistsDopamine D2 Receptor Antagonists +1
Target Protein:
D(2) dopamine receptorD(3) dopamine receptor5HT3 serotonin receptor
Waktu Paruh-
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ASC-JM-17 DB16931
small molecule | CAS: 1039760-91-2

Deskripsi belum tersedia.

Kategori:
AlkanesBenzene DerivativesCatechols +4
Waktu Paruh-
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Asciminib Approved DB12597
small molecule | CAS: 1492952-76-7

Asciminib is a tyrosine kinase inhibitor (TKI) used in the treatment of chronic-phase Philadelphia chromosome-positive chronic myeloid leukemia (Ph+ CML). More specifically, it is an inhibitor of the ABL1 kinase activity of the BCR-ABL1 fusion protein[L38995]…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBcr-Abl Tyrosine Kinase Inhibitors +26
Target Protein:
Tyrosine-protein kinase ABL1
Waktu ParuhThe terminal elimin…
Vol. DistribusiAt steady-state, th…
KlirensThe total apparent …
Genetik -
Ascorbic acid Approved DB00126
small molecule | CAS: 50-81-7

A six carbon compound related to glucose. It is found naturally in citrus fruits and many vegetables. Ascorbic acid is an essential nutrient in human diets, and necessary to maintain connective tissue and bone. Its biologically active form, vitamin C, functio…

Kategori:
Acids, AcyclicAlimentary Tract and MetabolismAntioxidants +20
Target Protein:
Solute carrier family 23 member 2Solute carrier family 23 member 1Hyaluronate lyase +23
Waktu Paruh16 days (3.4 hours …
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small molecule | CAS: 129499-78-1

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicCarbohydratesHydroxy Acids +1
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Ascorbyl phosphate Approved DB11352
small molecule

Ascorbyl phosphate is a synthetic form of Vitamin C and is found in different salt forms such as magnesium ascorbyl phosphate and sodium ascorbyl phosphate. These salts are present in cosmetic products at concentrations ranging from 0.001 % to 3% [A27211]. As…

Kategori:
Acids, AcyclicCarbohydratesHydroxy Acids +3
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Asenapine Approved DB06216
small molecule | CAS: 65576-45-6

Developed by Schering-Plough after its merger with Organon International, asenapine is a sublingually administered, atypical antipsychotic for treatment of schizophrenia and acute mania associated with bipolar disorder. Asenapine also belongs to the dibenzo-o…

Kategori:
Acid ReducersAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +41
Target Protein:
5-hydroxytryptamine receptor 2AD(2) dopamine receptor5-hydroxytryptamine receptor 1A +17
Waktu Paruh24 hours (range of …
Vol. Distribusi20-25 L/kg
Klirens-
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ASF-1075 DB05727
small molecule

Deskripsi belum tersedia.

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Asfotase alfa Approved DB09105
biotech | CAS: 1174277-80-5

Asfotase alfa is a first-in-class bone-targeted enzyme replacement therapy designed to address the underlying cause of hypophosphatasia (HPP)—deficient alkaline phosphatase (ALP). Hypophosphatasia is almost always fatal when severe skeletal disease is obvious…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsAntibodies +16
Target Protein:
Pyrophosphate
Waktu ParuhApproximately 5 day…
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ASI402 DB06373
biotech | CAS: 372075-37-1

ASI402 is a monoclonal antibody that targets an aberrantly glycosylated antigen Mucin 1. It is being investigated in cancers.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Mucin-1
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ASN90 DB17927
small molecule

Deskripsi belum tersedia.

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Asoprisnil DB06680
small molecule | CAS: 199396-76-4

Asoprisnil (J867) is a selective progesterone receptor modulator. It can be used to treat progesterone sensitive myomata.

Kategori:
AminesEstranesFused-Ring Compounds +2
Target Protein:
Progesterone receptor
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ASP-2138 DB18473
biotech

ASP-2138 is a bispecific antibody directed against CLDN18.2 and T cell receptor complex CD3

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ASP-3026 DB12729
small molecule | CAS: 1097917-15-1

ASP3026 has been used in trials studying the treatment of Solid Tumor, B-Cell Lymphoma, Advanced Malignancies, Positive for Anaplastic Lymphoma Kinase, and Positive for Proto-Oncogene Tyrosine-Protein Kinase ROS.

Kategori:
Sulfur Compounds
Target Protein:
ALK tyrosine kinase receptor
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ASP-7317 DB18549
biotech

ASP-7317 consists of human embryonic stem cell-derived retinal pigment epithelium cells.

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ASP-8731 DB17696
small molecule | CAS: 2488255-42-9

ASP-8731 is a novel BACH1 inhibitor that potentially induces fetal hemoglobin (HbF). Developed by Mitobridge, it is being investigated for the treatment of sickle cell disease.[L46093]

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Aspacytarabine DB17226
small molecule | CAS: 2098942-53-9

Deskripsi belum tersedia.

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biotech | CAS: 1349719-22-7

Asparaginase _Erwinia chrysanthemi_ is an asparaginase-specific enzyme derived from _Erwinia_ _chrysanthemi_ used as an anticancer agent. It works by depleting the stores of an important amino acid called asparagine, which is involved in DNA synthesis and cel…

Kategori:
AmidohydrolasesAntineoplastic AgentsAsparaginase +7
Waktu ParuhThe apparent half-l…
Vol. DistribusiThe volume of distr…
KlirensThe geometric mean …
Genetik -
biotech | CAS: 9015-68-3

Asparaginase derived from _Escherichia coli_ (L-asparagine amidohydrolase, EC 3.5.1.1) is an enzyme responsible for the metabolism of L-asparagine, by catalyzing L-asparagine into L-aspartic acid and ammonia. It also facilitates the production of oxaloacetate…

Kategori:
AmidohydrolasesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +7
Target Protein:
L-asparagine
Waktu ParuhPlasma half life of…
Vol. DistribusiApparent volume of …
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Asparagine Approved DB00174
small molecule | CAS: 70-47-3

A non-essential amino acid that is involved in the metabolic control of cell functions in nerve and brain tissue. It is biosynthesized from aspartic acid and ammonia by asparagine synthetase. (From Concise Encyclopedia Biochemistry and Molecular Biology, 3rd …

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +5
Target Protein:
Sodium-coupled neutral amino acid transportersNeutral amino acid transporter B(0)Asparagine synthetase [glutamine-hydrolyzing] +3
Waktu Paruh-
Vol. Distribusi-
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Aspartame DB00168
small molecule | CAS: 22839-47-0

Flavoring agent sweeter than sugar, metabolized as phenylalanine and aspartic acid.

Kategori:
Amino Acids, Peptides, and ProteinsCompounds used in a research, industrial, or household settingDiet, Food, and Nutrition +13
Target Protein:
Taste receptor type 1 member 3Taste receptor type 1 member 2Transient receptor potential cation channel subfamily V member 1
Waktu ParuhAt room temperature…
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biotech

Deskripsi belum tersedia.

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Astaxanthin DB06543
small molecule | CAS: 472-61-7

Astaxanthin is a keto-carotenoid in the terpenes class of chemical compounds. It is classified as a xanthophyll but it is a carotenoid with no vitamin A activity. It is found in the majority of aquatic organisms with red pigment. Astaxanthin has shown to medi…

Kategori:
AlkenesAnticoagulantsBiological Factors +9
Target Protein:
NF-kappa-B inhibitor alpha
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Astegolimab DB16386
biotech | CAS: 2173054-79-8

Astegolimab is under investigation in clinical trial NCT04386616 (A Study to Evaluate the Safety and Efficacy of MSTT1041A (Astegolimab) or UTTR1147A in Patients With Severe COVID-19 Pneumonia).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAnti-Inflammatory Agents +10
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Astemizole Approved DB00637
small molecule | CAS: 68844-77-9

Astemizole is a long-acting, non-sedating second generation antihistamine used in the treatment of allergy symptoms. It was withdrawn from market by the manufacturer in 1999 due to the potential to cause arrhythmias at high doses, especially when when taken …

Kategori:
Anti-Allergic AgentsAntihistamines for Systemic UseBenzimidazoles +27
Target Protein:
Histamine H1 receptorVoltage-gated inwardly rectifying potassium channel KCNH2Voltage-gated delayed rectifier potassium channel KCNH1 +1
Waktu Paruh1 day
Vol. Distribusi-
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Astodrimer DB11854
biotech | CAS: 1379746-42-5

Astodrimer has been used in trials studying the treatment and prevention of Bacterial Vaginosis. It is a lysine-based dendrimer with naphthalene disulfonic acid surface groups.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +10
Target Protein:
Envelope glycoprotein gp160
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small molecule

Deskripsi belum tersedia.

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AstraZeneca COVID-19 Vaccine Approved DB15656
biotech | CAS: 2420395-83-9

The AstraZeneca COVID-19 Vaccine (previously known as ChAdOx1 nCoV-19 or AZD1222) is one of several vaccines developed in 2020 for the prevention of COVID-19 caused by SARS-CoV-2.[L12669,L32649] The ChAdOx1 viral vector was developed at the University of Oxfo…

Kategori:
Biological ProductsComplex MixturesCOVID-19 Vaccines +6
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ASTX-029 DB18900
small molecule | CAS: 2095719-92-7

ASTX-029 is under investigation in clinical trial NCT03520075 (Study of ASTX029 in Subjects With Advanced Solid Tumors).

Kategori:
Heterocyclic Compounds, Fused-Ring
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Asunaprevir Approved DB11586
small molecule | CAS: 630420-16-5

Asunaprevir, also named BMS-650032, is a potent hepatitis C virus (HCV) NS3 protease inhibitor. It has been shown to have a very high efficacy in dual-combination regimens with daclatasvir in patients chronically infected with HCV genotype 1b.[A32528] It was …

Kategori:
AmidesAntiinfectives for Systemic UseAntiviral Agents +35
Target Protein:
Gag-Pol polyproteinGenome polyprotein
Waktu ParuhClinical pharmacoki…
Vol. DistribusiThe registered volu…
KlirensClinical pharmacoki…
Genetik -
Asundexian DB19088
small molecule | CAS: 2064121-65-7

Asundexian is under investigation in clinical trial NCT05686070 (A Study to Test Asundexian for Preventing a Stroke Caused by a Clot in Participants After an Acute Ischemic Stroke or After a High-risk Transient Ischemic Attack, a So-called Mini Stroke).

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +2
Target Protein:
Coagulation factor XI
Waktu Paruh-
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Asvasiran DB05638
biotech | CAS: 870094-26-1

Asvasiran is an siRNA that targets the respiratory syncytial virus (RSV) N gene and inhibits viral replication. It has the potential to treat or prevent RSV infection.

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AT-001 DB15121
small molecule | CAS: 1355612-71-3

AT-001 is under investigation in clinical trial NCT03062384 (AT-001 for Long-term Preservation of Brain Health in Aging).

Kategori:
Heterocyclic Compounds, Fused-RingPyridinesThiazoles
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AT-301 DB16507
biotech

AT-301 was under investigation in clinical trial NCT01675284 to evaluate the safety, reactogenicity, and humoral immune responses to an inactivated H5N1 influenza vaccine

Kategori:
Experimental Unapproved Treatments for COVID-19
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