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11793

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Halaman 47 / 236
Auriclosene DB12197
small molecule | CAS: 846056-87-9

Auriclosene has been used in trials studying the treatment of Impetigo, Bacterial Conjunctivitis, Asymptomatic Bacteriuria, and Adenoviral Conjunctivitis.

Kategori:
AlkanesAlkanesulfonic AcidsHydrocarbons, Acyclic +3
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Aurothioglucose Approved DB09121
small molecule | CAS: 12192-57-3

Aurothioglucose, also known as gold thioglucose, was formerly used to treat rheumatoid arthritis. Contemporary research on the effect of gold salts treatment began in 1935, primarily to reduce inflammation and to slow disease progression in patients with r…

Kategori:
Antiinflammatory and Antirheumatic ProductsAntirheumatic AgentsDrugs that are Mainly Renally Excreted +5
Target Protein:
Adenylate cyclase type 1Adenylate cyclase type 2Adenylate cyclase type 5
Waktu ParuhThe biological half…
Vol. DistribusiReadily accessible …
KlirensWhen a standard wee…
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Aurothioglycanide Approved DB19361
small molecule | CAS: 16925-51-2

Deskripsi belum tersedia.

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Aurotioprol DB13763
small molecule | CAS: 27279-43-2

Deskripsi belum tersedia.

Kategori:
AlcoholsAntiinflammatory and Antirheumatic ProductsAntirheumatic Agents +5
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AUTO3 DB17364
biotech

AUTO3 is bicistronic chimeric antigen receptor T-cell therapy investigated for acute lymphoblastic leukemia (ALL). It is an investigational chimeric antigen receptor (CAR) T cell treatment targeting CD19 and CD22.

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biotech | CAS: 2365453-34-3

Autogene cevumeran is an mRNA-based cancer vaccine targeting an unspecified amount of tumour-associated antigens. It is being investigated for cancers.

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biotech

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biotech

Autologous CD34+ hematopoietic stem and progenitor cells expressing adenosine deaminase is an investigational lentiviral gene therapy. It comprises autologous CD34+ hematopoietic stem and progenitor cells (HSPCs) that had been genetically modified ex vivo wit…

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biotech

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biotech

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biotech

Autologous DNP-conjugated tumour vaccine, or melanoma vaccine, is an investigational autologous cell vaccine technology for melanoma.[A254806]

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biotech

Autologous hematopoietic peripheral blood stem cells were tested in a clinical trial (NCT00424489) by Northwestern University for the treatment of refractory myasthenia gravis.

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biotech

Autologous non-hematopoietic peripheral blood stem cells have been created into a formulation for use in a clinical trial (NCT04473170) by the Abu Dhabi Stem Cells Center. The cells have the characterizations of CD90+, CD133+, Oct-4+, CD45-, and CD71-.[L16363]

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biotech

Autologous peripheral blood-derived CD34+ cells, or CLBS119 (a proprietary version being developed by Caladrius Biosciences, Inc.), are hematopoietic stem cells.[L27741] It is also a cell therapy being investigated by Caladrius Biosciences in the clinical tri…

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AUY922 DB11881
small molecule | CAS: 747412-64-2

AUY922 has been used in trials studying the treatment of Lymphoma, Breast Cancer, Metastatic Disease, Advanced Solid Tumors, and Hematologic Neoplasms, among others.

Kategori:
Benzene DerivativesHSP90 Heat-Shock Proteins, antagonists & inhibitorsPhenols
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AV-0113 DB18386
biotech

AV-0113 consists of IL-12 secreting dendritic cells loaded with autologous tumor lysate.

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AV-412 DB06021
small molecule | CAS: 451493-31-5

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Epidermal growth factor receptorReceptor tyrosine-protein kinase erbB-2
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AV-COVID-19 DB15802
biotech

AV-COVID-19 is a vaccine composed of autologous dendritic cells loaded with SARS-CoV-2 antigens and with or without Granulocyte-macrophage colony-stimulating factor (GM-CSF). The vaccine is created from the receiving patients’ isolated peripheral blood mon…

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AV608 DB05072
small molecule

AV608 is a NK-1 antagonist. It is developed for the treatment of Social anxiety disorder (SAD), irritable bowel syndrome (IBS) and overactive bladder (OAB).

Target Protein:
Substance-P receptor
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AVA-4746 DB18022
small molecule | CAS: 422268-99-3

Deskripsi belum tersedia.

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AVA-6000 DB17398
small molecule | CAS: 1841402-73-0

Deskripsi belum tersedia.

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Avacincaptad pegol Approved DB15165
biotech | CAS: 1613641-69-2

Avacincaptad pegol is an RNA aptamer covalently bound to a branched polyethylene glycol (PEG) molecule. It was developed to treat an advanced form of age-related macular degeneration (AMD) called geographic atrophy (GA).[L47696] AMD is the leading cause of vi…

Kategori:
Aptamers, NucleotideComplement Inactivating AgentsComplement Inactivator Proteins
Target Protein:
Complement C5
Waktu ParuhThe estimated appar…
Vol. DistribusiLimited information…
KlirensLimited information…
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Avacopan Approved DB15011
small molecule | CAS: 1346623-17-3

Anti-neutrophil cytoplasmic (auto)antibody (ANCA)-associated vasculitis (AAV) is a rare (estimated incidence of 3 cases per 100,000 per year) form of "pauci-immune" systemic small-vessel vasculitis typified by the presence of ANCAs in the serum.[A240249, A240…

Kategori:
AminesAntineoplastic and Immunomodulating AgentsComplement 5a Receptor Antagonist +22
Target Protein:
C5a anaphylatoxin chemotactic receptor 1
Waktu ParuhA single 30 mg dose…
Vol. DistribusiAvacopan has an app…
KlirensAvacopan has an est…
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Avadomide DB14857
small molecule | CAS: 1015474-32-4

Avadomide is under investigation in clinical trial NCT02031419 (Novel Combinations of CC-122, CC-223, CC-292, and Rituximab in Diffuse Large B-cell Lymphoma and Follicular Lymphoma).

Kategori:
Heterocyclic Compounds, Fused-RingPiperidinesQuinazolines
Target Protein:
Protein cereblon
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Avagacestat DB11893
small molecule | CAS: 1146699-66-2

Avagacestat has been investigated for the basic science and treatment of Alzheimer Disease.

Kategori:
AmidesAmyloid Precursor Protein Secretases, antagonists & inhibitorsEnzyme Inhibitors +4
Target Protein:
Gamma-secretase subunit APH-1ANicastrinGamma-secretase subunit APH-1B +2
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Avalglucosidase alfa Approved DB16099
biotech | CAS: 1802558-87-7

Avalglucosidase alfa, or NeoGAA, is a drug for enzyme replacement therapy specifically designed for Pompe disease, a rare inherited neuromuscular disorder caused by the deficiency of the alpha-glucosidase (GAA) enzyme. GAA is an essential enzyme that hydrolyz…

Kategori:
Alimentary Tract and MetabolismEnzyme Replacement TherapyEnzymes +2
Target Protein:
Cation-independent mannose-6-phosphate receptor
Waktu ParuhThe mean avalglucos…
Vol. DistribusiThe volume of distr…
KlirensThe mean avalglucos…
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biotech | CAS: 2227000-30-6

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
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Avanafil Approved DB06237
small molecule | CAS: 330784-47-9

Avanafil is a phosphodiesterase-5 (PDE5) inhibitor used in the treatment of erectile dysfunction. In comparison with other drugs of the same class, it shows greater selectivity for PDE5 over PDE6 than both [sildenafil] and [vardenafil] but less selectivity th…

Kategori:
BCRP/ABCG2 InhibitorsCytochrome P-450 CYP2C9 SubstratesCytochrome P-450 CYP3A Substrates +9
Target Protein:
cGMP-specific 3',5'-cyclic phosphodiesterase
Waktu ParuhStudies have demons…
Vol. DistribusiThe apparent volume…
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Avapritinib Approved DB15233
small molecule | CAS: 1703793-34-3

Avapritinib, or BLU-285,[A189327] is a selective tyrosine kinase inhibitor of KIT and platelet derived growth factor receptor alpha indicated for the treatment of unresectable, metastatic gastrointestinal stromal tumors and advanced systemic mastocytosis.[A18…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +17
Target Protein:
Platelet-derived growth factor receptor alphaMast/stem cell growth factor receptor Kit
Waktu ParuhThe half life of av…
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent o…
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Avasimibe DB06442
small molecule | CAS: 166518-60-1

Deskripsi belum tersedia.

Kategori:
AcetatesAcids, AcyclicAmides +14
Target Protein:
Liver carboxylesterase 1
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Avasopasem DB18481
small molecule

Deskripsi belum tersedia.

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small molecule | CAS: 435327-40-5

Avasopasem manganese, also known as GC4419, is a highly-selective small molecule mimetic of superoxide dismutase (SOD) being investigated for the reduction of radiation-induced severe oral mucositis.[L27246, L27256] This drug has potential application for rad…

Kategori:
AntioxidantsFree Radical Scavengers
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Avatrombopag Approved DB11995
small molecule | CAS: 570406-98-3

Avatrombopag (_Doptelet_), is an orally administered, small molecule thrombopoietin receptor (c-Mpl) agonist that increases platelet number without increasing platelet activation,[A33097,L2824] thereby decreasing the need for blood transfusions.[L2824] Patien…

Kategori:
BCRP/ABCG2 InhibitorsBlood and Blood Forming OrgansCytochrome P-450 CYP2C8 Inducers +14
Target Protein:
Thrombopoietin receptor
Waktu ParuhThe mean plasma eli…
Vol. DistribusiAvatrombopag has an…
KlirensThe mean (%CV) of t…
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AVB-101 DB18416
biotech

AVB-101 is a recombinant AAV9 vector encoding the human progranulin (PGRN) gene.

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Avdoralimab DB16392
biotech | CAS: 2226393-85-5

Avdoralimab is under investigation in clinical trial NCT04333914 (Prospective Study in Patients With Advanced or Metastatic Cancer and Sars-cov-2 Infection).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAnti-Inflammatory Agents +9
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AVE-2865 DB07396
small molecule | CAS: 648917-13-9

Deskripsi belum tersedia.

Target Protein:
Glycogen phosphorylase, liver form
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AVE9633 DB06318
biotech

AVE9633 is an anti-CD33 monoclonal antibody-DM4 conjugate.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAntibodies +14
Target Protein:
Myeloid cell surface antigen CD33
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Avelumab Approved DB11945
biotech | CAS: 1537032-82-8

Avelumab is a human IgG1 lambda monoclonal antibody that binds programmed cell death ligand-1 (PD-L1) to block its interaction with its receptors found on T cells and antigen-presenting cells.[A261496] Avelumab was first approved by the FDA on March 23, 2017.…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +19
Target Protein:
Programmed cell death 1 ligand 1
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe geometric mean …
KlirensThe total systemic …
Genetik -
Avenciguat DB18882
small molecule | CAS: 1579514-06-9

Avenciguat is under investigation in clinical trial NCT05282121 (A Study to Test Whether BI 685509 Alone or in Combination With Empagliflozin Helps People With Liver Cirrhosis Caused by Viral Hepatitis or Non-alcoholic Steatohepatitis (NASH) Who Have High Blo…

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Avexitide DB14806
small molecule | CAS: 133514-43-9

Avexitide is under investigation in clinical trial NCT02996812 (Evaluation of Single Ascending Doses of Subcutaneous Exendin 9-39 in Patients With Post-Bariatric Hypoglycemia).

Kategori:
Amino Acids, Peptides, and ProteinsGlucagon-Like Peptide 1Peptides
Target Protein:
Glucagon-like peptide 1 receptor
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AVI-014 DB17086
biotech

AVI-014 is a glycosylated, recombinant human granulocyte colony-stimulating factor (G-CSF).

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AVI-4065 DB05620
small molecule

AVI-4065, a phosphorodiamidate Morpholino oligomer (PMO), is an investigational antisense HCV drug. It was developed by Sarepta Therapeutics, Inc. After phase II trials it was cancelled due to lack of potency. [L2917]

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AVI-5126 DB05726
small molecule

AVI-526 is an improved formulation of [AVI-4557], developed for use on Vein Grafts before use in Heart by-Pass Graft Surgery. AVI-526 works by silencing a gene known as c-myc, a key regulatory gene involved in cardiovascular restenosis. The drug was under inv…

Kategori:
MorpholinesNucleic Acids, Nucleotides, and NucleosidesNucleotides +3
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AVI-7537 DB15433
biotech

AVI-7537 is an antisense molecule that binds to the Ebola virus mRNA to prevent the viral replication.[L46207] AVI-7537 is under investigation in clinical trial NCT01593072 (A Study to Assess the Safety, Tolerability and Pharmacokinetics of AVI-7537 in Health…

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Avibactam Approved DB09060
small molecule | CAS: 1192500-31-4

Avibactam is a non-?-lactam ?-lactamase inhibitor that is available in combination with ceftazidime (Avycaz). This combination was approved by the FDA on February 25, 2015 for the treatment of complicated intra-abdominal infections in combination with metroni…

Kategori:
Anti-Infective AgentsAza Compoundsbeta-Lactamase Inhibitors +2
Target Protein:
Beta-lactamase TEMBeta-lactamase CTX-MBeta-lactamase +7
Waktu ParuhCeftazidime-avibact…
Vol. DistribusiThe steady state vo…
KlirensAvibactam and cefta…
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AVID-200 DB18454
biotech | CAS: 2269485-28-9

AVID-200 is an Anti-transforming growth factor beta (TGF-?) trap fusion protein.

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Avidin DB15228
biotech | CAS: 110539-97-4

Avidin is under investigation in clinical trial NCT00345618 (Clinical Study Assessing Idrabiotaparinux Sodium Injections Once-weekly in Pulmonary Embolism Therapeutic Approach).

Kategori:
AlbuminsAmino Acids, Peptides, and ProteinsAnimal Proteins, Dietary +10
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Aviptadil DB06260
small molecule | CAS: 40077-57-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsErectile DysfunctionGastrointestinal Hormones +9
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Aviscumine DB12684
biotech | CAS: 223577-45-5

Cy 503 is under investigation in clinical trial NCT00658437 (Aviscumine for the Treatment of Malignant Melanoma Stage IV After Failure of Prior Therapy).

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsBiological Factors +12
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Avizakimab DB18842
biotech | CAS: 2229685-51-0

Avizakimab is under investigation in clinical trial NCT03371251 (Study of BOS161721 in Systemic Lupus Erythematosus (SLE) Patients on a Background of Limited Standard of Care).

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