Hasil Filter

14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (14063)

Halaman 46 / 282
small molecule | CAS: 41325-63-7

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Genetik -
small molecule | CAS: 88847-89-6

Deskripsi belum tersedia.

Kategori:
Adjuvants, ImmunologicDeoxyguanosineDeoxyribonucleosides +7
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small molecule

Deskripsi belum tersedia.

Target Protein:
P-proteinChorismate mutase AroHSecreted chorismate mutase
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small molecule

Deskripsi belum tersedia.

Target Protein:
Thiostrepton50S ribosomal protein L11
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8-iodo-guanine DB02985
small molecule

Deskripsi belum tersedia.

Target Protein:
Purine nucleoside phosphorylasePurine nucleoside phosphorylase
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small molecule

Deskripsi belum tersedia.

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8-oxo-dGMP DB02023
small molecule | CAS: 127027-50-3

Deskripsi belum tersedia.

Kategori:
Guanine NucleotidesHeterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and Nucleosides +4
Target Protein:
8-oxo-dGTP diphosphatase
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9(S)-HODE DB07302
small molecule | CAS: 73543-67-6

Deskripsi belum tersedia.

Target Protein:
Peroxisome proliferator-activated receptor gamma
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small molecule | CAS: 78111-17-8

A specific inhibitor of phosphoserine/threonine protein phosphatase 1 and 2a. It is also a potent tumor promoter. (Thromb Res 1992;67(4):345-54 & Cancer Res 1993;53(2):239-41)

Target Protein:
Dual specificity protein phosphatase 1Serine/threonine-protein phosphatase PP1-gamma catalytic subunit
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small molecule

Deskripsi belum tersedia.

Target Protein:
Immunoglobulin heavy constant gamma 1
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small molecule

Deskripsi belum tersedia.

Target Protein:
Purine nucleoside phosphorylase DeoD-type
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small molecule

Deskripsi belum tersedia.

Kategori:
Cholinesterase Inhibitors
Target Protein:
Cholinesterase
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small molecule

9-(4-hydroxybutyl)-N2-phenylguanine is a solid. This compound belongs to the hypoxanthines. These are compounds containing the purine derivative 1H-purin-6(9H)-one. 9-(4-hydroxybutyl)-n2-phenylguanine is known to target thymidine kinase.

Target Protein:
Thymidine kinase, cytosolicThymidine kinase
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small molecule

Deskripsi belum tersedia.

Target Protein:
Mitogen-activated protein kinase 10
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Purine nucleoside phosphorylase
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Purine nucleoside phosphorylase DeoD-type
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Purine nucleoside phosphorylase DeoD-type
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small molecule | CAS: 143205-42-9

9-(N-methyl-L-isoleucine)-cyclosporin A (NIM811) has been used in trials studying the treatment of Chronic Hepatitis C Genotype-1 Relapse.

Kategori:
Amino Acids, Peptides, and ProteinsCyclosporinsImmunosuppressive Agents +2
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small molecule

Deskripsi belum tersedia.

Target Protein:
CREB-binding protein
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small molecule

Deskripsi belum tersedia.

Target Protein:
Neuraminidase
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small molecule

9-amino-n-[3-(dimethylamino)propyl]acridine-4-carboxamide is an inactive derivative of the antitumour agents N-[2-(dimethylamino)ethyl]acridine-4-carboxamide (DACA) and 9-amino-DACA.

Target Protein:
DNA
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small molecule | CAS: 91421-43-1

Aminocamptothecin has been used in trials studying the treatment of Lymphoma, Gastric Cancer, Ovarian Cancer, Esophageal Cancer, and Ovarian Neoplasms, among others.

Kategori:
AlkaloidsAntineoplastic AgentsCytochrome P-450 CYP3A Substrates +3
Target Protein:
DNA topoisomerase 1
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Genetik -
small molecule

Deskripsi belum tersedia.

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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Purine nucleoside phosphorylase DeoD-type
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Heat shock protein HSP 90-alpha
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Heat shock protein HSP 90-alpha
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Heat shock protein HSP 90-alpha
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small molecule

Deskripsi belum tersedia.

Target Protein:
Heat shock protein HSP 90-alphaHeat shock protein HSP 90-beta
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small molecule

Deskripsi belum tersedia.

Target Protein:
Cathepsin K
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9-deazainosine DB02796
small molecule | CAS: 89458-19-5

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and NucleosidesNucleosides +3
Target Protein:
Purine nucleoside phosphorylase
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Purine nucleoside phosphorylase
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Wee1-like protein kinase
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Group IIE secretory phospholipase A2
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small molecule

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9-Methylguanine DB02489
small molecule | CAS: 5502-78-3

Deskripsi belum tersedia.

Kategori:
Cytochrome P-450 CYP1A2 SubstratesCytochrome P-450 SubstratesHeterocyclic Compounds, Fused-Ring +3
Target Protein:
Dihydroneopterin aldolase
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small molecule

Deskripsi belum tersedia.

Kategori:
Cholinesterase Inhibitors
Target Protein:
Cholinesterase
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9CUAB30 DB12316
small molecule | CAS: 205252-57-9

9 Cuab30 has been used in trials studying the treatment and prevention of HER2/Neu Positive, HER2/Neu Negative, No Evidence of Disease, Estrogen Receptor Negative, and estrogen receptor positive, among others.

Kategori:
Fatty AcidsLipids
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small molecule | CAS: 101860-00-8

?-Methylacetylfentanyl is an analog of fentanyl with opioid analgesic properties. It was categorized under the Schedule I in the US and it was illegally sold in early 1980. ?-Methylacetylfentanyl synthesis process is very similar to ?-methylfentanyl with the …

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?A?–Gas6 DB17069
biotech

?A?–Gas6 is a chimeric fusion protein being investigated in preclinical studies as an immunotherapeutic agent for Alzheimer's disease (AD). It is made of a single chain variable fragment (scFv) of an Amyloid ? (A?)-targeting monoclonal antibody fused with a t…

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small molecule

Deskripsi belum tersedia.

Target Protein:
Stromelysin-1
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A-16L DB18270
biotech | CAS: 410527-75-2

Deskripsi belum tersedia.

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A-620223 DB07330
small molecule | CAS: 272769-49-0

Deskripsi belum tersedia.

Target Protein:
Poly [ADP-ribose] polymerase 1
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A-674563 DB08568
small molecule | CAS: 552325-73-2

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingPyrazoles
Target Protein:
RAC-alpha serine/threonine-protein kinasecAMP-dependent protein kinase catalytic subunit alphacAMP-dependent protein kinase inhibitor alpha
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A-98881 DB02804
small molecule

Deskripsi belum tersedia.

Target Protein:
Gag-Pol polyprotein
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biotech | CAS: 1470038-56-2

A-dmDT390-bisFv(UCHT1) is under investigation in clinical trial NCT02943642 (Safety and Effectiveness of A-dmdt390-bisfv(ucht1) Fusion Protein in Subjects With Mycosis Fungoides).

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A166 DB17413
biotech

A166 is an antibody-drug conjugate composed of a novel cytotoxic drug (Duo-5, anti-microtubule agent) site-specifically conjugated to an anti-HER2 antibody (trastuzumab) via a stable protease-cleavable valine citrulline linker.

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AAG-1 DB17199
small molecule | CAS: 1204408-18-3

Deskripsi belum tersedia.

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AAV-AQP1 DB17417
biotech

Deskripsi belum tersedia.

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AAV1-FS344 DB17855
biotech

AAV1-FS344 is an investigational gene therapy developed by Milo Biotechnology to deliver follistatin, a potent myostatin inhibitor. It is being investigated for the treatment of Duchenne Muscular Dystrophy, Becker Muscular Dystrophy, and inclusion body myosit…

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biotech

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