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15718

Total database: 17430
Struktur (SMILES)
10762 (68.5%)
Target
7957 (50.6%)
Genomik
112 (0.7%)
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15718 (100.0%)

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Halaman 46 / 315
ADL 10-0101 DB05443
small molecule

ADL 10-0101 is a peripheral kappa opioid agonist analgesic product candidate. Preclinical trials of ADL 10-0101 have suggested that the compound may be effective for the treatment of inflammatory pain, itch and visceral pain. Because ADL 10-0101 does not cros…

Target Protein:
Kappa-type opioid receptor
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ADL-5859 DB18910
small molecule | CAS: 850305-06-5

ADL-5859 is under investigation in clinical trial NCT00626275 (Study Evaluating the Analgesic Efficacy and Safety of ADL5859 in Participants With Rheumatoid Arthritis).

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +4
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biotech | CAS: 2143579-02-4

Adlinacogene civaparvovec is an investigational _in vivo_ genome editing therapeutic product. It uses proprietary zinc finger nuclease (ZFN) genome editing to insert into the DNA of liver cells a copy of the F9 gene, which controls the production of Factor IX…

Kategori:
Adeno-associated Viral Vector Therapies
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Adomeglivant DB11704
small molecule | CAS: 1488363-78-5

Adomeglivant has been investigated for the basic science of Type 2 Diabetes.

Kategori:
Benzene Derivatives
Target Protein:
Glucagon receptor
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ADP-597 DB12084
small molecule | CAS: 897732-93-3

JNJ-38431055 has been used in trials studying the treatment of Diabetes Mellitus, Type 2.

Target Protein:
Glucose-dependent insulinotropic receptor
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AdPEDF DB05138
biotech

AdPEDF is under development for the treatment of wet age-related macular degeneration (AMD). It has been shown to rapidly elevate the intraocular AdPEDF protein levels in the eye, inhibit abnormal blood vessel growth, and cause abnormal blood vessels to regre…

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Adrabetadex DB15146
small molecule | CAS: 128446-35-5

Adrabetadex is under investigation in clinical trial NCT03887533 (Combined Intrathecal and Intravenous VTS-270 Therapy for Liver and Neurological Disease Associated With Niemann-Pick Disease, Type C1).

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Adrafinil DB08925
small molecule | CAS: 63547-13-7

Adrafinil is a mild central nervous system stimulating drug typically employed to relieve excessive sleepiness and inattention in geriatric patients. It is also been used off-label to prevent fatigue or falling asleep for extended periods of time. Adrafinil d…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-Agonists +10
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Adrenalone DB13394
small molecule | CAS: 99-45-6

Deskripsi belum tersedia.

Kategori:
AlcoholsAlimentary Tract and MetabolismAmines +16
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Adrenomedullin DB19102
biotech | CAS: 154835-90-2

Adrenomedullin is under investigation in clinical trial NCT06072118 (Adrenomedullin for CADASIL).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Asthmatic AgentsAntihypertensive Agents +13
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Adriforant DB15027
small molecule | CAS: 943057-12-3

Adriforant is under investigation in clinical trial NCT00992342 (A Phase 1 Study To Evaluate The Safety And Tolerability Of Different Doses Of PF-03893787 In Healthy Adult Volunteers).

Target Protein:
Histamine H4 receptor
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ADU-S100 DB14722
small molecule | CAS: 1638241-89-0

ADU-S100 (MIW815) is a synthetic cyclic dinucleotide (CDN) agonist (activator) of Stimulator of Interferon Genes (STING), a receptor crucial to activate the innate (endogenous) immune system. ADU-S100 (MIW815) activates all known human and mouse STINGs, and e…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotides
Target Protein:
Stimulator of interferon genes protein
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Aducanumab Approved DB12274
biotech | CAS: 1384260-65-4

Aducanumab, or BIIB037, is a monoclonal IgG1 antibody that targets extracellular amyloid-? plaques in the brain; similar to [gantenerumab], [bapineuzumab] and [solanezumab].[A235668,A235730] Aducanumab is a recombinant antibody derived from patients with slow…

Kategori:
Alzheimer Disease, drug therapyAmino Acids, Peptides, and ProteinsAmyloid Beta-directed Antibodies +11
Target Protein:
Amyloid-beta precursor protein
Waktu ParuhThe terminal half l…
Vol. DistribusiThe volume of distr…
KlirensA 10 mg/kg intraven…
Genetik -
ADVM-053 DB17592
biotech

Deskripsi belum tersedia.

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ADVM-062 DB18341
biotech

ADVM-062 is an adeno-associated virus vector carrying complementary deoxyribonucleic acid encoding the human long-wave-sensitive opsin 1 (AAV.7m8-L-opsin)

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ADX-10061 DB05419
small molecule | CAS: 128022-68-4

ADX10061 is a potent, selective antagonist of the dopamine D1 receptor. It is developed by Addex Pharmaceuticals for the treatment of nicotine dependence.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Neuron-specific vesicular protein calcyon
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ADX10059 DB05070
small molecule

ADX10059 is a metabotropic glutamate receptor 5 (mGluR5) negative allosteric modulator (NAM). The orally available small molecule drug candidate, which is highly specific for mGluR5, was discovered at Addex in 2003. It is developed for the treatment of GERD,…

Target Protein:
Metabotropic glutamate receptor 5
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ADXS-31164 DB17325
biotech

Deskripsi belum tersedia.

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Adze-1.17-CD40L DB18528
biotech

Deskripsi belum tersedia.

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Aedes taeniorhynchus Approved DB10691
biotech

Aedes taeniorhynchus allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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AEE-788 DB12558
small molecule | CAS: 497839-62-0

AEE788 has been used in trials studying the treatment of Cancer, Glioblastoma Multiforme, and Brain and Central Nervous System Tumors.

Kategori:
Heterocyclic Compounds, Fused-RingReceptors, Vascular Endothelial Growth Factor, antagonists & inhibitors
Target Protein:
Fibroblast growth factor receptor 2Fibroblast growth factor receptor 3
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AEG35156 DB06184
small molecule

A second-generation synthetic antisense oligonucleotide with potential antineoplastic activity. AEG35156 selectively blocks the cellular expression of X-linked inhibitor of apoptosis protein (XIAP), a pivotal inhibitor of apoptosis that is overexpressed in ma…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Target Protein:
E3 ubiquitin-protein ligase XIAP
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AEM-28 DB17642
biotech

AEM-28 is a 28 amino acid mimetic of apolipoprotein E being investigated for lipid disorders, such as homozygous familial hypercholesterolemia. It possesses anti-inflammatory properties.[A258764]

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AEM-28-14 DB17643
biotech

AEM-28-14 is an analog of [AEM-28], an apolipoprotein E mimetic peptide, with a 400 percent greater cholesterol-lowering efficacy and a several-fold increase in drug tolerability.[L45909] It is being investigated for lipid disorders such as homozygous familia…

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AEOL-10150 DB05874
small molecule | CAS: 286475-30-7

AEOL 10150 is developed by Aeolus as a therapeutic agents based on its proprietary small molecule catalytic antioxidants.

Kategori:
AntioxidantsBiological FactorsCoordination Complexes +3
Target Protein:
Superoxide dismutase [Cu-Zn]
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AER001 DB05078
small molecule

AER001, an IL4/13 receptor antagonist for severe asthma and eczema currently in Phase 2 studies.

Target Protein:
Interleukin-4 receptor subunit alphaInterleukin-13 receptor subunit alpha-2
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small molecule

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Target Protein:
Serine protease 1
Waktu Paruh-
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AF-710B DB16911
small molecule | CAS: 1235733-73-9

Deskripsi belum tersedia.

Kategori:
Sulfur CompoundsThiazoles
Target Protein:
Muscarinic acetylcholine receptor M1Sigma non-opioid intracellular receptor 1
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Afabicin DB15268
small molecule | CAS: 1518800-35-5

Afabicin is under investigation in clinical trial NCT03723551 (Study to Assess Safety, Tolerability and Efficacy of Afabicin in The Treatment of Participants With Bone or Joint Infection Due to Staphylococcus).

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsHeterocyclic Compounds, Fused-Ring
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Afamelanotide Approved DB04931
small molecule | CAS: 75921-69-6

Afamelanotide is a first-in-class, synthetic, 13-amino acid peptide analogue of the endogenous alpha melanocyte-stimulating hormone (?-MSH).[L9086] It differs structurally from its endogenous counterpart by only two amino acids - these structural differences …

Kategori:
Amino Acids, Peptides, and ProteinsCompounds used in a research, industrial, or household settingDermatologicals +11
Target Protein:
Melanocortin receptor 4Melanocyte-stimulating hormone receptor
Waktu ParuhThe half-life of af…
Vol. DistribusiThe apparent volume…
KlirensData regarding plas…
Genetik -
Afamitresgene autoleucel Approved DB18592
biotech

Afamitresgene autoleucel is a melanoma-associated antigen A4 (MAGE-A4)-directed genetically modified autologous T cell immunotherapy product consisting of CD4 and CD8 positive T cells transduced with a self-inactivating lentiviral vector (LV) expressing an af…

Kategori:
Autologous Cellular Immunotherapy
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Afasevikumab DB14798
biotech | CAS: 1589503-30-9

Afasevikumab is under investigation in clinical trial NCT01480310 (Study to Investigate the Safety, Pharmacokinetics, and Immunogenicity of Subcutaneous MCAF5352A in Healthy Volunteers).

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Afatinib Approved DB08916
small molecule | CAS: 850140-72-6

Afatinib is a 4-anilinoquinazoline tyrosine kinase inhibitor in the form of a dimaleate salt available as Boehringer Ingelheim's brand name Gilotrif [FDA Label]. For oral use, afatinib tablets are a first-line (initial) treatment for patients with metastatic …

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +11
Target Protein:
Epidermal growth factor receptorReceptor tyrosine-protein kinase erbB-2Receptor tyrosine-protein kinase erbB-4
Gen Terkait:
EGFR EGFR EGFR
Waktu ParuhAfatinib is elimina…
Vol. DistribusiThe volume of distr…
KlirensThe apparent total …
Genetik 3 Varian
Afegostat DB04545
small molecule | CAS: 169105-89-9

Deskripsi belum tersedia.

Kategori:
CarbohydratesGlycoside Hydrolases, antagonists & inhibitorsImines +2
Target Protein:
Lysosomal acid glucosylceramidaseEndoglucanase 5ABeta-glucosidase A +1
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Afelimomab DB04956
biotech | CAS: 156227-98-4

Afelimomab (also known as Fab 2 or MAK 195F) is an anti-TNF-? monoclonal antibody. Administration of 195F reduces the concentration of interleukin-6 in patients with sepsis.

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAntibodies +11
Target Protein:
Tumor necrosis factor
Waktu Paruh44.7 hours
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Affitope AD01 DB06086
biotech

Affitope AD01 is an investigational drug developed for immunization to treat Alzheimer's Disease. AD01 is a short peptide (7 amino acids in length) that induces Aß-targeting antibodies, therefore lowering Aß aggregates.

Target Protein:
Amyloid-beta precursor protein
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Aficamten DB18490
small molecule | CAS: 2364554-48-1

Deskripsi belum tersedia.

Target Protein:
Myosin-binding protein C, cardiac-type
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Afimetoran DB16580
small molecule | CAS: 2171019-55-7

Afimetoran is an immunomodulator and an antagonist of toll-like receptors 7 and 8.[L32018, L32023] It is also is under investigation in clinical trial NCT04269356 (Study to Assess the Way the Body Absorbs, Distributes, Breaks Down and Eliminates Radioactive B…

Target Protein:
Toll-like receptor 7Toll-like receptor 8
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Aflibercept Approved DB08885
biotech | CAS: 862111-32-8

Aflibercept is a recombinant protein composed of the binding domains of two human vascular endothelial growth factor (VEGF) receptors, VEGFR1 and VEGFR2, fused with the Fc region of human immunoglobulin gamma 1 (IgG1).[A261130] Structurally, Aflibercept is a …

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +16
Target Protein:
Vascular endothelial growth factor A, long formPlacenta growth factorVascular endothelial growth factor B
Waktu ParuhFor the intravitrea…
Vol. DistribusiThe volume of distr…
KlirensFollowing an hour o…
Genetik -
AFM-13 DB17404
biotech

Deskripsi belum tersedia.

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AFN-1252 DB12658
small molecule | CAS: 620175-39-5

AFN-1252 has been used in trials studying the treatment of Cellulitis, Burn Infection, Wound Infection, Cutaneous Abscess, and Skin and Subcutaneous Tissue Bacterial Infections.

Kategori:
Heterocyclic Compounds, Fused-RingPyrans
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Afoxolaner DB11369
small molecule | CAS: 1093861-60-9

Deskripsi belum tersedia.

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Afuresertib DB11648
small molecule | CAS: 1047644-62-1

Afuresertib has been used in trials studying the treatment of Cancer and Neoplasms, Haematologic.

Kategori:
AminesPolyaminesSulfur Compounds
Target Protein:
RAC-alpha serine/threonine-protein kinase
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AG-24322 DB13035
small molecule | CAS: 837364-57-5

AG-024322 has been used in trials studying the treatment of Neoplasms and Lymphoma, Non-Hodgkin.

Kategori:
CDC2 Protein Kinase, antagonists & inhibitorsCyclin-Dependent Kinase 2, antagonists & inhibitorsHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Cyclin-dependent kinase 2Cyclin-dependent kinase 4Cyclin-dependent kinase 1
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AG0301-COVID19 DB15856
biotech

AG0301-COVID19 is a vaccine candidate developed by AnGes Inc. and Osaka University. The candidate is a plasmid DNA vaccine developed using an intradermal gene transfer method targeting the SARS-CoV-2 spike protein. The gene transfer method increases the effic…

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AG0302-COVID19 DB16435
biotech

Sponsored by Anges, Inc. in Japan, the AG0302-COVID19 is a DNA-based vaccine that recently completed Phase I/II trials (NCT04527081)[A226813, L30548].

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AGA2115 DB17840
biotech

AGA2115 is a humanized bispecific antibody neutralizing both sclerostin and Dickkopf-1. Developed by Angitia Biopharmaceuticals, AGA2115 is being investigated for the treatment of osteogenesis imperfect.[L46646]

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Agalsidase alfa Approved DB15874
biotech

Agalsidase alfa is a recombinant human ?-galactosidase A similar to [agalsidase beta]. While patients generally do not experience a clinically significant difference in outcomes between the two drugs, some patients may experience greater benefit with agalsida…

Kategori:
Alimentary Tract and Metabolismalpha-Galactosidase, antagonists & inhibitorsAmino Acids, Peptides, and Proteins +9
Target Protein:
Globotriaosylceramide
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance for d…
Genetik -
Agalsidase beta Approved DB00103
biotech

Agalsidase beta is a recombinant human ?-galactosidase A similar to [agalsidase alfa]. While patients generally do not experience a clinically significant difference in outcomes between the two drugs, some patients may experience greater benefit with agalsida…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsEnzymes +7
Target Protein:
Globotriaosylceramide
Waktu Paruhagalsidase beta has…
Vol. DistribusiA 1 mg/kg dose of a…
KlirensA 1 mg/kg dose of a…
Genetik -
small molecule | CAS: 910562-20-8

Aganepag isopropyl is under investigation in clinical trial NCT01110499 (Safety and Efficacy of AGN-210961 Ophthalmic Solution Compared With Bimatoprost Ophthalmic Solution in Patients With Glaucoma or Ocular Hypertension).

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