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6694

Total database: 17430
Struktur (SMILES)
4518 (67.5%)
Target
3751 (56.0%)
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81 (1.2%)
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6694 (100.0%)

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Halaman 45 / 134
Davanat DB15311
small molecule | CAS: 916851-14-4

Davanat is under investigation in clinical trial NCT00054977 (Safety of GM-CT-01 With and Without 5-Fluorouracil in Patients With Solid Tumors).

Kategori:
CarbohydratesHexosesMonosaccharides +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Davesomeran Approved DB17091
biotech | CAS: 2798905-80-1

Davesomeran is a mRNA vaccine used in conjunction with [elasomeran] as part of the Moderna Bivalent COVID-19 vaccine. Similar to the previous Moderna COVID-19 vaccine, Moderna Bivalent vaccine encodes the full-length pre-fusion stabilized spike (S) protein to…

Kategori:
COVID-19 VaccinesVaccinesViral Vaccines
Waktu ParuhThere is limited ph…
Vol. DistribusiThere is limited ph…
KlirensThere is limited ph…
Genetik -
Davunetide DB12613
small molecule | CAS: 211439-12-2

Davunetide has been used in trials studying the treatment of Progressive Nonfluent Aphasia, Progressive Supranuclear Palsy, Predicted Tauopathies, Including, Corticobasal Degeneration Syndrome, and Frontotemporal Dementia With Parkinsonism Linked to Chromosom…

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dazodalibep DB19025
biotech | CAS: 2245953-10-8

Dazodalibep is under investigation in clinical trial NCT06104124 (A Study to Evaluate the Efficacy and Safety of Dazodalibep in Participants With Sjögren's Syndrome (SS) With Moderate-to-severe Systemic Disease Activity).

Waktu Paruh-
Vol. Distribusi-
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DCLL-9718S DB17392
biotech

DCLL9718S is an antibody-drug conjugate targeting C-type lectin-like molecule-1 (CLL-1). DCLL9718S is under investigation in clinical trial NCT03298516 (A Study of DCLL9718S in Participants With Relapsed or Refractory Acute Myeloid Leukemia (AML) or DCLL9718S…

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsGlobulins +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DCVax-L DB17580
biotech

DCVax-L is a personalized immunotherapy comprising an autologous vaccine with dendritic cells loaded _in vitro_ with autologous tumour lysate.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Deanol DB13352
small molecule | CAS: 108-01-0

Deanol is commonly referred to as 2-(dimethylamino)ethanol, dimethylaminoethanol (DMAE) or dimethylethanolamine (DMEA). It holds tertiary amine and primary alcohol groups as functional groups. Deanol has been used in the treatment of attention deficit-hyperac…

Kategori:
AlcoholsAminesAmino Alcohols +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Decitabine Approved DB01262
small molecule | CAS: 2353-33-5

Myelodysplastic syndromes (MDS) are a heterogeneous group of hematopoietic neoplasms with variable underlying etiology and presentation, including neutropenia and thrombocytopenia. Further mutations leading to increased proliferation of cancerous cells can ev…

Kategori:
AntimetabolitesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +18
Target Protein:
DNADNA (cytosine-5)-methyltransferase 1DNA (cytosine-5)-methyltransferase 3A +2
Waktu ParuhDecitabine has a ha…
Vol. DistribusiDecitabine as an ap…
KlirensDecitabine has a cl…
Genetik -
Decoquinate DB11394
small molecule | CAS: 18507-89-6

Decoquinate is used in veterinary to delay the growth and reproduction of coccidian parasites.

Kategori:
Anti-Infective AgentsAntiparasitic AgentsAntiprotozoals +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 20283-21-0

Deskripsi belum tersedia.

Target Protein:
SDS hydrolase SdsA1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Deferitazole DB13120
small molecule | CAS: 945635-15-4

Deferitazole is an iron chelator. It has been used in trials studying the treatment and basic science of Beta-thalassemia, Hepatic Impairment, Impaired Renal Function, Transfusional Iron Overload, and Iron Overload Due to Repeated Red Blood Cell Transfusions.

Kategori:
EthersIron Chelating AgentsSulfur Compounds
Target Protein:
Hemoglobin subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Defibrotide Approved DB04932
biotech | CAS: 83712-60-1

Defibrotide is the sodium salt of a mixture of single-stranded oligodeoxyribonucleotides derived from porcine mucosal DNA. It has been shown to have antithrombotic, anti-inflammatory and anti-ischemic properties (but without associated significant systemic an…

Kategori:
Anti-Inflammatory AgentsAnticoagulantsAntiplatelet agents +9
Target Protein:
Adenosine receptor A1Adenosine receptor A2aAdenosine receptor A2b
Waktu Paruht1/2-alpha = minute…
Vol. Distribusi-
Klirens-
Genetik -
Degarelix Approved DB06699
small molecule | CAS: 214766-78-6

Degarelix is used for the treatment of advanced prostate cancer. Degarelix is a synthetic peptide derivative drug which binds to gonadotropin-releasing hormone (GnRH) receptors in the pituitary gland and blocks interaction with GnRH. This antagonism reduces l…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +9
Target Protein:
Gonadotropin-releasing hormone receptor
Waktu ParuhTerminal half-life:…
Vol. DistribusiCentral compartment…
KlirensFollowing subcutane…
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Arginase-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 490-83-5

Dehydroascorbic acid is made from the oxidation of ascorbic acid. This reaction is reversible, but dehydroascorbic acid can instead undergo irreversible hydrolysis to 2,3-diketogulonic acid. Dehydroascorbic acid as well as ascorbic acid are both termed Vitami…

Kategori:
Acids, AcyclicCarbohydratesDiet, Food, and Nutrition +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dehydrocholic acid Approved DB11622
small molecule | CAS: 81-23-2

Dehydrocholic acid is a synthetic bile acid that was prepared from the oxidation of cholic acid with chromic acid [A33022]. It has been used for stimulation of biliary lipid secretion. The use of dehydrocholic acid in over-the-counter products has been discon…

Kategori:
Bile Acids and SaltsCholagogues and CholereticsCholanes +5
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Delafloxacin Approved DB11943
small molecule | CAS: 189279-58-1

Delafloxacin is a fluoroquinolone antibiotic which has been used in trials studying the treatment and basic science of Gonorrhea, Hepatic Impairment, Bacterial Skin Diseases, Skin Structure Infections, and Community Acquired Pneumonia, among others. It was ap…

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +21
Target Protein:
DNA topoisomerase 4 subunit ADNA gyrase subunit A
Waktu ParuhThe mean half life …
Vol. DistribusiThe steady sate vol…
KlirensThe mean total clea…
Genetik -
Delamanid Approved DB11637
small molecule | CAS: 681492-22-8

Delamanid is an anti-tuberculosis agent derived from the nitro-dihydro-imidazooxazole class of compounds that inhibits mycolic acid synthesis of bacterial cell wall [A31965]. It is used in the treatment of multidrug-resistant and extensively drug-resistant tu…

Kategori:
Antiinfectives for Systemic UseAntimycobacterialsCytochrome P-450 CYP3A Substrates +7
Waktu ParuhThe half life range…
Vol. DistribusiThe apparent volume…
Klirens-
Genetik -
Delandistrogene moxeparvovec Approved DB16802
biotech | CAS: 2305040-16-6

Delandistrogene moxeparvovec is an adeno-associated virus vector-based gene therapy developed by Sarepta Therapeutics. It was granted accelerated approval by the FDA on June 22, 2023, as the first gene therapy to treat Duchenne Muscular Dystrophy (DMD).[L4702…

Kategori:
Adeno-associated Viral Vector TherapiesMuscular Dystrophy, DuchenneMusculo-Skeletal System
Waktu ParuhNo information is a…
Vol. DistribusiThere is limited in…
KlirensNo information is a…
Genetik -
Delavirdine Approved DB00705
small molecule | CAS: 136817-59-9

A potent, non-nucleoside reverse transcriptase inhibitor with activity specific for HIV-1.

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +31
Target Protein:
Gag-Pol polyproteinReverse transcriptase/RNaseH
Waktu Paruh5.8 hours
Vol. Distribusi-
Klirens-
Genetik -
Delgocitinib DB16133
small molecule | CAS: 1263774-59-9

Delgocitinib is a pan-Janus kinase (JAK) inhibitor. After the first global approval in Japan,[A264693] delgocitinib was also approved by the European Commission on September 23, 2024.[L51913] It works to reduce the inflammatory response in inflammatory skin d…

Kategori:
Agents for Dermatitis, Excluding CorticosteroidsDermatologicalsOAT3/SLC22A8 Substrates +2
Target Protein:
Tyrosine-protein kinase JAK1Tyrosine-protein kinase JAK2Tyrosine-protein kinase JAK3 +1
Waktu ParuhFollowing repeated …
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2061938-98-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Iron(3+)-hydroxamate-binding protein FhuDFerrichrome-iron receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Delta-aminolevulinic acid dehydrataseGlycine amidinotransferase, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Demcizumab DB12734
biotech | CAS: 1243262-17-0

Demcizumab is under investigation for the treatment of Nonsquamous Nonsmall Cell Neoplasm of Lung.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Demecarium Approved DB00944
small molecule | CAS: 16505-84-3

Demecarium is an indirect-acting parasympathomimetic agent that is used to treat glaucoma. It is a cholinesterase inhibitor or an anticholinesterase. Cholinesterase inhibitors prolong the effect of acetylcholine, which is released at the neuroeffector junctio…

Kategori:
AminesAmmonium CompoundsAntiglaucoma Preparations and Miotics +9
Target Protein:
AcetylcholinesteraseCholinesterase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Demeclocycline Approved DB00618
small molecule | CAS: 127-33-3

A tetracycline analog having a 7-chloro and a 6-methyl. Because it is excreted more slowly than tetracycline, it maintains effective blood levels for longer periods of time.

Kategori:
Agents that produce neuromuscular block (indirect)Anti-Bacterial AgentsAnti-Infective Agents +8
Target Protein:
30S ribosomal proteinVasopressin V2 receptor
Waktu Paruh10-17 hours
Vol. Distribusi-
Klirens* Renal cl=35 mL/mi…
Genetik -
Demecolcine DB13318
small molecule | CAS: 477-30-5

Deskripsi belum tersedia.

Kategori:
AlkaloidsAntimitotic AgentsAntineoplastic Agents +5
Target Protein:
Microtubule-associated protein 1BMicrotubule-associated protein 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Demegestone DB13857
small molecule | CAS: 10116-22-0

Demegestone is a progesterone receptor agonist that was previously used to treat luteal insufficiency. It was previously marketed in France as Lutionex, but has since been discontinued.

Kategori:
Adrenal Cortex HormonesContraceptive Agents, FemaleContraceptives, Oral +15
Target Protein:
Progesterone receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Demoxytocin DB13798
small molecule | CAS: 113-78-0

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1009838-50-9

Demplatin pegraglumer is under investigation in clinical trial NCT02043288 (Combination Therapy With NC-6004 and Gemcitabine Versus Gemcitabine Alone in Pancreatic Cancer).

Kategori:
Amino AcidsAmino Acids, AcidicAmino Acids, Dicarboxylic +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

The recombinant chimeric DC vaccine is a subunit-based vaccine candidate investigated for safety and effectiveness against SARS-CoV-2-induced pneumonia. With a better safety profile than inactivated and live-attenuated virus and virus-vector vaccines, the rec…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Denecimig DB18426
biotech | CAS: 2488745-86-2

Delpacibart is a humanized, bispecific, bivalent monoclonal antibody against coagulation factor 9.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Kategori:
Biological ProductsComplex MixturesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DengueCide DB18546
biotech

DengueCide is a nonjugate of a dengue virus specific small chemical ligand and an amphiphilic PEG based polymer

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Denibulin DB05932
small molecule | CAS: 284019-34-7

Denibulin is a novel small molecule Vascular Disrupting Agent under development by MediciNova for treatment of solid tumor cancers.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Vascular endothelial growth factor A, long formVascular endothelial growth factor receptor 1Vascular endothelial growth factor receptor 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Denifanstat DB17576
small molecule | CAS: 1399177-37-7

Denifanstat is an orally bioavailable fatty acid synthase (FASN) inhibitor. Due to its antineoplastic activities, it is being investigated for various cancers.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Denileukin diftitox Approved DB00004
biotech | CAS: 173146-27-5

Denileukin diftitox is an IL2-receptor-directed cytotoxin, is a recombinant DNA-derived fusion protein composed of the amino acid sequences for diphtheria toxin fragments A and B (Met<sub>1</sub>-Thr<sub>387</sub>)-His and the sequence for human interleukin-2…

Kategori:
ADP Ribose TransferasesAmino Acids, Peptides, and ProteinsAntineoplastic Agents +15
Target Protein:
Interleukin-2 receptor subunit alphaInterleukin-2 receptor subunit beta
Waktu ParuhThe arithmetic mean…
Vol. DistribusiThe geometric mean …
KlirensThe geometric mean …
Genetik -
Denosumab Approved DB06643
biotech | CAS: 615258-40-7

Denosumab is a novel, fully human IgG2 monoclonal antibody specific to receptor activator of nuclear factor kappa-B ligand (RANKL), suppresses bone resorption via inhibiting RANK-mediated activation of osteoclasts. It is the first and currently the only RANKL…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +16
Target Protein:
Tumor necrosis factor ligand superfamily member 11
Waktu ParuhAfter C<sub>max</su…
Vol. DistribusiThe central volume …
KlirensNo information is a…
Genetik -
biotech

Dental pulp is a soft, connective tissue present in the dental crown of both third molar and first premolar teeth. Dental pulp stem cells (DPSCs) exhibit fibro-blast like plasticity and adherent properties. They are harvested through surgical extraction of wi…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Clavaminate synthase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Deoxycholic acid Approved DB03619
small molecule | CAS: 83-44-3

Deoxycholic acid is a a bile acid which emulsifies and solubilizes dietary fats in the intestine, and when injected subcutaneously, it disrupts cell membranes in adipocytes and destroys fat cells in that tissue. In April 2015, deoxycholic acid was approved by…

Kategori:
Bile Acids and SaltsBSEP/ABCB11 inducersCholagogues and Choleretics +9
Target Protein:
Proliferating cell nuclear antigenSteroid Delta-isomeraseCytochrome C +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 964-26-1

Deskripsi belum tersedia.

Kategori:
DeoxyribonucleotidesNucleic Acids, Nucleotides, and NucleosidesNucleotides +3
Target Protein:
Thymidylate synthaseDeoxyuridine 5'-triphosphate nucleotidohydrolaseThymidylate synthase +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Depatuxizumab DB12826
biotech | CAS: 1471999-69-5

Depatuxizumab has been used in trials studying the treatment and diagnostic of Adenocarcinoma and Advanced Solid Tumors.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Depemokimab DB18846
biotech | CAS: 2243274-14-6

Depemokimab is under investigation in clinical trial NCT05274750 (Efficacy and Safety of Depemokimab (GSK3511294) in Participants With Chronic Rhinosinusitis With Nasal Polyps).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Deracoxib DB11395
small molecule | CAS: 169590-41-4

Deracoxib is a non-steroidal anti-inflammatory drug of the coxib class, used in veterinary medicine to treat osteoarthritis in dogs. It is sold in tablets, which have added beefy flavour to increase palatability. Deramaxx received FDA approval in August 2002 …

Kategori:
AmidesAnalgesicsAnalgesics, Non-Narcotic +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Deramciclane DB06512
small molecule | CAS: 120444-71-5

Deramciclane (EGIS-3886) is used for the treatment of a number of anxiety disorders. Deramciclane differs from other anti anxiety medications in that it is not a benzodiazepine and so has a different structure and target. It antagonizes 5-HT2A receptors, agon…

Kategori:
Anti-Anxiety AgentsAnticonvulsantsAntidepressive Agents +17
Target Protein:
5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 2C
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Derazantinib DB14889
small molecule | CAS: 1234356-69-4

Derazantinib is under investigation in clinical trial NCT03230318 (Derazantinib in Subjects With FGFR2 Gene Fusion Positive Inoperable or Advanced Intrahepatic Cholangiocarcinoma).

Kategori:
AminesHeterocyclic Compounds, Fused-Ring
Target Protein:
Fibroblast growth factor receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 2201–2250 dari 6694
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