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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 45 / 236
AP-102 DB18206
small molecule | CAS: 846569-60-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AP-22408 DB01830
small molecule | CAS: 268741-43-1

Deskripsi belum tersedia.

Target Protein:
Proto-oncogene tyrosine-protein kinase SrcTyrosine-protein kinase Lck
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Apabetalone DB12000
small molecule | CAS: 1044870-39-4

Apabetalone has been investigated for the treatment of Diabetes, Atherosclerosis, and Coronary Artery Disease.

Kategori:
Heterocyclic Compounds, Fused-RingQuinazolines
Waktu Paruh-
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Genetik -
Apadamtase alfa Approved DB15164
biotech | CAS: 2086325-24-6

Thrombotic thrombocytopenic purpura (TTP) is a rare blood clotting disorder characterized by thrombocytopenia, microangiopathic hemolytic anemia, and various degrees of organ damage.[A262076] It may be inherited (congenital TTP; cTTP) or acquired due to autoa…

Kategori:
ADAM ProteinsADAMTS ProteinsAmino Acids, Peptides, and Proteins +12
Target Protein:
von Willebrand factor
Waktu ParuhFollowing the intra…
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2097132-02-8

Deskripsi belum tersedia.

Waktu Paruh-
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Apatorsen DB06094
biotech | CAS: 1002331-21-6

Apatorsen is a second generation antisense drug which in preclinical experiments, inhibits production of Heat Shock Protein 27 (Hsp27) a cell survival protein found at elevated levels in many human cancers including prostate, lung, breast, ovarian, bladder, r…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Target Protein:
Heat shock protein beta-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apc001 DB17819
biotech

Apc001 is an aptamer developed for the treatment of osteogenesis imperfecta.

Waktu Paruh-
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Genetik -
Apc001PE DB17902
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
APC8020 DB17228
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
APD-209 DB18759
small molecule | CAS: 1261156-82-4

Deskripsi belum tersedia.

Target Protein:
Beta-2 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
APD791 DB05227
small molecule

APD791 is an oral anti-thrombotic drug candidate being evaluated in a Phase 1 clinical trial by Arena. APD791 is intended to lower the risk of arterial thrombosis by reducing the amplification of platelet aggregation, arterial constriction and intimal hyperpl…

Kategori:
Acids, CarbocyclicAmidesAntidepressive Agents +8
Target Protein:
5-hydroxytryptamine receptor 2A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apelin DB18909
biotech | CAS: 372170-33-7

Apelin is under investigation in clinical trial NCT03449251 (A Series of Pilot Studies to Evaluate the Haemodynamic and Metabolic Effects of Apelin and Relaxin).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsIntercellular Signaling Peptides and Proteins +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
APG-1387 DB16095
small molecule | CAS: 1570231-89-8

APG-1387 is under investigation in clinical trial NCT04568265 (A Clinical Study of APG-1387 in Combination With Entecavir in Patients With Chronic Hepatitis B).

Kategori:
AmidesSulfonesSulfur Compounds
Target Protein:
E3 ubiquitin-protein ligase XIAPBaculoviral IAP repeat-containing protein 2Baculoviral IAP repeat-containing protein 3 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
APG-157 DB18683
small molecule

APG-157 consists of zinflavonoids being investigated for the treatment of cancers.

Waktu Paruh-
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Genetik -
Aphidicolin DB17742
small molecule | CAS: 38966-21-1

Aphidicolin is an antimitotic and antiviral metabolite of the mould _Cephalosporium aphidicola_. It inhibits DNA polymerase alpha and blocks DNA replication.[A259157, A259162]

Kategori:
Anti-Infective AgentsAntiviral AgentsDiterpenes +2
Target Protein:
DNA polymerase catalytic subunit
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Apigenin DB07352
small molecule | CAS: 520-36-5

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesFlavones +3
Target Protein:
Casein kinase II subunit alphaAldo-keto reductase family 1 member B1Cytochrome P450 1B1 +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apinocaltamide DB16241
small molecule | CAS: 1838651-58-3

Apinocaltamide is under investigation in clinical trial NCT03239691 (A Study to Evaluate the Effect of ACT-709478 in Photosensitive Epilepsy Patients).

Kategori:
AcetatesAcids, AcyclicAmides +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apitegromab DB16096
biotech | CAS: 2278276-46-1

Apitegromab is under investigation in clinical trial NCT03921528 (An Active Treatment Study of SRK-015 in Patients With Type 2 or Type 3 Spinal Muscular Atrophy).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apitolisib DB12180
small molecule | CAS: 1032754-93-0

Apitolisib has been used in trials studying the treatment of Solid Cancers, Breast Cancer, Prostate Cancer, Renal Cell Carcinoma, and Endometrial Carcinoma, among others.

Kategori:
Phosphatidylinositol 3-Kinases, antagonists & inhibitors
Target Protein:
Serine/threonine-protein kinase mTORPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apixaban Approved DB06605
small molecule | CAS: 503612-47-3

Apixaban is an oral, direct, and highly selective factor Xa (FXa) inhibitor of both free and bound FXa, as well as prothrombinase, independent of antithrombin III for the prevention and treatment of thromboembolic diseases[Label,A6897]. It is marketed under t…

Kategori:
AnticoagulantsAntithrombinsBCRP/ABCG2 Substrates +17
Target Protein:
Coagulation factor X
Waktu Paruh12.7±8.55h[Label,A1…
Vol. DistribusiApproximately 21L[L…
Klirens3.3L/h[Label] thoug…
Genetik -
APL-030 DB18735
small molecule

APL-030 is a orally-active small molecule inhibitor of GCN2.

Waktu Paruh-
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APL-502 DB17473
biotech | CAS: 2303884-58-2

APL 502 is a humanised immunoglobulin G1 (IgG1) monoclonal antibody targeting the programmed cell death-1 ligand-1 (PD-L1).

Waktu Paruh-
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Aplaviroc DB06497
small molecule | CAS: 461443-59-4

A spiro-diketo-piperazine; a potent noncompetitive allosteric antagonist of the CCR5 receptor with concomitantly potent antiviral effects for HIV-1.

Kategori:
Acids, CarbocyclicAnti-HIV AgentsAnti-Infective Agents +6
Target Protein:
C-C chemokine receptor type 5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aplindore DB06620
small molecule | CAS: 189681-70-7

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
D(2) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apolizumab DB06467
biotech | CAS: 267227-08-7

Apolizumab is a humanized monoclonal antibody that is being studied as a treatment for hematologic cancers.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Apomab DB15022
biotech | CAS: 1108170-71-3

Apomab is under investigation in clinical trial NCT00851136 (A Study of PRO95780 Administered in Combination With the FOLFOX Regimen and Bevacizumab in Patients With Previously Untreated, Locally Advanced, Recurrent, and Metastatic Colorectal Cancer (APM4566g…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apomine DB12276
small molecule | CAS: 126411-13-0

Apomine has been used in trials studying the treatment of Osteoporosis and Unspecified Adult Solid Tumor, Protocol Specific.

Kategori:
OrganophosphonatesOrganophosphorus Compounds
Target Protein:
Bile acid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apomorphine Approved DB00714
small molecule | CAS: 58-00-4

Apomorphine is a non-ergoline dopamine D2 agonist indicated to treat hypomobility associated with Parkinson's. It was first synthesized in 1845 and first used in Parkinson's disease in 1884.[A203618] Apomorphine has also been investigated as an emetic, a seda…

Kategori:
AlkaloidsAnti-Parkinson Agents (Dopamine Agonist)Anti-Parkinson Drugs +32
Target Protein:
D(4) dopamine receptorD(2) dopamine receptorD(3) dopamine receptor +11
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe apparent volume…
KlirensThe clearance of a …
Genetik -
small molecule | CAS: 42337-33-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apoptone DB06307
small molecule | CAS: 183387-50-0

Deskripsi belum tersedia.

Kategori:
AndrostanesFused-Ring CompoundsSteroids
Target Protein:
Apoptosis regulator Bcl-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
APR-2020 DB18497
biotech

APR-2020 is a CD34+ cells that have been transduced in vitro with a lentiviral vector carrying a codon-optimized sequence for expressing the wild type RPS19 protein

Waktu Paruh-
Vol. Distribusi-
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Genetik -
APR-548 DB17546
small molecule

APR-548 is an analog of [eprenetapopt] and a reactivator of mutant p53.

Waktu Paruh-
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Genetik -
Apraclonidine Approved DB00964
small molecule | CAS: 66711-21-5

Apraclonidine, also known as iopidine, is a sympathomimetic used in glaucoma therapy. It is an alpha2-adrenergic agonist.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +12
Target Protein:
Alpha-1A adrenergic receptorAlpha-2A adrenergic receptorAlpha-2B adrenergic receptor
Waktu Paruh8 hours
Vol. Distribusi-
Klirens-
Genetik -
Apramycin DB04626
small molecule | CAS: 37321-09-8

Apramycin is an aminoglycoside antibiotic and has a bactericidal action against many gram-negative bacteria. Apramycin is a structurally unique antibiotic that contains a bicyclic sugar moiety and a monosubstituted deoxystreptamine. It is not approved for use…

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +4
Target Protein:
16S ribosomal RNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apratastat DB13020
small molecule | CAS: 287405-51-0

Tmi 005 is under investigation in clinical trial NCT00095342 (Study Evaluating TMI-005 in Active Rheumatoid Arthritis).

Kategori:
Oxazines
Target Protein:
Interstitial collagenaseCollagenase 3Disintegrin and metalloproteinase domain-containing protein 17
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apremilast Approved DB05676
small molecule | CAS: 608141-41-9

Apremilast, also known as Otezla, is a phosphodiesterase 4 (PDE4) inhibitor used to treat various types of symptoms resulting from certain inflammatory autoimmune diseases. It belongs to the same drug class as [Roflumilast] and [Crisaborole].[A181244,L7495] I…

Kategori:
Agents reducing cytokine levelsAnti-Inflammatory AgentsAntineoplastic and Immunomodulating Agents +17
Target Protein:
Phosphodiesterase isozyme 4Cyclin-dependent kinase 4Cyclin-dependent kinase 6
Waktu ParuhThe average elimina…
Vol. DistribusiThe average apparen…
KlirensIn healthy patients…
Genetik -
Aprepitant Approved DB00673
small molecule | CAS: 170729-80-3

Aprepitant, an antiemetic, is a substance P/neurokinin 1 (NK1) receptor antagonist which, in combination with other antiemetic agents, is indicated for the prevention of acute and delayed nausea and vomiting associated with initial and repeat courses of highl…

Kategori:
Alimentary Tract and MetabolismAntiemeticsAntiemetics and Antinauseants +36
Target Protein:
Substance-P receptor
Waktu Paruh9-13 hours
Vol. Distribusi* 70 L
Klirens* Apparent plasma c…
Genetik -
Apricitabine DB12855
small molecule | CAS: 160707-69-7

Apricitabine has been used in trials studying the treatment of HIV Infections.

Kategori:
DeoxyribonucleosidesNucleic Acids, Nucleotides, and NucleosidesNucleosides +2
Target Protein:
Gag-Pol polyproteinReverse transcriptase/RNaseH
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apricot kernel oil Approved DB14324
biotech | CAS: 72869-69-3

Apricot kernel oil is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
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Genetik -
Apricoxib DB12378
small molecule | CAS: 197904-84-0

Apricoxib has been used in trials studying the treatment and prevention of Lung Cancer, Breast Cancer, Pancreatic Cancer, Non Small Cell Lung Cancer, and Metastatic Pancreatic Cancer, among others.

Kategori:
AmidesSulfonesSulfur Compounds
Target Protein:
Prostaglandin G/H synthase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aprindine DB01429
small molecule | CAS: 37640-71-4

Aprindine is a cardiac depressant used in arrhythmias.

Kategori:
Antiarrhythmic agentsAntiarrhythmics, Class IAntiarrhythmics, Class Ib +9
Target Protein:
Calmodulin-2Calmodulin-1Calmodulin-3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aprinocarsen DB06451
biotech | CAS: 151879-73-1

Aprinocarsen is a specific antisense oligonucleotide inhibitor of protein kinase C-alpha.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +3
Target Protein:
Protein kinase C alpha type
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aprobarbital DB01352
small molecule | CAS: 77-02-1

Aprobarbital is a barbiturate derivative synthesized in the 1920s by Ernst Preiswerk. It was determined that the substance was capable of demonstrating sedative, hypnotic, and anticonvulsant effects. A primary treatment indicated for the use of aprobarbital w…

Kategori:
Anticholinergic AgentsBarbiturates, PlainCentral Nervous System Depressants +10
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Gamma-aminobutyric acid receptor subunit alpha-2Gamma-aminobutyric acid receptor subunit alpha-3 +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aprocitentan Approved DB15059
small molecule | CAS: 1103522-45-7

Aprocitentan is a dual antagonist of endothelin receptors A and B used for treatment-resistant hypertension. It is the active metabolite of [macitentan]. Approximately 10-15% of patients with hypertension have resistant hypertension, defined as uncontrolle…

Kategori:
AmidesAntihypertensive AgentsBCRP/ABCG2 Inhibitors +26
Target Protein:
Endothelin-1 receptorEndothelin receptor type B
Waktu ParuhThe effective half-…
Vol. DistribusiThe apparent volume…
KlirensThe apparent cleara…
Genetik -
Apronalide Approved DB13221
small molecule | CAS: 528-92-7

Apronalide is approved in Japan. Apronalide has been withdrawn from the market in many other countries due to patient development of thrombocytopenic purpura [A174814].

Kategori:
AmidesCentral Nervous System DepressantsHypnotics and Sedatives +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aprotinin Approved DB06692
biotech | CAS: 9087-70-1

Aprotinin is a protein-based drug that is also known as bovine pancreatic trypsin inhibitor (BPTI). Since it demonstrates the capacity to slow fibrinolysis, it has been employed to reduce bleeding during complex surgery such as heart and liver surgery. For th…

Kategori:
Amino Acids, Peptides, and ProteinsAntifibrinolytic AgentsBlood and Blood Forming Organs +11
Target Protein:
Serine protease 1Chymotrypsinogen BPlasminogen +1
Waktu ParuhFollowing this dist…
Vol. Distribusi-
Klirens-
Genetik -
Apstatin DB04092
small molecule | CAS: 160470-73-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and Proteins
Target Protein:
Xaa-Pro aminopeptidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
APT-101 DB18003
small molecule | CAS: 2100848-01-7

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
Aptazapine DB09305
small molecule | CAS: 71576-40-4

Aptazapine (CGS-7525A) was a tetracyclic antidepressant developed in the 1980s. Aptazapine had noradrenergic and specific serotonergic activity. It antagonised ?2 adrenergic receptors approximately 10 times more effectively than mianserin, antagonised 5-HT2 r…

Kategori:
Antidepressive Agents, TetracyclicBenzazepinesHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
APTO-253 DB17143
small molecule | CAS: 916151-99-0

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Krueppel-like factor 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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