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2279

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866 (38.0%)
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1100 (48.3%)
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Halaman 44 / 46
Upanovimab DB16505
biotech | CAS: 2500633-46-3

Upanovimab (SCTA01) was under investigation in clinical trials (NCT04683328, NCT04644185, NCT04709328 and NCT05156645) to evaluate its safety and efficacy in patients with severe COVID-19

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Urabrelimab DB17209
biotech | CAS: 2249722-58-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Uracil C-13 DB16345
small molecule | CAS: 35803-45-3

Uracil C-13 is under investigation in clinical trial NCT01677338 (Phase 2 Study to Evaluate the Preliminary Performance of the C13-URA Breath Test Kit in Dyspeptic Subjects).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Urelumab DB12077
biotech | CAS: 934823-49-1

Urelumab has been used in trials studying the treatment of Leukemia, Multiple Myeloma, Malignant Tumors, and Cancer - Solid Tumors and B-Cell Non-Hodgkin's Lymphoma. Urelumab is a fully human antibody that targets CD137. The antibody product was developed usi…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Target Protein:
Tumor necrosis factor receptor superfamily member 9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Uric acid DB08844
small molecule | CAS: 69-93-2

Uric acid is the last product of purine metabolism in humans. The formation of uric acid is through the enzyme xanthine oxidase, which oxidizes oxypurines. Normally a small amount of uric acid is present in the body, but when there is an excess amount in the …

Kategori:
AlkaloidsAntioxidantsBiological Factors +6
Target Protein:
Glycogen phosphorylase, liver form
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Uridine triacetate Approved DB09144
small molecule | CAS: 4105-38-8

Uridine triacetate, formerly known as vistonuridine, is an orally active prodrug of the naturally occurring nucleoside uridine. It is used for the treatment of hereditary orotic aciduria (Xuriden), or for the emergency treatment of fluorouracil or capecitabin…

Kategori:
Acids, AcyclicAlimentary Tract and MetabolismFatty Acids +9
Waktu Paruh2 to 2.5 hours
Vol. DistribusiCirculating uridine…
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
UDP-glucose 4-epimerase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Urofollitropin Approved DB00094
biotech | CAS: 97048-13-0

Urofollitropin is a urinary-derived follicle-stimulating hormone (FSH) that is extracted and purified from human urine samples. It consists of two non-covalently linked, non-identical glycoproteins designated as the alpha- and beta- subunits. The alpha- and b…

Kategori:
Amino Acids, Peptides, and ProteinsGenito Urinary System and Sex HormonesGonadotropins +9
Target Protein:
Follicle-stimulating hormone receptor
Waktu ParuhCirculation half li…
Vol. DistribusiTime to peak in pla…
Klirens-
Genetik -
Ursodeoxycholic acid Approved DB01586
small molecule | CAS: 128-13-2

Ursodeoxycholic acid (UDCA), also known as ursodiol, is a naturally-occurring bile acid that constitutes a minor fraction of the human bile acid pool.[A256272,A256277] UDCA has been used to treat liver disease for decades: its first use in traditional medicin…

Kategori:
Alimentary Tract and MetabolismBile Acid PreparationsBile acids and derivatives +15
Target Protein:
Aldo-keto reductase family 1 member C2Biliverdin reductase ASolute carrier family 23 member 2 +1
Waktu ParuhThe estimated half-…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
Urtoxazumab DB17806
biotech | CAS: 502496-16-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ustekinumab Approved DB05679
biotech | CAS: 815610-63-0

Ustekinumab is a human immunoglobulin (Ig) G1 kappa monoclonal antibody directed against interleukin(IL)-12 and IL-23, which are cytokines that are involved in immune and inflammatory responses.[A187349] It was generated via recombinant human IL-12 immunizati…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +16
Target Protein:
Interleukin-23Interleukin-12 subunit beta
Waktu ParuhFollowing administr…
Vol. DistribusiThe total volume of…
KlirensThe median apparent…
Genetik -
UX053 DB18558
biotech

UX053 is an mRNA encoding the human glycogen debranching enzyme.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
V1003 DB05046
small molecule

V1003 is an intranasal formulation of buprenorphine, an opiate analgesic, for the management of post-operative pain in hospital and home settings. Buprenorphine is a well-known analgesic and the intranasal formulation has the potential to provide a convenient…

Target Protein:
Kappa-type opioid receptorMu-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VA-MENGOC-BC® DB15800
biotech

VA-MENGOC-BC is a meningococcal B and C vaccine and an outer membrane vesicle (OMV)-based vaccine. The OMVs contain over 100 proteins, and are derived from meningococcal group B and capsular polysaccharide of meningococcal group C. As there already exists a p…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Valaciclovir Approved DB00577
small molecule | CAS: 124832-26-4

Valaciclovir (valacyclovir), also known as _Valtrex_, is an antiviral drug that has been used to manage and treat various herpes infections for more than 2 decades. It was initially approved by the FDA in 1995 [FDA label] and marketed by GlaxoSmithKline [L56…

Kategori:
Acyclovir and prodrugAmino AcidsAmino Acids, Branched-Chain +19
Target Protein:
Thymidine kinaseDNA polymerase catalytic subunit
Waktu ParuhThe plasma eliminat…
Vol. DistribusiCerebrospinal fluid…
KlirensRenal clearance of …
Genetik -
Valerian Approved DB13196
biotech | CAS: 8057-49-6

Valerian is extracted from a herb that is a perennial flowering plant. Valerian root is reported to have sedative and anxiolytic effects however its mechanism of action is not completely understood. Valerian has been used in the treatment of conditions includ…

Kategori:
AngiospermsBiological ProductsCentral Nervous System Depressants +15
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Valganciclovir Approved DB01610
small molecule | CAS: 175865-60-8

Valganciclovir hydrochloride (Valcyte, manufactured by Roche) is an antiviral medication used to treat cytomegalovirus infections. As the L-valyl ester of ganciclovir, it is actually a prodrug for ganciclovir. After oral administration, it is rapidly converte…

Kategori:
Agents that reduce seizure thresholdAnti-Infective AgentsAntiinfectives for Systemic Use +13
Target Protein:
DNA polymerase catalytic subunitDNA
Waktu ParuhApproximately 4.08 …
Vol. Distribusi* 0.703 ± 0.134 L/kg
Klirens* 3.07+/- 0.64 mL/m…
Genetik -
Valnoctamide DB13099
small molecule | CAS: 4171-13-5

Valnoctamide has been used in trials studying the treatment of Mania and Schizoaffective Disorder, Manic Type.

Kategori:
Central Nervous System DepressantsHypnotics and SedativesNervous System +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Valoctocogene roxaparvovec Approved DB15561
biotech | CAS: 1819334-78-5

Valoctocogene roxaparvovec is an adeno-associated virus serotype 5 (AAV5) based gene therapy vector that expresses the B-domain deleted SQ form of human coagulation factor VIII (hFVIII-SQ).[L43282] The expression of hFVIII-SQ is driven by a liver-specific pro…

Kategori:
Adeno-associated Viral Vector TherapiesAmino Acids, Peptides, and ProteinsBiological Factors +9
Target Protein:
Coagulation factor VIII (F8)
Waktu Paruh-
Vol. Distribusi-
KlirensThe maximum time to…
Genetik -
Valproic acid Approved DB00313
small molecule | CAS: 99-66-1

Valproic acid, or valproate, is an fatty acid derivative and anticonvulsant originally synthesized in 1881 by Beverly S. Burton.[A178051] It enjoyed use as a popular organic solvent in industry and pharmaceutical manufacturing for nearly a century. In 1963, a…

Kategori:
Acids, AcyclicAnti-epileptic AgentAnticonvulsants +68
Target Protein:
4-aminobutyrate aminotransferase, mitochondrialGlycogen synthase kinase-3 alphaHistone deacetylase 9 +13
Gen Terkait:
POLG POLG
Waktu Paruh13-19 hours.[label]…
Vol. Distribusi11 L/1.73m<sup>2</s…
Klirens0.56 L/hr/m<sup>2</…
Genetik 2 Varian
Valsartan Approved DB00177
small molecule | CAS: 137862-53-4

Valsartan belongs to the angiotensin II receptor blocker (ARB) family of drugs, which also includes [telmisartan], [candesartan], [losartan], [olmesartan], and [irbesartan]. ARBs selectively bind to angiotensin receptor 1 (AT1) and prevent the protein angiote…

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +22
Target Protein:
Type-1 angiotensin II receptor
Waktu ParuhAfter intravenous (…
Vol. DistribusiThe steady-state vo…
KlirensFollowing intraveno…
Genetik -
Valziflocept DB17728
biotech | CAS: 1804910-11-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vamorolone Approved DB15114
small molecule | CAS: 13209-41-1

Vamorolone is a novel and fully synthetic glucocorticoid developed by Santhera Pharmaceuticals. It is used to manage inflammation and immune dysregulation in patients with Duchenne muscular dystrophy (DMD), a neuromuscular disorder characterized by the insidi…

Kategori:
Adrenal Cortex HormonesAnti-Inflammatory AgentsCorticosteroids +20
Target Protein:
Glucocorticoid receptorMineralocorticoid receptor
Waktu ParuhThe terminal elimin…
Vol. DistribusiBased on population…
KlirensBased on population…
Genetik -
biotech | CAS: 2382896-00-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vanoxerine DB03701
small molecule | CAS: 67469-69-6

Vanoxerine is a highly selective dopamine transporter antagonist. It was synthesized in the late 1970s and developed as a potential treatment for depression.[A19824] Vanoxerine was later evaluated as a potential treatment for cocaine addiction due to its abil…

Kategori:
Antiarrhythmic agentsCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +6
Target Protein:
Sodium-dependent dopamine transporterHERG human cardiac K+ channel
Waktu ParuhThe mean eliminatio…
Vol. DistribusiVanoxerine is capab…
KlirensAt 25, 75 and 125 m…
Genetik -
biotech

Live attenuated zoster vaccine is available as two products: Zostavax for the prevention of shingles in immunocompetent people over the age of 50, and Varivax for the prevention of chickenpox in individuals 12 months of age and older. While the two vaccines c…

Kategori:
Actively Acquired ImmunityAntiinfectives for Systemic UseBiological Products +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Recombinant zoster vaccine, manufactured as the product Shingrix by GlaxoSmithKline, is an adjuvanted non-live recombinant vaccine indicated for prevention of shingles. First approved in October 2017 by the Food and Drug Administration, Shingrix is the prefer…

Kategori:
VaccinesVaricella Zoster Vaccines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Varlilumab DB11930
biotech | CAS: 1393344-72-3

Varlilumab has been used in trials studying the treatment of MELANOMA, Skin Ulcer, Burkett's Lymphoma, Mantle cell lymphoma, and Any T-cell Malignancy, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Varlitinib DB05944
small molecule | CAS: 845272-21-1

Varlitinib is an oral, selective, reversible, small molecule tyrosine kinase inhibitor of both ErbB-2 (Her-2/neu) and EGFR. Over-expression of ErbB-2 and EGFR receptors in tumors is predictive of poor prognosis in cancer patients. Varlitinib has shown signifi…

Kategori:
Heterocyclic Compounds, Fused-RingSulfur Compounds
Target Protein:
Epidermal growth factor receptorReceptor tyrosine-protein kinase erbB-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 37221-79-7

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsCardiovascular AgentsCentral Nervous System Agents +13
Target Protein:
Vasoactive intestinal polypeptide receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VaxSyn DB17827
biotech

VaxSyn HIV-1 is a recombinant form of the HIV envelope protein gp 160 developed by MicroGeneSys and the National Institute of Allergy and Infectious Diseases (NIAID).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Vayarin Approved DB09328
biotech

Vayarin is a prescription medical food for the clinical dietary management of certain lipid imbalances blamed to be associated with attention deficit hyperactivity disorder (ADHD) in children. Vayarin contains _Lipirinen_, a proprietary composition containing…

Kategori:
Cytochrome P-450 CYP2E1 InhibitorsCytochrome P-450 CYP2E1 Inhibitors (strength unknown)Cytochrome P-450 Enzyme Inhibitors
Waktu ParuhAbout 2h [L1507]
Vol. Distribusi-
KlirensMainly in the feces…
Genetik -
VB10.16 DB17512
biotech

VB10.16 is a novel therapeutic antigen-presenting cell-targeting DNA vaccine developed to treat HPV16-positive cancers. It is composed of three parts, one encodes the E6/E7 fusion protein of human papillomavirus (HPV) type 16 (HPV16), a dimerization entity, a…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
VCN-01 DB18193
biotech

VCN-01 is an investigational, genetically modified human adenovirus encoding human PH20.

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Klirens-
Genetik -
Vedolizumab Approved DB09033
biotech | CAS: 943609-66-3

Vedolizumab is a recombinant humanized IgG1 monoclonal antibody directed against the human lymphocyte ?4?7 integrin, a key mediator of gastrointestinal inflammation implicated in diseases like ulcerative colitis or Crohn's disease.[L48216] ?4?7 integrin facil…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +15
Target Protein:
Integrin alpha-4Integrin beta-7
Waktu ParuhVedolizumab has a l…
Vol. DistribusiSerum apparent volu…
KlirensVedolizumab clearan…
Genetik -
Velafermin DB06493
small molecule | CAS: 697766-75-9

Velafermin was a novel investigational protein therapeutic, also known as fibroblast growth factor-20 (FGF-20), which promotes both epithelial and mesenchymal cell proliferation in vitro and has demonstrated activity in multiple animal models. Velafermin was …

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsIntercellular Signaling Peptides and Proteins +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Velaglucerase alfa Approved DB06720
biotech | CAS: 884604-91-5

Velaglucerase alfa is a gene-activated human recombinant glucocerebrosidase used for the treatment of Type 1 Gaucher disease, caused by a deficiency of the lysosomal enzyme glucocerebrosidase. Additionally, Velaglucerase alfa has also been investigated for us…

Kategori:
Alimentary Tract and MetabolismEnzymesEnzymes and Coenzymes +1
Target Protein:
Lysosomal acid glucosylceramidase
Waktu Paruh11-12 minutes.
Vol. DistribusiThe mean volume of …
KlirensMean clearance rang…
Genetik -
Veligrotug DB18976
biotech | CAS: 2728655-31-8

Veligrotug is under investigation in clinical trial NCT00791544 (Dose Finding Study of AVE1642 in Patients With Advanced or Metastatic Liver Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Velmanase alfa Approved DB12374
biotech | CAS: 1492823-75-2

Velmanase alfa is a recombinant human lysosomal alpha-mannosidase developed for enzyme replacement therapy to treat alpha-mannosidosis. Alpha-mannosidosis is a rare autosomal recessive lysosomal storage disorder. Patients with alpha-mannosidosis have a geneti…

Kategori:
Alimentary Tract and MetabolismEnzyme Replacement TherapyEnzymes +2
Waktu ParuhAt the end of intra…
Vol. DistribusiThe steady-state vo…
KlirensThe mean clearance …
Genetik -
Vemurafenib Approved DB08881
small molecule | CAS: 918504-65-1

Vemurafenib is a competitive kinase inhibitor with activity against BRAF kinase with mutations like V600E.[A31269] It exerts its function by binding to the ATP-binding domain of the mutant BRAF.[A31270] Vemurafenib was co-developed by Roche and Plexxikon and …

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +41
Target Protein:
Serine/threonine-protein kinase B-raf
Waktu ParuhThe elimination hal…
Vol. DistribusiThe estimation of t…
KlirensThe total body clea…
Genetik -
Venlafaxine Approved DB00285
small molecule | CAS: 93413-69-5

Venlafaxine is an antidepressant and a serotonin and norepinephrine reuptake inhibitor (SNRI). Its active metabolite, [desvenlafaxine], works by blocking the reuptake of serotonin and norepinephrine, which are key neurotransmitters in mood regulation. Venlafa…

Kategori:
Agents producing tachycardiaAgents that reduce seizure thresholdAmines +39
Target Protein:
Sodium-dependent serotonin transporterSodium-dependent noradrenaline transporterSodium-dependent dopamine transporter
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +2
Waktu ParuhThe apparent elimin…
Vol. DistribusiThe apparent volume…
KlirensMean ± SD plasma ap…
Genetik 5 Varian
Vepdegestrant DB19006
small molecule | CAS: 2229711-68-4

Vepdegestrant is under investigation in clinical trial NCT05909397 (A Study of ARV-471 (PF-07850327) Plus Palbociclib Versus Letrozole Plus Palbociclib in Participants With Estrogen Receptor Positive, Human Epidermal Growth Factor Negative Advanced Breast Can…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vepsitamab DB18211
biotech | CAS: 2413453-53-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vericiguat Approved DB15456
small molecule | CAS: 1350653-20-1

Vericiguat is a direct stimulator of soluble guanylate cyclase (sGC) used in the management of systolic heart failure to reduce mortality and hospitalizations.[L31153] A key component of the NO-sGC-cGMP signaling pathway that helps to regulate the cardiovascu…

Kategori:
BCRP/ABCG2 SubstratesCardiac TherapyGuanylate Cyclase Stimulators +8
Target Protein:
Retinal guanylyl cyclase 1Guanylate cyclase soluble subunit beta-1
Waktu ParuhIn patients with he…
Vol. DistribusiIn healthy subjects…
KlirensVericiguat is a low…
Genetik -
biotech | CAS: 295371-00-5

Verpasep caltespen is a recombinant chimeric protein composed of the heat shock protein 65 (Hsp65) from _Mycobacterium bovis_, and the human papilloma viral (HPV) protein E7. Hsp65, similar to other members of its family of proteins, elicits a strong immune r…

Target Protein:
Keratin, type II cytoskeletal 7E3 ubiquitin-protein ligase UBR4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Vespula germanica venom protein is an extract of Vespula germanica venom. Vespula germanica venom protein is used in allergenic testing.

Kategori:
Bee and Wasp VenomCell-mediated ImmunityIncreased Histamine Release +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vestronidase alfa Approved DB12366
biotech | CAS: 1638194-78-1

Vestronidase alfa, or vestronidase alfa-vjbk, is a recombinant human lysosomal beta glucuronidase that is a purified enzyme produced by recombinant DNA technology in a Chinese hamster ovary cell line. The enzyme is a homotetramer consisted of 4 monomers with …

Kategori:
Alimentary Tract and MetabolismEnzymesEnzymes and Coenzymes +3
Waktu ParuhAfter repeated dosi…
Vol. DistribusiAfter repeated dosi…
KlirensAfter repeated dosi…
Genetik -
VG161 DB18469
biotech

VG161 is an oncolytic virus therapy under investigation for the treatment of cholangiocarcinoma.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
VGB-R04 DB18615
biotech

VGB-R04 is an adeno-associated viral vector delivering human FIX Padua gene.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Vicriviroc DB06652
small molecule | CAS: 306296-47-9

Vicriviroc, also known as SCH 417690 and SCH-D, is currently in clinical trials for the management of HIV-1. This pyrimidine based drug inhibits the interaction of HIV-1 with CCR5, preventing viral entry into cells. This drug was developed by Schering-Plough.

Kategori:
Cytochrome P-450 CYP2C9 SubstratesCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +2
Target Protein:
C-C chemokine receptor type 5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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